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Found 63 with Last Name = 'xiao' and Initial = 'a'
TargetDiphosphomevalonate decarboxylase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287714((3R)-3-(fluoromethyl)-3-hydroxy-5-{[(phosphonatoox...)
Affinity DataKi:  37nMAssay Description:Compound was evaluated for its inhibitory activity against Mevalonate 5-pyrophosphate decarboxylaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDiphosphomevalonate decarboxylase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287713([methyl(2-{[(phosphonatooxy)phosphinato]oxy}ethyl)...)
Affinity DataKi:  750nMAssay Description:Compound was evaluated for its inhibitory activity against Mevalonate 5-pyrophosphate decarboxylaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDiphosphomevalonate decarboxylase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287710((2S)-1-({[(phosphonatooxy)phosphinato]oxy}acetyl)p...)
Affinity DataIC50:  9nMAssay Description:Compound was evaluated for its inhibitory activity against Mevalonate 5-pyrophosphate decarboxylaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDiphosphomevalonate decarboxylase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287715((2R)-1-({[(phosphonatooxy)phosphinato]oxy}acetyl)p...)
Affinity DataIC50:  15nMAssay Description:Compound was evaluated for its inhibitory activity against Mevalonate 5-pyrophosphate decarboxylaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDiphosphomevalonate decarboxylase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287715((2R)-1-({[(phosphonatooxy)phosphinato]oxy}acetyl)p...)
Affinity DataIC50:  15nMAssay Description:Compound was evaluated for its inhibitory activity against MevPP decarboxylaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50016496(CHEMBL3260241)
Affinity DataIC50:  30nMAssay Description:Inhibition of PLK1 (unknown origin) using RRRDELMEASFADQEAKV as substrate after 20 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50016508(CHEMBL3260249)
Affinity DataIC50:  90nMAssay Description:Inhibition of PLK1 (unknown origin) using RRRDELMEASFADQEAKV as substrate after 20 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50016502(CHEMBL3260248)
Affinity DataIC50:  120nMAssay Description:Inhibition of PLK1 (unknown origin) using RRRDELMEASFADQEAKV as substrate after 20 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiphosphomevalonate decarboxylase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287712([(2-{[(phosphonatooxy)phosphinato]oxy}ethyl)thio]a...)
Affinity DataIC50:  150nMAssay Description:Compound was evaluated for its inhibitory activity against Mevalonate 5-pyrophosphate decarboxylaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50016495(CHEMBL3260236)
Affinity DataIC50:  190nMAssay Description:Inhibition of PLK1 (unknown origin) using RRRDELMEASFADQEAKV as substrate after 20 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50016501(CHEMBL3260247)
Affinity DataIC50:  190nMAssay Description:Inhibition of PLK1 (unknown origin) using RRRDELMEASFADQEAKV as substrate after 20 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiphosphomevalonate decarboxylase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287711([methyl({[(phosphonatooxy)phosphinato]oxy}acetyl)a...)
Affinity DataIC50:  300nMAssay Description:Compound was evaluated for its inhibitory activity against MevPP decarboxylaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50016498(CHEMBL3260243)
Affinity DataIC50:  590nMAssay Description:Inhibition of PLK1 (unknown origin) using RRRDELMEASFADQEAKV as substrate after 20 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50016500(CHEMBL3260246)
Affinity DataIC50:  1.05E+3nMAssay Description:Inhibition of PLK1 (unknown origin) using RRRDELMEASFADQEAKV as substrate after 20 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50016499(CHEMBL3260244)
Affinity DataIC50:  1.55E+3nMAssay Description:Inhibition of PLK1 (unknown origin) using RRRDELMEASFADQEAKV as substrate after 20 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50016497(CHEMBL3260242)
Affinity DataIC50:  1.55E+3nMAssay Description:Inhibition of PLK1 (unknown origin) using RRRDELMEASFADQEAKV as substrate after 20 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50016509(CHEMBL3260250)
Affinity DataIC50:  2.31E+3nMAssay Description:Inhibition of PLK1 (unknown origin) using RRRDELMEASFADQEAKV as substrate after 20 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50423984(CHEMBL2313419)
Affinity DataIC50:  8.40E+3nMAssay Description:Inhibition of PTP1B (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSialidase(Vibrio cholerae)
University of California-Davis

