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Found 131 with Last Name = 'aman' and Initial = 'am'
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
University Of Toronto At Mississauga

Curated by ChEMBL
LigandPNGBDBM50446144(CHEMBL3108911)
Affinity DataKi:  1.00E+4nMAssay Description:Competitive binding affinity to STAT3 SH2 domain (unknown origin) assessed as inhibition of interaction with FAMpYLPQTV after 15 to 30 mins by fluore...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
University Of Toronto At Mississauga

Curated by ChEMBL
LigandPNGBDBM50446145(CHEMBL3108910)
Affinity DataKi:  1.00E+4nMAssay Description:Competitive binding affinity to STAT3 SH2 domain (unknown origin) assessed as inhibition of interaction with FAMpYLPQTV after 15 to 30 mins by fluore...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
University Of Toronto At Mississauga

Curated by ChEMBL
LigandPNGBDBM50446146(CHEMBL3108909)
Affinity DataKi:  1.00E+4nMAssay Description:Competitive binding affinity to STAT3 SH2 domain (unknown origin) assessed as inhibition of interaction with FAMpYLPQTV after 15 to 30 mins by fluore...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50412352(CHEMBL5278336)
Affinity DataIC50:  800nMAssay Description:Inhibition of AChE in organophosphate-susceptible clone of Schizaphis graminum OSS adult or last-instar nymphs homogenates assessed as bimolecular ra...More data for this Ligand-Target Pair
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50412352(CHEMBL5278336)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of AChE in organophosphate-resistant clone of Schizaphis graminum OR1 adult or last-instar nymphs homogenates assessed as bimolecular rate...More data for this Ligand-Target Pair
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50412352(CHEMBL5278336)
Affinity DataIC50:  2.60E+4nMAssay Description:Inhibition of AChE in organophosphate-susceptible clone of Schizaphis graminum OSS adult or last-instar nymphs homogenates assessed as bimolecular ra...More data for this Ligand-Target Pair
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50412352(CHEMBL5278336)
Affinity DataIC50:  4.60E+4nMAssay Description:Inhibition of AChE in organophosphate-resistant clone of Schizaphis graminum OR1 adult or last-instar nymphs homogenates assessed as bimolecular rate...More data for this Ligand-Target Pair
TargetSignal transducer and activator of transcription 5A(Homo sapiens (Human))
University Of Toronto At Mississauga

Curated by ChEMBL
LigandPNGBDBM50446146(CHEMBL3108909)
Affinity DataKd:  464nMAssay Description:Binding affinity to His-tagged STAT5 (unknown origin) by SPR spectroscopic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
University Of Toronto At Mississauga

