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Found 42 with Last Name = 'basile' and Initial = 'as'
TargetTranslocator protein(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50054125((E)-2-(2-(4-chlorophenyl)-1,2-dihydro-1-oxo-3H-pyr...)
Affinity DataIC50:  0.700nMAssay Description:Displacement of [3H]-PK11195 from rat kidney peripheral benzodiazepine receptor (type 1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50054126((E)-N-(4-chlorophenyl)-2-(2-(4-chlorophenyl)-1-oxo...)
Affinity DataIC50:  1.10nMAssay Description:Displacement of [3H]-PK11195 from rat kidney peripheral benzodiazepine receptor (type 1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50054125((E)-2-(2-(4-chlorophenyl)-1,2-dihydro-1-oxo-3H-pyr...)
Affinity DataIC50:  1.70nMAssay Description:Displacement of [3H]-Ro-5-4864 from rat kidney peripheral benzodiazepine receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM22032(1-(2-chlorophenyl)-N-methyl-N-(1-methylpropyl)isoq...)
Affinity DataIC50:  1.80nMAssay Description:Binding affinity against peripheral benzodiazepine receptor( PBR).More data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50054125((E)-2-(2-(4-chlorophenyl)-1,2-dihydro-1-oxo-3H-pyr...)
Affinity DataIC50:  1.90nMAssay Description:Binding affinity against peripheral benzodiazepine receptor( PBR).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50054126((E)-N-(4-chlorophenyl)-2-(2-(4-chlorophenyl)-1-oxo...)
Affinity DataIC50:  2.10nMAssay Description:Displacement of [3H]-Ro-5-4864 from rat kidney peripheral benzodiazepine receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50054125((E)-2-(2-(4-chlorophenyl)-1,2-dihydro-1-oxo-3H-pyr...)
Affinity DataIC50:  2.30nMAssay Description:Displacement of [3H]-Ro-5-4864 from rat cerebral cortex peripheral benzodiazepine receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50054126((E)-N-(4-chlorophenyl)-2-(2-(4-chlorophenyl)-1-oxo...)
Affinity DataIC50:  2.40nMAssay Description:Displacement of [3H]-PK11195 from rat cerebral cortex peripheral benzodiazepine receptor (type 1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50054128(2-[2-(4-Chloro-phenyl)-1-oxo-1,2-dihydro-pyrrolo[3...)
Affinity DataIC50:  2.70nMAssay Description:Displacement of [3H]-PK11195 from rat kidney peripheral benzodiazepine receptor (type 1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50054126((E)-N-(4-chlorophenyl)-2-(2-(4-chlorophenyl)-1-oxo...)
Affinity DataIC50:  3.20nMAssay Description:Binding affinity against peripheral benzodiazepine receptor( PBR).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50054127(2-[6-Chloro-2-(4-chloro-phenyl)-1,8a-dihydro-imida...)
Affinity DataIC50:  3.90nMAssay Description:Binding affinity against peripheral benzodiazepine receptor( PBR).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50054126((E)-N-(4-chlorophenyl)-2-(2-(4-chlorophenyl)-1-oxo...)
Affinity DataIC50:  4.5nMAssay Description:Displacement of [3H]-Ro-5-4864 from rat cerebral cortex peripheral benzodiazepine receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50054128(2-[2-(4-Chloro-phenyl)-1-oxo-1,2-dihydro-pyrrolo[3...)
Affinity DataIC50:  4.90nMAssay Description:Displacement of [3H]-PK11195 from rat cerebral cortex peripheral benzodiazepine receptor (type 1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM22041(2-[6-chloro-2-(4-chlorophenyl)imidazo[1,2-a]pyridi...)
Affinity DataIC50:  7nMAssay Description:Binding affinity against peripheral benzodiazepine receptor( PBR).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50054125((E)-2-(2-(4-chlorophenyl)-1,2-dihydro-1-oxo-3H-pyr...)
Affinity DataIC50:  9.80nMAssay Description:Displacement of [3H]-PK11195 from rat cerebral cortex peripheral benzodiazepine receptor (type 1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50054125((E)-2-(2-(4-chlorophenyl)-1,2-dihydro-1-oxo-3H-pyr...)
Affinity DataIC50:  14nMAssay Description:Displacement of [3H]-PK11195 from rat kidney peripheral benzodiazepine receptor (type 2)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50054128(2-[2-(4-Chloro-phenyl)-1-oxo-1,2-dihydro-pyrrolo[3...)
Affinity DataIC50:  40nMAssay Description:Binding affinity against peripheral benzodiazepine receptor( PBR).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50054128(2-[2-(4-Chloro-phenyl)-1-oxo-1,2-dihydro-pyrrolo[3...)
Affinity DataIC50:  40nMAssay Description:Binding affinity against peripheral benzodiazepine receptor( PBR).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50054128(2-[2-(4-Chloro-phenyl)-1-oxo-1,2-dihydro-pyrrolo[3...)
Affinity DataIC50:  120nMAssay Description:Displacement of [3H]-Ro-5-4864 from rat cerebral cortex peripheral benzodiazepine receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50054126((E)-N-(4-chlorophenyl)-2-(2-(4-chlorophenyl)-1-oxo...)
Affinity DataIC50:  140nMAssay Description:Displacement of [3H]-PK11195 from rat kidney peripheral benzodiazepine receptor (type 2)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50054130((E)-2-(2-(4-chlorophenyl)-1-oxo-1,2-dihydropyrrolo...)
