Affinity DataIC50: 0.0500nMAssay Description:Inhibition of porcine DPP4More data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Inhibition of Abl1 kinase (unknown origin) using Tyr 6 peptide as substrate assessed as residual enzyme activity after every 10 secs measured for 10 ...More data for this Ligand-Target Pair
Affinity DataIC50: 0.270nMAssay Description:Inhibition of porcine DPP4 using H-Gly-Pro-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.400nMAssay Description:Inhibition of Abl1 kinase (unknown origin) using Tyr 6 peptide as substrate assessed as residual enzyme activity after every 10 secs measured for 10 ...More data for this Ligand-Target Pair
Affinity DataIC50: 0.600nMAssay Description:Inhibition of wild type Abl1 kinase (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 0.730nMAssay Description:Inhibition of porcine DPP4 using H-Gly-Pro-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibition of Abl2 kinase (unknown origin) using Tyr 6 peptide as substrate assessed as residual enzyme activity after every 10 secs measured for 10 ...More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibition of wild type Abl1 kinase (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibition of porcine DPP4More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibition of Abl1 kinase (unknown origin) using Tyr 6 peptide as substrate assessed as residual enzyme activity after every 10 secs measured for 10 ...More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibition of wild type Abl1 kinase (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.10nMAssay Description:Inhibition of human DPP4 using H-Gly-Pro-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60nMAssay Description:Inhibition of porcine DPP4 using H-Gly-Pro-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60nMAssay Description:Inhibition of wild type Abl1 kinase (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.60nMAssay Description:Inhibition of human DPP4 using H-Gly-Pro-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibition of Abl2 kinase (unknown origin) using Tyr 6 peptide as substrate assessed as residual enzyme activity after every 10 secs measured for 10 ...More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibition of Abl1 kinase (unknown origin) using Tyr 6 peptide as substrate assessed as residual enzyme activity after every 10 secs measured for 10 ...More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of Abl2 kinase (unknown origin) using Tyr 6 peptide as substrate assessed as residual enzyme activity after every 10 secs measured for 10 ...More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibition of recombinant C-terminal His10-tagged human Hepsin (R45 to L17 residues) D161E/ R162K double mutant expressed in mouse NS0 cells using Bo...More data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibition of Abl2 kinase (unknown origin) using Tyr 6 peptide as substrate assessed as residual enzyme activity after every 10 secs measured for 10 ...More data for this Ligand-Target Pair
Affinity DataIC50: 6.30nMAssay Description:Binding affinity for human tachykinin receptor 2 expressed in CHO cells using [125I]- NKA radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 6.30nMAssay Description:Binding affinity for human tachykinin receptor 2 expressed in CHO cells using [125I]- NKA radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 6.40nMAssay Description:Binding affinity for human tachykinin receptor 2 expressed in CHO cells using [125I]- NKA radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 6.5nMAssay Description:Binding affinity for human tachykinin receptor 2 expressed in CHO cells using [125I]- NKA radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 6.5nMAssay Description:Inhibition of porcine DPP4 using H-Gly-Pro-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6.60nMAssay Description:Binding affinity for human tachykinin receptor 2 expressed in CHO cells using [125I]- NKA radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 6.70nMAssay Description:Binding affinity for human tachykinin receptor 2 expressed in CHO cells using [125I]- NKA radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 6.80nMAssay Description:Binding affinity for human tachykinin receptor 2 expressed in CHO cells using [125I]- NKA radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 6.80nMAssay Description:Binding affinity for human tachykinin receptor 2 expressed in CHO cells using [125I]- NKA radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: <7nMAssay Description:Binding affinity for human tachykinin receptor 2 expressed in CHO cells using [125I]- NKA radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Inhibition of Abl1 kinase (unknown origin) using Tyr 6 peptide as substrate assessed as residual enzyme activity after every 10 secs measured for 10 ...More data for this Ligand-Target Pair
Affinity DataIC50: 7.10nMAssay Description:Binding affinity for human tachykinin receptor 2 expressed in CHO cells using [125I]- NKA radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 7.20nMAssay Description:Binding affinity for human tachykinin receptor 2 expressed in CHO cells using [125I]- NKA radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 7.30nMAssay Description:Binding affinity for human tachykinin receptor 2 expressed in CHO cells using [125I]- NKA radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 7.40nMAssay Description:Binding affinity for human tachykinin receptor 2 expressed in CHO cells using [125I]- NKA radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 7.5nMAssay Description:Binding affinity for human tachykinin receptor 2 expressed in CHO cells using [125I]- NKA radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 7.70nMAssay Description:Binding affinity for human tachykinin receptor 2 expressed in CHO cells using [125I]- NKA radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 7.70nMAssay Description:Binding affinity for human tachykinin receptor 2 expressed in CHO cells using [125I]- NKA radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Inhibition of Abl2 kinase (unknown origin) using Tyr 6 peptide as substrate assessed as residual enzyme activity after every 10 secs measured for 10 ...More data for this Ligand-Target Pair
Affinity DataIC50: 8.10nMAssay Description:Binding affinity for human tachykinin receptor 2 expressed in CHO cells using [125I]- NKA radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 8.40nMAssay Description:Binding affinity for human tachykinin receptor 2 expressed in CHO cells using [125I]- NKA radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 8.90nMAssay Description:Binding affinity for human tachykinin receptor 2 expressed in CHO cells using [125I]- NKA radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 8.90nMAssay Description:Binding affinity for human tachykinin receptor 2 expressed in CHO cells using [125I]- NKA radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 8.90nMAssay Description:Binding affinity towards human Tachykinin receptor 2 using [125I]- NKA radioligand expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Inhibition of porcine DPP4More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of Abl2 kinase (unknown origin) using Tyr 6 peptide as substrate assessed as residual enzyme activity after every 10 secs measured for 10 ...More data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Inhibition of human DPP4 using H-Gly-Pro-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Inhibition of Abl2 kinase (unknown origin) using Tyr 6 peptide as substrate assessed as residual enzyme activity after every 10 secs measured for 10 ...More data for this Ligand-Target Pair