Affinity DataIC50: 4nMAssay Description:Inhibition of CypD (unknown origin) PPIase activity using N-Suc-AAPF-p-nitroanilide as substrate preincubated with enzyme for 10 mins followed by chy...More data for this Ligand-Target Pair
Affinity DataIC50: 60nMAssay Description:Displacement of fluorescein labelled cyclosporine A derivative from human recombinant CypD (30 to 207 residues) expressed in Escherichia coli cells i...More data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Homo sapiens (Human))
Università
Curated by ChEMBL
Università
Curated by ChEMBL
Affinity DataIC50: 150nMAssay Description:Inhibition of (-)-[3H]- D-888 binding to L-type calcium channels in kitten heart ventricle membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 190nMAssay Description:Displacement of fluorescein labelled cyclosporine A derivative from human recombinant CypD (30 to 207 residues) expressed in Escherichia coli cells i...More data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Homo sapiens (Human))
Università
Curated by ChEMBL
Università
Curated by ChEMBL
Affinity DataIC50: 260nMAssay Description:Inhibition of (-)-[3H]- D-888 binding to L-type calcium channels in kitten heart ventricle membranesMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Homo sapiens (Human))
Università
Curated by ChEMBL
Università
Curated by ChEMBL
Affinity DataIC50: 540nMAssay Description:Inhibition of (-)-[3H]- D-888 binding to L-type calcium channels in kitten heart ventricle membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 600nMAssay Description:Inhibition of CypD (unknown origin) PPIase activity using N-Suc-AAPF-p-nitroanilide as substrate preincubated with enzyme for 10 mins followed by chy...More data for this Ligand-Target Pair
Affinity DataIC50: 735nMAssay Description:Displacement of fluorescein labelled cyclosporine A derivative from human recombinant CypD (30 to 207 residues) expressed in Escherichia coli cells i...More data for this Ligand-Target Pair
Affinity DataIC50: 1.35E+3nMAssay Description:Displacement of fluorescein labelled cyclosporine A derivative from human recombinant CypD (30 to 207 residues) expressed in Escherichia coli cells i...More data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of CypD (unknown origin) PPIase activity using N-Suc-AAPF-p-nitroanilide as substrate preincubated with enzyme for 10 mins followed by chy...More data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+3nMAssay Description:Displacement of fluorescein labelled cyclosporine A derivative from human recombinant CypD (30 to 207 residues) expressed in Escherichia coli cells i...More data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+3nMAssay Description:Displacement of fluorescein labelled cyclosporine A derivative from human recombinant CypD (30 to 207 residues) expressed in Escherichia coli cells i...More data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Displacement of fluorescein labelled cyclosporine A derivative from human recombinant CypD (30 to 207 residues) expressed in Escherichia coli cells i...More data for this Ligand-Target Pair
Affinity DataIC50: 2.80E+3nMAssay Description:Displacement of fluorescein labelled cyclosporine A derivative from human recombinant CypD (30 to 207 residues) expressed in Escherichia coli cells i...More data for this Ligand-Target Pair
Affinity DataIC50: 3.50E+3nMAssay Description:Displacement of fluorescein labelled cyclosporine A derivative from human recombinant CypD (30 to 207 residues) expressed in Escherichia coli cells i...More data for this Ligand-Target Pair
Affinity DataIC50: 3.60E+3nMAssay Description:Displacement of fluorescein labelled cyclosporine A derivative from human recombinant CypD (30 to 207 residues) expressed in Escherichia coli cells i...More data for this Ligand-Target Pair
Affinity DataIC50: 4.10E+3nMAssay Description:Displacement of fluorescein labelled cyclosporine A derivative from human recombinant CypD (30 to 207 residues) expressed in Escherichia coli cells i...More data for this Ligand-Target Pair
Affinity DataIC50: 7.40E+3nMAssay Description:Inhibition of CypD (unknown origin) PPIase activity using N-Suc-AAPF-p-nitroanilide as substrate preincubated with enzyme for 10 mins followed by chy...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of fluorescein labelled cyclosporine A derivative from human recombinant CypD (30 to 207 residues) expressed in Escherichia coli cells i...More data for this Ligand-Target Pair
