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Found 679 with Last Name = 'joshi' and Initial = 'aa'
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50485121(CHEMBL2030954)
Affinity DataKi:  0.400nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli using DABCYL-Abu-Ser-Gln-ASN-Tyr-Pro-Ile-Val-Gln-EDANS as substrate preincubated for 20 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50485126(CHEMBL2030953)
Affinity DataKi:  0.700nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli using DABCYL-Abu-Ser-Gln-ASN-Tyr-Pro-Ile-Val-Gln-EDANS as substrate preincubated for 20 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50485120(CHEMBL2030952)
Affinity DataKi:  0.800nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli using DABCYL-Abu-Ser-Gln-ASN-Tyr-Pro-Ile-Val-Gln-EDANS as substrate preincubated for 20 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50485130(CHEMBL2031103)
Affinity DataKi:  0.800nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli using DABCYL-Abu-Ser-Gln-ASN-Tyr-Pro-Ile-Val-Gln-EDANS as substrate preincubated for 20 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50485118(CHEMBL2030950)
Affinity DataKi:  1.70nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli using DABCYL-Abu-Ser-Gln-ASN-Tyr-Pro-Ile-Val-Gln-EDANS as substrate preincubated for 20 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50485122(CHEMBL2030955)
Affinity DataKi:  1.70nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli using DABCYL-Abu-Ser-Gln-ASN-Tyr-Pro-Ile-Val-Gln-EDANS as substrate preincubated for 20 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50485119(CHEMBL2030951)
Affinity DataKi:  2nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli using DABCYL-Abu-Ser-Gln-ASN-Tyr-Pro-Ile-Val-Gln-EDANS as substrate preincubated for 20 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50485116(CHEMBL2030946)
Affinity DataKi:  2.10nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli using DABCYL-Abu-Ser-Gln-ASN-Tyr-Pro-Ile-Val-Gln-EDANS as substrate preincubated for 20 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM13934(Atazanavir | BMS 232632 | CGP 73547 | CHEMBL1163 |...)
Affinity DataKi:  2.70nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli using DABCYL-Abu-Ser-Gln-ASN-Tyr-Pro-Ile-Val-Gln-EDANS as substrate preincubated for 20 min...More data for this Ligand-Target Pair
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50485131(CHEMBL2031101)
Affinity DataKi:  4.20nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli using DABCYL-Abu-Ser-Gln-ASN-Tyr-Pro-Ile-Val-Gln-EDANS as substrate preincubated for 20 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50485124(CHEMBL2031100)
Affinity DataKi:  5.30nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli using DABCYL-Abu-Ser-Gln-ASN-Tyr-Pro-Ile-Val-Gln-EDANS as substrate preincubated for 20 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50485114(CHEMBL2031102)
Affinity DataKi:  6.30nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli using DABCYL-Abu-Ser-Gln-ASN-Tyr-Pro-Ile-Val-Gln-EDANS as substrate preincubated for 20 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50485129(CHEMBL2030949)
Affinity DataKi:  6.40nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli using DABCYL-Abu-Ser-Gln-ASN-Tyr-Pro-Ile-Val-Gln-EDANS as substrate preincubated for 20 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50485123(CHEMBL2031099)
Affinity DataKi:  12nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli using DABCYL-Abu-Ser-Gln-ASN-Tyr-Pro-Ile-Val-Gln-EDANS as substrate preincubated for 20 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50485128(CHEMBL2030956)
Affinity DataKi:  13nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli using DABCYL-Abu-Ser-Gln-ASN-Tyr-Pro-Ile-Val-Gln-EDANS as substrate preincubated for 20 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
The University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50133217(CHEMBL3634917)
Affinity DataKi:  29nMAssay Description:Displacement of [3H]diprenorphine from rat kappa-opioid receptor expressed in CHO cells after 90 mins by scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
The University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50133220(CHEMBL3634920)
Affinity DataKi:  44nMAssay Description:Displacement of [3H]diprenorphine from rat kappa-opioid receptor expressed in CHO cells after 90 mins by scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
The University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50133221(CHEMBL3634921)
Affinity DataKi:  62nMAssay Description:Displacement of [3H]diprenorphine from rat kappa-opioid receptor expressed in CHO cells after 90 mins by scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
The University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50133260(CHEMBL3634927)
Affinity DataKi:  69nMAssay Description:Displacement of [3H]diprenorphine from rat kappa-opioid receptor expressed in CHO cells after 90 mins by scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
The University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50012153(zyklophin)
Affinity DataKi:  95nMAssay Description:Displacement of [3H]diprenorphine from rat kappa-opioid receptor expressed in CHO cells after 90 mins by scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
The University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50133217(CHEMBL3634917)
Affinity DataKi:  157nMAssay Description:Displacement of [3H]DAMGO from rat mu-opioid receptor expressed in CHO cells after 90 mins by scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
The University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50133218(CHEMBL3634918)
Affinity DataKi:  160nMAssay Description:Displacement of [3H]diprenorphine from rat kappa-opioid receptor expressed in CHO cells after 90 mins by scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
The University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50133256(CHEMBL3632647)
Affinity DataKi:  168nMAssay Description:Displacement of [3H]diprenorphine from rat kappa-opioid receptor expressed in CHO cells after 90 mins by scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
The University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50133263(CHEMBL3634929)
Affinity DataKi:  222nMAssay Description:Displacement of [3H]diprenorphine from rat kappa-opioid receptor expressed in CHO cells after 90 mins by scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
The University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50133255(CHEMBL3634926)
Affinity DataKi:  293nMAssay Description:Displacement of [3H]diprenorphine from rat kappa-opioid receptor expressed in CHO cells after 90 mins by scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
The University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50133219(CHEMBL3634919)
