Affinity DataKi: 1.90nMAssay Description:Displacement of [3H]CCPA from recombinant human adenosine A1 receptor expressed in CHO cell membranes after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Displacement of [3H]CCPA from recombinant human adenosine A1 receptor expressed in CHO cell membranes after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 3.5nMAssay Description:Displacement of [3H]CCPA from recombinant human adenosine A1 receptor expressed in CHO cell membranes after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 4.40nMAssay Description:Displacement of [3H]CCPA from recombinant human adenosine A1 receptor expressed in CHO cell membranes after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Displacement of [3H]CCPA from recombinant human adenosine A1 receptor expressed in CHO cell membranes after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Displacement of [3H]CCPA from recombinant human adenosine A1 receptor expressed in CHO cell membranes after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Displacement of [3H]CCPA from recombinant human adenosine A1 receptor expressed in CHO cell membranes after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Displacement of [3H]CCPA from recombinant human adenosine A1 receptor expressed in CHO cell membranes after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Displacement of [3H]CCPA from recombinant human adenosine A1 receptor expressed in CHO cell membranes after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 59nMAssay Description:Displacement of [3H]CCPA from recombinant human adenosine A1 receptor expressed in CHO cell membranes after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 91nMAssay Description:Displacement of [3H]CCPA from recombinant human adenosine A1 receptor expressed in CHO cell membranes after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 115nMAssay Description:Displacement of [3H]CCPA from recombinant human adenosine A1 receptor expressed in CHO cell membranes after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 136nMAssay Description:Displacement of [3H]HEMADO from recombinant human adenosine A3 receptor expressed in CHO cell membranes after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 139nMAssay Description:Displacement of [3H]CCPA from recombinant human adenosine A1 receptor expressed in CHO cell membranes after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 139nMAssay Description:Displacement of [3H]HEMADO from recombinant human adenosine A3 receptor expressed in CHO cell membranes after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 158nMAssay Description:Displacement of [3H]CCPA from recombinant human adenosine A1 receptor expressed in CHO cell membranes after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 232nMAssay Description:Displacement of [3H]HEMADO from recombinant human adenosine A3 receptor expressed in CHO cell membranes after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 343nMAssay Description:Displacement of [3H]HEMADO from recombinant human adenosine A3 receptor expressed in CHO cell membranes after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 438nMAssay Description:Displacement of [3H]CCPA from recombinant human adenosine A1 receptor expressed in CHO cell membranes after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 491nMAssay Description:Displacement of [3H]CCPA from recombinant human adenosine A1 receptor expressed in CHO cell membranes after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 562nMAssay Description:Displacement of [3H]HEMADO from recombinant human adenosine A3 receptor expressed in CHO cell membranes after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 636nMAssay Description:Displacement of [3H]HEMADO from recombinant human adenosine A3 receptor expressed in CHO cell membranes after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 667nMAssay Description:Displacement of [3H]HEMADO from recombinant human adenosine A3 receptor expressed in CHO cell membranes after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 996nMAssay Description:Displacement of [3H]HEMADO from recombinant human adenosine A3 receptor expressed in CHO cell membranes after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+3nMAssay Description:Displacement of [3H]HEMADO from recombinant human adenosine A3 receptor expressed in CHO cell membranes after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 1.10E+3nMAssay Description:Displacement of [3H]HEMADO from recombinant human adenosine A3 receptor expressed in CHO cell membranes after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 1.20E+3nMAssay Description:Displacement of [3H]HEMADO from recombinant human adenosine A3 receptor expressed in CHO cell membranes after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 1.36E+3nMAssay Description:Displacement of [3H]NECA from recombinant human adenosine A2A receptor expressed in CHO cell membranes after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 1.45E+3nMAssay Description:Displacement of [3H]HEMADO from recombinant human adenosine A3 receptor expressed in CHO cell membranes after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 1.96E+3nMAssay Description:Displacement of [3H]NECA from recombinant human adenosine A2A receptor expressed in CHO cell membranes after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 2.73E+3nMAssay Description:Displacement of [3H]HEMADO from recombinant human adenosine A3 receptor expressed in CHO cell membranes after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 4.32E+3nMAssay Description:Displacement of [3H]NECA from recombinant human adenosine A2A receptor expressed in CHO cell membranes after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 5.09E+3nMAssay Description:Displacement of [3H]NECA from recombinant human adenosine A2A receptor expressed in CHO cell membranes after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 5.28E+3nMAssay Description:Displacement of [3H]HEMADO from recombinant human adenosine A3 receptor expressed in CHO cell membranes after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 5.45E+3nMAssay Description:Displacement of [3H]HEMADO from recombinant human adenosine A3 receptor expressed in CHO cell membranes after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 5.64E+3nMAssay Description:Displacement of [3H]HEMADO from recombinant human adenosine A3 receptor expressed in CHO cell membranes after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 5.87E+3nMAssay Description:Displacement of [3H]NECA from recombinant human adenosine A2A receptor expressed in CHO cell membranes after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 6.83E+3nMAssay Description:Displacement of [3H]NECA from recombinant human adenosine A2A receptor expressed in CHO cell membranes after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 8.68E+3nMAssay Description:Displacement of [3H]NECA from recombinant human adenosine A2A receptor expressed in CHO cell membranes after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 9.43E+3nMAssay Description:Displacement of [3H]NECA from recombinant human adenosine A2A receptor expressed in CHO cell membranes after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 1.02E+4nMAssay Description:Displacement of [3H]NECA from recombinant human adenosine A2A receptor expressed in CHO cell membranes after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 1.04E+4nMAssay Description:Displacement of [3H]NECA from recombinant human adenosine A2A receptor expressed in CHO cell membranes after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 1.05E+4nMAssay Description:Displacement of [3H]NECA from recombinant human adenosine A2A receptor expressed in CHO cell membranes after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 1.19E+4nMAssay Description:Displacement of [3H]NECA from recombinant human adenosine A2A receptor expressed in CHO cell membranes after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 1.45E+4nMAssay Description:Displacement of [3H]NECA from recombinant human adenosine A2A receptor expressed in CHO cell membranes after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 1.96E+4nMAssay Description:Displacement of [3H]NECA from recombinant human adenosine A2A receptor expressed in CHO cell membranes after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 2.86E+4nMAssay Description:Displacement of [3H]NECA from recombinant human adenosine A2A receptor expressed in CHO cell membranes after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]NECA from recombinant human adenosine A2A receptor expressed in CHO cell membranes after 3 hrsMore data for this Ligand-Target Pair
Affinity DataIC50: 701nMAssay Description:Antagonist activity at recombinant human adenosine A3 receptor expressed in CHO cell membranes assessed as inhibition of forskolin-stimulated adenyly...More data for this Ligand-Target Pair
Affinity DataIC50: 1.91E+3nMAssay Description:Antagonist activity at recombinant human adenosine A3 receptor expressed in CHO cell membranes assessed as inhibition of forskolin-stimulated adenyly...More data for this Ligand-Target Pair