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Found 2063 with Last Name = 'almansa-rosales' and Initial = 'c'
TargetSigma non-opioid intracellular receptor 1(Mus musculus (Mouse))
Laboratorios Del Dr. Esteve

US Patent
LigandPNGBDBM50077877(CHEMBL3417042 | US9611229, 2)
Affinity DataKi:  4.80nMAssay Description:Brain membrane preparation and binding assays for the 61-receptor were performed as described (DeHaven-Hudkins, D. L., L. C. Fleissner, and F. Y. For...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Laboratorios Del Dr. Esteve

US Patent
LigandPNGBDBM287137(1-(1-(2-(azepan- 1-yl)ethyl)-1H- pyrazolo[3,4- d]p...)
Affinity DataKi:  6.70nMpH: 7.4Assay Description:Brain membrane preparation and binding assays for the σ1-receptor were performed as described (DeHaven-Hudkins, D. L., L. C. Fleissner, and F. Y...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma non-opioid intracellular receptor 1(Mus musculus (Mouse))
Laboratorios Del Dr. Esteve

US Patent
LigandPNGBDBM50077891(CHEMBL3417066 | US9611229, 12)
Affinity DataKi:  8.70nMAssay Description:Brain membrane preparation and binding assays for the 61-receptor were performed as described (DeHaven-Hudkins, D. L., L. C. Fleissner, and F. Y. For...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Laboratorios Del Dr. Esteve

US Patent
LigandPNGBDBM287087(N-(1-(2-(azepan-1-yl)ethyl)-1H-pyrazolo[3,4-d]pyri...)
Affinity DataKi:  9.20nMpH: 7.4Assay Description:Brain membrane preparation and binding assays for the σ1-receptor were performed as described (DeHaven-Hudkins, D. L., L. C. Fleissner, and F. Y...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Laboratorios Del Dr. Esteve

US Patent
LigandPNGBDBM287138(1-(1-(2-(azepan- 1-yl)ethyl)-1H- pyrazolo[3,4- d]p...)
Affinity DataKi:  9.20nMpH: 7.4Assay Description:Brain membrane preparation and binding assays for the σ1-receptor were performed as described (DeHaven-Hudkins, D. L., L. C. Fleissner, and F. Y...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Laboratorios Del Dr. Esteve

US Patent
LigandPNGBDBM287101(N-(1-(2-(Azepan-1- yl)ethyl)-1H-pyrazolo[3,4- d]py...)
Affinity DataKi:  9.40nMpH: 7.4Assay Description:Brain membrane preparation and binding assays for the σ1-receptor were performed as described (DeHaven-Hudkins, D. L., L. C. Fleissner, and F. Y...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Laboratorios Del Dr. Esteve

US Patent
LigandPNGBDBM393445(2-(azepan-1- yl)-1-(3,4- dihydro- pyrazino[1,2- a]...)
Affinity DataKi:  10.2nMAssay Description:To investigate binding properties of sigma 1 receptor ligands to human sigma 1 receptor, transfected HEK-293 membranes and [3H](+)-pentazocine (Perki...More data for this Ligand-Target Pair
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In DepthDetails US Patent
TargetSigma non-opioid intracellular receptor 1(Mus musculus (Mouse))
Laboratorios Del Dr. Esteve

US Patent
LigandPNGBDBM50077886(CHEMBL3417058 | US9611229, 9)
Affinity DataKi:  10.3nMAssay Description:Brain membrane preparation and binding assays for the 61-receptor were performed as described (DeHaven-Hudkins, D. L., L. C. Fleissner, and F. Y. For...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSigma non-opioid intracellular receptor 1(Mus musculus (Mouse))
Laboratorios Del Dr. Esteve

US Patent
LigandPNGBDBM314366(N-(2-(azepan-1- yl)ethyl)-1-(1- adamantyl)-1H- 1,2...)
Affinity DataKi:  10.8nMAssay Description:Brain membrane preparation and binding assays for the 61-receptor were performed as described (DeHaven-Hudkins, D. L., L. C. Fleissner, and F. Y. For...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Laboratorios Del Dr. Esteve

US Patent
LigandPNGBDBM393458(3-(azepan-1- yl)-1-(3,4- dihydro- pyrazino[1,2- a]...)
Affinity DataKi:  10.9nMAssay Description:To investigate binding properties of sigma 1 receptor ligands to human sigma 1 receptor, transfected HEK-293 membranes and [3H](+)-pentazocine (Perki...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Laboratorios Del Dr. Esteve

US Patent
LigandPNGBDBM287111(N-(1-(2-(azepan-1- yl)ethyl)-1H-pyrazolo[3,4- d]py...)
Affinity DataKi:  11.1nMpH: 7.4Assay Description:Brain membrane preparation and binding assays for the σ1-receptor were performed as described (DeHaven-Hudkins, D. L., L. C. Fleissner, and F. Y...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma non-opioid intracellular receptor 1(Mus musculus (Mouse))
Laboratorios Del Dr. Esteve

US Patent
LigandPNGBDBM50077899(CHEMBL3417052 | US9611229, 13)
Affinity DataKi:  11.7nMAssay Description:Brain membrane preparation and binding assays for the 61-receptor were performed as described (DeHaven-Hudkins, D. L., L. C. Fleissner, and F. Y. For...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Laboratorios Del Dr. Esteve

US Patent
LigandPNGBDBM287140(N-(1-(2-(4-tert- butylpiperidin-1-yl)ethyl)- 1H-py...)
Affinity DataKi:  12.2nMpH: 7.4Assay Description:Brain membrane preparation and binding assays for the σ1-receptor were performed as described (DeHaven-Hudkins, D. L., L. C. Fleissner, and F. Y...More data for this Ligand-Target Pair
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TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Laboratorios Del Dr. Esteve

US Patent
LigandPNGBDBM287088(N-(1-[2-(Piperidin-1- yl)ethyl]-1H-pyrazolo[3,4- d...)
Affinity DataKi:  12.7nMpH: 7.4Assay Description:Brain membrane preparation and binding assays for the σ1-receptor were performed as described (DeHaven-Hudkins, D. L., L. C. Fleissner, and F. Y...More data for this Ligand-Target Pair
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TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Laboratorios Del Dr. Esteve

US Patent
LigandPNGBDBM287135(1-(1-(2-(azepan-1-yl)ethyl)-1H-pyrazolo[3,4-d]pyri...)
Affinity DataKi:  12.8nMpH: 7.4Assay Description:Brain membrane preparation and binding assays for the σ1-receptor were performed as described (DeHaven-Hudkins, D. L., L. C. Fleissner, and F. Y...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Laboratorios Del Dr. Esteve

US Patent
LigandPNGBDBM287097(N-(1-(2-(Azepan-1- yl)ethyl)-1H-pyrazolo[3,4- d]py...)
Affinity DataKi:  13.1nMpH: 7.4Assay Description:Brain membrane preparation and binding assays for the σ1-receptor were performed as described (DeHaven-Hudkins, D. L., L. C. Fleissner, and F. Y...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetSigma non-opioid intracellular receptor 1(Mus musculus (Mouse))
Laboratorios Del Dr. Esteve

US Patent
LigandPNGBDBM50077905(CHEMBL3417068 | US9611229, 33)
Affinity DataKi:  13.4nMAssay Description:Brain membrane preparation and binding assays for the 61-receptor were performed as described (DeHaven-Hudkins, D. L., L. C. Fleissner, and F. Y. For...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Laboratorios Del Dr. Esteve

US Patent
LigandPNGBDBM393447(2-(4-benzyl- piperidin- 1-yl)-1-(3,4- dihydro- pyr...)
Affinity DataKi:  14.4nMAssay Description:To investigate binding properties of sigma 1 receptor ligands to human sigma 1 receptor, transfected HEK-293 membranes and [3H](+)-pentazocine (Perki...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Laboratorios Del Dr. Esteve

US Patent
LigandPNGBDBM393453(2-(azepan-1- yl)-1-(8- fluoro-3,4- dihydro- pyrazi...)
Affinity DataKi:  14.6nMAssay Description:To investigate binding properties of sigma 1 receptor ligands to human sigma 1 receptor, transfected HEK-293 membranes and [3H](+)-pentazocine (Perki...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Laboratorios Del Dr. Esteve

US Patent
LigandPNGBDBM287136(1-(1-(2-(azepan- 1-yl)ethyl)-1H- pyrazolo[3,4- d]p...)
Affinity DataKi:  14.9nMpH: 7.4Assay Description:Brain membrane preparation and binding assays for the σ1-receptor were performed as described (DeHaven-Hudkins, D. L., L. C. Fleissner, and F. Y...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Laboratorios Del Dr. Esteve

US Patent
LigandPNGBDBM287103(N-(1-(2-(Azepan-1- yl)ethyl)-1H-pyrazolo[3,4- d]py...)
Affinity DataKi:  15nMpH: 7.4Assay Description:Brain membrane preparation and binding assays for the σ1-receptor were performed as described (DeHaven-Hudkins, D. L., L. C. Fleissner, and F. Y...More data for this Ligand-Target Pair
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TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Laboratorios Del Dr. Esteve

US Patent
LigandPNGBDBM287107(N-(1-(2-(azepan-1- yl)ethyl)-1H-pyrazolo[3,4- d]py...)
Affinity DataKi:  16.4nMpH: 7.4Assay Description:Brain membrane preparation and binding assays for the σ1-receptor were performed as described (DeHaven-Hudkins, D. L., L. C. Fleissner, and F. Y...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Laboratorios Del Dr. Esteve

US Patent
LigandPNGBDBM287119(1-(1-(2-(Azepan-1- yl)ethyl)-1H- pyrazolo[3,4- d]p...)
Affinity DataKi:  21.2nMpH: 7.4Assay Description:Brain membrane preparation and binding assays for the σ1-receptor were performed as described (DeHaven-Hudkins, D. L., L. C. Fleissner, and F. Y...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Laboratorios Del Dr. Esteve

US Patent
LigandPNGBDBM287139(1-(1-(2-(azepan- 1-yl)ethyl)-1H- pyrazolo[3,4- d]p...)
Affinity DataKi:  21.8nMpH: 7.4Assay Description:Brain membrane preparation and binding assays for the σ1-receptor were performed as described (DeHaven-Hudkins, D. L., L. C. Fleissner, and F. Y...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Laboratorios Del Dr. Esteve

US Patent
LigandPNGBDBM393461(4-(azepan-1- yl)-1-(8- fluoro-3,4- dihydro- pyrazi...)
Affinity DataKi:  21.9nMAssay Description:To investigate binding properties of sigma 1 receptor ligands to human sigma 1 receptor, transfected HEK-293 membranes and [3H](+)-pentazocine (Perki...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Laboratorios Del Dr. Esteve

US Patent
LigandPNGBDBM393457(1-(8-fluoro- 3,4- dihydro- pyrazino[1,2- a]indol- ...)
Affinity DataKi:  22.2nMAssay Description:To investigate binding properties of sigma 1 receptor ligands to human sigma 1 receptor, transfected HEK-293 membranes and [3H](+)-pentazocine (Perki...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma non-opioid intracellular receptor 1(Mus musculus (Mouse))
Laboratorios Del Dr. Esteve

US Patent
LigandPNGBDBM50077892(CHEMBL3417067 | US9611229, 15)
Affinity DataKi:  23.3nMAssay Description:Brain membrane preparation and binding assays for the 61-receptor were performed as described (DeHaven-Hudkins, D. L., L. C. Fleissner, and F. Y. For...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Laboratorios Del Dr. Esteve

US Patent
LigandPNGBDBM287132(1-(1-(2-(azepan-1- yl)ethyl)-1H- pyrazolo[3,4- d]p...)
Affinity DataKi:  23.4nMpH: 7.4Assay Description:Brain membrane preparation and binding assays for the σ1-receptor were performed as described (DeHaven-Hudkins, D. L., L. C. Fleissner, and F. Y...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Laboratorios Del Dr. Esteve

US Patent
LigandPNGBDBM393455(1-(10-methyl- 3,4- dihydro- pyrazino[1,2- a]indol-...)
Affinity DataKi:  24nMAssay Description:To investigate binding properties of sigma 1 receptor ligands to human sigma 1 receptor, transfected HEK-293 membranes and [3H](+)-pentazocine (Perki...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Laboratorios Del Dr. Esteve

US Patent
LigandPNGBDBM287129(1-(1-(2-(azepan-1- yl)ethyl)-1H- pyrazolo[3,4- d]p...)
Affinity DataKi:  24nMpH: 7.4Assay Description:Brain membrane preparation and binding assays for the σ1-receptor were performed as described (DeHaven-Hudkins, D. L., L. C. Fleissner, and F. Y...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Laboratorios Del Dr. Esteve

US Patent
LigandPNGBDBM287093(N-(1-(2-(piperidin-1- yl)ethyl)-1H-pyrazolo[3,4- d...)
Affinity DataKi:  24.4nMpH: 7.4Assay Description:Brain membrane preparation and binding assays for the σ1-receptor were performed as described (DeHaven-Hudkins, D. L., L. C. Fleissner, and F. Y...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Laboratorios Del Dr. Esteve

US Patent
LigandPNGBDBM393448(2-(azepan-1- yl)-1-(3,4- dihydro- pyrazino[1,2- a]...)
Affinity DataKi:  24.8nMAssay Description:To investigate binding properties of sigma 1 receptor ligands to human sigma 1 receptor, transfected HEK-293 membranes and [3H](+)-pentazocine (Perki...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Laboratorios Del Dr. Esteve

US Patent
LigandPNGBDBM393451(2-(4- benzyl- piperidin-1-yl)- 1-(3,4- dihydro- py...)
Affinity DataKi:  25nMAssay Description:To investigate binding properties of sigma 1 receptor ligands to human sigma 1 receptor, transfected HEK-293 membranes and [3H](+)-pentazocine (Perki...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Laboratorios Del Dr. Esteve

US Patent
LigandPNGBDBM393466(2-(4- cyclohexyl- piperazin-1- yl)- 1-(8-fluoro- 3...)
Affinity DataKi:  25.6nMAssay Description:To investigate binding properties of sigma 1 receptor ligands to human sigma 1 receptor, transfected HEK-293 membranes and [3H](+)-pentazocine (Perki...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Laboratorios Del Dr. Esteve

US Patent
LigandPNGBDBM393456(2-(4- benzyl- piperidin- 1-yl)-1- (10-methyl- 3,4-...)
Affinity DataKi:  26.2nMAssay Description:To investigate binding properties of sigma 1 receptor ligands to human sigma 1 receptor, transfected HEK-293 membranes and [3H](+)-pentazocine (Perki...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Laboratorios Del Dr. Esteve

US Patent
LigandPNGBDBM287128(1-(1-(2-(azepan-1- yl)ethyl)-1H- pyrazolo[3,4- d]p...)
Affinity DataKi:  27.9nMpH: 7.4Assay Description:Brain membrane preparation and binding assays for the σ1-receptor were performed as described (DeHaven-Hudkins, D. L., L. C. Fleissner, and F. Y...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Laboratorios Del Dr. Esteve

US Patent
LigandPNGBDBM393460(1-(3,4- dihydro- pyrazino[1,2- a]indol- 2(1H)-yl)-...)
Affinity DataKi:  28.8nMAssay Description:To investigate binding properties of sigma 1 receptor ligands to human sigma 1 receptor, transfected HEK-293 membranes and [3H](+)-pentazocine (Perki...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Laboratorios Del Dr. Esteve

US Patent
LigandPNGBDBM287130(1-(1-(2-(azepan-1- yl)ethyl)-1H- pyrazolo[3,4- d]p...)
Affinity DataKi:  29nMpH: 7.4Assay Description:Brain membrane preparation and binding assays for the σ1-receptor were performed as described (DeHaven-Hudkins, D. L., L. C. Fleissner, and F. Y...More data for this Ligand-Target Pair
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TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Laboratorios Del Dr. Esteve

US Patent
LigandPNGBDBM393448(2-(azepan-1- yl)-1-(3,4- dihydro- pyrazino[1,2- a]...)
Affinity DataKi:  29.6nMAssay Description:To investigate binding properties of sigma 1 receptor ligands to human sigma 1 receptor, transfected HEK-293 membranes and [3H](+)-pentazocine (Perki...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetSigma non-opioid intracellular receptor 1(Mus musculus (Mouse))
Laboratorios Del Dr. Esteve

US Patent
LigandPNGBDBM50077878(CHEMBL3417043 | US9611229, 3)
Affinity DataKi:  31.1nMAssay Description:Brain membrane preparation and binding assays for the 61-receptor were performed as described (DeHaven-Hudkins, D. L., L. C. Fleissner, and F. Y. For...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSigma non-opioid intracellular receptor 1(Mus musculus (Mouse))
Laboratorios Del Dr. Esteve

