Compile Data Set for Download or QSAR
maximum 50k data
Found 161 with Last Name = 'scribner' and Initial = 'a'
TargetcGMP-dependent protein kinase(Eimeria tenella)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50210476((2,5-difluorobenzyl)-{4-[7-dimethylaminomethyl-2-(...)
Affinity DataIC50:  0.0260nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinase by Ten_K assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50182369(4-(2-(4-fluorophenyl)-7-(1-methylpiperidin-4-yl)H-...)
Affinity DataIC50:  0.0400nMAssay Description:Inhibitory activity against PKGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50182369(4-(2-(4-fluorophenyl)-7-(1-methylpiperidin-4-yl)H-...)
Affinity DataIC50:  0.0440nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50265424(2-{4-[3-(2-Aminopyrimidin-4-yl)-2-(4-fluorophenyl)...)
Affinity DataIC50:  0.0440nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50182369(4-(2-(4-fluorophenyl)-7-(1-methylpiperidin-4-yl)H-...)
Affinity DataIC50:  0.0440nMAssay Description:Inhibition of Eimeria tenella parasite-specific cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50182367(4-(2-(4-fluorophenyl)-7-(piperidin-4-yl)H-imidazo[...)
Affinity DataIC50:  0.0460nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50182367(4-(2-(4-fluorophenyl)-7-(piperidin-4-yl)H-imidazo[...)
Affinity DataIC50:  0.0500nMAssay Description:Inhibitory activity against PKGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50210490((2-chlorobenzyl)-{4-[7-dimethylaminomethyl-2-(4-fl...)
Affinity DataIC50:  0.0560nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinase by Ten_K assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50210473((3,4-difluorobenzyl)-{4-[7-dimethylaminomethyl-2-(...)
Affinity DataIC50:  0.0600nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinase by Ten_K assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50210479((2,6-difluorobenzyl)-{4-[7-dimethylaminomethyl-2-(...)
Affinity DataIC50:  0.0600nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinase by Ten_K assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50210495(CHEMBL251184 | cyclopropylmethyl{4-[7-dimethylamin...)
Affinity DataIC50:  0.0640nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinase by Ten_K assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50265419(4-[7-(1-Dimethylaminobutyl)-2-(4-fluorophenyl)imid...)
Affinity DataIC50:  0.0650nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50265425(2-{4-[3-(2-Aminopyrimidin-4-yl)-2-(4-fluorophenyl)...)
Affinity DataIC50:  0.0650nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50210517(CHEMBL249527 | {4-[7-dimethylaminomethyl-2-(4-fluo...)
Affinity DataIC50:  0.0660nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinase by Ten_K assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50265397(4-[7-(1-Dimethylaminoethyl)-2-(4-fluorophenyl)imid...)
Affinity DataIC50:  0.0670nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50265397(4-[7-(1-Dimethylaminoethyl)-2-(4-fluorophenyl)imid...)
Affinity DataIC50:  0.0670nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50265430(4-[2-(4-Fluorophenyl)-7-(1-phenethylpiperidin-4-yl...)
Affinity DataIC50:  0.0700nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50210508(CHEMBL250791 | cyclopropyl{4-[7-dimethylaminomethy...)
Affinity DataIC50:  0.0800nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinase by Ten_K assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50210494(CHEMBL250601 | {4-[7-dimethylaminomethyl-2-(4-fluo...)
Affinity DataIC50:  0.0800nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinase by Ten_K assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50182359(CHEMBL379059 | N-benzyl-4-(7-((dimethylamino)methy...)
Affinity DataIC50:  0.0810nMAssay Description:Inhibitory activity against PKGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50210489(CHEMBL249526 | {4-[7-dimethylaminomethyl-2-(4-fluo...)
Affinity DataIC50:  0.0830nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinase by Ten_K assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50210493(CHEMBL401102 | {4-[7-dimethylaminomethyl-2-(4-fluo...)
Affinity DataIC50:  0.0870nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinase by Ten_K assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50210478(CHEMBL249326 | {4-[7-dimethylaminomethyl-2-(4-fluo...)
Affinity DataIC50:  0.0900nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinase by Ten_K assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50265427(4-[7-(1-Cyclopropylmethylpiperidin-4-yl)-2-(4-fluo...)
Affinity DataIC50:  0.0950nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50210511(4-[2-(2,4-difluorophenyl)-7-dimethylaminomethylimi...)
