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Found 62 with Last Name = 'szabó' and Initial = 'c'
TargetAdenosine receptor A1(Homo sapiens (Human))
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50085658((2R,3R,4S,5R)-2-(2-Chloro-6-cyclopentylamino-purin...)
Affinity DataKi:  0.830nMAssay Description:Displacement of [3H]-CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50141447(CHEMBL279391 | N-[6-Cyclopentylamino-9-((2R,3R,4S,...)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]-CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50141452(3-Cyclopentyl-N-[6-cyclopentylamino-9-((2R,3R,4S,5...)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]-CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50085658((2R,3R,4S,5R)-2-(2-Chloro-6-cyclopentylamino-purin...)
Affinity DataKi:  42nMAssay Description:Displacement of [3H]-NECA from human adenosine A3 receptor in stably transfected HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50141455(CHEMBL285251 | N-[6-Amino-9-((2R,3R,4S,5R)-3,4-dih...)
Affinity DataKi:  71nMAssay Description:Displacement of [3H]-CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50141453(2-Cyclohexyl-N-[9-((2R,3R,4S,5R)-3,4-dihydroxy-5-h...)
Affinity DataKi:  181nMAssay Description:Displacement of [3H]-NECA from human adenosine A3 receptor in stably transfected HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50141453(2-Cyclohexyl-N-[9-((2R,3R,4S,5R)-3,4-dihydroxy-5-h...)
Affinity DataKi:  207nMAssay Description:Displacement of [3H]-CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50141451(CHEMBL36786 | N-[6-Amino-9-((2R,3R,4S,5R)-3,4-dihy...)
Affinity DataKi:  252nMAssay Description:Displacement of [3H]-CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50141449(CHEMBL36789 | N-[6-Amino-9-((2R,3R,4S,5R)-3,4-dihy...)
Affinity DataKi:  342nMAssay Description:Displacement of [3H]-CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50141456(CHEMBL289982 | N-[6-Amino-9-((2R,3R,4S,5R)-3,4-dih...)
Affinity DataKi:  432nMAssay Description:Displacement of [3H]-CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50141450(CHEMBL36320 | N-[6-Amino-9-((2R,3R,4S,5R)-3,4-dihy...)
Affinity DataKi:  733nMAssay Description:Displacement of [3H]-CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50141455(CHEMBL285251 | N-[6-Amino-9-((2R,3R,4S,5R)-3,4-dih...)
Affinity DataKi:  900nMAssay Description:Displacement of [3H]-NECA from human adenosine A3 receptor in stably transfected HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50141448((2S,3S,4R,5R)-5-[6-Amino-2-(3-cyclopentyl-propiony...)
Affinity DataKi:  1.01E+3nMAssay Description:Displacement of [3H]-NECA from human adenosine A3 receptor in stably transfected HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50141451(CHEMBL36786 | N-[6-Amino-9-((2R,3R,4S,5R)-3,4-dihy...)
Affinity DataKi:  1.04E+3nMAssay Description:Displacement of [3H]-NECA from human adenosine A3 receptor in stably transfected HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50141450(CHEMBL36320 | N-[6-Amino-9-((2R,3R,4S,5R)-3,4-dihy...)
Affinity DataKi:  1.06E+3nMAssay Description:Displacement of [3H]-NECA from human adenosine A3 receptor in stably transfected HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50141449(CHEMBL36789 | N-[6-Amino-9-((2R,3R,4S,5R)-3,4-dihy...)
Affinity DataKi:  1.23E+3nMAssay Description:Displacement of [3H]-NECA from human adenosine A3 receptor in stably transfected HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50141447(CHEMBL279391 | N-[6-Cyclopentylamino-9-((2R,3R,4S,...)
Affinity DataKi:  1.25E+3nMAssay Description:Displacement of [3H]-NECA from human adenosine A3 receptor in stably transfected HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50141452(3-Cyclopentyl-N-[6-cyclopentylamino-9-((2R,3R,4S,5...)
Affinity DataKi:  1.41E+3nMAssay Description:Displacement of [3H]-NECA from human adenosine A3 receptor in stably transfected HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50141454(CHEMBL288258 | Cyclohexanecarboxylic acid [6-amino...)
Affinity DataKi:  1.62E+3nMAssay Description:Displacement of [3H]-CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50141454(CHEMBL288258 | Cyclohexanecarboxylic acid [6-amino...)
Affinity DataKi:  1.78E+3nMAssay Description:Displacement of [3H]-NECA from human adenosine A2A receptor in stably transfected CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50141450(CHEMBL36320 | N-[6-Amino-9-((2R,3R,4S,5R)-3,4-dihy...)
Affinity DataKi:  1.94E+3nMAssay Description:Displacement of [3H]-NECA from human adenosine A2A receptor in stably transfected CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50141451(CHEMBL36786 | N-[6-Amino-9-((2R,3R,4S,5R)-3,4-dihy...)
Affinity DataKi:  2.00E+3nMAssay Description:Displacement of [3H]-NECA from human adenosine A2A receptor in stably transfected CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50141452(3-Cyclopentyl-N-[6-cyclopentylamino-9-((2R,3R,4S,5...)
Affinity DataKi:  2.18E+3nMAssay Description:Displacement of [3H]-NECA from human adenosine A2A receptor in stably transfected CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50085658((2R,3R,4S,5R)-2-(2-Chloro-6-cyclopentylamino-purin...)
Affinity DataKi:  2.27E+3nMAssay Description:Displacement of [3H]-NECA from human adenosine A2A receptor in stably transfected CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50141449(CHEMBL36789 | N-[6-Amino-9-((2R,3R,4S,5R)-3,4-dihy...)
Affinity DataKi:  2.41E+3nMAssay Description:Displacement of [3H]-NECA from human adenosine A2A receptor in stably transfected CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50141456(CHEMBL289982 | N-[6-Amino-9-((2R,3R,4S,5R)-3,4-dih...)
Affinity DataKi:  2.71E+3nMAssay Description:Displacement of [3H]-NECA from human adenosine A3 receptor in stably transfected HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50141454(CHEMBL288258 | Cyclohexanecarboxylic acid [6-amino...)
Affinity DataKi:  2.76E+3nMAssay Description:Displacement of [3H]-NECA from human adenosine A3 receptor in stably transfected HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50141455(CHEMBL285251 | N-[6-Amino-9-((2R,3R,4S,5R)-3,4-dih...)
Affinity DataKi:  4.10E+3nMAssay Description:Displacement of [3H]-NECA from human adenosine A2A receptor in stably transfected CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50141456(CHEMBL289982 | N-[6-Amino-9-((2R,3R,4S,5R)-3,4-dih...)
Affinity DataKi:  4.57E+3nMAssay Description:Displacement of [3H]-NECA from human adenosine A2A receptor in stably transfected CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50141448((2S,3S,4R,5R)-5-[6-Amino-2-(3-cyclopentyl-propiony...)
Affinity DataKi:  5.45E+3nMAssay Description:Displacement of [3H]-CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50141447(CHEMBL279391 | N-[6-Cyclopentylamino-9-((2R,3R,4S,...)
Affinity DataKi:  5.66E+3nMAssay Description:Displacement of [3H]-NECA from human adenosine A2A receptor in stably transfected CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50141453(2-Cyclohexyl-N-[9-((2R,3R,4S,5R)-3,4-dihydroxy-5-h...)
Affinity DataKi:  7.75E+3nMAssay Description:Displacement of [3H]-NECA from human adenosine A2A receptor in stably transfected CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50141448((2S,3S,4R,5R)-5-[6-Amino-2-(3-cyclopentyl-propiony...)
Affinity DataKi:  1.08E+4nMAssay Description:Displacement of [3H]-NECA from human adenosine A2A receptor in stably transfected CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Mus musculus)
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50322362(2-(4-((2S,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-3,4-...)
