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Found 167 with Last Name = 'spadaro' and Initial = 'a'
TargetMu-type opioid receptor(Homo sapiens (Human))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50534063(CHEMBL4575464)
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]DAMGO from MOR in HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50000296(CHEMBL441765 | CHEMBL482811 | U-50488H | US1149237...)
Affinity DataKi:  0.600nMAssay Description:Displacement of [3H]U69593 from rat KOR expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University of Catania

Curated by ChEMBL
LigandPNGBDBM21015((2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl...)
Affinity DataKi:  0.600nMAssay Description:Displacement of [3H]DAMGO from MOR in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50142692(CHEMBL3759092)
Affinity DataKi:  0.830nMAssay Description:Displacement of [3H]DAMGO from MOR in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University of Catania

Curated by ChEMBL
LigandPNGBDBM21008((4S,7S,13S)-13-[(2S)-2-amino-3-(4-hydroxyphenyl)pr...)
Affinity DataKi:  1.70nMAssay Description:Displacement of [3H]DPDPE from human DOR expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50534068(CHEMBL4466859)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]Diprenorphine from human MOR expressed in HEK293 cell membranes by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50142692(CHEMBL3759092)
Affinity DataKi:  29nMAssay Description:Displacement of [3H]DPDPE from human DOR expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50534064(CHEMBL4442357)
Affinity DataKi:  84nMAssay Description:Displacement of [3H]DAMGO from MOR in HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50534065(CHEMBL4545050)
Affinity DataKi:  96nMAssay Description:Displacement of [3H]DAMGO from MOR in HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50142692(CHEMBL3759092)
Affinity DataKi:  110nMAssay Description:Displacement of [3H]U69593 from rat KOR expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50534067(CHEMBL4453773)
Affinity DataKi:  160nMAssay Description:Displacement of [3H]DAMGO from MOR in HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50534063(CHEMBL4575464)
Affinity DataKi:  190nMAssay Description:Displacement of [3H]U69593 from rat KOR expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50534067(CHEMBL4453773)
Affinity DataKi:  370nMAssay Description:Displacement of [3H]U69593 from rat KOR expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50534066(CHEMBL4562025)
Affinity DataKi:  380nMAssay Description:Displacement of [3H]DAMGO from MOR in HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50534063(CHEMBL4575464)
Affinity DataKi:  440nMAssay Description:Displacement of [3H]DPDPE from human DOR expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50534062(CHEMBL4464491)
Affinity DataKi:  470nMAssay Description:Displacement of [3H]DAMGO from MOR in HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50534064(CHEMBL4442357)
Affinity DataKi:  680nMAssay Description:Displacement of [3H]U69593 from rat KOR expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50534066(CHEMBL4562025)
Affinity DataKi:  900nMAssay Description:Displacement of [3H]U69593 from rat KOR expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50534067(CHEMBL4453773)
Affinity DataKi:  1.40E+3nMAssay Description:Displacement of [3H]DPDPE from human DOR expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50534062(CHEMBL4464491)
Affinity DataKi:  1.90E+3nMAssay Description:Displacement of [3H]U69593 from rat KOR expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50534064(CHEMBL4442357)
Affinity DataKi:  2.90E+3nMAssay Description:Displacement of [3H]DPDPE from human DOR expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50534066(CHEMBL4562025)
Affinity DataKi:  2.90E+3nMAssay Description:Displacement of [3H]DPDPE from human DOR expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50534062(CHEMBL4464491)
Affinity DataKi:  7.90E+3nMAssay Description:Displacement of [3H]DPDPE from human DOR expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50534068(CHEMBL4466859)
Affinity DataKi: <1.00E+4nMAssay Description:Displacement of [3H]Diprenorphine from human KOR expressed in HEK293 cell membranes by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50396085(CHEMBL2170762)
Affinity DataIC50:  5nMAssay Description:Inhibition of human placenta 17beta-HSD1 cytosolic fraction using unlabelled and [2,4,6,7-3H]estrone as substrate after 10 mins by HPLC analysis in p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50299643(2-Fluoro-4-[5-(3-hydroxyphenyl)-2-thienyl]phenol |...)
Affinity DataIC50:  8nMAssay Description:Inhibition of human placental 17betaHSD1 by radiodetection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50396084(CHEMBL2170750)
Affinity DataIC50:  11nMAssay Description:Inhibition of 17beta-HSD1 in human T47D cells using unlabelled and [2,4,6,7-3H]estrone as substrate preincubated for 30 mins prior to substrate addit...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50396081(CHEMBL2170753)
Affinity DataIC50:  13nMAssay Description:Inhibition of human placenta 17beta-HSD1 cytosolic fraction using unlabelled and [2,4,6,7-3H]estrone as substrate after 10 mins by HPLC analysis in p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50396084(CHEMBL2170750)
Affinity DataIC50:  13nMAssay Description:Inhibition of human placenta 17beta-HSD1 cytosolic fraction using unlabelled and [2,4,6,7-3H]estrone as substrate after 10 mins by HPLC analysis in p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50396087(CHEMBL2170747)
Affinity DataIC50:  13nMAssay Description:Inhibition of human placenta 17beta-HSD1 cytosolic fraction using unlabelled and [2,4,6,7-3H]estrone as substrate after 10 mins by HPLC analysis in p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50299656(2-Fluoro-4-[5-(4-fluoro-3-hydroxyphenyl)thien-2-yl...)
