Affinity DataIC50: 0.0600nMAssay Description:Binding affinity to AT2 in rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 0.220nMAssay Description:Binding affinity to AT2 in rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 0.220nMAssay Description:Binding affinity to AT2 in rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 0.220nMAssay Description:Binding affinity to AT2 in rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 0.220nMAssay Description:Binding affinity to AT2 in rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 0.220nMAssay Description:Binding affinity to AT2 in rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 0.220nMAssay Description:Binding affinity to AT2 in rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 0.220nMAssay Description:Binding affinity to AT2 in rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 0.460nMAssay Description:Binding affinity to AT2 in rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 0.460nMAssay Description:Binding affinity to AT2 in rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Binding affinity to AT2 in rat brainMore data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
Hibercell
Curated by ChEMBL
Hibercell
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibition of human His-tagged PERK expressed in Escherichia coli assessed as eIF2alpha phosphorylation by TR-FRET assayMore data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
Hibercell
Curated by ChEMBL
Hibercell
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibition of human His-tagged PERK expressed in Escherichia coli assessed as eIF2alpha phosphorylation by TR-FRET assayMore data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
Hibercell
Curated by ChEMBL
Hibercell
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibition of human His-tagged PERK expressed in Escherichia coli assessed as eIF2alpha phosphorylation by TR-FRET assayMore data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
Hibercell
Curated by ChEMBL
Hibercell
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibition of human His-tagged PERK expressed in Escherichia coli assessed as eIF2alpha phosphorylation by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.5nMAssay Description:Inhibition of angiotensin II (unknown origin)More data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
Hibercell
Curated by ChEMBL
Hibercell
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Inhibition of human His-tagged PERK expressed in Escherichia coli assessed as eIF2alpha phosphorylation by TR-FRET assayMore data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
Hibercell
Curated by ChEMBL
Hibercell
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Inhibition of human His-tagged PERK expressed in Escherichia coli assessed as eIF2alpha phosphorylation by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibition of rat adrenal cortex angiotensin IIMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibition of rat adrenal cortex angiotensin IIMore data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
Hibercell
Curated by ChEMBL
Hibercell
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Inhibition of human His-tagged PERK expressed in Escherichia coli assessed as eIF2alpha phosphorylation by TR-FRET assayMore data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
Hibercell
Curated by ChEMBL
Hibercell
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Inhibition of human His-tagged PERK expressed in Escherichia coli assessed as eIF2alpha phosphorylation by TR-FRET assayMore data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
Hibercell
Curated by ChEMBL
Hibercell
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Inhibition of human His-tagged PERK expressed in Escherichia coli assessed as eIF2alpha phosphorylation by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Inhibition of eIF2alpha (unknown origin) assessed as eIF2alpha phosphorylation by TR-FRET assayMore data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
Hibercell
Curated by ChEMBL
Hibercell
Curated by ChEMBL
Affinity DataIC50: 9nMAssay Description:Inhibition of human His-tagged PERK expressed in Escherichia coli assessed as eIF2alpha phosphorylation by TR-FRET assayMore data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
Hibercell
Curated by ChEMBL
Hibercell
Curated by ChEMBL
Affinity DataIC50: 9nMAssay Description:Inhibition of human His-tagged PERK expressed in Escherichia coli assessed as eIF2alpha phosphorylation by TR-FRET assayMore data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
Hibercell
Curated by ChEMBL
Hibercell
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Inhibition of human His-tagged PERK expressed in Escherichia coli assessed as eIF2alpha phosphorylation by TR-FRET assayMore data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
Hibercell
Curated by ChEMBL
Hibercell
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Inhibition of human His-tagged PERK expressed in Escherichia coli assessed as eIF2alpha phosphorylation by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Inhibition of rat adrenal cortex angiotensin IIMore data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Inhibition of rat adrenal cortex angiotensin IIMore data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Inhibition of rat adrenal cortex angiotensin IIMore data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Inhibition of eIF2alpha (unknown origin) assessed as eIF2alpha phosphorylation by TR-FRET assayMore data for this Ligand-Target Pair
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