Affinity DataIC50: 7nMAssay Description:Displacement of [3H]WIN35428 from human DAT transfected cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 7.20nMAssay Description:Displacement of [3H]WIN35428 from human DAT transfected cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Displacement of [3H]WIN35428 from human DAT transfected cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Displacement of [3H]WIN35428 from human DAT transfected cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:Displacement of [3H]WIN35428 from human DAT transfected cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 32.7nMAssay Description:Displacement of [3H]WIN35428 from human DAT transfected cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of mouse full length GST-tagged BRAF V600E mutant using recombinant human His6-tagged MEK1 as substrate preincubated for 1 hr followed by ...More data for this Ligand-Target Pair
Affinity DataIC50: 43.5nMAssay Description:Displacement of [3H]WIN35428 from human DAT transfected cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 46.6nMAssay Description:Displacement of [3H]WIN35428 from human DAT transfected cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 49nMAssay Description:Displacement of [3H]WIN35428 from human DAT transfected cell membraneMore data for this Ligand-Target Pair
TargetCysteine proteinase falcipain 3(Plasmodium falciparum)
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataIC50: 60nMAssay Description:Inhibition of Plasmodium falciparum cysteine protease falcipain-3More data for this Ligand-Target Pair
Affinity DataIC50: 65nMAssay Description:Displacement of [3H]WIN35428 from human DAT transfected cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 66.5nMAssay Description:Displacement of [3H]WIN35428 from human DAT transfected cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 69.2nMAssay Description:Displacement of [3H]WIN35428 from human DAT transfected cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:Inhibition of His6-tagged recombinant EGFR cytoplasmic domain (645 to 1186 residues) (unknown origin) expressed in baculovirus infected Sf9 insect ce...More data for this Ligand-Target Pair
TargetCysteine proteinase falcipain 2a(Plasmodium falciparum)
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataIC50: 80nMAssay Description:Inhibition of Plasmodium falciparum cysteine protease falcipain-2More data for this Ligand-Target Pair
Affinity DataIC50: 101nMAssay Description:Displacement of [3H]WIN35428 from human DAT transfected cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 126nMAssay Description:Displacement of [3H]WIN35428 from human DAT transfected cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:Displacement of [3H]WIN35428 from human DAT transfected cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 139nMAssay Description:Displacement of [3H]WIN35428 from human DAT transfected cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 155nMAssay Description:Displacement of [3H]WIN35428 from human DAT transfected cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 157nMAssay Description:Displacement of [3H]WIN35428 from human DAT transfected cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 238nMAssay Description:Displacement of [3H]WIN35428 from human DAT transfected cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 269nMAssay Description:Displacement of [3H]WIN35428 from human DAT transfected cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 332nMAssay Description:Displacement of [3H]WIN35428 from human DAT transfected cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 456nMAssay Description:Displacement of [3H]WIN35428 from human DAT transfected cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 497nMAssay Description:Displacement of [3H]WIN35428 from human DAT transfected cell membraneMore data for this Ligand-Target Pair
TargetCysteine proteinase falcipain 3(Plasmodium falciparum)
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataIC50: 520nMAssay Description:Inhibition of Plasmodium falciparum cysteine protease falcipain-3More data for this Ligand-Target Pair
TargetCysteine proteinase falcipain 3(Plasmodium falciparum)
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataIC50: 540nMAssay Description:Inhibition of Plasmodium falciparum cysteine protease falcipain-3More data for this Ligand-Target Pair
Affinity DataIC50: 540nMAssay Description:Displacement of [3H]citalopram from human SERT expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 670nMAssay Description:Displacement of [3H]WIN35428 from human DAT transfected cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 755nMAssay Description:Displacement of [3H]citalopram from human SERT expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 766nMAssay Description:Displacement of [3H]citalopram from human SERT expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
TargetCysteine proteinase falcipain 3(Plasmodium falciparum)
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataIC50: 910nMAssay Description:Inhibition of Plasmodium falciparum cysteine protease falcipain-3More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [3H]WIN35428 from human DAT transfected cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [3H]citalopram from human SERT expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [3H]WIN35428 from human DAT transfected cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [3H]citalopram from human SERT expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
TargetCysteine proteinase falcipain 2a(Plasmodium falciparum)
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of Plasmodium falciparum cysteine protease falcipain-2More data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of His6-tagged recombinant EGFR cytoplasmic domain (645 to 1186 residues) (unknown origin) expressed in baculovirus infected Sf9 insect ce...More data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of His6-tagged recombinant EGFR cytoplasmic domain (645 to 1186 residues) (unknown origin) expressed in baculovirus infected Sf9 insect ce...More data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+3nMAssay Description:Displacement of [3H]citalopram from human SERT expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+3nMAssay Description:Displacement of [3H]WIN35428 from human DAT transfected cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+3nMAssay Description:Displacement of [3H]WIN35428 from human DAT transfected cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of His6-tagged recombinant EGFR cytoplasmic domain (645 to 1186 residues) (unknown origin) expressed in baculovirus infected Sf9 insect ce...More data for this Ligand-Target Pair
TargetCysteine proteinase falcipain 2a(Plasmodium falciparum)
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataIC50: 3.25E+3nMAssay Description:Inhibition of Plasmodium falciparum cysteine protease falcipain-2More data for this Ligand-Target Pair
TargetCysteine proteinase falcipain 3(Plasmodium falciparum)
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataIC50: 3.56E+3nMAssay Description:Inhibition of Plasmodium falciparum cysteine protease falcipain-3More data for this Ligand-Target Pair
Affinity DataIC50: >4.00E+3nMAssay Description:Displacement of [3H]citalopram from human SERT expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
TargetCysteine proteinase falcipain 2a(Plasmodium falciparum)
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataIC50: 4.42E+3nMAssay Description:Inhibition of Plasmodium falciparum cysteine protease falcipain-2More data for this Ligand-Target Pair
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition of mouse full length GST-tagged BRAF V600E mutant using recombinant human His6-tagged MEK1 as substrate preincubated for 1 hr followed by ...More data for this Ligand-Target Pair