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Found 64 with Last Name = 'shilkar' and Initial = 'd'
TargetGenome polyprotein(Dengue virus 2)
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50588190(CHEMBL5170076)
Affinity DataKi:  1.40E+3nMAssay Description:Binding affinity to DENV2 NS2B/NS3 protease assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGenome polyprotein(Dengue virus 2)
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50588190(CHEMBL5170076)
Affinity DataKi:  1.40E+3nMAssay Description:Inhibition of DENV2 NS2B-NS3 proteaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGenome polyprotein(Dengue virus 2)
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50513213(CHEMBL3344303)
Affinity DataKi:  2.00E+3nMAssay Description:Inhibition of DENV2 NS2B-NS3 proteaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGenome polyprotein(Dengue virus 2)
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50513213(CHEMBL3344303)
Affinity DataKi:  2.00E+3nMAssay Description:Binding affinity to DENV2 NS2B/NS3 protease assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGenome polyprotein(Dengue virus 2)
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50588187(CHEMBL5194503)
Affinity DataKi:  5.30E+3nMAssay Description:Binding affinity to DENV2 NS2B/NS3 protease assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGenome polyprotein(Dengue virus 2)
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50588187(CHEMBL5194503)
Affinity DataKi:  5.30E+3nMAssay Description:Inhibition of DENV2 NS2B-NS3 proteaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGenome polyprotein(Dengue virus 2)
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50513887(CHEMBL4458555)
Affinity DataKi:  1.21E+4nMAssay Description:Inhibition of DENV2 NS2B-NS3 proteaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGenome polyprotein(Dengue virus 2)
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50513887(CHEMBL4458555)
Affinity DataKi:  1.21E+4nMAssay Description:Binding affinity to DENV2 NS2B/NS3 protease assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGenome polyprotein(Dengue virus 2)
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50588189(CHEMBL5206550)
Affinity DataKi:  1.50E+4nMAssay Description:Inhibition of DENV2 NS2B-NS3 proteaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGenome polyprotein(Dengue virus 2)
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50588189(CHEMBL5206550)
Affinity DataKi:  1.50E+4nMAssay Description:Binding affinity to DENV2 NS2B/NS3 protease assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGenome polyprotein(Dengue virus 2)
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50026784(CHEMBL2440339)
Affinity DataKi:  1.56E+4nMAssay Description:Binding affinity to DENV2 NS2B/NS3 protease assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGenome polyprotein(Dengue virus 2)
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50026784(CHEMBL2440339)
Affinity DataKi:  1.56E+4nMAssay Description:Inhibition of DENV2 NS2B-NS3 proteaseMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGenome polyprotein(Dengue virus 2)
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50588188(CHEMBL5200710)
Affinity DataKi:  1.70E+4nMAssay Description:Binding affinity to DENV2 NS2B/NS3 protease assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGenome polyprotein(Dengue virus 2)
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50588188(CHEMBL5200710)
Affinity DataKi:  1.70E+4nMAssay Description:Inhibition of DENV2 NS2B-NS3 proteaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGenome polyprotein(Dengue virus 2)
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM4355((2E)-2-cyano-3-(4-hydroxyphenyl)prop-2-enamide | C...)
Affinity DataKi:  3.57E+4nMAssay Description:Binding affinity to DENV2 NS2B/NS3 protease assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGenome polyprotein(Dengue virus 2)
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM4355((2E)-2-cyano-3-(4-hydroxyphenyl)prop-2-enamide | C...)
Affinity DataKi:  3.57E+4nMAssay Description:Inhibition of DENV2 NS2B-NS3 proteaseMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGenome polyprotein(Dengue virus 2)
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50588191(ALEXIDINE HYDROCHLORIDE | Alexidine dihydrochlorid...)
Affinity DataKi:  4.10E+4nMAssay Description:Inhibition of DENV2 NS2B-NS3 proteaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGenome polyprotein(Dengue virus 2)
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50588191(ALEXIDINE HYDROCHLORIDE | Alexidine dihydrochlorid...)
Affinity DataKi:  4.10E+4nMAssay Description:Binding affinity to DENV2 NS2B/NS3 protease assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGenome polyprotein(Dengue virus 2)
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50588186(CHEMBL403278 | SN-20440)
Affinity DataKi:  4.40E+4nMAssay Description:Binding affinity to DENV2 NS2B/NS3 protease assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGenome polyprotein(Dengue virus 2)
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50588186(CHEMBL403278 | SN-20440)
Affinity DataKi:  4.40E+4nMAssay Description:Inhibition of DENV2 NS2B-NS3 proteaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGenome polyprotein(Dengue virus 2)
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50588192(Revolution | SELAMECTIN | Selamectin | UK-124,114 ...)
Affinity DataKi:  6.30E+4nMAssay Description:Binding affinity to DENV2 NS2B/NS3 protease assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGenome polyprotein(Dengue virus 2)
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50588192(Revolution | SELAMECTIN | Selamectin | UK-124,114 ...)
