TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
National Institute On Drug Abuse
Curated by PDSP Ki Database
National Institute On Drug Abuse
Curated by PDSP Ki Database
TargetNicotinic acetylcholine receptor(RAT)
National Institute On Drug Abuse
Curated by PDSP Ki Database
National Institute On Drug Abuse
Curated by PDSP Ki Database
TargetNicotinic acetylcholine receptor(RAT)
National Institute On Drug Abuse
Curated by PDSP Ki Database
National Institute On Drug Abuse
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
National Institute On Drug Abuse
Curated by PDSP Ki Database
National Institute On Drug Abuse
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
National Institute On Drug Abuse
Curated by PDSP Ki Database
National Institute On Drug Abuse
Curated by PDSP Ki Database
TargetNicotinic acetylcholine receptor(RAT)
National Institute On Drug Abuse
Curated by PDSP Ki Database
National Institute On Drug Abuse
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Affinity DataKi: 0.0100nMAssay Description:Binding affinity to Nicotinic acetylcholine receptor alpha4-beta2 using +/-[3H]epibatidine as radioligand in rat brainMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit beta-4(Rattus norvegicus (Rat))
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Affinity DataKi: 0.0200nMAssay Description:Binding affinity to Nicotinic acetylcholine receptor alpha3-beta4 using +/-[3H]epibatidine as radioligand in pig adrenal glandMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
National Institute On Drug Abuse
Curated by PDSP Ki Database
National Institute On Drug Abuse
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Affinity DataKi: 0.0400nMAssay Description:Binding affinity to Nicotinic acetylcholine receptor alpha4-beta2 using +/-[3H]epibatidine as radioligand in rat brainMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3(Rattus norvegicus (Rat))
National Institute On Drug Abuse
Curated by PDSP Ki Database
National Institute On Drug Abuse
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Affinity DataKi: 0.0500nMAssay Description:Binding affinity to Nicotinic acetylcholine receptor alpha4-beta2 using +/-[3H]epibatidine as radioligand in rat brainMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3(Rattus norvegicus (Rat))
National Institute On Drug Abuse
Curated by PDSP Ki Database
National Institute On Drug Abuse
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Affinity DataKi: 0.140nMAssay Description:Binding affinity to Nicotinic acetylcholine receptor alpha4-beta2 using +/-[3H]epibatidine as radioligand in rat brainMore data for this Ligand-Target Pair
TargetNicotinic acetylcholine receptor(RAT)
National Institute On Drug Abuse
Curated by PDSP Ki Database
National Institute On Drug Abuse
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
National Institute On Drug Abuse
Curated by PDSP Ki Database
National Institute On Drug Abuse
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
National Institute On Drug Abuse
Curated by PDSP Ki Database
National Institute On Drug Abuse
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Affinity DataKi: 0.840nMAssay Description:Binding affinity to Nicotinic acetylcholine receptor alpha4-beta2 using +/-[3H]epibatidine as radioligand in rat brainMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Affinity DataKi: 0.950nMAssay Description:Binding affinity to subtype Nicotinic acetylcholine receptor alpha7 using [3H]-MLA as radioligand in rat brainMore data for this Ligand-Target Pair
TargetNicotinic acetylcholine receptor(RAT)
National Institute On Drug Abuse
Curated by PDSP Ki Database
National Institute On Drug Abuse
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Affinity DataKi: 1.10nMAssay Description:Binding affinity to Nicotinic acetylcholine receptor alpha4-beta2 using +/-[3H]epibatidine as radioligand in rat brainMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit beta-4(Rattus norvegicus (Rat))
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Affinity DataKi: 1.30nMAssay Description:Binding affinity to Nicotinic acetylcholine receptor alpha3-beta4 using +/-[3H]epibatidine as radioligand in pig adrenal glandMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit beta-4(Rattus norvegicus (Rat))
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Affinity DataKi: 2.5nMAssay Description:Binding affinity to Nicotinic acetylcholine receptor alpha3-beta4 using +/-[3H]epibatidine as radioligand in pig adrenal glandMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University Of Bonn
Curated by ChEMBL
University Of Bonn
Curated by ChEMBL
Affinity DataKi: 2.90nMAssay Description:Displacement of [3H]nicotine from alpha4beta2 nAChR expressed in human SH-EP1 clonal cell membranes after 2 to 3 hrs by liquid scintillation counting...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Affinity DataKi: 4nMAssay Description:Binding affinity to subtype Nicotinic acetylcholine receptor alpha-7 using [125I]-alpha-BTX as radioligand in rat brainMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
