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Found 127 with Last Name = 'sheri' and Initial = 'a'
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50334386(2beta-(3-Methylisoxazol-5-yl)-3beta-(4-fluoropheny...)
Affinity DataIC50:  7nMAssay Description:Displacement of [3H]WIN35428 from human DAT transfected cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50334387(2beta-(4-Methylisoxazol-5-yl)-3beta-(4-chloropheny...)
Affinity DataIC50:  7.20nMAssay Description:Displacement of [3H]WIN35428 from human DAT transfected cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50334385(2beta-(3-Methylisoxazol-5-yl)-3beta-Phenyl-8-thiab...)
Affinity DataIC50:  12nMAssay Description:Displacement of [3H]WIN35428 from human DAT transfected cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50334388(2beta-(4-Methylisoxazol-5-yl)-3beta-(4-bromophenyl...)
Affinity DataIC50:  14nMAssay Description:Displacement of [3H]WIN35428 from human DAT transfected cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50334376(2beta-(3-Methylisoxazol-5-yl)-3alpha-(4-fluorophen...)
Affinity DataIC50:  22nMAssay Description:Displacement of [3H]WIN35428 from human DAT transfected cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50334377(2beta-(3-Methylisoxazol-5-yl)-3alpha-(4-chlorophen...)
Affinity DataIC50:  32.7nMAssay Description:Displacement of [3H]WIN35428 from human DAT transfected cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Mus musculus)
Nahda University

Curated by ChEMBL
LigandPNGBDBM5446(CHEMBL553 | ERLOTINIB HYDROCHLORIDE | Erlotinib | ...)
Affinity DataIC50:  40nMAssay Description:Inhibition of mouse full length GST-tagged BRAF V600E mutant using recombinant human His6-tagged MEK1 as substrate preincubated for 1 hr followed by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50334389(2beta-(4-Methylisoxazol-5-yl)-3beta-(3,4-dichlorop...)
Affinity DataIC50:  43.5nMAssay Description:Displacement of [3H]WIN35428 from human DAT transfected cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50334378(2beta-(3-Methylisoxazol-5-yl)-3alpha-(4-bromopheny...)
Affinity DataIC50:  46.6nMAssay Description:Displacement of [3H]WIN35428 from human DAT transfected cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50334391(2beta-(3-Phenylisoxazol-5-yl)-3beta-(4-fluoropheny...)
Affinity DataIC50:  49nMAssay Description:Displacement of [3H]WIN35428 from human DAT transfected cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine proteinase falcipain 3(Plasmodium falciparum)
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50448248(CHEMBL3120847)
Affinity DataIC50:  60nMAssay Description:Inhibition of Plasmodium falciparum cysteine protease falcipain-3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50334375(2beta-(3-Methylisoxazol-5-yl)-3alpha-phenyl-8-thia...)
Affinity DataIC50:  65nMAssay Description:Displacement of [3H]WIN35428 from human DAT transfected cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50334399(2-(3-Phenylisoxazol-5-yl)-3-(4-chlorophenyl)-8-thi...)
Affinity DataIC50:  66.5nMAssay Description:Displacement of [3H]WIN35428 from human DAT transfected cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50334396(2-(3-Methylisoxazol-5-yl)-3-(3,4-dichlorophenyl)-8...)
Affinity DataIC50:  69.2nMAssay Description:Displacement of [3H]WIN35428 from human DAT transfected cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Nahda University