Affinity DataIC50: 2.80E+4nMAssay Description:Inhibition of CypD (unknown origin) PPIase activity using N-Suc-AAPF-p-nitroanilide as substrate preincubated with enzyme for 10 mins followed by chy...More data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Displacement of fluorescein labelled cyclosporine A derivative from human recombinant CypD (30 to 207 residues) expressed in Escherichia coli cells i...More data for this Ligand-Target Pair
Affinity DataIC50: 4.40E+4nMAssay Description:Displacement of fluorescein labelled cyclosporine A derivative from human recombinant CypD (30 to 207 residues) expressed in Escherichia coli cells i...More data for this Ligand-Target Pair
Affinity DataIC50: 5.40E+4nMAssay Description:Displacement of fluorescein labelled cyclosporine A derivative from human recombinant CypD (30 to 207 residues) expressed in Escherichia coli cells i...More data for this Ligand-Target Pair
Affinity DataIC50: 8.00E+4nMAssay Description:Displacement of fluorescein labelled cyclosporine A derivative from human recombinant CypD (30 to 207 residues) expressed in Escherichia coli cells i...More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Displacement of fluorescein labelled cyclosporine A derivative from human recombinant CypD (30 to 207 residues) expressed in Escherichia coli cells i...More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Displacement of fluorescein labelled cyclosporine A derivative from human recombinant CypD (30 to 207 residues) expressed in Escherichia coli cells i...More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Displacement of fluorescein labelled cyclosporine A derivative from human recombinant CypD (30 to 207 residues) expressed in Escherichia coli cells i...More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Displacement of fluorescein labelled cyclosporine A derivative from human recombinant CypD (30 to 207 residues) expressed in Escherichia coli cells i...More data for this Ligand-Target Pair
Affinity DataIC50: 4.90E+5nMAssay Description:Displacement of fluorescein labelled cyclosporine A derivative from human recombinant CypD (30 to 207 residues) expressed in Escherichia coli cells i...More data for this Ligand-Target Pair
Affinity DataIC50: 8.70E+5nMAssay Description:Displacement of fluorescein labelled cyclosporine A derivative from human recombinant CypD (30 to 207 residues) expressed in Escherichia coli cells i...More data for this Ligand-Target Pair
TargetATP-binding cassette sub-family C member 9(Rattus norvegicus)
Heinrich-Heine-Universit£T
Curated by ChEMBL
Heinrich-Heine-Universit£T
Curated by ChEMBL
Affinity DataKd: 17nMAssay Description:Binding affinity to the sulfonylurea receptor 2A (SUR2A) in purified membranes of rat-heart myocytesMore data for this Ligand-Target Pair
Affinity DataKd: 30nMAssay Description:Binding affinity to CypD (unknown origin) assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
TargetATP-binding cassette sub-family C member 9(Rattus norvegicus)
Heinrich-Heine-Universit£T
Curated by ChEMBL
Heinrich-Heine-Universit£T
Curated by ChEMBL
Affinity DataKd: 8.32E+3nMAssay Description:Binding affinity towards Sulfonylurea receptor 2B (SUR2B) in cultured rat aortic smooth muscle cells (SMC)More data for this Ligand-Target Pair
TargetATP-binding cassette sub-family C member 9(Rattus norvegicus)
Heinrich-Heine-Universit£T
Curated by ChEMBL
Heinrich-Heine-Universit£T
Curated by ChEMBL
Affinity DataKd: 20nMAssay Description:Binding affinity to the sulfonylurea receptor 2A (SUR2A) in purified membranes of rat-heart myocytesMore data for this Ligand-Target Pair
TargetATP-binding cassette sub-family C member 9(Rattus norvegicus)
Heinrich-Heine-Universit£T
Curated by ChEMBL
Heinrich-Heine-Universit£T
Curated by ChEMBL
Affinity DataKd: 138nMAssay Description:Binding affinity to the sulfonylurea receptor 2A (SUR2A) in purified membranes of rat-heart myocytesMore data for this Ligand-Target Pair
TargetATP-binding cassette sub-family C member 9(Rattus norvegicus)
Heinrich-Heine-Universit£T
Curated by ChEMBL
Heinrich-Heine-Universit£T
Curated by ChEMBL
Affinity DataKd: 6.61E+3nMAssay Description:Binding affinity to the sulfonylurea receptor 2A (SUR2A) in purified membranes of rat-heart myocytesMore data for this Ligand-Target Pair
TargetATP-binding cassette sub-family C member 9(Rattus norvegicus)
Heinrich-Heine-Universit£T
Curated by ChEMBL
Heinrich-Heine-Universit£T
Curated by ChEMBL
Affinity DataKd: 66nMAssay Description:Binding affinity to the sulfonylurea receptor 2A (SUR2A) in purified membranes of rat-heart myocytesMore data for this Ligand-Target Pair
