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Found 109 with Last Name = 'chamberlin' and Initial = 'ar'
TargetProtein phosphatase 1B(Homo sapiens (Human))
University Of California Irvine

Curated by ChEMBL
LigandPNGBDBM50135699((10S,13S,18S,19S,22R)-8-Isobutyl-18-((1E,3E)-(5S,6...)
Affinity DataIC50:  0.300nMAssay Description:Inhibitory concentration of the compound against protein phosphatase 1 (PP1) using phosphorylase-a assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase 2A catalytic subunit alpha isoform(Bos taurus)
University Of California Irvine

Curated by ChEMBL
LigandPNGBDBM50135699((10S,13S,18S,19S,22R)-8-Isobutyl-18-((1E,3E)-(5S,6...)
Affinity DataIC50:  0.300nMAssay Description:Inhibitory concentration of the compound against protein phosphatase 1 (PP1) using phosphorylase-a assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase 1B(Homo sapiens (Human))
University Of California Irvine

Curated by ChEMBL
LigandPNGBDBM50135699((10S,13S,18S,19S,22R)-8-Isobutyl-18-((1E,3E)-(5S,6...)
Affinity DataIC50:  3nMAssay Description:Inhibitory concentration of the compound against protein phosphatase 2A (PP2A) using phosphorylase-a assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase 2A catalytic subunit alpha isoform(Bos taurus)
University Of California Irvine

Curated by ChEMBL
LigandPNGBDBM50135699((10S,13S,18S,19S,22R)-8-Isobutyl-18-((1E,3E)-(5S,6...)
Affinity DataIC50:  3nMAssay Description:Inhibitory concentration against protein phosphatase 2A (PP2A) using pNPP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase 2A 55 kDa regulatory subunit B(Gallus gallus)
University Of California Irvine

Curated by ChEMBL
LigandPNGBDBM50061067(15-(3-Guanidino-propyl)-8-isobutyl-18-((1E,3E)-6-m...)
Affinity DataIC50:  3nMAssay Description:Inhibitory concentration of the compound required against protein phosphatase 2A using pNPP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase 1A(Homo sapiens (Human))
University Of California Irvine

Curated by ChEMBL
LigandPNGBDBM50061067(15-(3-Guanidino-propyl)-8-isobutyl-18-((1E,3E)-6-m...)
Affinity DataIC50:  3nMAssay Description:Inhibitory concentration of the compound required against protein phosphatase 1 using pNPP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase 2A catalytic subunit alpha isoform(Bos taurus)
University Of California Irvine

Curated by ChEMBL
LigandPNGBDBM50135691((R)-2-((4E,6E)-(2S,3S,8S,9S)-3-Acetylamino-9-metho...)
Affinity DataIC50:  160nMAssay Description:Inhibitory concentration of the compound against protein phosphatase 2A (PP2A) using phosphorylase-a assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50083523((1-Benzyl-1H-quinolin-4-ylidene)-pentyl-amine | CH...)
Affinity DataIC50:  200nMAssay Description:Displacement of [125I]- ChTX from human T cell voltage-gated potassium channel subunit Kv1.3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
University Of California Irvine

Curated by ChEMBL
LigandPNGBDBM50176903(CHEMBL3814877)
Affinity DataIC50:  210nMAssay Description:Inhibition of C-terminal four-histidine tagged human CYP3A4delta3 to 24 residues expressed in Escherichia coli assessed as 7-benzyloxy-4-(trifluorome...More data for this Ligand-Target Pair
TargetProtein phosphatase 1B(Homo sapiens (Human))
University Of California Irvine

Curated by ChEMBL
LigandPNGBDBM50090505((1R,2S,6R,7S)-2,6-Dimethyl-4,10-dioxa-tricyclo[5.2...)
Affinity DataIC50:  430nMAssay Description:Inhibitory activity against protein phosphatase-1 from rabbit skeletal muscleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase 2A activator(Homo sapiens (Human))
University Of California Irvine

Curated by ChEMBL
LigandPNGBDBM50127377(10-[3,9-dimethyl-8-(3-methyl-4-oxopentyl)-(9R)-1,7...)
Affinity DataIC50:  500nMAssay Description:Inhibition of protein phosphatase 2A (PP2A) was determined by standard phosphorylase a inhibition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase 2A catalytic subunit alpha isoform(Bos taurus)
University Of California Irvine

Curated by ChEMBL
LigandPNGBDBM50135697(((4E,6E)-(2S,3S,8S,9S)-3-Acetylamino-9-methoxy-2,6...)
Affinity DataIC50:  500nMAssay Description:Inhibitory concentration of the compound against protein phosphatase 2A (PP2A) using phosphorylase-a assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
University Of California Irvine

Curated by ChEMBL
LigandPNGBDBM50176904(CHEMBL3814479)
Affinity DataIC50:  520nMAssay Description:Inhibition of C-terminal four-histidine tagged human CYP3A4delta3 to 24 residues expressed in Escherichia coli assessed as 7-benzyloxy-4-(trifluorome...More data for this Ligand-Target Pair
TargetProtein phosphatase 1B(Homo sapiens (Human))
University Of California Irvine

Curated by ChEMBL
LigandPNGBDBM50366474(NORCANTHARIDIN)
Affinity DataIC50:  570nMAssay Description:Inhibitory activity against protein phosphatase-1 from rabbit skeletal muscleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase 1B(Homo sapiens (Human))
University Of California Irvine

Curated by ChEMBL
LigandPNGBDBM50135691((R)-2-((4E,6E)-(2S,3S,8S,9S)-3-Acetylamino-9-metho...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibitory concentration against protein phosphatase 1 (PP1) using pNPP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50083514(4-[(E)-2-(3,4-Bis-benzyloxy-phenyl)-vinyl]-4'-chlo...)
Affinity DataIC50:  2.90E+3nMAssay Description:Displacement of [125I]- ChTX from human T cell voltage-gated potassium channel subunit Kv1.3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50083518(4'-Chloro-4-((E)-4-phenyl-but-1-enyl)-biphenyl-2-c...)
Affinity DataIC50:  3.20E+3nMAssay Description:Displacement of [125I]- ChTX from human T cell voltage-gated potassium channel subunit Kv1.3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50083522(4'-Chloro-4-[(E)-2-(4-chloro-3-fluoro-phenyl)-viny...)
Affinity DataIC50:  3.70E+3nMAssay Description:Displacement of [125I]- ChTX from human T cell voltage-gated potassium channel subunit Kv1.3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50083515(2-({4'-chloro-4-[(E)-2-(4-fluorophenyl)vinyl]-1,1'...)
Affinity DataIC50:  3.90E+3nMAssay Description:Displacement of [125I]- ChTX from human T cell voltage-gated potassium channel subunit Kv1.3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50083513(4'-Chloro-4-((E)-4-phenyl-but-1-enyl)-biphenyl-2-c...)
Affinity DataIC50:  4.00E+3nMAssay Description:Displacement of [125I]- ChTX from human T cell voltage-gated potassium channel subunit Kv1.3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase 2A activator(Homo sapiens (Human))
University Of California Irvine

Curated by ChEMBL
LigandPNGBDBM50127375((E)-(R)-4-Hydroxy-2-methyl-hex-2-enedioic acid 6-{...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of protein phosphatase 2A (PP2A) was determined by standard phosphorylase a inhibition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50083511(4'-Chloro-4-((E)-3-phenyl-propenyl)-biphenyl-2-car...)
Affinity DataIC50:  5.60E+3nMAssay Description:Displacement of [125I]- ChTX from human T cell voltage-gated potassium channel subunit Kv1.3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase 1B(Homo sapiens (Human))
University Of California Irvine

Curated by ChEMBL
LigandPNGBDBM50135697(((4E,6E)-(2S,3S,8S,9S)-3-Acetylamino-9-methoxy-2,6...)
Affinity DataIC50:  5.60E+3nMAssay Description:Inhibitory concentration of the compound against protein phosphatase 1 (PP1) using phosphorylase-a assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50083516(4'-Chloro-4-((E)-3-phenyl-propenyl)-biphenyl-2-car...)
Affinity DataIC50:  5.80E+3nMAssay Description:Displacement of [125I]- ChTX from human T cell voltage-gated potassium channel subunit Kv1.3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50083519(4'-Chloro-4-((E)-3-phenyl-propenyl)-biphenyl-2-car...)
Affinity DataIC50:  6.10E+3nMAssay Description:Displacement of [125I]- ChTX from human T cell voltage-gated potassium channel subunit Kv1.3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase 2A catalytic subunit alpha isoform(Bos taurus)
University Of California Irvine