Curated by ChEMBL
LigandPNGBDBM5446(CHEMBL553 | ERLOTINIB HYDROCHLORIDE | Erlotinib | ...)
Affinity DataIC50:  70nMAssay Description:Inhibition of His6-tagged recombinant EGFR cytoplasmic domain (645 to 1186 residues) (unknown origin) expressed in baculovirus infected Sf9 insect ce...More data for this Ligand-Target Pair
TargetCysteine proteinase falcipain 2a(Plasmodium falciparum)
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50448248(CHEMBL3120847)
Affinity DataIC50:  80nMAssay Description:Inhibition of Plasmodium falciparum cysteine protease falcipain-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50334379(2beta-(3-Methylisoxazol-5-yl)-3alpha-(3,4-dichloro...)
Affinity DataIC50:  101nMAssay Description:Displacement of [3H]WIN35428 from human DAT transfected cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50334400(2-(3-Phenylisoxazol-5-yl)-3-(4-bromophenyl)-8-thia...)
Affinity DataIC50:  126nMAssay Description:Displacement of [3H]WIN35428 from human DAT transfected cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50334382(2beta-(3-Phenylisoxazol-5-yl)-3alpha-(4-chlorophen...)
Affinity DataIC50:  130nMAssay Description:Displacement of [3H]WIN35428 from human DAT transfected cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50334395(2-(3-Methylisoxazol-5-yl)-3-(4-bromophenyl)-8-thia...)
Affinity DataIC50:  139nMAssay Description:Displacement of [3H]WIN35428 from human DAT transfected cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50334394(2-(3-Methylisoxazol-5-yl)-3-(4-chlorophenyl)-8-thi...)
Affinity DataIC50:  155nMAssay Description:Displacement of [3H]WIN35428 from human DAT transfected cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50334390(2beta-(3-Phenylisoxazol-5-yl)-3beta-phenyl-8-thiab...)
Affinity DataIC50:  157nMAssay Description:Displacement of [3H]WIN35428 from human DAT transfected cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50334383(2beta-(3-Phenylisoxazol-5-yl)-3alpha-(4-bromopheny...)
Affinity DataIC50:  238nMAssay Description:Displacement of [3H]WIN35428 from human DAT transfected cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50334392(2beta-(3-Phenylisoxazol-5-yl)-3beta-(3,4-dichlorop...)
Affinity DataIC50:  269nMAssay Description:Displacement of [3H]WIN35428 from human DAT transfected cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50334374(2-(3-Phenylisoxazol-5-yl)-3-(3,4-dichlorophenyl)-8...)
Affinity DataIC50:  332nMAssay Description:Displacement of [3H]WIN35428 from human DAT transfected cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50334381(2beta-(3-Phenylisoxazol-5-yl)-3alpha-(4-fluorophen...)
Affinity DataIC50:  456nMAssay Description:Displacement of [3H]WIN35428 from human DAT transfected cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50334384(2beta-(3-Phenylisoxazol-5-yl)-3alpha-(3,4-dichloro...)
Affinity DataIC50:  497nMAssay Description:Displacement of [3H]WIN35428 from human DAT transfected cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine proteinase falcipain 3(Plasmodium falciparum)
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50448247(CHEMBL3120848)
Affinity DataIC50:  520nMAssay Description:Inhibition of Plasmodium falciparum cysteine protease falcipain-3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine proteinase falcipain 3(Plasmodium falciparum)
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50448261(CHEMBL3120834)
Affinity DataIC50:  540nMAssay Description:Inhibition of Plasmodium falciparum cysteine protease falcipain-3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50084717((+)-(1R,2R,3S,5S)-methyl 3-(benzoyloxy)-8-methyl-8...)
Affinity DataIC50:  540nMAssay Description:Displacement of [3H]citalopram from human SERT expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50084717((+)-(1R,2R,3S,5S)-methyl 3-(benzoyloxy)-8-methyl-8...)
Affinity DataIC50:  670nMAssay Description:Displacement of [3H]WIN35428 from human DAT transfected cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50334388(2beta-(4-Methylisoxazol-5-yl)-3beta-(4-bromophenyl...)
Affinity DataIC50:  755nMAssay Description:Displacement of [3H]citalopram from human SERT expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50334389(2beta-(4-Methylisoxazol-5-yl)-3beta-(3,4-dichlorop...)
Affinity DataIC50:  766nMAssay Description:Displacement of [3H]citalopram from human SERT expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine proteinase falcipain 3(Plasmodium falciparum)
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50448260(CHEMBL3120835)
Affinity DataIC50:  910nMAssay Description:Inhibition of Plasmodium falciparum cysteine protease falcipain-3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50334380(2beta-(3-Phenylisoxazol-5-yl)-3alpha-phenyl-8-thia...)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [3H]WIN35428 from human DAT transfected cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50334386(2beta-(3-Methylisoxazol-5-yl)-3beta-(4-fluoropheny...)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [3H]citalopram from human SERT expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50334393(2-(3-Methylisoxazol-5-yl)-3-(4-fluorophenyl)-8-thi...)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [3H]WIN35428 from human DAT transfected cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50334387(2beta-(4-Methylisoxazol-5-yl)-3beta-(4-chloropheny...)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [3H]citalopram from human SERT expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine proteinase falcipain 2a(Plasmodium falciparum)
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50448247(CHEMBL3120848)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of Plasmodium falciparum cysteine protease falcipain-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Nahda University

