TargetVesicular acetylcholine transporter(Torpedo californica)
University of Minnesota
Curated by ChEMBL
University of Minnesota
Curated by ChEMBL
Affinity DataKi: 0.00650nMAssay Description:In vitro binding affinity to vesamicol receptor using [3H]-vesamicol.More data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University of Minnesota
Curated by ChEMBL
University of Minnesota
Curated by ChEMBL
Affinity DataKi: 0.0500nMAssay Description:In vitro binding affinity to vesamicol receptor using [3H]-vesamicol.More data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University of Minnesota
Curated by ChEMBL
University of Minnesota
Curated by ChEMBL
Affinity DataKi: 0.0550nMAssay Description:In vitro binding affinity to vesamicol receptor using [3H]-vesamicol.More data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University of Minnesota
Curated by ChEMBL
University of Minnesota
Curated by ChEMBL
Affinity DataKi: 0.0630nMAssay Description:In vitro binding affinity to vesamicol receptor using [3H]-vesamicol.More data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University of Minnesota
Curated by ChEMBL
University of Minnesota
Curated by ChEMBL
Affinity DataKi: 0.121nMAssay Description:In vitro binding affinity to vesamicol receptor using [3H]-vesamicol.More data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University of Minnesota
Curated by ChEMBL
University of Minnesota
Curated by ChEMBL
Affinity DataKi: 0.147nMAssay Description:In vitro binding affinity to vesamicol receptor using [3H]-vesamicol.More data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University of Minnesota
Curated by ChEMBL
University of Minnesota
Curated by ChEMBL
Affinity DataKi: 0.212nMAssay Description:In vitro binding affinity to vesamicol receptor using [3H]-vesamicol.More data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University of Minnesota
Curated by ChEMBL
University of Minnesota
Curated by ChEMBL
Affinity DataKi: 0.248nMAssay Description:In vitro binding affinity to vesamicol receptor using [3H]-vesamicol.More data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University of Minnesota
Curated by ChEMBL
University of Minnesota
Curated by ChEMBL
Affinity DataKi: 0.264nMAssay Description:In vitro binding affinity to vesamicol receptor using [3H]-vesamicol.More data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University of Minnesota
Curated by ChEMBL
University of Minnesota
Curated by ChEMBL
Affinity DataKi: 0.271nMAssay Description:In vitro binding affinity to vesamicol receptor using [3H]-vesamicol.More data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University of Minnesota
Curated by ChEMBL
University of Minnesota
Curated by ChEMBL
Affinity DataKi: 0.360nMAssay Description:In vitro binding affinity to vesamicol receptor using [3H]-vesamicol.More data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University of Minnesota
Curated by ChEMBL
University of Minnesota
Curated by ChEMBL
Affinity DataKi: 0.360nMAssay Description:In vitro binding affinity to vesamicol receptor using [3H]-vesamicol.More data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University of Minnesota
Curated by ChEMBL
University of Minnesota
Curated by ChEMBL
Affinity DataKi: 0.410nMAssay Description:In vitro binding affinity to vesamicol receptor using [3H]-vesamicol.More data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University of Minnesota
Curated by ChEMBL
University of Minnesota
Curated by ChEMBL
Affinity DataKi: 0.638nMAssay Description:In vitro binding affinity to vesamicol receptor using [3H]-vesamicol.More data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University of Minnesota
Curated by ChEMBL
University of Minnesota
Curated by ChEMBL
Affinity DataKi: 0.660nMAssay Description:In vitro binding affinity to vesamicol receptor using [3H]-vesamicol.More data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University of Minnesota
Curated by ChEMBL
University of Minnesota
Curated by ChEMBL
Affinity DataKi: 0.762nMAssay Description:In vitro binding affinity to vesamicol receptor using [3H]-vesamicol.More data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University of Minnesota
Curated by ChEMBL
University of Minnesota
Curated by ChEMBL
Affinity DataKi: 0.798nMAssay Description:In vitro binding affinity to vesamicol receptor using [3H]-vesamicol.More data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University of Minnesota
Curated by ChEMBL
University of Minnesota
Curated by ChEMBL
Affinity DataKi: 0.800nMAssay Description:In vitro binding affinity to vesamicol receptor using [3H]-vesamicol.More data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University of Minnesota
Curated by ChEMBL
University of Minnesota
Curated by ChEMBL
Affinity DataKi: 0.856nMAssay Description:In vitro binding affinity to vesamicol receptor using [3H]-vesamicol.More data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University of Minnesota
Curated by ChEMBL
University of Minnesota
Curated by ChEMBL
Affinity DataKi: 0.980nMAssay Description:In vitro binding affinity to vesamicol receptor using [3H]-vesamicol.More data for this Ligand-Target Pair