Curated by ChEMBL
LigandPNGBDBM4706((2R,3R,4S)-3-acetamido-4-hydroxy-2-[(1R,2R)-1,2,3-...)
Affinity DataIC50:  8.60E+3nMAssay Description:Inhibition of Vibrio cholerae sialidase using Neu5Acalpha2-3GalbetapNP as substrate after 30 mins by colorimetric assayMore data for this Ligand-Target Pair
TargetSialidase A(Streptococcus pneumoniae)
University of California-Davis

Curated by ChEMBL
LigandPNGBDBM4706((2R,3R,4S)-3-acetamido-4-hydroxy-2-[(1R,2R)-1,2,3-...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of Streptococcus pneumoniae NanA using Neu5Acalpha2-3GalbetapNP as substrate after 30 mins by colorimetric assayMore data for this Ligand-Target Pair
TargetSialidase(Vibrio cholerae)
University of California-Davis

Curated by ChEMBL
LigandPNGBDBM50466472(CHEMBL4289476)
Affinity DataIC50:  1.09E+4nMAssay Description:Inhibition of Vibrio cholerae sialidase using Neu5Acalpha2-3GalbetapNP as substrate after 30 mins by colorimetric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50423983(CHEMBL2313420)
Affinity DataIC50:  1.31E+4nMAssay Description:Inhibition of PTP1B (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSialidase(Vibrio cholerae)
University of California-Davis

Curated by ChEMBL
LigandPNGBDBM50466474(CHEMBL4282280)
Affinity DataIC50:  1.35E+4nMAssay Description:Inhibition of Vibrio cholerae sialidase using Neu5Acalpha2-3GalbetapNP as substrate after 30 mins by colorimetric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50423991(CHEMBL2313414)
Affinity DataIC50:  1.52E+4nMAssay Description:Inhibition of PTP1B (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSialidase-2(Homo sapiens (Human))
University of California-Davis

Curated by ChEMBL
LigandPNGBDBM4706((2R,3R,4S)-3-acetamido-4-hydroxy-2-[(1R,2R)-1,2,3-...)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibition of recombinant human cytosolic sialidase NEU2 using Neu5Acalpha2-3GalbetapNP as substrate after 30 mins by colorimetric assayMore data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50423982(GYPENSAPOGENIN A)
Affinity DataIC50:  1.97E+4nMAssay Description:Inhibition of PTP1B (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSialidase(Vibrio cholerae)
University of California-Davis

Curated by ChEMBL
LigandPNGBDBM50331692((2R,3R,4S)-3-acetamido-2-((1R,2R)-3-azido-1,2-dihy...)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of Vibrio cholerae sialidase using Neu5Acalpha2-3GalbetapNP as substrate after 30 mins by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSialidase(Clostridium perfringens)
University of California-Davis

Curated by ChEMBL
LigandPNGBDBM4706((2R,3R,4S)-3-acetamido-4-hydroxy-2-[(1R,2R)-1,2,3-...)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of Clostridium perfringens sialidase using Neu5Acalpha2-3GalbetapNP as substrate after 30 mins by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50115732(CHEMBL294467 | Sodium vanadate)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibition of PTP1B (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50423994(CHEMBL2313421 | Gypensapogenin E)
Affinity DataIC50:  2.30E+4nMAssay Description:Inhibition of PTP1B (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50423990(20(S)-Protopanaxadiol | CHEMBL375563)
Affinity DataIC50:  2.36E+4nMAssay Description:Inhibition of PTP1B (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50423981(GYPENSAPOGENIN B)
Affinity DataIC50:  2.45E+4nMAssay Description:Inhibition of PTP1B (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50423992(CHEMBL2313423 | Gypensapogenin G)
Affinity DataIC50:  2.45E+4nMAssay Description:Inhibition of PTP1B (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50423985(CHEMBL2313418)
Affinity DataIC50:  2.78E+4nMAssay Description:Inhibition of PTP1B (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSialidase(Vibrio cholerae)
University of California-Davis

Curated by ChEMBL
LigandPNGBDBM50466473(CHEMBL4278803)
Affinity DataIC50:  2.89E+4nMAssay Description:Inhibition of Vibrio cholerae sialidase using Neu5Acalpha2-3GalbetapNP as substrate after 30 mins by colorimetric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSialidase A(Streptococcus pneumoniae)
University of California-Davis

Curated by ChEMBL
LigandPNGBDBM50331692((2R,3R,4S)-3-acetamido-2-((1R,2R)-3-azido-1,2-dihy...)
Affinity DataIC50:  4.43E+4nMAssay Description:Inhibition of Streptococcus pneumoniae NanA using Neu5Acalpha2-3GalbetapNP as substrate after 30 mins by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50423993(CHEMBL2313422 | Gypensapogenin F)
Affinity DataIC50:  4.90E+4nMAssay Description:Inhibition of PTP1B (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50423980(GYPENSAPOGENIN C)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of PTP1B (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50423989(CHEMBL2313415)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of PTP1B (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50423988(CHEMBL2313416)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of PTP1B (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50423986(GYPENSAPOGENIN D)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of PTP1B (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50423987(CHEMBL2313417)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of PTP1B (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSialidase(Clostridium perfringens)
University of California-Davis

Curated by ChEMBL
LigandPNGBDBM50331692((2R,3R,4S)-3-acetamido-2-((1R,2R)-3-azido-1,2-dihy...)
Affinity DataIC50:  5.90E+4nMAssay Description:Inhibition of Clostridium perfringens sialidase using Neu5Acalpha2-3GalbetapNP as substrate after 30 mins by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSialidase A(Streptococcus pneumoniae)
University of California-Davis

Curated by ChEMBL
LigandPNGBDBM50466472(CHEMBL4289476)
Affinity DataIC50:  6.56E+4nMAssay Description:Inhibition of Streptococcus pneumoniae NanA using Neu5Acalpha2-3GalbetapNP as substrate after 30 mins by colorimetric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSialidase(Clostridium perfringens)
University of California-Davis

Curated by ChEMBL
LigandPNGBDBM50466474(CHEMBL4282280)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibition of Clostridium perfringens sialidase using Neu5Acalpha2-3GalbetapNP as substrate after 30 mins by colorimetric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSialidase(Clostridium perfringens)
University of California-Davis

Curated by ChEMBL
LigandPNGBDBM50466472(CHEMBL4289476)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibition of Clostridium perfringens sialidase using Neu5Acalpha2-3GalbetapNP as substrate after 30 mins by colorimetric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSialidase(Clostridium perfringens)
University of California-Davis

Curated by ChEMBL
LigandPNGBDBM50466473(CHEMBL4278803)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibition of Clostridium perfringens sialidase using Neu5Acalpha2-3GalbetapNP as substrate after 30 mins by colorimetric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSialidase A(Streptococcus pneumoniae)
University of California-Davis

Curated by ChEMBL
LigandPNGBDBM50466474(CHEMBL4282280)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibition of Streptococcus pneumoniae NanA using Neu5Acalpha2-3GalbetapNP as substrate after 30 mins by colorimetric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSialidase-2(Homo sapiens (Human))
University of California-Davis

Curated by ChEMBL
LigandPNGBDBM50331692((2R,3R,4S)-3-acetamido-2-((1R,2R)-3-azido-1,2-dihy...)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibition of recombinant human cytosolic sialidase NEU2 using Neu5Acalpha2-3GalbetapNP as substrate after 30 mins by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSialidase A(Streptococcus pneumoniae)
University of California-Davis

Curated by ChEMBL
LigandPNGBDBM50466473(CHEMBL4278803)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibition of Streptococcus pneumoniae NanA using Neu5Acalpha2-3GalbetapNP as substrate after 30 mins by colorimetric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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