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Found 57 with Last Name = 'pearce' and Initial = 'cj'
TargetMitogen-activated protein kinase kinase kinase 7(Homo sapiens (Human))
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50042034((5Z)-7-Oxozeaenol | 5Z-7-Oxozeaenol | CHEBI:67559 ...)
Affinity DataIC50:  8.10nMAssay Description:Inhibition of TAK1 (unknown origin) expressed in sf9 cells assessed as 32P level incorporation into myelin basic protein incubated for 5 mins at 30 d...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 7(Homo sapiens (Human))
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50042034((5Z)-7-Oxozeaenol | 5Z-7-Oxozeaenol | CHEBI:67559 ...)
Affinity DataIC50:  11nMAssay Description:Inhibition of TAK1 (unknown origin)More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 2 group C member 2/TGF-beta-activated kinase 1 and MAP3K7-binding protein 1(Homo sapiens (Human))
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50129131(CHEBI:83275 | Hypothemycin | US10434085, Compound ...)
Affinity DataIC50:  30nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged TAK1 (1 to 303 residues)/TAB1 (437 to end residues) expressed in baculovirus infected Sf9 insec...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMitogen-activated protein kinase kinase kinase 7(Homo sapiens (Human))
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50129131(CHEBI:83275 | Hypothemycin | US10434085, Compound ...)
Affinity DataIC50:  33nMAssay Description:Inhibition of TAK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscription factor p65(Homo sapiens (Human))
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50196926(CHEMBL438139 | Rocaglamide | US10085988, Compound ...)
Affinity DataIC50:  75nMAssay Description:Inhibition of NFkappa p65 isolated from nuclear extract of human HeLa cells by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 7(Homo sapiens (Human))
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50129130(CHEMBL3629241)
Affinity DataIC50:  77nMAssay Description:Inhibition of TAK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50593519(CHEMBL5204252)
Affinity DataIC50:  96nMAssay Description:Inhibition of chymotrypsin-like activity of human erythrocytes 20S proteasome using Suc-LLVY-AMC as substrate and measured by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTranscription factor p65(Homo sapiens (Human))
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50336457((3S,5Z,8S,9R,11E)-8,9,16-trihydroxy-14-methoxy-3-m...)
Affinity DataIC50:  250nMAssay Description:Inhibition of NFkappa p65 isolated from nuclear extract of human HeLa cells by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 7(Homo sapiens (Human))
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50129129(CHEMBL3629242 | US10434085, Compound 7)
Affinity DataIC50:  360nMAssay Description:Inhibition of TAK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 7(Homo sapiens (Human))
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50129128(CHEMBL3629243 | US10434085, Compound 10)
Affinity DataIC50:  380nMAssay Description:Inhibition of TAK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 2 group C member 2/TGF-beta-activated kinase 1 and MAP3K7-binding protein 1(Homo sapiens (Human))
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50594358(CHEMBL5204235)
Affinity DataIC50:  380nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged TAK1 (1 to 303 residues)/TAB1 (437 to end residues) expressed in baculovirus infected Sf9 insec...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNuclear receptor subfamily 2 group C member 2/TGF-beta-activated kinase 1 and MAP3K7-binding protein 1(Homo sapiens (Human))
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50594353(CHEMBL5174288)
Affinity DataIC50:  430nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged TAK1 (1 to 303 residues)/TAB1 (437 to end residues) expressed in baculovirus infected Sf9 insec...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNuclear receptor subfamily 2 group C member 2/TGF-beta-activated kinase 1 and MAP3K7-binding protein 1(Homo sapiens (Human))
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50594354(CHEMBL5186931)
Affinity DataIC50:  450nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged TAK1 (1 to 303 residues)/TAB1 (437 to end residues) expressed in baculovirus infected Sf9 insec...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNuclear receptor subfamily 2 group C member 2/TGF-beta-activated kinase 1 and MAP3K7-binding protein 1(Homo sapiens (Human))
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50594367(CHEMBL5207996)
Affinity DataIC50:  500nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged TAK1 (1 to 303 residues)/TAB1 (437 to end residues) expressed in baculovirus infected Sf9 insec...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNuclear receptor subfamily 2 group C member 2/TGF-beta-activated kinase 1 and MAP3K7-binding protein 1(Homo sapiens (Human))
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50594360(CHEMBL5173905)
Affinity DataIC50:  630nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged TAK1 (1 to 303 residues)/TAB1 (437 to end residues) expressed in baculovirus infected Sf9 insec...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNuclear receptor subfamily 2 group C member 2/TGF-beta-activated kinase 1 and MAP3K7-binding protein 1(Homo sapiens (Human))
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50594364(CHEMBL5185893)
Affinity DataIC50:  700nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged TAK1 (1 to 303 residues)/TAB1 (437 to end residues) expressed in baculovirus infected Sf9 insec...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNuclear receptor subfamily 2 group C member 2/TGF-beta-activated kinase 1 and MAP3K7-binding protein 1(Homo sapiens (Human))
