Affinity DataKi: 0.800nMAssay Description:Competitive reversible inhibition of DPP4 (unknown origin)More data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
The Oregon Health Sciences University
Curated by PDSP Ki Database
The Oregon Health Sciences University
Curated by PDSP Ki Database
Affinity DataKi: 2nMAssay Description:Binding affinity for dipeptidyl-peptidase IVMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
The Oregon Health Sciences University
Curated by PDSP Ki Database
The Oregon Health Sciences University
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
The Oregon Health Sciences University
Curated by PDSP Ki Database
The Oregon Health Sciences University
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
The Oregon Health Sciences University
Curated by PDSP Ki Database
The Oregon Health Sciences University
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
The Oregon Health Sciences University
Curated by PDSP Ki Database
The Oregon Health Sciences University
Curated by PDSP Ki Database
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
The Oregon Health Sciences University
Curated by PDSP Ki Database
The Oregon Health Sciences University
Curated by PDSP Ki Database
Affinity DataKi: 64nMAssay Description:Inhibitory concentration against dipeptidyl-peptidase IVMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
The Oregon Health Sciences University
Curated by PDSP Ki Database
The Oregon Health Sciences University
Curated by PDSP Ki Database
TargetAlpha-2C adrenergic receptor(RAT)
The Oregon Health Sciences University
Curated by PDSP Ki Database
The Oregon Health Sciences University
Curated by PDSP Ki Database
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
The Oregon Health Sciences University
Curated by PDSP Ki Database
The Oregon Health Sciences University
Curated by PDSP Ki Database
Affinity DataKi: 125nMAssay Description:Inhibition of quiescent cell proline dipeptidase (QPP)More data for this Ligand-Target Pair
Affinity DataKi: 126nMAssay Description:Binding affinity for dipeptidyl-peptidase IVMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
The Oregon Health Sciences University
Curated by PDSP Ki Database
The Oregon Health Sciences University
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
The Oregon Health Sciences University
Curated by PDSP Ki Database
The Oregon Health Sciences University
Curated by PDSP Ki Database
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
The Oregon Health Sciences University
Curated by PDSP Ki Database
The Oregon Health Sciences University
Curated by PDSP Ki Database
TargetAlpha-2C adrenergic receptor(RAT)
The Oregon Health Sciences University
Curated by PDSP Ki Database
The Oregon Health Sciences University
Curated by PDSP Ki Database
TargetAlpha-2C adrenergic receptor(RAT)
The Oregon Health Sciences University
Curated by PDSP Ki Database
The Oregon Health Sciences University
Curated by PDSP Ki Database
TargetAlpha-2C adrenergic receptor(RAT)
The Oregon Health Sciences University
Curated by PDSP Ki Database
The Oregon Health Sciences University
Curated by PDSP Ki Database
TargetAlpha-2C adrenergic receptor(RAT)
The Oregon Health Sciences University
Curated by PDSP Ki Database
The Oregon Health Sciences University
Curated by PDSP Ki Database
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck
Curated by ChEMBL
Merck
Curated by ChEMBL
Affinity DataKi: 1.90E+3nMAssay Description:Binding affinity for Potassium channel HERG Kv11.1More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck
Curated by ChEMBL
Merck
Curated by ChEMBL
Affinity DataKi: 2.80E+3nMAssay Description:Binding affinity for Potassium channel HERG Kv11.1More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck
Curated by ChEMBL
Merck
Curated by ChEMBL
Affinity DataKi: 2.80E+3nMAssay Description:Binding affinity of the compound towards human ERG potassium ion channel was determinedMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck
Curated by ChEMBL
Merck
Curated by ChEMBL
Affinity DataKi: 5.30E+3nMAssay Description:Binding affinity of the compound towards human ERG potassium ion channel was determinedMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck
Curated by ChEMBL
Merck
Curated by ChEMBL
Affinity DataKi: 5.50E+3nMAssay Description:Binding affinity of the compound towards human ERG potassium ion channel was determinedMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck
Curated by ChEMBL
Merck
Curated by ChEMBL
Affinity DataKi: 5.70E+3nMAssay Description:Binding affinity for Potassium channel HERG Kv11.1More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck
Curated by ChEMBL
Merck
Curated by ChEMBL
Affinity DataKi: 5.70E+3nMAssay Description:Binding affinity of the compound towards human ERG potassium ion channel was determinedMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck
Curated by ChEMBL
Merck
Curated by ChEMBL
Affinity DataKi: 5.90E+3nMAssay Description:Binding affinity for Potassium channel HERG Kv11.1More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck
Curated by ChEMBL
Merck
Curated by ChEMBL
Affinity DataKi: 5.90E+3nMAssay Description:Binding affinity of the compound towards human ERG potassium ion channel was determinedMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck
Curated by ChEMBL
Merck
Curated by ChEMBL
Affinity DataKi: 6.00E+3nMAssay Description:Binding affinity of the compound towards human ERG potassium ion channel was determinedMore data for this Ligand-Target Pair
TargetAlpha-2C adrenergic receptor(RAT)
The Oregon Health Sciences University
Curated by PDSP Ki Database
The Oregon Health Sciences University
Curated by PDSP Ki Database
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck
Curated by ChEMBL
Merck
Curated by ChEMBL
Affinity DataKi: 1.60E+4nMAssay Description:Binding affinity of the compound towards human ERG potassium ion channel was determinedMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck
Curated by ChEMBL
Merck
Curated by ChEMBL
Affinity DataKi: 1.70E+4nMAssay Description:Binding affinity for Potassium channel HERG Kv11.1More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck
Curated by ChEMBL
Merck
Curated by ChEMBL
Affinity DataKi: 1.90E+4nMAssay Description:Binding affinity of the compound towards human ERG potassium ion channel was determinedMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck
Curated by ChEMBL
Merck
Curated by ChEMBL
Affinity DataKi: 2.20E+4nMAssay Description:Binding affinity for Potassium channel HERG Kv11.1More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck
Curated by ChEMBL
Merck
Curated by ChEMBL
Affinity DataKi: 2.80E+4nMAssay Description:Binding affinity of the compound towards human ERG potassium ion channel was determinedMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck
Curated by ChEMBL
Merck
Curated by ChEMBL
Affinity DataKi: 2.90E+4nMAssay Description:Binding affinity of the compound towards human ERG potassium ion channel was determinedMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck
Curated by ChEMBL
Merck
Curated by ChEMBL
Affinity DataKi: 3.50E+4nMAssay Description:Binding affinity for Potassium channel HERG Kv11.1More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck
Curated by ChEMBL
Merck
Curated by ChEMBL
Affinity DataKi: 3.50E+4nMAssay Description:Binding affinity of the compound towards human ERG potassium ion channel was determinedMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck
Curated by ChEMBL
Merck
Curated by ChEMBL
Affinity DataKi: 3.70E+4nMAssay Description:Binding affinity of the compound towards human ERG potassium ion channel was determinedMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck
Curated by ChEMBL
Merck
Curated by ChEMBL
Affinity DataKi: 3.90E+4nMAssay Description:Binding affinity of the compound towards human ERG potassium ion channel was determinedMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck
Curated by ChEMBL
Merck
Curated by ChEMBL
Affinity DataKi: 4.00E+4nMAssay Description:Binding affinity of the compound towards human ERG potassium ion channel was determinedMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck
Curated by ChEMBL
Merck
Curated by ChEMBL
Affinity DataKi: 4.00E+4nMAssay Description:Binding affinity for Potassium channel HERG Kv11.1More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck
Curated by ChEMBL
Merck
Curated by ChEMBL
Affinity DataKi: 4.20E+4nMAssay Description:Binding affinity of the compound towards human ERG potassium ion channel was determinedMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck
Curated by ChEMBL
Merck
Curated by ChEMBL
Affinity DataKi: 4.30E+4nMAssay Description:Binding affinity of the compound towards human ERG potassium ion channel was determinedMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck
Curated by ChEMBL
Merck
Curated by ChEMBL
Affinity DataKi: 4.90E+4nMAssay Description:Binding affinity of the compound towards human ERG potassium ion channel was determinedMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck
Curated by ChEMBL
Merck
Curated by ChEMBL
Affinity DataKi: 5.20E+4nMAssay Description:Binding affinity of the compound towards human ERG potassium ion channel was determinedMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck
Curated by ChEMBL
Merck
Curated by ChEMBL
Affinity DataKi: 7.30E+4nMAssay Description:Binding affinity of the compound towards human ERG potassium ion channel was determinedMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck
Curated by ChEMBL
Merck
Curated by ChEMBL
Affinity DataKi: >9.00E+4nMAssay Description:Binding affinity of the compound towards human ERG potassium ion channel was determinedMore data for this Ligand-Target Pair