Curated by ChEMBL
LigandPNGBDBM50135691((R)-2-((4E,6E)-(2S,3S,8S,9S)-3-Acetylamino-9-metho...)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibitory concentration against protein phosphatase 2A (PP2A) using pNPP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase 2A catalytic subunit alpha isoform(Bos taurus)
University Of California Irvine

Curated by ChEMBL
LigandPNGBDBM50135700((S)-2-((4E,6E)-(2S,3S,8S,9S)-3-Acetylamino-9-metho...)
Affinity DataIC50:  7.80E+3nMAssay Description:Inhibitory concentration of the compound against protein phosphatase 2A (PP2A) using phosphorylase-a assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50083517(4'-Chloro-4-[(E)-2-(2-fluoro-phenyl)-vinyl]-biphen...)
Affinity DataIC50:  8.00E+3nMAssay Description:Displacement of [125I]- ChTX from human T cell voltage-gated potassium channel subunit Kv1.3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase 2A activator(Homo sapiens (Human))
University Of California Irvine

Curated by ChEMBL
LigandPNGBDBM50366883(TAUTOMYCIN)
Affinity DataIC50:  9.40E+3nMAssay Description:Inhibition of protein phosphatase 2A (PP2A) was determined by standard phosphorylase a inhibition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50083512(4'-Chloro-4-[(E)-2-(4-fluoro-phenyl)-vinyl]-biphen...)
Affinity DataIC50:  9.70E+3nMAssay Description:Displacement of [125I]- ChTX from human T cell voltage-gated potassium channel subunit Kv1.3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50083520(4-[(E)-2-(4-Benzyloxy-phenyl)-vinyl]-4'-chloro-bip...)
Affinity DataIC50:  9.90E+3nMAssay Description:Displacement of [125I]- ChTX from human T cell voltage-gated potassium channel subunit Kv1.3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase 2A catalytic subunit alpha isoform(Bos taurus)
University Of California Irvine

Curated by ChEMBL
LigandPNGBDBM50135696((2R,5S)-1-((4E,6E)-(2S,3S,8S,9S)-3-Acetylamino-9-m...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibitory concentration against protein phosphatase 2A (PP2A) using pNPP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50083521(4'-Chloro-4-[(E)-2-(3-chloro-phenyl)-vinyl]-biphen...)
Affinity DataIC50:  1.01E+4nMAssay Description:Displacement of [125I]- ChTX from human T cell voltage-gated potassium channel subunit Kv1.3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase 1B(Homo sapiens (Human))
University Of California Irvine

Curated by ChEMBL
LigandPNGBDBM50143522((1S,4R)-3-(3-Carboxy-phenylcarbamoyl)-7-oxa-bicycl...)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibitory activity against protein phosphatase-1 from rabbit skeletal muscleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase 1B(Homo sapiens (Human))
University Of California Irvine

Curated by ChEMBL
LigandPNGBDBM50143517((1S,4R)-3-(3-Methoxycarbonyl-phenylcarbamoyl)-7-ox...)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibitory activity against protein phosphatase-1 from rabbit skeletal muscleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase 2A 55 kDa regulatory subunit B(Gallus gallus)
University Of California Irvine

Curated by ChEMBL
LigandPNGBDBM50135676((S)-2-[(R)-2-(2-{[(R)-4-((4E,6E)-(2S,3S,8S,9S)-3-A...)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibitory concentration of the compound required against protein phosphatase 2A using pNPP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase 2A 55 kDa regulatory subunit B(Gallus gallus)
University Of California Irvine

Curated by ChEMBL
LigandPNGBDBM50135679((S)-2-[(R)-2-(2-{[(R)-4-((4E,6E)-(2S,3S,8S,9S)-3-A...)
Affinity DataIC50:  1.70E+4nMAssay Description:Inhibitory concentration of the compound required against protein phosphatase 2A using pNPP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase 1B(Homo sapiens (Human))
University Of California Irvine

Curated by ChEMBL
LigandPNGBDBM50143509((1S,4R)-3-Dimethylcarbamoyl-7-oxa-bicyclo[2.2.1]he...)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibitory activity against protein phosphatase-1 from rabbit skeletal muscleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase 2A 55 kDa regulatory subunit B(Gallus gallus)
University Of California Irvine