Affinity DataIC50:  0.100nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinase by Ten_K assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50210500(CHEMBL251589 | {4-[7-dimethylaminomethyl-2-(4-fluo...)
Affinity DataIC50:  0.100nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinase by Ten_K assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50248496(2-(4-(2-(4-fluorophenyl)-3-(pyridin-4-yl)-1H-indol...)
Affinity DataIC50:  0.100nMAssay Description:Inhibition of Eimeria tenella parasite-specific cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50210514(CHEMBL399257 | cyclopentyl{4-[7-dimethylaminomethy...)
Affinity DataIC50:  0.102nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinase by Ten_K assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50265421(4-[7-(1-Dimethylamino-1-methyl-ethyl)-2-(4-fluorop...)
Affinity DataIC50:  0.110nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50182362(4-(7-((dimethylamino)methyl)-2-(4-fluorophenyl)H-i...)
Affinity DataIC50:  0.110nMAssay Description:Inhibitory activity against PKGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50182362(4-(7-((dimethylamino)methyl)-2-(4-fluorophenyl)H-i...)
Affinity DataIC50:  0.110nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50210486((3,5-difluorobenzyl)-{4-[7-dimethylaminomethyl-2-(...)
Affinity DataIC50:  0.110nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinase by Ten_K assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50265402(4-[7-[1-(3,3-Dimethylbutyl)piperidin-4-yl)-2-(4-fl...)
Affinity DataIC50:  0.110nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50265429(4-[7-(1-Benzylpiperidin-4-yl)-2-(4-fluorophenyl)-i...)
Affinity DataIC50:  0.110nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50265404(4-(7-(1-ethylpiperidin-4-yl)-2-(4-fluorophenyl)imi...)
Affinity DataIC50:  0.110nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50210505(CHEMBL399258 | cyclohexyl-{4-[7-dimethylaminomethy...)
Affinity DataIC50:  0.120nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinase by Ten_K assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50210488((2,3-difluorobenzyl)-{4-[7-dimethylaminomethyl-2-(...)
Affinity DataIC50:  0.120nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinase by Ten_K assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50265403(4-{2-(4-Fluorophenyl)-7-[1-(2-methylpentyl)piperid...)
Affinity DataIC50:  0.120nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50265426(4-[2-(4-Fluorophenyl)-7-(1-isobutylpiperidin-4-yl)...)
Affinity DataIC50:  0.120nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50210482(CHEMBL398887 | {4-[7-dimethylaminomethyl-2-(4-fluo...)
Affinity DataIC50:  0.121nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinase by Ten_K assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50182355(4-(7-((dimethylamino)methyl)-2-(4-fluorophenyl)H-i...)
Affinity DataIC50:  0.130nMAssay Description:Inhibitory activity against PKGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50210499(CHEMBL400896 | {4-[7-dimethylaminomethyl-2-(4-fluo...)
Affinity DataIC50:  0.130nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinase by Ten_K assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50182355(4-(7-((dimethylamino)methyl)-2-(4-fluorophenyl)H-i...)
Affinity DataIC50:  0.130nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinase by Ten_K assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50265428(4-[2-(4-Fluorophenyl)-7-(1-hexylpiperidin-4-yl)-im...)
Affinity DataIC50:  0.130nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50265401(4-{2-(4-Fluorophenyl)-7-[1-(2-methylbutyl)piperidi...)
Affinity DataIC50:  0.130nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50265398(4-[7-(1-Dimethylaminopropyl)-2-(4-fluorophenyl)-im...)
Affinity DataIC50:  0.130nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50265420(4-[7-(1-Amino-1-methyl-ethyl)-2-(4-fluorophenyl)-i...)
Affinity DataIC50:  0.145nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50182361(4-(7-((dimethylamino)methyl)-2-(4-fluorophenyl)H-i...)
Affinity DataIC50:  0.150nMAssay Description:Inhibitory activity against PKGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50248451(2-(4-fluorophenyl)-6-(1-methylpiperidin-4-yl)-3-(p...)
Affinity DataIC50:  0.150nMAssay Description:Inhibition of Eimeria tenella parasite-specific cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50248450(2-(4-fluorophenyl)-6-(piperidin-4-yl)-3-(pyridin-4...)
Affinity DataIC50:  0.150nMAssay Description:Inhibition of Eimeria tenella parasite-specific cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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