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50594356(CHEMBL5179846)
Affinity DataIC50:  720nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged TAK1 (1 to 303 residues)/TAB1 (437 to end residues) expressed in baculovirus infected Sf9 insec...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTranscription factor p65(Homo sapiens (Human))
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50347543(CHEMBL1801948)
Affinity DataIC50:  750nMAssay Description:Inhibition of NFkappa p65 isolated from nuclear extract of human HeLa cells by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase 2A(Homo sapiens (Human))
University of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50530867(CHEMBL4472654)
Affinity DataIC50:  800nMAssay Description:Inhibition of human recombinant MLL1 using [3H]S-adenosyl-methionine as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase 2A(Homo sapiens (Human))
University of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50530867(CHEMBL4472654)
Affinity DataIC50:  800nMAssay Description:Inhibition of human recombinant MLL1 using [3H]S-adenosyl-methionine as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 2 group C member 2/TGF-beta-activated kinase 1 and MAP3K7-binding protein 1(Homo sapiens (Human))
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50594365(CHEMBL5186989)
Affinity DataIC50:  820nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged TAK1 (1 to 303 residues)/TAB1 (437 to end residues) expressed in baculovirus infected Sf9 insec...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNuclear receptor subfamily 2 group C member 2/TGF-beta-activated kinase 1 and MAP3K7-binding protein 1(Homo sapiens (Human))
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50594361(CHEMBL5174742)
Affinity DataIC50:  820nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged TAK1 (1 to 303 residues)/TAB1 (437 to end residues) expressed in baculovirus infected Sf9 insec...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase kinase kinase 7(Homo sapiens (Human))
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50129127(CHEMBL3629244)
Affinity DataIC50:  990nMAssay Description:Inhibition of TAK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 2 group C member 2/TGF-beta-activated kinase 1 and MAP3K7-binding protein 1(Homo sapiens (Human))
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50594377(CHEMBL5183713)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged TAK1 (1 to 303 residues)/TAB1 (437 to end residues) expressed in baculovirus infected Sf9 insec...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNuclear receptor subfamily 2 group C member 2/TGF-beta-activated kinase 1 and MAP3K7-binding protein 1(Homo sapiens (Human))
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50594378(CHEMBL5174017)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged TAK1 (1 to 303 residues)/TAB1 (437 to end residues) expressed in baculovirus infected Sf9 insec...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNuclear receptor subfamily 2 group C member 2/TGF-beta-activated kinase 1 and MAP3K7-binding protein 1(Homo sapiens (Human))
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50594376(CHEMBL5207341)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged TAK1 (1 to 303 residues)/TAB1 (437 to end residues) expressed in baculovirus infected Sf9 insec...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNuclear receptor subfamily 2 group C member 2/TGF-beta-activated kinase 1 and MAP3K7-binding protein 1(Homo sapiens (Human))
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50594375(CHEMBL5181612)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged TAK1 (1 to 303 residues)/TAB1 (437 to end residues) expressed in baculovirus infected Sf9 insec...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNuclear receptor subfamily 2 group C member 2/TGF-beta-activated kinase 1 and MAP3K7-binding protein 1(Homo sapiens (Human))
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50594374(CHEMBL5203686)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged TAK1 (1 to 303 residues)/TAB1 (437 to end residues) expressed in baculovirus infected Sf9 insec...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNuclear receptor subfamily 2 group C member 2/TGF-beta-activated kinase 1 and MAP3K7-binding protein 1(Homo sapiens (Human))
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50594373(CHEMBL5198327)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged TAK1 (1 to 303 residues)/TAB1 (437 to end residues) expressed in baculovirus infected Sf9 insec...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNuclear receptor subfamily 2 group C member 2/TGF-beta-activated kinase 1 and MAP3K7-binding protein 1(Homo sapiens (Human))
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50594372(CHEMBL5188253)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged TAK1 (1 to 303 residues)/TAB1 (437 to end residues) expressed in baculovirus infected Sf9 insec...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNuclear receptor subfamily 2 group C member 2/TGF-beta-activated kinase 1 and MAP3K7-binding protein 1(Homo sapiens (Human))
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50594371(CHEMBL5190572)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged TAK1 (1 to 303 residues)/TAB1 (437 to end residues) expressed in baculovirus infected Sf9 insec...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNuclear receptor subfamily 2 group C member 2/TGF-beta-activated kinase 1 and MAP3K7-binding protein 1(Homo sapiens (Human))