Curated by ChEMBL
LigandPNGBDBM50135677((R)-2-((4E,6E)-(2S,3S,8S,9S)-3-Acetylamino-9-metho...)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibitory concentration of the compound required against protein phosphatase 2A using pNPP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase 2A 55 kDa regulatory subunit B(Gallus gallus)
University Of California Irvine

Curated by ChEMBL
LigandPNGBDBM50135681((R)-2-((4E,6E)-(2S,3S,8S,9S)-3-Amino-9-methoxy-2,6...)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibitory concentration of the compound required against protein phosphatase 2A using pNPP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase 2A catalytic subunit alpha isoform(Bos taurus)
University Of California Irvine

Curated by ChEMBL
LigandPNGBDBM50135687((R)-1-((4E,6E)-(2S,3S,8S,9S)-3-Acetylamino-9-metho...)
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibitory concentration against protein phosphatase 2A (PP2A) using pNPP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase 1B(Homo sapiens (Human))
University Of California Irvine

Curated by ChEMBL
LigandPNGBDBM50135691((R)-2-((4E,6E)-(2S,3S,8S,9S)-3-Acetylamino-9-metho...)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibitory concentration against protein phosphatase 1 (PP1) using pNPP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase 1B(Homo sapiens (Human))
University Of California Irvine

Curated by ChEMBL
LigandPNGBDBM50143515(Benzoic acid (1S,2R,6S,7R,8R)-3,5-dioxo-4,10-dioxa...)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibitory activity against protein phosphatase-1 from rabbit skeletal muscleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase 2A 55 kDa regulatory subunit B(Gallus gallus)
University Of California Irvine

Curated by ChEMBL
LigandPNGBDBM50135675((R)-2-((4E,6E)-(2S,3S,8S,9S)-3-Acetylamino-9-metho...)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibitory concentration of the compound required against protein phosphatase 2A using pNPP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase 2A activator(Homo sapiens (Human))
University Of California Irvine

Curated by ChEMBL
LigandPNGBDBM50127378((S)-2-Hydroxy-2-methyl-succinic acid 4-{(1R,2S,3R,...)
Affinity DataIC50:  2.90E+4nMAssay Description:Inhibition of protein phosphatase 2A (PP2A) was determined by standard phosphorylase a inhibition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase 1B(Homo sapiens (Human))
University Of California Irvine

Curated by ChEMBL
LigandPNGBDBM50143516((1S,4R)-3-(4-Ethoxycarbonyl-phenylcarbamoyl)-7-oxa...)
Affinity DataIC50:  2.90E+4nMAssay Description:Inhibitory activity against protein phosphatase-1 from rabbit skeletal muscleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
University Of California Irvine

Curated by ChEMBL
LigandPNGBDBM50176905(CHEMBL3814345)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibition of C-terminal four-histidine tagged human CYP3A4delta3 to 24 residues expressed in Escherichia coli assessed as 7-benzyloxy-4-(trifluorome...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase 2A catalytic subunit alpha isoform(Bos taurus)
University Of California Irvine

Curated by ChEMBL
LigandPNGBDBM50135685((2S,5S)-1-((4E,6E)-(2S,3S,8S,9S)-3-Acetylamino-9-m...)
Affinity DataIC50: >3.90E+4nMAssay Description:Inhibitory concentration against protein phosphatase 2A (PP2A) using pNPP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase 1A(Homo sapiens (Human))
University Of California Irvine

Curated by ChEMBL
LigandPNGBDBM50135681((R)-2-((4E,6E)-(2S,3S,8S,9S)-3-Amino-9-methoxy-2,6...)
Affinity DataIC50:  4.50E+4nMAssay Description:Inhibitory concentration of the compound required against protein phosphatase 1 using pNPP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase 1B(Homo sapiens (Human))
University Of California Irvine

Curated by ChEMBL
LigandPNGBDBM50143512((1S,4R)-3-(4-Chloro-phenylcarbamoyl)-7-oxa-bicyclo...)
Affinity DataIC50:  4.90E+4nMAssay Description:Inhibitory activity against protein phosphatase-1 from rabbit skeletal muscleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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