Affinity DataIC50:  150nMAssay Description:Binding affinity against peripheral benzodiazepine receptor( PBR).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50054128(2-[2-(4-Chloro-phenyl)-1-oxo-1,2-dihydro-pyrrolo[3...)
Affinity DataIC50:  160nMAssay Description:Displacement of [3H]-PK11195 from rat kidney peripheral benzodiazepine receptor (type 2)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50054128(2-[2-(4-Chloro-phenyl)-1-oxo-1,2-dihydro-pyrrolo[3...)
Affinity DataIC50:  210nMAssay Description:Displacement of [3H]-PK11195 from rat cerebral cortex peripheral benzodiazepine receptor (type 2)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50054134(2-[6-(4-Chloro-phenyl)-5-oxo-5,6-dihydro-pyrrolo[3...)
Affinity DataIC50:  290nMAssay Description:Binding affinity against peripheral benzodiazepine receptor( PBR).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50054125((E)-2-(2-(4-chlorophenyl)-1,2-dihydro-1-oxo-3H-pyr...)
Affinity DataIC50:  320nMAssay Description:Displacement of [3H]-PK11195 from rat cerebral cortex peripheral benzodiazepine receptor (type 2)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50054126((E)-N-(4-chlorophenyl)-2-(2-(4-chlorophenyl)-1-oxo...)
Affinity DataIC50:  610nMAssay Description:Displacement of [3H]-PK11195 from rat cerebral cortex peripheral benzodiazepine receptor (type 2)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50454429(CHEMBL2111919)
Affinity DataIC50: >1.00E+3nMAssay Description:Binding affinity against peripheral benzodiazepine receptor( PBR).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50054132(2-[6-(4-Chloro-phenyl)-5-oxo-6,7-dihydro-5H-pyrrol...)
Affinity DataIC50: >1.00E+3nMAssay Description:Binding affinity against peripheral benzodiazepine receptor( PBR).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50054140((E)-N-benzyl-2-(2-(4-chlorophenyl)-1-oxo-1,2-dihyd...)
Affinity DataIC50: >1.00E+3nMAssay Description:Binding affinity against peripheral benzodiazepine receptor( PBR).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50054131(2-[2-(4-Chloro-phenyl)-1-oxo-2,3-dihydro-1H-pyrrol...)
Affinity DataIC50: >1.00E+3nMAssay Description:Binding affinity against peripheral benzodiazepine receptor( PBR).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50054138((E)-N-benzyl-2-(2-(4-chlorophenyl)-1-oxo-1,2-dihyd...)
Affinity DataIC50: >1.00E+3nMAssay Description:Binding affinity against peripheral benzodiazepine receptor( PBR).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50054129(2-[2-(4-Chloro-phenyl)-1-oxo-2,3-dihydro-1H-pyrrol...)
Affinity DataIC50: >1.00E+3nMAssay Description:Binding affinity against peripheral benzodiazepine receptor( PBR).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50054133(6-(4-Chloro-phenyl)-6,7-dihydro-pyrrolo[3,4-b]pyri...)
Affinity DataIC50: >1.00E+3nMAssay Description:Binding affinity against peripheral benzodiazepine receptor( PBR).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50054135(2-[6-(4-Chloro-phenyl)-5-oxo-6,7-dihydro-5H-pyrrol...)
Affinity DataIC50:  1.60E+3nMAssay Description:Binding affinity against peripheral benzodiazepine receptor( PBR).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50054137(2-[6-(4-Chloro-phenyl)-5-oxo-5,6-dihydro-pyrrolo[3...)
Affinity DataIC50:  3.30E+4nMAssay Description:Binding affinity against peripheral benzodiazepine receptor( PBR).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50058155((R)-3-{4-[Bis-(2-chloro-ethyl)-amino]-phenyl}-2-[4...)
Affinity DataIC50:  3.27E+5nMAssay Description:The compound was tested for binding affinity against PBR(peripheral benzodiazepine receptor) in normal rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50058155((R)-3-{4-[Bis-(2-chloro-ethyl)-amino]-phenyl}-2-[4...)
Affinity DataIC50:  3.27E+5nMAssay Description:The compound was tested for binding affinity against PBR(peripheral benzodiazepine receptor) in normal rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50058155((R)-3-{4-[Bis-(2-chloro-ethyl)-amino]-phenyl}-2-[4...)
Affinity DataIC50:  3.90E+5nMAssay Description:Binding affinity for PBR (peripheral benzodiazepine receptor) in rat RG-2 glioma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50027835(7-Chloro-5-phenyl-1,3-dihydro-benzo[e][1,4]diazepi...)
Affinity DataIC50:  5.20E+5nMAssay Description:The compound was tested for binding affinity against PBR(peripheral benzodiazepine receptor) in normal rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM22040(4 -chlorodiazepam | 4' Cl-diazepam | 7-chloro-...)
Affinity DataKd:  1.30E+3nMAssay Description:Binding affinity constant for Benzodiazepine receptor in normal rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM22040(4 -chlorodiazepam | 4' Cl-diazepam | 7-chloro-...)
Affinity DataKd:  3.5nMAssay Description:Binding affinity constant for Benzodiazepine receptor in rat RG-2 glioma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM22040(4 -chlorodiazepam | 4' Cl-diazepam | 7-chloro-...)
Affinity DataKd:  4.00E+3nMAssay Description:Binding affinity constant for Benzodiazepine receptor in rat C6 glioma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed