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Found 275 with Last Name = 'schilke' and Initial = 'h'
TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM50610836(MSC-4381)
Affinity DataKi:  11nMAssay Description:Binding affinity to full-length C-terminal GFP-tagged human MCT4 incubated for 1 hrs by fluorescence cross-correlation spectroscopy analysisMore data for this Ligand-Target Pair
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TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM50610833(CHEMBL5276884)
Affinity DataKi:  11nMAssay Description:Binding affinity to full-length C-terminal GFP-tagged human MCT4 incubated for 1 hrs by fluorescence cross-correlation spectroscopy analysisMore data for this Ligand-Target Pair
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TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM50610834(CHEMBL5279064)
Affinity DataKi:  16nMAssay Description:Binding affinity to full-length C-terminal GFP-tagged human MCT4 incubated for 1 hrs by fluorescence cross-correlation spectroscopy analysisMore data for this Ligand-Target Pair
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TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM50610830(CHEMBL5267752)
Affinity DataKi:  17nMAssay Description:Binding affinity to full-length C-terminal GFP-tagged human MCT4 incubated for 1 hrs by fluorescence cross-correlation spectroscopy analysisMore data for this Ligand-Target Pair
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TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM50610837(CHEMBL5281492)
Affinity DataKi:  17nMAssay Description:Binding affinity to full-length C-terminal GFP-tagged human MCT4 incubated for 1 hrs by fluorescence cross-correlation spectroscopy analysisMore data for this Ligand-Target Pair
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TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM50610835(CHEMBL5267349)
Affinity DataKi:  17nMAssay Description:Binding affinity to full-length C-terminal GFP-tagged human MCT4 incubated for 1 hrs by fluorescence cross-correlation spectroscopy analysisMore data for this Ligand-Target Pair
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TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM50610826(CHEMBL5287351)
Affinity DataKi:  29nMAssay Description:Binding affinity to full-length C-terminal GFP-tagged human MCT4 incubated for 1 hrs by fluorescence cross-correlation spectroscopy analysisMore data for this Ligand-Target Pair
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TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM50610827(CHEMBL5287780)
Affinity DataKi:  32nMAssay Description:Binding affinity to full-length C-terminal GFP-tagged human MCT4 incubated for 1 hrs by fluorescence cross-correlation spectroscopy analysisMore data for this Ligand-Target Pair
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TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM50610824(CHEMBL5268966)
Affinity DataKi:  37nMAssay Description:Binding affinity to full-length C-terminal GFP-tagged human MCT4 incubated for 1 hrs by fluorescence cross-correlation spectroscopy analysisMore data for this Ligand-Target Pair
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TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM50610829(CHEMBL5288904)
Affinity DataKi:  51nMAssay Description:Binding affinity to full-length C-terminal GFP-tagged human MCT4 incubated for 1 hrs by fluorescence cross-correlation spectroscopy analysisMore data for this Ligand-Target Pair
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TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM50610831(CHEMBL5265956)
Affinity DataKi:  56nMAssay Description:Binding affinity to full-length C-terminal GFP-tagged human MCT4 incubated for 1 hrs by fluorescence cross-correlation spectroscopy analysisMore data for this Ligand-Target Pair
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TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM50610825(CHEMBL5266104)
Affinity DataKi:  99nMAssay Description:Binding affinity to full-length C-terminal GFP-tagged human MCT4 incubated for 1 hrs by fluorescence cross-correlation spectroscopy analysisMore data for this Ligand-Target Pair
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TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM50610828(CHEMBL5271816)
Affinity DataKi:  222nMAssay Description:Binding affinity to full-length C-terminal GFP-tagged human MCT4 incubated for 1 hrs by fluorescence cross-correlation spectroscopy analysisMore data for this Ligand-Target Pair
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TargetMonocarboxylate transporter 4(Mus musculus)TBA
LigandPNGBDBM50610868(CHEMBL5282978)
Affinity DataKi:  301nMAssay Description:Binding affinity to full-length C-terminal GFP-tagged mouse MCT4 incubated for 1 hrs by fluorescence cross-correlation spectroscopy analysisMore data for this Ligand-Target Pair
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TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50615065(CHEMBL5280227)
Affinity DataIC50:  2nMAssay Description:Inhibition of human full length GST-tagged WEE1 expressed in insect cells incubated for 15 mins followed by ATP addition by ADP Glo luminescent assayMore data for this Ligand-Target Pair
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TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50615031(CHEMBL5281815)
Affinity DataIC50:  2.30nMAssay Description:Inhibition of human full length GST-tagged WEE1 expressed in insect cells incubated for 15 mins followed by ATP addition by ADP Glo luminescent assayMore data for this Ligand-Target Pair
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TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50615046(CHEMBL5289001)
Affinity DataIC50:  2.30nMAssay Description:Inhibition of human full length GST-tagged WEE1 expressed in insect cells incubated for 15 mins followed by ATP addition by ADP Glo luminescent assayMore data for this Ligand-Target Pair
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TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM21998(6-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-5-{[(4S)-...)