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50594370(CHEMBL5208768)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged TAK1 (1 to 303 residues)/TAB1 (437 to end residues) expressed in baculovirus infected Sf9 insec...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNuclear receptor subfamily 2 group C member 2/TGF-beta-activated kinase 1 and MAP3K7-binding protein 1(Homo sapiens (Human))
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50594369(CHEMBL5173639)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged TAK1 (1 to 303 residues)/TAB1 (437 to end residues) expressed in baculovirus infected Sf9 insec...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNuclear receptor subfamily 2 group C member 2/TGF-beta-activated kinase 1 and MAP3K7-binding protein 1(Homo sapiens (Human))
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50594366(CHEMBL5188775)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged TAK1 (1 to 303 residues)/TAB1 (437 to end residues) expressed in baculovirus infected Sf9 insec...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNuclear receptor subfamily 2 group C member 2/TGF-beta-activated kinase 1 and MAP3K7-binding protein 1(Homo sapiens (Human))
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50594363(CHEMBL5196408)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged TAK1 (1 to 303 residues)/TAB1 (437 to end residues) expressed in baculovirus infected Sf9 insec...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNuclear receptor subfamily 2 group C member 2/TGF-beta-activated kinase 1 and MAP3K7-binding protein 1(Homo sapiens (Human))
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50594362(CHEMBL5187912)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged TAK1 (1 to 303 residues)/TAB1 (437 to end residues) expressed in baculovirus infected Sf9 insec...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNuclear receptor subfamily 2 group C member 2/TGF-beta-activated kinase 1 and MAP3K7-binding protein 1(Homo sapiens (Human))
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50594357(CHEMBL5203951)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged TAK1 (1 to 303 residues)/TAB1 (437 to end residues) expressed in baculovirus infected Sf9 insec...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNuclear receptor subfamily 2 group C member 2/TGF-beta-activated kinase 1 and MAP3K7-binding protein 1(Homo sapiens (Human))
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50594355(CHEMBL5196981)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged TAK1 (1 to 303 residues)/TAB1 (437 to end residues) expressed in baculovirus infected Sf9 insec...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNuclear receptor subfamily 2 group C member 2/TGF-beta-activated kinase 1 and MAP3K7-binding protein 1(Homo sapiens (Human))
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50594359(CHEMBL5185951)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged TAK1 (1 to 303 residues)/TAB1 (437 to end residues) expressed in baculovirus infected Sf9 insec...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase kinase kinase 7(Homo sapiens (Human))
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50129126((5E)-7-Oxozeaenol | CHEBI:67558 | CHEMBL1801950 | ...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of TAK1 (unknown origin)More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 2 group C member 2/TGF-beta-activated kinase 1 and MAP3K7-binding protein 1(Homo sapiens (Human))
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50594368(CHEMBL5186228)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged TAK1 (1 to 303 residues)/TAB1 (437 to end residues) expressed in baculovirus infected Sf9 insec...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase kinase kinase 7(Homo sapiens (Human))
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50129125(CHEMBL3629245 | US10434085, Compound 6)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of TAK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 7(Homo sapiens (Human))
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50347546(CHEMBL1801951 | US10434085, Compound LL-Z164-1)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of TAK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM14361((R,S)-Rolipram | 4-(3-cyclopentyloxy-4-methoxy-phe...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of human PDE4B2More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 7(Homo sapiens (Human))
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50129124(CHEMBL3629246 | US10434085, Compound 8)
Affinity DataIC50:  8.90E+3nMAssay Description:Inhibition of TAK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 7(Homo sapiens (Human))
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50347544(US10434085, Compound zeaenol | ZEAENOL)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of TAK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscription factor p65(Homo sapiens (Human))
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50336457((3S,5Z,8S,9R,11E)-8,9,16-trihydroxy-14-methoxy-3-m...)
Affinity DataIC50:  1.15E+4nMAssay Description:Inhibition of NFkappa p65 isolated from nuclear extract of human HeLa cells by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50428912(Betulinan C | CHEMBL2331809)
Affinity DataIC50:  1.70E+4nMAssay Description:Inhibition of human PDE4B2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 7(Homo sapiens (Human))
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50129085(CHEMBL3334712)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of TAK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 7(Homo sapiens (Human))
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50129083(CHEMBL3628303)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of TAK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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