TargetNicotinic acetylcholine receptor(RAT)
National Institute On Drug Abuse
Curated by PDSP Ki Database
National Institute On Drug Abuse
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit beta-4(Rattus norvegicus (Rat))
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Affinity DataKi: 6.20nMAssay Description:Binding affinity to Nicotinic acetylcholine receptor alpha3-beta4 using +/-[3H]epibatidine as radioligand in pig adrenal glandMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-9(RAT)
National Institute On Drug Abuse
Curated by PDSP Ki Database
National Institute On Drug Abuse
Curated by PDSP Ki Database
TargetNicotinic acetylcholine receptor(RAT)
National Institute On Drug Abuse
Curated by PDSP Ki Database
National Institute On Drug Abuse
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-9(RAT)
National Institute On Drug Abuse
Curated by PDSP Ki Database
National Institute On Drug Abuse
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University Of Bonn
Curated by ChEMBL
University Of Bonn
Curated by ChEMBL
Affinity DataKi: 9.90nMAssay Description:Displacement of [3H]nicotine from alpha4beta2 nAChR expressed in human SH-EP1 clonal cell membranes after 2 to 3 hrs by liquid scintillation counting...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Affinity DataKi: >10nMAssay Description:Binding affinity to subtype Nicotinic acetylcholine receptor alpha7 using [3H]-MLA as radioligand in rat brainMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University Of Bonn
Curated by ChEMBL
University Of Bonn
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Displacement of [3H]nicotine from alpha4beta2 nAChR expressed in human SH-EP1 clonal cell membranes after 2 to 3 hrs by liquid scintillation counting...More data for this Ligand-Target Pair
TargetNicotinic acetylcholine receptor(RAT)
National Institute On Drug Abuse
Curated by PDSP Ki Database
National Institute On Drug Abuse
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:Binding affinity to subtype Nicotinic acetylcholine receptor alpha7 using [3H]-MLA as radioligand in rat brainMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Binding affinity to Nicotinic acetylcholine receptor alpha4-beta2 using +/-[3H]epibatidine as radioligand in rat brainMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Binding affinity to subtype Nicotinic acetylcholine receptor alpha7 using [3H]-MLA as radioligand in rat brainMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University Of Bonn
Curated by ChEMBL
University Of Bonn
Curated by ChEMBL
Affinity DataKi: 17nMAssay Description:Binding affinity to alpha4beta2 nAChR (unknown origin)More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Affinity DataKi: 19nMAssay Description:Binding affinity to Nicotinic acetylcholine receptor alpha4-beta2 using +/-[3H]epibatidine as radioligand in rat brainMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit beta-4(Rattus norvegicus (Rat))
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Affinity DataKi: 19nMAssay Description:Binding affinity to Nicotinic acetylcholine receptor alpha3-beta4 using +/-[3H]epibatidine as radioligand in pig adrenal glandMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University Of Bonn
Curated by ChEMBL
University Of Bonn
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Displacement of [3H]nicotine from alpha4beta2 nAChR expressed in human SH-EP1 clonal cell membranes after 2 to 3 hrs by liquid scintillation counting...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University Of Bonn
Curated by ChEMBL
University Of Bonn
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Displacement of [3H]nicotine from alpha4beta2 nAChR expressed in human SH-EP1 clonal cell membranes after 2 to 3 hrs by liquid scintillation counting...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit beta-4(Rattus norvegicus (Rat))
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Binding affinity to Nicotinic acetylcholine receptor alpha3-beta4 using +/-[3H]epibatidine as radioligand in pig adrenal glandMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University Of Bonn
Curated by ChEMBL
University Of Bonn
Curated by ChEMBL
Affinity DataKi: 34nMAssay Description:Binding affinity to alpha4beta2 nAChR (unknown origin)More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University Of Bonn
Curated by ChEMBL
University Of Bonn
Curated by ChEMBL
Affinity DataKi: 44nMAssay Description:Displacement of [3H]nicotine from alpha4beta2 nAChR expressed in human SH-EP1 clonal cell membranes after 2 to 3 hrs by liquid scintillation counting...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3(Rattus norvegicus (Rat))
National Institute On Drug Abuse
Curated by PDSP Ki Database
National Institute On Drug Abuse
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-3(Rattus norvegicus (Rat))
National Institute On Drug Abuse
Curated by PDSP Ki Database
National Institute On Drug Abuse
Curated by PDSP Ki Database