Affinity DataIC50: 0.300nMAssay Description:Inhibitory concentration of the compound against protein phosphatase 1 (PP1) using phosphorylase-a assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase 2A catalytic subunit alpha isoform(Bos taurus)
University Of California Irvine
Curated by ChEMBL
University Of California Irvine
Curated by ChEMBL
Affinity DataIC50: 0.300nMAssay Description:Inhibitory concentration of the compound against protein phosphatase 1 (PP1) using phosphorylase-a assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibitory concentration of the compound against protein phosphatase 2A (PP2A) using phosphorylase-a assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase 2A catalytic subunit alpha isoform(Bos taurus)
University Of California Irvine
Curated by ChEMBL
University Of California Irvine
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibitory concentration against protein phosphatase 2A (PP2A) using pNPP assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase 2A 55 kDa regulatory subunit B(Gallus gallus)
University Of California Irvine
Curated by ChEMBL
University Of California Irvine
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibitory concentration of the compound required against protein phosphatase 2A using pNPP assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibitory concentration of the compound required against protein phosphatase 1 using pNPP assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase 2A catalytic subunit alpha isoform(Bos taurus)
University Of California Irvine
Curated by ChEMBL
University Of California Irvine
Curated by ChEMBL
Affinity DataIC50: 160nMAssay Description:Inhibitory concentration of the compound against protein phosphatase 2A (PP2A) using phosphorylase-a assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Displacement of [125I]- ChTX from human T cell voltage-gated potassium channel subunit Kv1.3More data for this Ligand-Target Pair
Affinity DataIC50: 210nMAssay Description:Inhibition of C-terminal four-histidine tagged human CYP3A4delta3 to 24 residues expressed in Escherichia coli assessed as 7-benzyloxy-4-(trifluorome...More data for this Ligand-Target Pair
Affinity DataIC50: 430nMAssay Description:Inhibitory activity against protein phosphatase-1 from rabbit skeletal muscleMore data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase 2A activator(Homo sapiens (Human))
University Of California Irvine
Curated by ChEMBL
University Of California Irvine
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibition of protein phosphatase 2A (PP2A) was determined by standard phosphorylase a inhibition assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase 2A catalytic subunit alpha isoform(Bos taurus)
University Of California Irvine
Curated by ChEMBL
University Of California Irvine
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibitory concentration of the compound against protein phosphatase 2A (PP2A) using phosphorylase-a assayMore data for this Ligand-Target Pair
Affinity DataIC50: 520nMAssay Description:Inhibition of C-terminal four-histidine tagged human CYP3A4delta3 to 24 residues expressed in Escherichia coli assessed as 7-benzyloxy-4-(trifluorome...More data for this Ligand-Target Pair
Affinity DataIC50: 570nMAssay Description:Inhibitory activity against protein phosphatase-1 from rabbit skeletal muscleMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory concentration against protein phosphatase 1 (PP1) using pNPP assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 2.90E+3nMAssay Description:Displacement of [125I]- ChTX from human T cell voltage-gated potassium channel subunit Kv1.3More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 3.20E+3nMAssay Description:Displacement of [125I]- ChTX from human T cell voltage-gated potassium channel subunit Kv1.3More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 3.70E+3nMAssay Description:Displacement of [125I]- ChTX from human T cell voltage-gated potassium channel subunit Kv1.3More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 3.90E+3nMAssay Description:Displacement of [125I]- ChTX from human T cell voltage-gated potassium channel subunit Kv1.3More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 4.00E+3nMAssay Description:Displacement of [125I]- ChTX from human T cell voltage-gated potassium channel subunit Kv1.3More data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase 2A activator(Homo sapiens (Human))
University Of California Irvine
Curated by ChEMBL
University Of California Irvine
Curated by ChEMBL
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of protein phosphatase 2A (PP2A) was determined by standard phosphorylase a inhibition assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 5.60E+3nMAssay Description:Displacement of [125I]- ChTX from human T cell voltage-gated potassium channel subunit Kv1.3More data for this Ligand-Target Pair
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibitory concentration of the compound against protein phosphatase 1 (PP1) using phosphorylase-a assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 5.80E+3nMAssay Description:Displacement of [125I]- ChTX from human T cell voltage-gated potassium channel subunit Kv1.3More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 6.10E+3nMAssay Description:Displacement of [125I]- ChTX from human T cell voltage-gated potassium channel subunit Kv1.3More data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase 2A catalytic subunit alpha isoform(Bos taurus)
University Of California Irvine
Curated by ChEMBL
University Of California Irvine
Curated by ChEMBL
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibitory concentration against protein phosphatase 2A (PP2A) using pNPP assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase 2A catalytic subunit alpha isoform(Bos taurus)
University Of California Irvine
Curated by ChEMBL
University Of California Irvine
Curated by ChEMBL
Affinity DataIC50: 7.80E+3nMAssay Description:Inhibitory concentration of the compound against protein phosphatase 2A (PP2A) using phosphorylase-a assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 8.00E+3nMAssay Description:Displacement of [125I]- ChTX from human T cell voltage-gated potassium channel subunit Kv1.3More data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase 2A activator(Homo sapiens (Human))
University Of California Irvine
Curated by ChEMBL
University Of California Irvine
Curated by ChEMBL
Affinity DataIC50: 9.40E+3nMAssay Description:Inhibition of protein phosphatase 2A (PP2A) was determined by standard phosphorylase a inhibition assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 9.70E+3nMAssay Description:Displacement of [125I]- ChTX from human T cell voltage-gated potassium channel subunit Kv1.3More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 9.90E+3nMAssay Description:Displacement of [125I]- ChTX from human T cell voltage-gated potassium channel subunit Kv1.3More data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase 2A catalytic subunit alpha isoform(Bos taurus)
University Of California Irvine
Curated by ChEMBL
University Of California Irvine
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory concentration against protein phosphatase 2A (PP2A) using pNPP assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 1.01E+4nMAssay Description:Displacement of [125I]- ChTX from human T cell voltage-gated potassium channel subunit Kv1.3More data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibitory activity against protein phosphatase-1 from rabbit skeletal muscleMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibitory activity against protein phosphatase-1 from rabbit skeletal muscleMore data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase 2A 55 kDa regulatory subunit B(Gallus gallus)
University Of California Irvine
Curated by ChEMBL
University Of California Irvine
Curated by ChEMBL
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibitory concentration of the compound required against protein phosphatase 2A using pNPP assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase 2A 55 kDa regulatory subunit B(Gallus gallus)
University Of California Irvine
Curated by ChEMBL
University Of California Irvine
Curated by ChEMBL
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibitory concentration of the compound required against protein phosphatase 2A using pNPP assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibitory activity against protein phosphatase-1 from rabbit skeletal muscleMore data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase 2A 55 kDa regulatory subunit B(Gallus gallus)
University Of California Irvine
Curated by ChEMBL
University Of California Irvine
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibitory concentration of the compound required against protein phosphatase 2A using pNPP assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase 2A 55 kDa regulatory subunit B(Gallus gallus)
University Of California Irvine
Curated by ChEMBL
University Of California Irvine
Curated by ChEMBL
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibitory concentration of the compound required against protein phosphatase 2A using pNPP assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase 2A catalytic subunit alpha isoform(Bos taurus)
University Of California Irvine
Curated by ChEMBL
University Of California Irvine
Curated by ChEMBL
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibitory concentration against protein phosphatase 2A (PP2A) using pNPP assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibitory concentration against protein phosphatase 1 (PP1) using pNPP assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibitory activity against protein phosphatase-1 from rabbit skeletal muscleMore data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase 2A 55 kDa regulatory subunit B(Gallus gallus)
University Of California Irvine
Curated by ChEMBL
University Of California Irvine
Curated by ChEMBL
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibitory concentration of the compound required against protein phosphatase 2A using pNPP assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase 2A activator(Homo sapiens (Human))
University Of California Irvine
Curated by ChEMBL
University Of California Irvine
Curated by ChEMBL
Affinity DataIC50: 2.90E+4nMAssay Description:Inhibition of protein phosphatase 2A (PP2A) was determined by standard phosphorylase a inhibition assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.90E+4nMAssay Description:Inhibitory activity against protein phosphatase-1 from rabbit skeletal muscleMore data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of C-terminal four-histidine tagged human CYP3A4delta3 to 24 residues expressed in Escherichia coli assessed as 7-benzyloxy-4-(trifluorome...More data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase 2A catalytic subunit alpha isoform(Bos taurus)
University Of California Irvine
Curated by ChEMBL
University Of California Irvine
Curated by ChEMBL
Affinity DataIC50: >3.90E+4nMAssay Description:Inhibitory concentration against protein phosphatase 2A (PP2A) using pNPP assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.50E+4nMAssay Description:Inhibitory concentration of the compound required against protein phosphatase 1 using pNPP assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.90E+4nMAssay Description:Inhibitory activity against protein phosphatase-1 from rabbit skeletal muscleMore data for this Ligand-Target Pair
![](/img/powered_by_small.gif)