US Patent
LigandPNGBDBM50077881(CHEMBL3417047 | US9611229, 47)
Affinity DataKi:  31.4nMAssay Description:Brain membrane preparation and binding assays for the 61-receptor were performed as described (DeHaven-Hudkins, D. L., L. C. Fleissner, and F. Y. For...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSigma non-opioid intracellular receptor 1(Mus musculus (Mouse))
Laboratorios Del Dr. Esteve

US Patent
LigandPNGBDBM50077889(CHEMBL3417061 | US9611229, 37)
Affinity DataKi:  32.7nMAssay Description:Brain membrane preparation and binding assays for the 61-receptor were performed as described (DeHaven-Hudkins, D. L., L. C. Fleissner, and F. Y. For...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Laboratorios Del Dr. Esteve

US Patent
LigandPNGBDBM287116(N-(1-(3-(azepan-1- yl)propyl)-1H-pyrazolo[3,4- d]p...)
Affinity DataKi:  32.7nMpH: 7.4Assay Description:Brain membrane preparation and binding assays for the σ1-receptor were performed as described (DeHaven-Hudkins, D. L., L. C. Fleissner, and F. Y...More data for this Ligand-Target Pair
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TargetSigma non-opioid intracellular receptor 1(Mus musculus (Mouse))
Laboratorios Del Dr. Esteve

US Patent
LigandPNGBDBM314373(1-(3-fluorophenyl)-N- (2-(pyrrolidin-1- yl)ethyl)-...)
Affinity DataKi:  34.6nMAssay Description:Brain membrane preparation and binding assays for the 61-receptor were performed as described (DeHaven-Hudkins, D. L., L. C. Fleissner, and F. Y. For...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetSigma non-opioid intracellular receptor 1(Mus musculus (Mouse))
Laboratorios Del Dr. Esteve

US Patent
LigandPNGBDBM314290(1-(3,4- dichlorobenzyl)-N- (3-(piperidin-1- yl)pro...)
Affinity DataKi:  34.8nMAssay Description:Brain membrane preparation and binding assays for the 61-receptor were performed as described (DeHaven-Hudkins, D. L., L. C. Fleissner, and F. Y. For...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma non-opioid intracellular receptor 1(Mus musculus (Mouse))
Laboratorios Del Dr. Esteve

US Patent
LigandPNGBDBM50077888(CHEMBL3417060 | US9611229, 18)
Affinity DataKi:  35.4nMAssay Description:Brain membrane preparation and binding assays for the 61-receptor were performed as described (DeHaven-Hudkins, D. L., L. C. Fleissner, and F. Y. For...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSigma non-opioid intracellular receptor 1(Mus musculus (Mouse))
Laboratorios Del Dr. Esteve

US Patent
LigandPNGBDBM50077883(CHEMBL3417054 | US9611229, 32)
Affinity DataKi:  36.3nMAssay Description:Brain membrane preparation and binding assays for the 61-receptor were performed as described (DeHaven-Hudkins, D. L., L. C. Fleissner, and F. Y. For...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Laboratorios Del Dr. Esteve

US Patent
LigandPNGBDBM393463(2-(4- cyclohexyl- piperazin-1- yl)- 1-(3,4- dihydr...)
Affinity DataKi:  37.6nMAssay Description:To investigate binding properties of sigma 1 receptor ligands to human sigma 1 receptor, transfected HEK-293 membranes and [3H](+)-pentazocine (Perki...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Laboratorios Del Dr. Esteve

US Patent
LigandPNGBDBM393446(1-(3,4- dihydro- pyrazino[1,2- a]indol- 2(1H)-yl)-...)
Affinity DataKi:  39.8nMAssay Description:To investigate binding properties of sigma 1 receptor ligands to human sigma 1 receptor, transfected HEK-293 membranes and [3H](+)-pentazocine (Perki...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Laboratorios Del Dr. Esteve

US Patent
LigandPNGBDBM287126(1-(1-(2-(azepan-1- yl)ethyl)-1H- pyrazolo[3,4- d]p...)
Affinity DataKi:  41.4nMpH: 7.4Assay Description:Brain membrane preparation and binding assays for the σ1-receptor were performed as described (DeHaven-Hudkins, D. L., L. C. Fleissner, and F. Y...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
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