Affinity DataKi: 0.990nMAssay Description:Tested for binding affinity against dopamine receptor D3 expressed in Sf9 cells.More data for this Ligand-Target Pair
Affinity DataKi: 0.990nMAssay Description:Tested for the inhibitory activity against Dopamine D3 receptor in infected Sf9 cellsMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University of Minnesota
Curated by ChEMBL
University of Minnesota
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:In vitro binding affinity to vesamicol receptor using [3H]-vesamicol.More data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Tested for binding affinity against dopamine receptor D3 expressed in Sf9 cells.More data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University of Minnesota
Curated by ChEMBL
University of Minnesota
Curated by ChEMBL
Affinity DataKi: 1.40nMAssay Description:In vitro binding affinity to vesamicol receptor using [3H]-vesamicol.More data for this Ligand-Target Pair
Affinity DataKi: 1.68nMAssay Description:tested for the inhibitory activity against sigma receptor rat cerebellarMore data for this Ligand-Target Pair
Affinity DataKi: 1.85nMAssay Description:Tested for the inhibitory activity against Dopamine D3 receptor in infected Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Tested for inhibition of the binding of [125I]NCQ298 to dopamine receptor D3More data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Tested for the inhibitory activity against Dopamine D3 receptor in infected Sf9 cellsMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University of Minnesota
Curated by ChEMBL
University of Minnesota
Curated by ChEMBL
Affinity DataKi: 2.60nMAssay Description:In vitro binding affinity to vesamicol receptor using [3H]-vesamicol.More data for this Ligand-Target Pair
Affinity DataKi: 2.90nMAssay Description:Tested for inhibition of the binding of [125I]NCQ298 to dopamine receptor D3More data for this Ligand-Target Pair
Affinity DataKi: 2.90nMAssay Description:Tested for the inhibitory activity against Dopamine D3 receptor in infected Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.20nMAssay Description:Tested for the inhibitory activity against sigma receptor rat cerebellarMore data for this Ligand-Target Pair
Affinity DataKi: 3.60nMAssay Description:Tested for the inhibitory activity against D2H (high-affinity states) receptor in infected HEK 293 cells.More data for this Ligand-Target Pair
Affinity DataKi: 3.90nMAssay Description:Tested for binding affinity against dopamine receptor D3 expressed in Sf9 cells.More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
University of Pennsylvania
Curated by ChEMBL
University of Pennsylvania
Curated by ChEMBL
Affinity DataKi: 5.10nMAssay Description:Tested for the inhibitory activity against 5-hydroxytryptamine 1A receptor in rat hippocampalMore data for this Ligand-Target Pair
Affinity DataKi: 5.70nMAssay Description:Tested for binding affinity against dopamine receptor D3 expressed in Sf9 cells.More data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University of Minnesota
Curated by ChEMBL
University of Minnesota
Curated by ChEMBL
Affinity DataKi: 5.80nMAssay Description:In vitro binding affinity to vesamicol receptor using [3H]-vesamicol.More data for this Ligand-Target Pair
Affinity DataKi: 6.60nMAssay Description:Tested for the inhibitory activity against D2H (high-affinity states) receptor in infected HEK 293 cells.More data for this Ligand-Target Pair
Affinity DataKi: 6.69nMAssay Description:Tested for the inhibitory activity against Dopamine D3 receptor in infected Sf9 cellsMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University of Minnesota
Curated by ChEMBL
University of Minnesota
Curated by ChEMBL
Affinity DataKi: 6.93nMAssay Description:In vitro binding affinity to vesamicol receptor using [3H]-vesamicol.More data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University of Minnesota
Curated by ChEMBL
University of Minnesota
Curated by ChEMBL
Affinity DataKi: 7.59nMAssay Description:In vitro binding affinity to vesamicol receptor using [3H]-vesamicol.More data for this Ligand-Target Pair
Affinity DataKi: 8.90nMAssay Description:Inhibition of human carbonic anhydrase 2 preincubated for 10 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Inhibition of human carbonic anhydrase 2 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataKi: 9.10nMAssay Description:Inhibition of human carbonic anhydrase 2 preincubated for 10 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
Affinity DataKi: 9.30nMAssay Description:Tested for binding affinity against dopamine receptor D3 expressed in Sf9 cells.More data for this Ligand-Target Pair
Affinity DataKi: 9.60nMAssay Description:Inhibition of human carbonic anhydrase 2 preincubated for 10 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
Affinity DataKi: 9.70nMAssay Description:Tested for the inhibitory activity against D2H (high-affinity states) receptor in infected HEK 293 cells.More data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Inhibition of human carbonic anhydrase 2 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Inhibition of human carbonic anhydrase 2 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
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