Curated by ChEMBL
LigandPNGBDBM50446146(CHEMBL3108909)
Affinity DataKd:  300nMAssay Description:Binding affinity to His-tagged STAT3 (unknown origin) by SPR spectroscopic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50411266(CHEMBL5284285)
Affinity DataKd:  1.30E+5nMAssay Description:Inhibition of carbonic anhydrase 2 assessed as inhibition of carbon dioxide hydrationMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50411267(CHEMBL5269641)
Affinity DataKd:  2.70E+5nMAssay Description:Inhibition of carbonic anhydrase 2 assessed as inhibition of carbon dioxide hydrationMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50411268(CHEMBL5267700)
Affinity DataKd:  1.10E+5nMAssay Description:Inhibition of carbonic anhydrase 2 assessed as inhibition of carbon dioxide hydrationMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50411269(CHEMBL5275351)
Affinity DataKd:  1.70E+5nMAssay Description:Inhibition of carbonic anhydrase 2 assessed as inhibition of carbon dioxide hydrationMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50411270(CHEMBL5272566)
Affinity DataKd:  3.30E+4nMAssay Description:Inhibition of carbonic anhydrase 2 assessed as inhibition of carbon dioxide hydrationMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50411271(CHEMBL5267112)
Affinity DataKd:  9.00E+3nMAssay Description:Inhibition of carbonic anhydrase 2 assessed as inhibition of carbon dioxide hydrationMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50411272(CHEMBL5266658)
Affinity DataKd:  3.40E+4nMAssay Description:Inhibition of carbonic anhydrase 2 assessed as inhibition of carbon dioxide hydrationMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50411273(CHEMBL5273203)
Affinity DataKd:  8.00E+3nMAssay Description:Inhibition of carbonic anhydrase 2 assessed as inhibition of carbon dioxide hydrationMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50411274(CHEMBL5282322)
Affinity DataKd:  3.10E+4nMAssay Description:Inhibition of carbonic anhydrase 2 assessed as inhibition of carbon dioxide hydrationMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50411309(CHEMBL5276559)
Affinity DataKd:  1.20E+4nMAssay Description:Inhibition of carbonic anhydrase 2 assessed as inhibition of carbon dioxide hydrationMore data for this Ligand-Target Pair
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50411310(CHEMBL5273690)
Affinity DataKd:  9.40E+4nMAssay Description:Inhibition of carbonic anhydrase 2 assessed as inhibition of carbon dioxide hydrationMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50411330(CHEMBL5282333)
Affinity DataKd:  1.50E+5nMAssay Description:Inhibition of carbonic anhydrase 2 assessed as inhibition of carbon dioxide hydrationMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50411331(CHEMBL5270273)
Affinity DataKd:  5.40E+4nMAssay Description:Inhibition of carbonic anhydrase 2 assessed as inhibition of carbon dioxide hydrationMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50411332(CHEMBL5270844)
Affinity DataKd:  9.00E+4nMAssay Description:Inhibition of carbonic anhydrase 2 assessed as inhibition of carbon dioxide hydrationMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50411349(CHEMBL5285781)
Affinity DataKd:  9.20E+4nMAssay Description:Inhibition of carbonic anhydrase 2 assessed as inhibition of carbon dioxide hydrationMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50411350(CHEMBL5283991)
Affinity DataKd:  8.70E+4nMAssay Description:Inhibition of carbonic anhydrase 2 assessed as inhibition of carbon dioxide hydrationMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50411351(CHEMBL5290299)
Affinity DataKd:  6.10E+4nMAssay Description:Inhibition of carbonic anhydrase 2 assessed as inhibition of carbon dioxide hydrationMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50411352(CHEMBL5285743)
Affinity DataKd:  1.30E+5nMAssay Description:Inhibition of carbonic anhydrase 2 assessed as inhibition of carbon dioxide hydrationMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50411353(CHEMBL5274321)
Affinity DataKd:  2.20E+5nMAssay Description:Inhibition of carbonic anhydrase 2 assessed as inhibition of carbon dioxide hydrationMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50411354(CHEMBL5273898)
Affinity DataKd:  8.00E+4nMAssay Description:Inhibition of carbonic anhydrase 2 assessed as inhibition of carbon dioxide hydrationMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50411355(CHEMBL5282155)
Affinity DataKd:  3.80E+4nMAssay Description:Inhibition of carbonic anhydrase 2 assessed as inhibition of carbon dioxide hydrationMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50411357(CHEMBL5290717)
Affinity DataKd:  4.50E+4nMAssay Description:Inhibition of carbonic anhydrase 2 assessed as inhibition of carbon dioxide hydrationMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50411358(CHEMBL5268053)
Affinity DataKd:  3.40E+4nMAssay Description:Inhibition of carbonic anhydrase 2 assessed as inhibition of carbon dioxide hydrationMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50411359(CHEMBL5284407)
Affinity DataKd:  1.50E+5nMAssay Description:Inhibition of carbonic anhydrase 2 assessed as inhibition of carbon dioxide hydrationMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50411360(CHEMBL5268432)
Affinity DataKd:  2.50E+4nMAssay Description:Inhibition of carbonic anhydrase 2 assessed as inhibition of carbon dioxide hydrationMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50411363(CHEMBL5277702)
Affinity DataKd:  1.90E+4nMAssay Description:Inhibition of carbonic anhydrase 2 assessed as inhibition of carbon dioxide hydrationMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50411432(CHEMBL5266727)
Affinity DataKd:  4.00E+4nMAssay Description:Inhibition of carbonic anhydrase 2 assessed as inhibition of carbon dioxide hydrationMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50411433(CHEMBL5285627)
Affinity DataKd:  2.30E+4nMAssay Description:Inhibition of carbonic anhydrase 2 assessed as inhibition of carbon dioxide hydrationMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50411434(CHEMBL5281654)
Affinity DataKd:  2.10E+4nMAssay Description:Inhibition of carbonic anhydrase 2 assessed as inhibition of carbon dioxide hydrationMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50411438(CHEMBL5265979)
Affinity DataKd:  2.20E+4nMAssay Description:Inhibition of carbonic anhydrase 2 assessed as inhibition of carbon dioxide hydrationMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50411440(CHEMBL5274675)
Affinity DataKd:  7.90E+4nMAssay Description:Inhibition of carbonic anhydrase 2 assessed as inhibition of carbon dioxide hydrationMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50411561(CHEMBL5266393)
Affinity DataKd:  1.80E+4nMAssay Description:Inhibition of carbonic anhydrase 2 assessed as inhibition of carbon dioxide hydrationMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50411964(CHEMBL5290467)
Affinity DataKd:  3.90E+4nMAssay Description:Inhibition of carbonic anhydrase 2 assessed as inhibition of carbon dioxide hydrationMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50411965(CHEMBL5269269)
Affinity DataKd:  3.10E+4nMAssay Description:Inhibition of carbonic anhydrase 2 assessed as inhibition of carbon dioxide hydrationMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50411968(CHEMBL5268349)
Affinity DataKd:  8.20E+4nMAssay Description:Inhibition of carbonic anhydrase 2 assessed as inhibition of carbon dioxide hydrationMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50411969(CHEMBL5290098)
Affinity DataKd:  4.20E+4nMAssay Description:Inhibition of carbonic anhydrase 2 assessed as inhibition of carbon dioxide hydrationMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50411970(CHEMBL5286035)
Affinity DataKd:  4.70E+4nMAssay Description:Inhibition of carbonic anhydrase 2 assessed as inhibition of carbon dioxide hydrationMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50411971(CHEMBL5289065)
Affinity DataKd:  5.90E+4nMAssay Description:Inhibition of carbonic anhydrase 2 assessed as inhibition of carbon dioxide hydrationMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50411972(CHEMBL5271929)
Affinity DataKd:  9.00E+3nMAssay Description:Binding affinity to human CD69 receptor expressed in Escherichia coli by equilibrium dialysisMore data for this Ligand-Target Pair
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50411973(CHEMBL5286558)
Affinity DataKd:  2.10E+5nMAssay Description:Binding affinity to human monomeric CD69 receptor expressed in Escherichia coli by equilibrium dialysisMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50411974(CHEMBL5288864)
Affinity DataKd: >1.00E+6nMAssay Description:Binding affinity to human dimeric CD69 receptor expressed in Escherichia coli by equilibrium dialysisMore data for this Ligand-Target Pair
In DepthDetails PubMed
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