Affinity DataIC50:  45nMAssay Description:Tested for inhibition of poly(ADP-ribose) polymerase-1 (PARP-1) in mouse using Cell protection assayMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Mus musculus)
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50366893(CHEMBL607649)
Affinity DataIC50:  100nMAssay Description:Tested for inhibition of poly(ADP-ribose) polymerase-1 (PARP-1) in mouse using Cell protection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Mus musculus)
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50366900(CHEMBL608792)
Affinity DataIC50:  250nMAssay Description:Tested for inhibition of poly(ADP-ribose) polymerase-1 (PARP-1) in mouse using Cell protection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Mus musculus)
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50366902(CHEMBL607648)
Affinity DataIC50:  450nMAssay Description:Tested for inhibition of poly(ADP-ribose) polymerase-1 (PARP-1) in mouse using Cell protection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Mus musculus)
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50366904(CHEMBL607928)
Affinity DataIC50:  700nMAssay Description:Tested for inhibition of poly(ADP-ribose) polymerase-1 (PARP-1) in mouse using Cell protection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Mus musculus)
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50366895(CHEMBL607633)
Affinity DataIC50:  700nMAssay Description:Tested for inhibition of poly(ADP-ribose) polymerase-1 (PARP-1) in mouse using Cell protection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Mus musculus)
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50366901(CHEMBL608232)
Affinity DataIC50:  900nMAssay Description:Tested for inhibition of poly(ADP-ribose) polymerase-1 (PARP-1) in mouse using Cell protection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Mus musculus)
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50366897(CHEMBL607650)
Affinity DataIC50:  1.90E+3nMAssay Description:Tested for inhibition of poly(ADP-ribose) polymerase-1 (PARP-1) in mouse using Cell protection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Mus musculus)
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50366898(CHEMBL608784)
Affinity DataIC50:  2.00E+3nMAssay Description:Tested for inhibition of poly(ADP-ribose) polymerase-1 (PARP-1) in mouse using Cell protection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Mus musculus)
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50366903(CHEMBL607634)
Affinity DataIC50:  3.00E+3nMAssay Description:Tested for inhibition of poly(ADP-ribose) polymerase-1 (PARP-1) in mouse using Cell protection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Mus musculus)
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50366892(CHEMBL608783)
Affinity DataIC50:  3.00E+3nMAssay Description:Tested for inhibition of poly(ADP-ribose) polymerase-1 (PARP-1) in mouse using Cell protection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Mus musculus)
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50137382(2-(6-Methylamino-purin-9-yl)-N-(1-oxo-2,3-dihydro-...)
Affinity DataIC50:  3.00E+3nMAssay Description:Tested for inhibition of poly(ADP-ribose) polymerase-1 (PARP-1) in mouse using Cell protection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Mus musculus)
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50137371(2-Benzoimidazol-1-yl-N-(1-oxo-2,3-dihydro-1H-isoin...)
Affinity DataIC50:  3.00E+3nMAssay Description:Tested for inhibition of poly(ADP-ribose) polymerase-1 (PARP-1) in mouse using Cell protection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Mus musculus)
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50137378(CHEMBL424399 | N-[(3S,4R)-5-(6-Amino-purin-9-yl)-3...)
Affinity DataIC50:  5.00E+3nMAssay Description:Tested for inhibition of poly(ADP-ribose) polymerase-1 (PARP-1) in mouse using Cell protection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Mus musculus)
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50366899(CHEMBL607657)
Affinity DataIC50:  1.00E+4nMAssay Description:Tested for inhibition of poly(ADP-ribose) polymerase-1 (PARP-1) in mouse using Cell protection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Mus musculus)
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50137359(2-Ethylamino-N-(1-oxo-2,3-dihydro-1H-isoindol-4-yl...)
Affinity DataIC50:  1.80E+4nMAssay Description:Tested for inhibition of poly(ADP-ribose) polymerase-1 (PARP-1) in mouse using Cell protection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Mus musculus)
Inotek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50137376(CHEMBL537836 | N-(1-Oxo-2,3-dihydro-1H-isoindol-4-...)
Affinity DataIC50:  1.80E+4nMAssay Description:Tested for inhibition of poly(ADP-ribose) polymerase-1 (PARP-1) in mouse using Cell protection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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