TargetATP-binding cassette sub-family C member 9(Rattus norvegicus)
Heinrich-Heine-Universit£T
Curated by ChEMBL
Heinrich-Heine-Universit£T
Curated by ChEMBL
Affinity DataKd: 10nMAssay Description:Binding affinity towards Sulfonylurea receptor 2B (SUR2B) in cultured rat aortic smooth muscle cells (SMC)More data for this Ligand-Target Pair
TargetATP-binding cassette sub-family C member 9(Rattus norvegicus)
Heinrich-Heine-Universit£T
Curated by ChEMBL
Heinrich-Heine-Universit£T
Curated by ChEMBL
Affinity DataKd: 1.59E+3nMAssay Description:Binding affinity towards Sulfonylurea receptor 2B (SUR2B) in cultured rat aortic smooth muscle cells (SMC)More data for this Ligand-Target Pair
TargetATP-binding cassette sub-family C member 9(Rattus norvegicus)
Heinrich-Heine-Universit£T
Curated by ChEMBL
Heinrich-Heine-Universit£T
Curated by ChEMBL
Affinity DataKd: 7.10nMAssay Description:Binding affinity towards Sulfonylurea receptor 2B (SUR2B) in cultured rat aortic smooth muscle cells (SMC)More data for this Ligand-Target Pair
TargetATP-binding cassette sub-family C member 9(Rattus norvegicus)
Heinrich-Heine-Universit£T
Curated by ChEMBL
Heinrich-Heine-Universit£T
Curated by ChEMBL
Affinity DataKd: 11nMAssay Description:Binding affinity towards Sulfonylurea receptor 2B (SUR2B) in cultured rat aortic smooth muscle cells (SMC)More data for this Ligand-Target Pair
TargetATP-binding cassette sub-family C member 9(Rattus norvegicus)
Heinrich-Heine-Universit£T
Curated by ChEMBL
Heinrich-Heine-Universit£T
Curated by ChEMBL
Affinity DataKd: 3.16E+3nMAssay Description:Binding affinity to the sulfonylurea receptor 2A (SUR2A) in purified membranes of rat-heart myocytesMore data for this Ligand-Target Pair
TargetATP-binding cassette sub-family C member 9(Rattus norvegicus)
Heinrich-Heine-Universit£T
Curated by ChEMBL
Heinrich-Heine-Universit£T
Curated by ChEMBL
Affinity DataKd: 4.47E+3nMAssay Description:Binding affinity to the sulfonylurea receptor 2A (SUR2A) in purified membranes of rat-heart myocytesMore data for this Ligand-Target Pair
TargetATP-binding cassette sub-family C member 9(Rattus norvegicus)
Heinrich-Heine-Universit£T
Curated by ChEMBL
Heinrich-Heine-Universit£T
Curated by ChEMBL
Affinity DataKd: 23nMAssay Description:Binding affinity towards Sulfonylurea receptor 2B (SUR2B) in cultured rat aortic smooth muscle cells (SMC)More data for this Ligand-Target Pair
TargetATP-binding cassette sub-family C member 9(Rattus norvegicus)
Heinrich-Heine-Universit£T
Curated by ChEMBL
Heinrich-Heine-Universit£T
Curated by ChEMBL
Affinity DataKd: 1.00E+3nMAssay Description:Binding affinity towards Sulfonylurea receptor 2B (SUR2B) in cultured rat aortic smooth muscle cells (SMC)More data for this Ligand-Target Pair
TargetATP-binding cassette sub-family C member 9(Rattus norvegicus)
Heinrich-Heine-Universit£T
Curated by ChEMBL
Heinrich-Heine-Universit£T
Curated by ChEMBL
Affinity DataKd: 65nMAssay Description:Binding affinity towards Sulfonylurea receptor 2B (SUR2B) in cultured rat aortic smooth muscle cells (SMC)More data for this Ligand-Target Pair
TargetATP-binding cassette sub-family C member 9(Rattus norvegicus)
Heinrich-Heine-Universit£T
Curated by ChEMBL
Heinrich-Heine-Universit£T
Curated by ChEMBL
Affinity DataKd: 15nMAssay Description:Binding affinity to the sulfonylurea receptor 2A (SUR2A) in purified membranes of rat-heart myocytesMore data for this Ligand-Target Pair
TargetATP-binding cassette sub-family C member 9(Rattus norvegicus)
Heinrich-Heine-Universit£T
Curated by ChEMBL
Heinrich-Heine-Universit£T
Curated by ChEMBL
Affinity DataKd: 5.62E+3nMAssay Description:Binding affinity to the sulfonylurea receptor 2A (SUR2A) in purified membranes of rat-heart myocytesMore data for this Ligand-Target Pair
TargetATP-binding cassette sub-family C member 9(Rattus norvegicus)
Heinrich-Heine-Universit£T
Curated by ChEMBL
Heinrich-Heine-Universit£T
Curated by ChEMBL
Affinity DataKd: 457nMAssay Description:Binding affinity towards Sulfonylurea receptor 2B (SUR2B) in cultured rat aortic smooth muscle cells (SMC)More data for this Ligand-Target Pair
TargetATP-binding cassette sub-family C member 9(Rattus norvegicus)
Heinrich-Heine-Universit£T
Curated by ChEMBL
Heinrich-Heine-Universit£T
Curated by ChEMBL
Affinity DataKd: 363nMAssay Description:Binding affinity to the sulfonylurea receptor 2A (SUR2A) in purified membranes of rat-heart myocytesMore data for this Ligand-Target Pair