Affinity DataKi:  326nMAssay Description:Displacement of [3H]diprenorphine from rat kappa-opioid receptor expressed in CHO cells after 90 mins by scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
The University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50133222(CHEMBL3634922)
Affinity DataKi:  346nMAssay Description:Displacement of [3H]diprenorphine from rat kappa-opioid receptor expressed in CHO cells after 90 mins by scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
The University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50133262(CHEMBL3634928)
Affinity DataKi:  403nMAssay Description:Displacement of [3H]diprenorphine from rat kappa-opioid receptor expressed in CHO cells after 90 mins by scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
The University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50133266(CHEMBL3634930)
Affinity DataKi:  410nMAssay Description:Displacement of [3H]diprenorphine from rat kappa-opioid receptor expressed in CHO cells after 90 mins by scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
The University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50133216(CHEMBL3634916)
Affinity DataKi:  412nMAssay Description:Displacement of [3H]diprenorphine from rat kappa-opioid receptor expressed in CHO cells after 90 mins by scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
The University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50133252(CHEMBL3634923)
Affinity DataKi:  516nMAssay Description:Displacement of [3H]diprenorphine from rat kappa-opioid receptor expressed in CHO cells after 90 mins by scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50485125(CHEMBL2030944)
Affinity DataKi:  760nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli using DABCYL-Abu-Ser-Gln-ASN-Tyr-Pro-Ile-Val-Gln-EDANS as substrate preincubated for 20 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50485115(CHEMBL2030945)
Affinity DataKi:  800nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli using DABCYL-Abu-Ser-Gln-ASN-Tyr-Pro-Ile-Val-Gln-EDANS as substrate preincubated for 20 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50485127(CHEMBL2030948)
Affinity DataKi:  940nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli using DABCYL-Abu-Ser-Gln-ASN-Tyr-Pro-Ile-Val-Gln-EDANS as substrate preincubated for 20 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50485117(CHEMBL2030947)
Affinity DataKi:  1.20E+3nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli using DABCYL-Abu-Ser-Gln-ASN-Tyr-Pro-Ile-Val-Gln-EDANS as substrate preincubated for 20 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
The University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50133218(CHEMBL3634918)
Affinity DataKi:  1.49E+3nMAssay Description:Displacement of [3H]DAMGO from rat mu-opioid receptor expressed in CHO cells after 90 mins by scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
The University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50133254(CHEMBL3634925)
Affinity DataKi:  1.75E+3nMAssay Description:Displacement of [3H]diprenorphine from rat kappa-opioid receptor expressed in CHO cells after 90 mins by scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
The University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50133216(CHEMBL3634916)
Affinity DataKi:  2.44E+3nMAssay Description:Displacement of [3H]DAMGO from rat mu-opioid receptor expressed in CHO cells after 90 mins by scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
The University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50133256(CHEMBL3632647)
Affinity DataKi:  2.55E+3nMAssay Description:Displacement of [3H]DAMGO from rat mu-opioid receptor expressed in CHO cells after 90 mins by scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
The University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50133266(CHEMBL3634930)
Affinity DataKi:  2.61E+3nMAssay Description:Displacement of [3H]DAMGO from rat mu-opioid receptor expressed in CHO cells after 90 mins by scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
The University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50133262(CHEMBL3634928)
Affinity DataKi:  3.20E+3nMAssay Description:Displacement of [3H]DAMGO from rat mu-opioid receptor expressed in CHO cells after 90 mins by scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
The University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50133253(CHEMBL3634924)
Affinity DataKi:  4.01E+3nMAssay Description:Displacement of [3H]diprenorphine from rat kappa-opioid receptor expressed in CHO cells after 90 mins by scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
The University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50012153(zyklophin)
Affinity DataKi:  4.38E+3nMAssay Description:Displacement of [3H]DAMGO from rat mu-opioid receptor expressed in CHO cells after 90 mins by scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
The University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50133263(CHEMBL3634929)
Affinity DataKi:  8.26E+3nMAssay Description:Displacement of [3H]DAMGO from rat mu-opioid receptor expressed in CHO cells after 90 mins by scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
The University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50133221(CHEMBL3634921)
Affinity DataKi:  8.47E+3nMAssay Description:Displacement of [3H]DAMGO from rat mu-opioid receptor expressed in CHO cells after 90 mins by scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
The University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50133252(CHEMBL3634923)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]DAMGO from rat mu-opioid receptor expressed in CHO cells after 90 mins by scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
The University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50133255(CHEMBL3634926)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]DAMGO from rat mu-opioid receptor expressed in CHO cells after 90 mins by scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
The University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50133253(CHEMBL3634924)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]DAMGO from rat mu-opioid receptor expressed in CHO cells after 90 mins by scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
The University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50133222(CHEMBL3634922)
Affinity DataKi:  1.06E+4nMAssay Description:Displacement of [3H]DAMGO from rat mu-opioid receptor expressed in CHO cells after 90 mins by scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
The University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50133220(CHEMBL3634920)
Affinity DataKi:  1.09E+4nMAssay Description:Displacement of [3H]DAMGO from rat mu-opioid receptor expressed in CHO cells after 90 mins by scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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