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Found 29 with Last Name = 'tapparelli' and Initial = 'c'
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291335((R)-7-(4-Carbamimidoyl-benzoylamino)-3-[3-(4-metho...)
Affinity DataIC50:  0.360nMAssay Description:Inhibition of fibrinogen binding to immobilized human glycoprotein alpha IIb beta3 integrinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291333((R)-7-(4-Carbamimidoyl-benzoylamino)-3-(2-naphthal...)
Affinity DataIC50:  0.360nMAssay Description:Inhibition of fibrinogen binding to GPllb/IIIa receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291336((S)-3-(3-Adamantan-1-yl-propionylamino)-6-[2-(4-ca...)
Affinity DataIC50:  0.370nMAssay Description:Inhibition of fibrinogen binding to immobilized human glycoprotein alpha IIb beta3 integrinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291340((R)-7-(4-Carbamimidoyl-benzoylamino)-3-(3-methyl-b...)
Affinity DataIC50:  0.540nMAssay Description:Inhibition of fibrinogen binding to immobilized human glycoprotein alpha IIb beta3 integrinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291334((R)-7-(4-Carbamimidoyl-benzoylamino)-3-[2-(4-metho...)
Affinity DataIC50:  1nMAssay Description:Inhibition of fibrinogen binding to immobilized human glycoprotein alpha IIb beta3 integrinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291337((S)-6-[2-(4-Carbamimidoyl-phenyl)-acetylamino]-3-[...)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of fibrinogen binding to immobilized human glycoprotein alpha IIb beta3 integrinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291339((S)-6-[2-(4-Carbamimidoyl-phenyl)-acetylamino]-3-(...)
Affinity DataIC50:  1.70nMAssay Description:Inhibition of fibrinogen binding to immobilized human glycoprotein alpha IIb beta3 integrinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282124((S)-N-((S)-Adamantan-1-yl-carboxy-methyl)-3-{(S)-3...)
Affinity DataIC50:  2nMAssay Description:Inhibition of fibrinogen binding to purified immobilized alpha IIb beta3 integrin isolated from membranes of human blood platelets.More data for this Ligand-Target Pair
In DepthDetails Article
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291342((S)-3-(2-Adamantan-1-yl-acetylamino)-6-[2-(4-carba...)
Affinity DataIC50:  2.20nMAssay Description:Inhibition of fibrinogen binding to immobilized human glycoprotein alpha IIb beta3 integrinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282126((S)-N-((S)-2-Adamantan-1-yl-1-carboxy-ethyl)-3-{(S...)
Affinity DataIC50:  5nMAssay Description:Inhibition of fibrinogen binding to purified immobilized alpha IIb beta3 integrin isolated from membranes of human blood platelets.More data for this Ligand-Target Pair
In DepthDetails Article
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291338((S)-6-[2-(4-Carbamimidoyl-phenyl)-acetylamino]-3-(...)
Affinity DataIC50:  7.60nMAssay Description:Inhibition of fibrinogen binding to immobilized human glycoprotein alpha IIb beta3 integrinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291331((S)-6-[2-(4-Carbamimidoyl-phenyl)-acetylamino]-3-i...)
Affinity DataIC50:  7.90nMAssay Description:Inhibition of fibrinogen binding to immobilized human glycoprotein alpha IIb beta3 integrinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282121((S)-3-{(S)-3-[2-(4-Carbamimidoyl-phenyl)-acetylami...)
Affinity DataIC50:  20nMAssay Description:Inhibition of fibrinogen binding to purified immobilized alpha IIb beta3 integrin isolated from membranes of human blood platelets.More data for this Ligand-Target Pair
In DepthDetails Article
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282119((S)-N-((S)-2-Adamantan-1-yl-1-methoxycarbonyl-ethy...)
Affinity DataIC50:  20nMAssay Description:Inhibition of fibrinogen binding to purified immobilized alpha IIb beta3 integrin isolated from membranes of human blood platelets.More data for this Ligand-Target Pair
In DepthDetails Article
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282122((S)-2-((S)-2-{(S)-3-[2-(4-Carbamimidoyl-phenyl)-ac...)
Affinity DataIC50:  40nMAssay Description:Inhibition of fibrinogen binding to purified immobilized alpha IIb beta3 integrin isolated from membranes of human blood platelets.More data for this Ligand-Target Pair
In DepthDetails Article
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282116((S)-2-{(S)-2-[2-((S)-2-Benzyloxycarbonylamino-5-gu...)
Affinity DataIC50:  110nMAssay Description:Inhibition of fibrinogen binding to purified immobilized alpha IIb beta3 integrin isolated from membranes of human blood platelets.More data for this Ligand-Target Pair
In DepthDetails Article
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282127((S)-3-{(S)-3-[2-(4-Carbamimidoyl-phenyl)-acetylami...)
Affinity DataIC50:  120nMAssay Description:Inhibition of fibrinogen binding to purified immobilized alpha IIb beta3 integrin isolated from membranes of human blood platelets.More data for this Ligand-Target Pair
In DepthDetails Article
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282132((S)-3-[2-((S)-2-Benzyloxycarbonylamino-5-guanidino...)
Affinity DataIC50:  270nMAssay Description:Inhibition of fibrinogen binding to purified immobilized alpha IIb beta3 integrin isolated from membranes of human blood platelets.More data for this Ligand-Target Pair
In DepthDetails Article
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282120((S)-N-((S)-2-Adamantan-1-yl-1-methoxycarbonyl-ethy...)
Affinity DataIC50:  510nMAssay Description:Inhibition of fibrinogen binding to purified immobilized alpha IIb beta3 integrin isolated from membranes of human blood platelets.More data for this Ligand-Target Pair
In DepthDetails Article
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282117((S)-2-{(S)-2-[(S)-3-((S)-2-Benzyloxycarbonylamino-...)
Affinity DataIC50:  560nMAssay Description:Inhibition of fibrinogen binding to purified immobilized alpha IIb beta3 integrin isolated from membranes of human blood platelets.More data for this Ligand-Target Pair
In DepthDetails Article
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282129((S)-3-[(S)-3-((S)-2-Benzyloxycarbonylamino-5-guani...)
Affinity DataIC50:  770nMAssay Description:Inhibition of fibrinogen binding to purified immobilized alpha IIb beta3 integrin isolated from membranes of human blood platelets.More data for this Ligand-Target Pair
In DepthDetails Article
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282130((S)-3-[(S)-3-((S)-2-Benzyloxycarbonylamino-5-guani...)
Affinity DataIC50:  1.07E+3nMAssay Description:Inhibition of fibrinogen binding to purified immobilized alpha IIb beta3 integrin isolated from membranes of human blood platelets.More data for this Ligand-Target Pair
In DepthDetails Article
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282131((S)-3-[(S)-3-((S)-2-Benzyloxycarbonylamino-5-guani...)
Affinity DataIC50:  1.22E+3nMAssay Description:Inhibition of fibrinogen binding to purified immobilized alpha IIb beta3 integrin isolated from membranes of human blood platelets.More data for this Ligand-Target Pair
In DepthDetails Article
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291332(CHEMBL162760 | Ornithine sulfonamide)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of fibrinogen binding to immobilized human glycoprotein alpha IIb beta3 integrinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291341((S)-5-[2-(4-Carbamimidoyl-phenyl)-acetylamino]-2-(...)
Affinity DataIC50:  4.80E+4nMAssay Description:Inhibition of fibrinogen binding to immobilized human glycoprotein alpha IIb beta3 integrinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282118((S)-3-[(S)-2-((S)-2-Benzyloxycarbonylamino-5-guani...)
Affinity DataIC50:  7.80E+4nMAssay Description:Inhibition of fibrinogen binding to purified immobilized alpha IIb beta3 integrin isolated from membranes of human blood platelets.More data for this Ligand-Target Pair
In DepthDetails Article
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282125((S)-3-[(R)-3-((S)-2-Benzyloxycarbonylamino-5-guani...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of fibrinogen binding to purified immobilized alpha IIb beta3 integrin isolated from membranes of human blood platelets.More data for this Ligand-Target Pair
In DepthDetails Article
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282128((S)-2-((R)-2-{(S)-3-[2-(4-Carbamimidoyl-phenyl)-ac...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of fibrinogen binding to purified immobilized alpha IIb beta3 integrin isolated from membranes of human blood platelets.More data for this Ligand-Target Pair
In DepthDetails Article
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282123((S)-3-[(R)-2-((S)-2-Benzyloxycarbonylamino-5-guani...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of fibrinogen binding to purified immobilized alpha IIb beta3 integrin isolated from membranes of human blood platelets.More data for this Ligand-Target Pair
In DepthDetails Article