Affinity DataKi: 0.0800nMAssay Description:Displacement of [3H]DAMGO from rat brain MOR after 2 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0800nMAssay Description:Displacement of [3H]DAMGO from rat brain MOR after 2 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0900nMAssay Description:Displacement of [3H]DAMGO from rat brain MOR after 2 hrsMore data for this Ligand-Target Pair
Targetkappa-type opioid receptor isoform 1(Frog)
Biological Research Center of Hungarian Academy of Sciences
Curated by PDSP Ki Database
Biological Research Center of Hungarian Academy of Sciences
Curated by PDSP Ki Database
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
Biological Research Center of Hungarian Academy of Sciences
Curated by PDSP Ki Database
Biological Research Center of Hungarian Academy of Sciences
Curated by PDSP Ki Database
Targetkappa-type opioid receptor isoform 1(Frog)
Biological Research Center of Hungarian Academy of Sciences
Curated by PDSP Ki Database
Biological Research Center of Hungarian Academy of Sciences
Curated by PDSP Ki Database
Targetkappa-type opioid receptor isoform 1(Frog)
Biological Research Center of Hungarian Academy of Sciences
Curated by PDSP Ki Database
Biological Research Center of Hungarian Academy of Sciences
Curated by PDSP Ki Database
Affinity DataKi: 0.100nMAssay Description:Displacement of [3H]DAMGO from rat brain MOR after 2 hrsMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University of Arizona
Curated by PDSP Ki Database
University of Arizona
Curated by PDSP Ki Database
Affinity DataKi: 0.140nMAssay Description:Displacement of [3H]DAMGO from rat brain MOR after 2 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 0.150nMAssay Description:Displacement of [3H]DAMGO from rat brain MOR after 2 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 0.150nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membranes after 2 hrsMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
Biological Research Center of Hungarian Academy of Sciences
Curated by PDSP Ki Database
Biological Research Center of Hungarian Academy of Sciences
Curated by PDSP Ki Database
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Vrije Universiteit Brussel
Curated by ChEMBL
Vrije Universiteit Brussel
Curated by ChEMBL
Affinity DataKi: 0.280nMAssay Description:Displacement of [3H]DSLET from rat brain DOR after 2 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 0.280nMAssay Description:Displacement of [3H]DAMGO from rat brain MOR after 2 hrsMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
Biological Research Center of Hungarian Academy of Sciences
Curated by PDSP Ki Database
Biological Research Center of Hungarian Academy of Sciences
Curated by PDSP Ki Database
Affinity DataKi: 0.370nMAssay Description:Displacement of [3H]DAMGO from rat brain MOR after 2 hrsMore data for this Ligand-Target Pair
Targetkappa-type opioid receptor isoform 1(Frog)
Biological Research Center of Hungarian Academy of Sciences
Curated by PDSP Ki Database
Biological Research Center of Hungarian Academy of Sciences
Curated by PDSP Ki Database
Affinity DataKi: 0.416nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membranes after 2 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 0.420nMAssay Description:Displacement of [3H]DAMGO from rat brain MOR after 2 hrsMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Vrije Universiteit Brussel
Curated by ChEMBL
Vrije Universiteit Brussel
Curated by ChEMBL
Affinity DataKi: 0.480nMAssay Description:Displacement of [3H]DSLET from rat brain DOR after 2 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Displacement of [3H]SP from human recombinant NK1 receptor expressed in CHO cells after 20 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
Biological Research Center of Hungarian Academy of Sciences
Curated by PDSP Ki Database
Biological Research Center of Hungarian Academy of Sciences
Curated by PDSP Ki Database
Affinity DataKi: 0.5nMAssay Description:Displacement of [3H]SP from human NK1 receptor expressed in CHO cells after 20 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
Biological Research Center of Hungarian Academy of Sciences
Curated by PDSP Ki Database
Biological Research Center of Hungarian Academy of Sciences
Curated by PDSP Ki Database
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Vrije Universiteit Brussel
Curated by ChEMBL
Vrije Universiteit Brussel
Curated by ChEMBL
Affinity DataKi: 0.550nMAssay Description:Displacement of [3H]DSLET from rat brain DOR after 2 hrsMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Vrije Universiteit Brussel
Curated by ChEMBL
Vrije Universiteit Brussel
Curated by ChEMBL
Affinity DataKi: 0.600nMAssay Description:Displacement of [3H]DSLET from rat brain DOR after 2 hrsMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
Biological Research Center of Hungarian Academy of Sciences
Curated by PDSP Ki Database
Biological Research Center of Hungarian Academy of Sciences
Curated by PDSP Ki Database
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Vrije Universiteit Brussel
Curated by ChEMBL
Vrije Universiteit Brussel
Curated by ChEMBL
Affinity DataKi: 0.600nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membranes after 2 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 0.620nMAssay Description:Displacement of [3H]DAMGO from rat brain MOR after 2 hrsMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Vrije Universiteit Brussel
Curated by ChEMBL
Vrije Universiteit Brussel
Curated by ChEMBL
Affinity DataKi: 0.620nMAssay Description:Displacement of [3H]DSLET from rat brain DOR after 2 hrsMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University of Arizona
Curated by PDSP Ki Database
University of Arizona
Curated by PDSP Ki Database
Targetkappa-type opioid receptor isoform 1(Frog)
Biological Research Center of Hungarian Academy of Sciences
Curated by PDSP Ki Database
Biological Research Center of Hungarian Academy of Sciences
Curated by PDSP Ki Database
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University of Arizona
Curated by PDSP Ki Database
University of Arizona
Curated by PDSP Ki Database
Targetkappa-type opioid receptor isoform 1(Frog)
Biological Research Center of Hungarian Academy of Sciences
Curated by PDSP Ki Database
Biological Research Center of Hungarian Academy of Sciences
Curated by PDSP Ki Database
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
Biological Research Center of Hungarian Academy of Sciences
Curated by PDSP Ki Database
Biological Research Center of Hungarian Academy of Sciences
Curated by PDSP Ki Database
Affinity DataKi: 1.30nMAssay Description:Displacement of [3H]DAMGO from rat brain MOR after 2 hrsMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Vrije Universiteit Brussel
Curated by ChEMBL
Vrije Universiteit Brussel
Curated by ChEMBL
Affinity DataKi: 1.70nMAssay Description:Displacement of [3H]DSLET from rat brain DOR after 2 hrsMore data for this Ligand-Target Pair
Targetkappa-type opioid receptor isoform 1(Frog)
Biological Research Center of Hungarian Academy of Sciences
Curated by PDSP Ki Database
Biological Research Center of Hungarian Academy of Sciences
Curated by PDSP Ki Database
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Vrije Universiteit Brussel
Curated by ChEMBL
Vrije Universiteit Brussel
Curated by ChEMBL
Affinity DataKi: 2.10nMAssay Description:Displacement of [3H]DSLET from rat brain DOR after 2 hrsMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
Biological Research Center of Hungarian Academy of Sciences
Curated by PDSP Ki Database
Biological Research Center of Hungarian Academy of Sciences
Curated by PDSP Ki Database
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
Biological Research Center of Hungarian Academy of Sciences
Curated by PDSP Ki Database
Biological Research Center of Hungarian Academy of Sciences
Curated by PDSP Ki Database
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Vrije Universiteit Brussel
Curated by ChEMBL
Vrije Universiteit Brussel
Curated by ChEMBL
Affinity DataKi: 2.40nMAssay Description:Displacement of [3H]DSLET from rat brain DOR after 2 hrsMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
Biological Research Center of Hungarian Academy of Sciences
Curated by PDSP Ki Database
Biological Research Center of Hungarian Academy of Sciences
Curated by PDSP Ki Database
Targetkappa-type opioid receptor isoform 1(Frog)
Biological Research Center of Hungarian Academy of Sciences
Curated by PDSP Ki Database
Biological Research Center of Hungarian Academy of Sciences
Curated by PDSP Ki Database
Targetkappa-type opioid receptor isoform 1(Frog)
Biological Research Center of Hungarian Academy of Sciences
Curated by PDSP Ki Database
Biological Research Center of Hungarian Academy of Sciences
Curated by PDSP Ki Database
Targetkappa-type opioid receptor isoform 1(Frog)
Biological Research Center of Hungarian Academy of Sciences
Curated by PDSP Ki Database
Biological Research Center of Hungarian Academy of Sciences
Curated by PDSP Ki Database
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
Biological Research Center of Hungarian Academy of Sciences
Curated by PDSP Ki Database
Biological Research Center of Hungarian Academy of Sciences
Curated by PDSP Ki Database