Found 39 with Last Name = 's?czewski' and Initial = 'f' TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
Medical University of Gdansk
Curated by ChEMBL
Medical University of Gdansk
Curated by ChEMBL
Affinity DataKi: 14nMAssay Description:Displacement of [3H]RX821002 from alpha2-adrenoceptor in Sprague-Dawley rat brain membranes after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
Medical University of Gdansk
Curated by ChEMBL
Medical University of Gdansk
Curated by ChEMBL
Affinity DataKi: 26nMAssay Description:Displacement of [3H]RX821002 from alpha2-adrenoceptor in Sprague-Dawley rat brain membranes after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
Medical University of Gdansk
Curated by ChEMBL
Medical University of Gdansk
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:Displacement of [3H]RX821002 from alpha2-adrenoceptor in Sprague-Dawley rat brain membranes after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
Medical University of Gdansk
Curated by ChEMBL
Medical University of Gdansk
Curated by ChEMBL
Affinity DataKi: 31nMAssay Description:Displacement of [3H]RX821002 from alpha2-adrenoceptor in Sprague-Dawley rat brain membranes after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
Medical University of Gdansk
Curated by ChEMBL
Medical University of Gdansk
Curated by ChEMBL
Affinity DataKi: 32nMAssay Description:Displacement of [3H]RX821002 from alpha2-adrenoceptor in Sprague-Dawley rat brain membranes after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Medical University of Gdansk
Curated by ChEMBL
Medical University of Gdansk
Curated by ChEMBL
Affinity DataKi: 33nMAssay Description:Displacement of [3H]RS-79948-197 from human alpha2A adrenoceptor expressed in CHO-K1 cells after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Medical University of Gdansk
Curated by ChEMBL
Medical University of Gdansk
Curated by ChEMBL
Affinity DataKi: 52nMAssay Description:Displacement of [3H]RS-79948-197 from human alpha2A adrenoceptor expressed in CHO-K1 cells after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
Medical University of Gdansk
Curated by ChEMBL
Medical University of Gdansk
Curated by ChEMBL
Affinity DataKi: 64nMAssay Description:Displacement of [3H]RX821002 from alpha2-adrenoceptor in Sprague-Dawley rat brain membranes after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Medical University of Gdansk
Curated by ChEMBL
Medical University of Gdansk
Curated by ChEMBL
Affinity DataKi: 65nMAssay Description:Displacement of [3H]RS-79948-197 from human alpha2A adrenoceptor expressed in CHO-K1 cells after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Medical University of Gdansk
Curated by ChEMBL
Medical University of Gdansk
Curated by ChEMBL
Affinity DataKi: 72nMAssay Description:Displacement of [3H]RS-79948-197 from human alpha2B adrenoceptor expressed in CHO-K1 cells after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Medical University of Gdansk
Curated by ChEMBL
Medical University of Gdansk
Curated by ChEMBL
Affinity DataKi: 79nMAssay Description:Displacement of [3H]RS-79948-197 from human alpha2B adrenoceptor expressed in CHO-K1 cells after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Medical University of Gdansk
Curated by ChEMBL
Medical University of Gdansk
Curated by ChEMBL
Affinity DataKi: 158nMAssay Description:Displacement of [3H]RS-79948-197 from human alpha2B adrenoceptor expressed in CHO-K1 cells after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
Medical University of Gdansk
Curated by ChEMBL
Medical University of Gdansk
Curated by ChEMBL
Affinity DataKi: 187nMAssay Description:Displacement of [3H]RX821002 from alpha2-adrenoceptor in Sprague-Dawley rat brain membranes after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
Medical University of Gdansk
Curated by ChEMBL
Medical University of Gdansk
Curated by ChEMBL
Affinity DataKi: 416nMAssay Description:Displacement of [3H]RX821002 from alpha2-adrenoceptor in Sprague-Dawley rat brain membranes after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Medical University of Gdansk
Curated by ChEMBL
Medical University of Gdansk
Curated by ChEMBL
Affinity DataKi: 476nMAssay Description:Displacement of [3H]prazosin from alpha1-adrenoceptor in Sprague-Dawley rat brain membranes after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Medical University of Gdansk
Curated by ChEMBL
Medical University of Gdansk
Curated by ChEMBL
Affinity DataKi: 518nMAssay Description:Displacement of [3H]prazosin from alpha1-adrenoceptor in Sprague-Dawley rat brain membranes after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Medical University of Gdansk
Curated by ChEMBL
Medical University of Gdansk
Curated by ChEMBL
Affinity DataKi: 535nMAssay Description:Displacement of [3H]prazosin from alpha1-adrenoceptor in Sprague-Dawley rat brain membranes after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Medical University of Gdansk
Curated by ChEMBL
Medical University of Gdansk
Curated by ChEMBL
Affinity DataKi: 600nMAssay Description:Displacement of [3H]RS-79948-197 from human alpha2C adrenoceptor expressed in CHO-K1 cells after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Medical University of Gdansk
Curated by ChEMBL
Medical University of Gdansk
Curated by ChEMBL
Affinity DataKi: 640nMAssay Description:Displacement of [3H]RS-79948-197 from human alpha2C adrenoceptor expressed in CHO-K1 cells after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Medical University of Gdansk
Curated by ChEMBL
Medical University of Gdansk
Curated by ChEMBL
Affinity DataKi: 918nMAssay Description:Displacement of [3H]prazosin from alpha1-adrenoceptor in Sprague-Dawley rat brain membranes after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Medical University of Gdansk
Curated by ChEMBL
Medical University of Gdansk
Curated by ChEMBL
Affinity DataKi: 1.20E+3nMAssay Description:Displacement of [3H]RS-79948-197 from human alpha2C adrenoceptor expressed in CHO-K1 cells after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Medical University of Gdansk
Curated by ChEMBL
Medical University of Gdansk
Curated by ChEMBL
Affinity DataKi: 1.63E+3nMAssay Description:Displacement of [3H]prazosin from alpha1-adrenoceptor in Sprague-Dawley rat brain membranes after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Medical University of Gdansk
Curated by ChEMBL
Medical University of Gdansk
Curated by ChEMBL
Affinity DataKi: 2.32E+3nMAssay Description:Displacement of [3H]prazosin from alpha1-adrenoceptor in Sprague-Dawley rat brain membranes after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
Medical University of Gdansk
Curated by ChEMBL
Medical University of Gdansk
Curated by ChEMBL
Affinity DataKi: 3.72E+3nMAssay Description:Displacement of [3H]RX821002 from alpha2-adrenoceptor in Sprague-Dawley rat brain membranes after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Medical University of Gdansk
Curated by ChEMBL
Medical University of Gdansk
Curated by ChEMBL
Affinity DataKi: 3.81E+3nMAssay Description:Displacement of [3H]prazosin from alpha1-adrenoceptor in Sprague-Dawley rat brain membranes after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Medical University of Gdansk
Curated by ChEMBL
Medical University of Gdansk
Curated by ChEMBL
Affinity DataKi: 1.98E+4nMAssay Description:Displacement of [3H]prazosin from alpha1-adrenoceptor in Sprague-Dawley rat brain membranes after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 92nMAssay Description:Displacement of [3H]2BF1 from imidazoline I1 receptor in Sprague-Dawley rat kidney membranes after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 1.77E+3nMAssay Description:Displacement of [3H]2BF1 from imidazoline I1 receptor in Sprague-Dawley rat kidney membranes after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 2.42E+3nMAssay Description:Displacement of [3H]2BF1 from imidazoline I1 receptor in Sprague-Dawley rat kidney membranes after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 5.83E+3nMAssay Description:Displacement of [3H]2BF1 from imidazoline I1 receptor in Sprague-Dawley rat kidney membranes after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 7.74E+3nMAssay Description:Displacement of [3H]2BF1 from imidazoline I1 receptor in Sprague-Dawley rat kidney membranes after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 1.48E+4nMAssay Description:Displacement of [3H]2BF1 from imidazoline I1 receptor in Sprague-Dawley rat kidney membranes after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 2.07E+4nMAssay Description:Displacement of [3H]2BF1 from imidazoline I1 receptor in Sprague-Dawley rat kidney membranes after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 3.35E+4nMAssay Description:Displacement of [3H]2BF1 from imidazoline I1 receptor in Sprague-Dawley rat kidney membranes after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 5.46E+4nMAssay Description:Displacement of [3H]2BF1 from imidazoline I1 receptor in Sprague-Dawley rat kidney membranes after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Medical University of Gdansk
Curated by ChEMBL
Medical University of Gdansk
Curated by ChEMBL
Affinity DataEC50: 200nMAssay Description:Agonist activity at human alpha2A adrenoceptor expressed in CHO-K1 cells after 30 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Medical University of Gdansk
Curated by ChEMBL
Medical University of Gdansk
Curated by ChEMBL
Affinity DataEC50: 129nMAssay Description:Agonist activity at human alpha2A adrenoceptor expressed in CHO-K1 cells after 30 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Medical University of Gdansk
Curated by ChEMBL
Medical University of Gdansk
Curated by ChEMBL
Affinity DataEC50: 39nMAssay Description:Agonist activity at human alpha2A adrenoceptor expressed in CHO-K1 cells after 30 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Medical University of Gdansk
Curated by ChEMBL
Medical University of Gdansk
Curated by ChEMBL
Affinity DataEC50: 93nMAssay Description:Agonist activity at human alpha2A adrenoceptor expressed in CHO-K1 cells after 30 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