Affinity DataKi:  6.30E+4nMAssay Description:Inhibition of DENV2 NS2B-NS3 proteaseMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGenome polyprotein(Dengue virus 2)
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50409816(ABAMECTIN)
Affinity DataKi:  7.90E+4nMAssay Description:Binding affinity to DENV2 NS2B/NS3 protease assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGenome polyprotein(Dengue virus 2)
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50409816(ABAMECTIN)
Affinity DataKi:  7.90E+4nMAssay Description:Inhibition of DENV2 NS2B-NS3 proteaseMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGenome polyprotein(Dengue virus 2)
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50588195(CHEMBL5188858)
Affinity DataIC50:  0.480nMAssay Description:Inhibition of DENV NS2B/NS3 proMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGenome polyprotein(Dengue virus 2)
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50588184(CHEMBL5206054)
Affinity DataIC50:  15nMAssay Description:Inhibition of DENV2 NS2B-NS3 protease using Boc-Gly-Arg-7-amino-4-methylcoumarin as substrate preincubated for 10 mins followed by substrate addition...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGenome polyprotein(Dengue virus 2)
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50588185(CHEMBL5205657)
Affinity DataIC50:  16nMAssay Description:Inhibition of DENV2 NS2B-NS3 protease using Boc-Gly-Arg-7-amino-4-methylcoumarin as substrate preincubated for 10 mins followed by substrate addition...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGenome polyprotein(Dengue virus 2)
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50185449((-)-panduratin A | CHEMBL379110 | panduratin A)
Affinity DataIC50:  57nMAssay Description:Inhibition of DENV2 NS2B-NS3 protease using Boc-Gly-Arg-7-amino-4-methylcoumarin as substrate preincubated for 10 mins followed by substrate addition...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGenome polyprotein(Dengue virus 2)
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM60986(MLS001335996 | SMR000857330 | TANNIC ACID | cid_16...)
Affinity DataIC50:  130nMAssay Description:Inhibition of Dengue Virus 4 recombinant NS2B-NS3 protease expressed in Escherichia coli using Bz-Nle-Arg-Arg-AMC as substrate incubated for 30 minsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGenome polyprotein(Dengue virus 2)
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM60986(MLS001335996 | SMR000857330 | TANNIC ACID | cid_16...)
Affinity DataIC50:  130nMAssay Description:Inhibition of Dengue Virus 3 recombinant NS2B-NS3 protease expressed in Escherichia coli using Bz-Nle-Arg-Arg-AMC as substrate incubated for 30 minsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGenome polyprotein(Dengue virus 2)
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM60986(MLS001335996 | SMR000857330 | TANNIC ACID | cid_16...)
Affinity DataIC50:  130nMAssay Description:Inhibition of Dengue Virus 2 recombinant NS2B-NS3 protease expressed in Escherichia coli using Bz-Nle-Arg-Arg-AMC as substrate incubated for 30 minsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGenome polyprotein(Dengue virus 2)
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM60986(MLS001335996 | SMR000857330 | TANNIC ACID | cid_16...)
Affinity DataIC50:  130nMAssay Description:Inhibition of Dengue Virus 1 recombinant NS2B-NS3 protease expressed in Escherichia coli using Bz-Nle-Arg-Arg-AMC as substrate incubated for 30 minsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGenome polyprotein(Dengue virus 2)
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50588181(CHEMBL5194226)
Affinity DataIC50:  380nMAssay Description:Inhibition of DENV-2 NS2B/NS3 protease expressed in Escherichia coli XL1 using Boc-GRR-MCA as substrate preincubated for 10 mins followed by substrat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGenome polyprotein(Dengue virus 2)
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50588175(CHEMBL5177343)
Affinity DataIC50:  500nMAssay Description:Inhibition of DENV2 NS2B-NS3 protease using fluorophore-tagged Bz-nKRR-AMC as substrate preincubated for 30 mins followed by substrate addition measu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGenome polyprotein(Dengue virus 2)
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50108877((3,4-Dihydroxy-5-nitro-phenyl)-p-tolyl-methanone |...)
Affinity DataIC50:  640nMAssay Description:Inhibition of Dengue Virus 3 recombinant NS2B-NS3 protease expressed in Escherichia coli using Bz-Nle-Arg-Arg-AMC as substrate incubated for 30 minsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGenome polyprotein(Dengue virus 2)
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50108877((3,4-Dihydroxy-5-nitro-phenyl)-p-tolyl-methanone |...)
Affinity DataIC50:  640nMAssay Description:Inhibition of Dengue Virus 4 recombinant NS2B-NS3 protease expressed in Escherichia coli using Bz-Nle-Arg-Arg-AMC as substrate incubated for 30 minsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGenome polyprotein(Dengue virus 2)
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50108877((3,4-Dihydroxy-5-nitro-phenyl)-p-tolyl-methanone |...)
Affinity DataIC50:  640nMAssay Description:Inhibition of Dengue Virus 1 recombinant NS2B-NS3 protease expressed in Escherichia coli using Bz-Nle-Arg-Arg-AMC as substrate incubated for 30 minsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGenome polyprotein(Dengue virus 2)
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50108877((3,4-Dihydroxy-5-nitro-phenyl)-p-tolyl-methanone |...)
Affinity DataIC50:  640nMAssay Description:Inhibition of Dengue Virus 2 recombinant NS2B-NS3 protease expressed in Escherichia coli using Bz-Nle-Arg-Arg-AMC as substrate incubated for 30 minsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGenome polyprotein(Dengue virus 2)
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50509461(CHEMBL4440832)
Affinity DataIC50:  990nMAssay Description:Inhibition of DENV3 NS2B-NS3 protease using PhAc-Lys-Arg-Arg-AMC as substrate incubated for 10 mins by fluorometric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGenome polyprotein(Dengue virus 2)
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50588176(CHEMBL5172831)
Affinity DataIC50:  2.90E+3nMAssay Description:Inhibition of DENV2 NS2B-NS3 protease using fluorophore-tagged Bz-nKRR-AMC as substrate preincubated for 30 mins followed by substrate addition measu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGenome polyprotein(Dengue virus 2)
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50482((5Z)-5-(3-bromo-4,5-dihydroxy-benzylidene)-2-(p-to...)
Affinity DataIC50:  2.94E+3nMAssay Description:Inhibition of Dengue Virus 4 recombinant NS2B-NS3 protease expressed in Escherichia coli using Bz-Nle-Arg-Arg-AMC as substrate incubated for 30 minsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGenome polyprotein(Dengue virus 2)
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50482((5Z)-5-(3-bromo-4,5-dihydroxy-benzylidene)-2-(p-to...)
Affinity DataIC50:  2.94E+3nMAssay Description:Inhibition of Dengue Virus 1 recombinant NS2B-NS3 protease expressed in Escherichia coli using Bz-Nle-Arg-Arg-AMC as substrate incubated for 30 minsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGenome polyprotein(Dengue virus 2)
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50482((5Z)-5-(3-bromo-4,5-dihydroxy-benzylidene)-2-(p-to...)
Affinity DataIC50:  2.94E+3nMAssay Description:Inhibition of Dengue Virus 3 recombinant NS2B-NS3 protease expressed in Escherichia coli using Bz-Nle-Arg-Arg-AMC as substrate incubated for 30 minsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGenome polyprotein(Dengue virus 2)
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50482((5Z)-5-(3-bromo-4,5-dihydroxy-benzylidene)-2-(p-to...)
Affinity DataIC50:  2.94E+3nMAssay Description:Inhibition of Dengue Virus 2 recombinant NS2B-NS3 protease expressed in Escherichia coli using Bz-Nle-Arg-Arg-AMC as substrate incubated for 30 minsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGenome polyprotein(Dengue virus 2)
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50525246(CHEMBL4522006)
Affinity DataIC50:  3.60E+3nMAssay Description:Inhibition of DENV2 NS2B-NS3 protease using Boc-Gly-Arg-Arg-7-amino-4-methylcoumarin as substrate incubated for 10 mins by fluorometric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGenome polyprotein(Dengue virus 2)
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50509461(CHEMBL4440832)
Affinity DataIC50:  4.20E+3nMAssay Description:Inhibition of DENV2 NS2B-NS3 protease using Boc-Gly-Arg-Arg-7-amino-4-methylcoumarin as substrate incubated for 10 mins by fluorometric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGenome polyprotein(Dengue virus 2)
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50588177(CHEMBL5192980)
Affinity DataIC50:  5.40E+3nMAssay Description:Inhibition of DENV3 NS2B-NS3 protease using PhAc-Lys-Arg-Arg-AMC as substrate incubated for 10 mins by fluorometric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGenome polyprotein(Dengue virus 2)
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50588180(CHEMBL5190426)
Affinity DataIC50:  5.95E+3nMAssay Description:Inhibition of DENV-2 NS2bNS3 proMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGenome polyprotein(Dengue virus 2)
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50525246(CHEMBL4522006)
Affinity DataIC50:  9.10E+3nMAssay Description:Inhibition of DENV3 NS2B-NS3 protease using PhAc-Lys-Arg-Arg-AMC as substrate incubated for 10 mins by fluorometric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGenome polyprotein(Dengue virus 2)
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50525248(CHEMBL4450411)
Affinity DataIC50:  1.23E+4nMAssay Description:Inhibition of DENV3 NS2B-NS3 protease using PhAc-Lys-Arg-Arg-AMC as substrate incubated for 10 mins by fluorometric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
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