TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
Oslo University Hospital
Curated by ChEMBL
Oslo University Hospital
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibition of TNKS2 (unknown origin) by NAD+-dependent autopoly(ADP ribosyl)lation assayMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
Oslo University Hospital
Curated by ChEMBL
Oslo University Hospital
Curated by ChEMBL
Affinity DataIC50: 43nMAssay Description:Inhibition of TNKS2 (unknown origin) by NAD+-dependent autopoly(ADP ribosyl)lation assayMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-1(Homo sapiens (Human))
Oslo University Hospital
Curated by ChEMBL
Oslo University Hospital
Curated by ChEMBL
Affinity DataIC50: 46nMAssay Description:Inhibition of TNSK1 (unknown origin) by NAD+-dependent autopoly(ADP ribosyl)lation assayMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
Oslo University Hospital
Curated by ChEMBL
Oslo University Hospital
Curated by ChEMBL
Affinity DataIC50: 51nMAssay Description:Inhibition of TNKS2 (unknown origin) by NAD+-dependent autopoly(ADP ribosyl)lation assayMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
Oslo University Hospital
Curated by ChEMBL
Oslo University Hospital
Curated by ChEMBL
Affinity DataIC50: 54nMAssay Description:Inhibition of TNKS2 (unknown origin) by NAD+-dependent autopoly(ADP ribosyl)lation assayMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
Oslo University Hospital
Curated by ChEMBL
Oslo University Hospital
Curated by ChEMBL
Affinity DataIC50: 290nMAssay Description:Inhibition of TNKS2 (unknown origin) by NAD+-dependent autopoly(ADP ribosyl)lation assayMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
Oslo University Hospital
Curated by ChEMBL
Oslo University Hospital
Curated by ChEMBL
Affinity DataIC50: 460nMAssay Description:Inhibition of TNKS2 (unknown origin) by NAD+-dependent autopoly(ADP ribosyl)lation assayMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
Oslo University Hospital
Curated by ChEMBL
Oslo University Hospital
Curated by ChEMBL
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of TNKS2 (unknown origin) by NAD+-dependent autopoly(ADP ribosyl)lation assayMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
Oslo University Hospital
Curated by ChEMBL
Oslo University Hospital
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of TNKS2 (unknown origin) by NAD+-dependent autopoly(ADP ribosyl)lation assayMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
Oslo University Hospital
Curated by ChEMBL
Oslo University Hospital
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of TNKS2 (unknown origin) by NAD+-dependent autopoly(ADP ribosyl)lation assayMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
Oslo University Hospital
Curated by ChEMBL
Oslo University Hospital
Curated by ChEMBL
Affinity DataIC50: 1.23E+4nMAssay Description:Inhibition of TNKS2 (unknown origin) by NAD+-dependent autopoly(ADP ribosyl)lation assayMore data for this Ligand-Target Pair
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair