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Found 141 with Last Name = 'koolpe' and Initial = 'ga'
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Sri International

Curated by ChEMBL
LigandPNGBDBM50020515(2-(Hydroxyimino-methyl)-3-methyl-1-(naphthalen-1-y...)
Affinity DataKi:  3.50E+3nMAssay Description:Compound was tested for the competitive inhibition of phosphorylation of Eel acetylcholinesterase (AChE)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Sri International

Curated by ChEMBL
LigandPNGBDBM50020529(2-(Hydroxyimino-methyl)-3-methyl-1-(3-phenyl-propo...)
Affinity DataKi:  4.00E+3nMAssay Description:Compound was tested for the competitive inhibition of phosphonylation of Eel acetylcholinesterase (AChE)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Sri International

Curated by ChEMBL
LigandPNGBDBM50020521(2-(Hydroxyimino-methyl)-3-methyl-1-(1,2,2-trimethy...)
Affinity DataKi:  7.60E+3nMAssay Description:Compound was tested for the competitive inhibition of phosphonylation of Eel acetylcholinesterase (AChE)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Sri International

Curated by ChEMBL
LigandPNGBDBM50020514(2-(Hydroxyimino-methyl)-1-methoxymethyl-3-methyl-3...)
Affinity DataKi:  4.80E+4nMAssay Description:Compound was tested for the competitive inhibition of phosphorylation of Eel acetylcholinesterase (AChE)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Sri International

Curated by ChEMBL
LigandPNGBDBM50011780(2-[(E)-(hydroxyimino)methyl]-1-methylpyridinium ch...)
Affinity DataKi:  1.27E+5nMAssay Description:Compound was tested for the competitive inhibition of phosphorylation of Eel acetylcholinesterase (AChE)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Sri International

Curated by ChEMBL
LigandPNGBDBM50020522(1-(((4-carbamoylpyridinium-1-yl)methoxy)methyl)-2-...)
Affinity DataKi:  2.29E+5nMAssay Description:Compound was tested for the competitive inhibition of phosphonylation of Eel acetylcholinesterase (AChE)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225687(CHEMBL611128)
Affinity DataIC50:  2nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the presence of 100 mM NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225687(CHEMBL611128)
Affinity DataIC50:  2nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the presence of 100 mM NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225681(CHEMBL611395)
Affinity DataIC50:  2.30nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the absence of NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225681(CHEMBL611395)
Affinity DataIC50:  3.5nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the presence of 100 mM NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225687(CHEMBL611128)
Affinity DataIC50:  4nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the absence of NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225687(CHEMBL611128)
Affinity DataIC50:  4nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the absence of NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225684(CHEMBL610611)
Affinity DataIC50:  6nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the absence of NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225690(CHEMBL610808)
Affinity DataIC50:  6nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the presence of 100 mM NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225683(CHEMBL610807)
Affinity DataIC50:  7nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the presence of 100 mM NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225685(CHEMBL175344)
Affinity DataIC50:  8nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the absence of NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225690(CHEMBL610808)
Affinity DataIC50:  10nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the absence of NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225692(CHEMBL610612)
Affinity DataIC50:  10nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the absence of NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225692(CHEMBL610612)
Affinity DataIC50:  10nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the presence of 100 mM NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225683(CHEMBL610807)
Affinity DataIC50:  10nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the absence of NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225254(CHEMBL610531)
Affinity DataIC50:  12.5nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the absence of NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225254(CHEMBL610531)
Affinity DataIC50:  12.5nMAssay Description:In vitro binding affinity against opioid receptor using 1 nM [3H]- Naltrexone in the presence of 100 mM NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225254(CHEMBL610531)
Affinity DataIC50:  13nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the absence of NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225254(CHEMBL610531)
Affinity DataIC50:  13nMAssay Description:In vitro binding affinity against opioid receptor using 1 nM [3H]- Naltrexone in the presence of 100 mM NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225254(CHEMBL610531)
Affinity DataIC50:  15nMAssay Description:In vitro binding affinity against opioid receptor using 1 nM of [3H]- Naltrexone in the absence of NaClMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225254(CHEMBL610531)
Affinity DataIC50:  15nMAssay Description:In vitro binding affinity against opioid receptor using 1 nM of [3H]- Naltrexone in the absence of NaClMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225682(CHEMBL174530)
Affinity DataIC50:  15nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the absence of NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225254(CHEMBL610531)
Affinity DataIC50:  15nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the presence of 100 mM NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225254(CHEMBL610531)
Affinity DataIC50:  15nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the presence of 100 mM NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225693(CHEMBL369657)
Affinity DataIC50:  30nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the absence of NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225255(CHEMBL2310924)
Affinity DataIC50:  35nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the absence of NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225255(CHEMBL2310924)
Affinity DataIC50:  35nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the absence of NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225688(CHEMBL611391)
Affinity DataIC50:  40nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the absence of NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225689(CHEMBL611392)
Affinity DataIC50:  50nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the presence of 100 mM NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225685(CHEMBL175344)
Affinity DataIC50:  60nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the presence of 100 mM NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225688(CHEMBL611391)
Affinity DataIC50:  70nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the presence of 100 mM NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225686(CHEMBL367540)
Affinity DataIC50:  70nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the absence of NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225689(CHEMBL611392)
Affinity DataIC50:  100nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the absence of NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225255(CHEMBL2310924)
Affinity DataIC50:  115nMAssay Description:In vitro binding affinity against opioid receptor using 1 nM of [3H]- Naltrexone in the absence of NaClMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225255(CHEMBL2310924)
Affinity DataIC50:  115nMAssay Description:In vitro binding affinity against opioid receptor using 1 nM of [3H]- Naltrexone in the absence of NaClMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225691(CHEMBL174268)
Affinity DataIC50:  200nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the absence of NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225682(CHEMBL174530)
Affinity DataIC50:  200nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the presence of 100 mM NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225255(CHEMBL2310924)
Affinity DataIC50:  250nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the presence of 100 mM NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225255(CHEMBL2310924)
Affinity DataIC50:  250nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the presence of 100 mM NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225693(CHEMBL369657)
Affinity DataIC50:  500nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the presence of 100 mM NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225255(CHEMBL2310924)
Affinity DataIC50:  880nMAssay Description:In vitro binding affinity against opioid receptor using 1 nM [3H]- Naltrexone in the presence of 100 mM NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225255(CHEMBL2310924)
Affinity DataIC50:  880nMAssay Description:In vitro binding affinity against opioid receptor using 1 nM [3H]- Naltrexone in the presence of 100 mM NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225691(CHEMBL174268)
Affinity DataIC50: >1.00E+3nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the presence of 100 mM NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225686(CHEMBL367540)
Affinity DataIC50:  1.00E+3nMAssay Description:In vitro opioid receptor binding competition against 1 nM [3H]- Naltrexone in the presence of 100 mM NaCl.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Sri International

Curated by ChEMBL
LigandPNGBDBM50020516(2-(3-{2-[2-hydroxy-(E)-1-methenylimino]-1-methyl-1...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of eel acetylcholinesterase (AChE) activity by 50% More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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