Affinity DataIC50:  17nMAssay Description:Inhibition of human placental 17betaHSD1 by radiodetection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50396080(CHEMBL2170754)
Affinity DataIC50:  27nMAssay Description:Inhibition of human placenta 17beta-HSD1 cytosolic fraction using unlabelled and [2,4,6,7-3H]estrone as substrate after 10 mins by HPLC analysis in p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50396089(CHEMBL2170759)
Affinity DataIC50:  29nMAssay Description:Inhibition of human placenta 17beta-HSD1 cytosolic fraction using unlabelled and [2,4,6,7-3H]estrone as substrate after 10 mins by HPLC analysis in p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50299655(2-Fluoro-4-[5-(3-fluoro-5-hydroxyphenyl)thien-2-yl...)
Affinity DataIC50:  29nMAssay Description:Inhibition of human placental 17betaHSD1 by radiodetection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50396087(CHEMBL2170747)
Affinity DataIC50:  37nMAssay Description:Inhibition of 17beta-HSD1 in human T47D cells using unlabelled and [2,4,6,7-3H]estrone as substrate preincubated for 30 mins prior to substrate addit...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50396083(CHEMBL2170751)
Affinity DataIC50:  38nMAssay Description:Inhibition of human placenta 17beta-HSD1 cytosolic fraction using unlabelled and [2,4,6,7-3H]estrone as substrate after 10 mins by HPLC analysis in p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50299659(4-[5-(3-Hydroxyphenyl)-2-thienyl]-2-(trifluorometh...)
Affinity DataIC50:  38nMAssay Description:Inhibition of human placental 17betaHSD1 by radiodetection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50299651(3-Fluoro-5-[5-(4-hydroxyphenyl)-2-thienyl]phenol |...)
Affinity DataIC50:  42nMAssay Description:Inhibition of human placental 17betaHSD1 by radiodetection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50396086(CHEMBL2170761)
Affinity DataIC50:  44nMAssay Description:Inhibition of human placenta 17beta-HSD1 cytosolic fraction using unlabelled and [2,4,6,7-3H]estrone as substrate after 10 mins by HPLC analysis in p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50299633(4-[5-(3-Hydroxyphenyl)-2-thienyl)-2-methyl]phenol ...)
Affinity DataIC50:  46nMAssay Description:Inhibition of human placental 17betaHSD1 by radiodetection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM25831(4-[2-(3-hydroxyphenyl)-1,3-thiazol-5-yl]phenol | h...)
Affinity DataIC50:  50nMAssay Description:Inhibition of human placental 17betaHSD1 by radiodetection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50299654(4-Fluoro-1,1':4',1''-terphenyl-3,3''-diol | CHEMBL...)
Affinity DataIC50:  51nMAssay Description:Inhibition of human placental 17betaHSD1 by radiodetection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50299653(2,6-Difluoro-4-[5-(3-hydroxyphenyl)-2-thienyl]phen...)
Affinity DataIC50:  56nMAssay Description:Inhibition of human placental 17betaHSD1 by radiodetection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 2(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50396083(CHEMBL2170751)
Affinity DataIC50:  59nMAssay Description:Inhibition of human placenta 17beta-HSD2 microsomal fraction using unlabelled and [2,4,6,7-3H]estradiol as substrate after 20 mins by HPLC analysis i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50299645(4-[5-(3-Hydroxyphenyl)-3-thienyl]-2-methylphenol |...)
Affinity DataIC50:  64nMAssay Description:Inhibition of human placental 17betaHSD1 by radiodetection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50299647(2-Fluoro-4-[5-(3-hydroxyphenyl)-3-thienyl]phenol |...)
Affinity DataIC50:  64nMAssay Description:Inhibition of human placental 17betaHSD1 by radiodetection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM25850(3-[5-(4-hydroxyphenyl)thiophen-2-yl]phenol | hydro...)
Affinity DataIC50:  69nMAssay Description:Inhibition of human placental 17betaHSD1 by radiodetection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50396089(CHEMBL2170759)
Affinity DataIC50:  73nMAssay Description:Inhibition of 17beta-HSD1 in human T47D cells using unlabelled and [2,4,6,7-3H]estrone as substrate preincubated for 30 mins prior to substrate addit...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM25855(3-[4-(4-hydroxyphenyl)thiophen-2-yl]phenol | hydro...)
Affinity DataIC50:  77nMAssay Description:Inhibition of human placental 17betaHSD1 by radiodetection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50396079(CHEMBL2170755)
Affinity DataIC50:  78nMAssay Description:Inhibition of human placenta 17beta-HSD1 cytosolic fraction using unlabelled and [2,4,6,7-3H]estrone as substrate after 10 mins by HPLC analysis in p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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