Curated by ChEMBL
LigandPNGBDBM50468896(CHEMBL4279008)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of His6-tagged recombinant EGFR cytoplasmic domain (645 to 1186 residues) (unknown origin) expressed in baculovirus infected Sf9 insect ce...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Nahda University

Curated by ChEMBL
LigandPNGBDBM50468892(CHEMBL4289274)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of His6-tagged recombinant EGFR cytoplasmic domain (645 to 1186 residues) (unknown origin) expressed in baculovirus infected Sf9 insect ce...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50334379(2beta-(3-Methylisoxazol-5-yl)-3alpha-(3,4-dichloro...)
Affinity DataIC50: >2.00E+3nMAssay Description:Displacement of [3H]citalopram from human SERT expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50334398(2-(3-Phenylisoxazol-5-yl)-3-(4-fluorophenyl)-8-thi...)
Affinity DataIC50: >2.00E+3nMAssay Description:Displacement of [3H]WIN35428 from human DAT transfected cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50334373(2-(3-Methylisoxazol-5-yl)-3-phenyl-8-thiabicyclo[3...)
Affinity DataIC50: >2.00E+3nMAssay Description:Displacement of [3H]WIN35428 from human DAT transfected cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Nahda University

Curated by ChEMBL
LigandPNGBDBM50468891(CHEMBL4286943)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibition of His6-tagged recombinant EGFR cytoplasmic domain (645 to 1186 residues) (unknown origin) expressed in baculovirus infected Sf9 insect ce...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCysteine proteinase falcipain 2a(Plasmodium falciparum)
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50448253(CHEMBL3120842)
Affinity DataIC50:  3.25E+3nMAssay Description:Inhibition of Plasmodium falciparum cysteine protease falcipain-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine proteinase falcipain 3(Plasmodium falciparum)
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50448246(CHEMBL3120849)
Affinity DataIC50:  3.56E+3nMAssay Description:Inhibition of Plasmodium falciparum cysteine protease falcipain-3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50334378(2beta-(3-Methylisoxazol-5-yl)-3alpha-(4-bromopheny...)
Affinity DataIC50: >4.00E+3nMAssay Description:Displacement of [3H]citalopram from human SERT expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine proteinase falcipain 2a(Plasmodium falciparum)
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50448260(CHEMBL3120835)
Affinity DataIC50:  4.42E+3nMAssay Description:Inhibition of Plasmodium falciparum cysteine protease falcipain-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Mus musculus)
Nahda University

Curated by ChEMBL
LigandPNGBDBM50468896(CHEMBL4279008)
Affinity DataIC50:  4.70E+3nMAssay Description:Inhibition of mouse full length GST-tagged BRAF V600E mutant using recombinant human His6-tagged MEK1 as substrate preincubated for 1 hr followed by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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