Affinity DataIC50:  2.5nMAssay Description:Inhibition of human MCT4 in human SNU-398 cells assessed as inhibition of radioactive lactate efflux preincubated for 30 mins followed by D(+)glucose...More data for this Ligand-Target Pair
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TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))TBA
LigandPNGBDBM50402023(BI 6727 | VOLASERTIB)
Affinity DataIC50:  2.5nMAssay Description:Inhibition of human N-terminal His6-tagged recombinant full-length PLK1 expressed in baculovirus infected Sf9 cells incubated for 15 mins followed by...More data for this Ligand-Target Pair
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50615034(CHEMBL5288130)
Affinity DataIC50:  2.60nMAssay Description:Inhibition of human full length GST-tagged WEE1 expressed in insect cells incubated for 15 mins followed by ATP addition by ADP Glo luminescent assayMore data for this Ligand-Target Pair
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TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50615037(CHEMBL5285844)
Affinity DataIC50:  2.80nMAssay Description:Inhibition of human full length GST-tagged WEE1 expressed in insect cells incubated for 15 mins followed by ATP addition by ADP Glo luminescent assayMore data for this Ligand-Target Pair
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TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50615029(CHEMBL5272346)
Affinity DataIC50:  2.80nMAssay Description:Inhibition of human full length GST-tagged WEE1 expressed in insect cells incubated for 15 mins followed by ATP addition by ADP Glo luminescent assayMore data for this Ligand-Target Pair
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TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50615030(CHEMBL5286243)
Affinity DataIC50:  2.90nMAssay Description:Inhibition of human full length GST-tagged WEE1 expressed in insect cells incubated for 15 mins followed by ATP addition by ADP Glo luminescent assayMore data for this Ligand-Target Pair
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TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50615032(CHEMBL5268938)
Affinity DataIC50:  2.90nMAssay Description:Inhibition of human full length GST-tagged WEE1 expressed in insect cells incubated for 15 mins followed by ATP addition by ADP Glo luminescent assayMore data for this Ligand-Target Pair
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TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM518537(2-Allyl-1-(6-(2-hydroxypropan-2-yl)pyridin-2-yl)-6...)
Affinity DataIC50:  2.90nMAssay Description:Inhibition of human full length GST-tagged WEE1 expressed in insect cells incubated for 15 mins followed by ATP addition by ADP Glo luminescent assayMore data for this Ligand-Target Pair
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TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50240826(AZD-1775 | MK-1775 | US11124518, Example AZD1775 |...)
Affinity DataIC50:  3nMAssay Description:Inhibition of human full length GST-tagged WEE1 expressed in insect cells incubated for 15 mins followed by ATP addition by ADP Glo luminescent assayMore data for this Ligand-Target Pair
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50615063(CHEMBL5285363)
Affinity DataIC50:  3.20nMAssay Description:Inhibition of human full length GST-tagged WEE1 expressed in insect cells incubated for 15 mins followed by ATP addition by ADP Glo luminescent assayMore data for this Ligand-Target Pair
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TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM518536(2-Allyl-6-((4,4-dimethyl-1,2,3,4-tetrahydroisoquin...)
Affinity DataIC50:  3.30nMAssay Description:Inhibition of human full length GST-tagged WEE1 expressed in insect cells incubated for 15 mins followed by ATP addition by ADP Glo luminescent assayMore data for this Ligand-Target Pair
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TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50615039(CHEMBL5280668)
Affinity DataIC50:  3.30nMAssay Description:Inhibition of human full length GST-tagged WEE1 expressed in insect cells incubated for 15 mins followed by ATP addition by ADP Glo luminescent assayMore data for this Ligand-Target Pair
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TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50615052(CHEMBL5283530)
Affinity DataIC50:  3.30nMAssay Description:Inhibition of human full length GST-tagged WEE1 expressed in insect cells incubated for 15 mins followed by ATP addition by ADP Glo luminescent assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50615051(CHEMBL5285960)
Affinity DataIC50:  3.70nMAssay Description:Inhibition of human full length GST-tagged WEE1 expressed in insect cells incubated for 15 mins followed by ATP addition by ADP Glo luminescent assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50615036(CHEMBL5269559)
Affinity DataIC50:  3.80nMAssay Description:Inhibition of human full length GST-tagged WEE1 expressed in insect cells incubated for 15 mins followed by ATP addition by ADP Glo luminescent assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50615054(CHEMBL5289458)
Affinity DataIC50:  3.80nMAssay Description:Inhibition of human full length GST-tagged WEE1 expressed in insect cells incubated for 15 mins followed by ATP addition by ADP Glo luminescent assayMore data for this Ligand-Target Pair
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TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50615040(CHEMBL5289015)
Affinity DataIC50:  4.10nMAssay Description:Inhibition of human full length GST-tagged WEE1 expressed in insect cells incubated for 15 mins followed by ATP addition by ADP Glo luminescent assayMore data for this Ligand-Target Pair
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TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50615066(CHEMBL5266595)
Affinity DataIC50:  4.20nMAssay Description:Inhibition of human full length GST-tagged WEE1 expressed in insect cells incubated for 15 mins followed by ATP addition by ADP Glo luminescent assayMore data for this Ligand-Target Pair
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TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50615050(CHEMBL5274253)
Affinity DataIC50:  4.30nMAssay Description:Inhibition of human full length GST-tagged WEE1 expressed in insect cells incubated for 15 mins followed by ATP addition by ADP Glo luminescent assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50615035(CHEMBL5291431)
Affinity DataIC50:  4.5nMAssay Description:Inhibition of human full length GST-tagged WEE1 expressed in insect cells incubated for 15 mins followed by ATP addition by ADP Glo luminescent assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50615024(CHEMBL5291362)
Affinity DataIC50:  4.5nMAssay Description:Inhibition of human full length GST-tagged WEE1 expressed in insect cells incubated for 15 mins followed by ATP addition by ADP Glo luminescent assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50615064(CHEMBL5290136)
Affinity DataIC50:  4.60nMAssay Description:Inhibition of human full length GST-tagged WEE1 expressed in insect cells incubated for 15 mins followed by ATP addition by ADP Glo luminescent assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50615038(CHEMBL5267993)
Affinity DataIC50:  4.60nMAssay Description:Inhibition of human full length GST-tagged WEE1 expressed in insect cells incubated for 15 mins followed by ATP addition by ADP Glo luminescent assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50615033(CHEMBL5269511)
Affinity DataIC50:  4.80nMAssay Description:Inhibition of human full length GST-tagged WEE1 expressed in insect cells incubated for 15 mins followed by ATP addition by ADP Glo luminescent assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50615025(CHEMBL5269631)
Affinity DataIC50:  4.80nMAssay Description:Inhibition of human full length GST-tagged WEE1 expressed in insect cells incubated for 15 mins followed by ATP addition by ADP Glo luminescent assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50615060(CHEMBL5277502)
Affinity DataIC50:  4.90nMAssay Description:Inhibition of human full length GST-tagged WEE1 expressed in insect cells incubated for 15 mins followed by ATP addition by ADP Glo luminescent assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50615056(CHEMBL5266147)
Affinity DataIC50:  4.90nMAssay Description:Inhibition of human full length GST-tagged WEE1 expressed in insect cells incubated for 15 mins followed by ATP addition by ADP Glo luminescent assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50615053(CHEMBL5291191)
Affinity DataIC50:  5.30nMAssay Description:Inhibition of human full length GST-tagged WEE1 expressed in insect cells incubated for 15 mins followed by ATP addition by ADP Glo luminescent assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50615059(CHEMBL5286445)
Affinity DataIC50:  5.40nMAssay Description:Inhibition of human full length GST-tagged WEE1 expressed in insect cells incubated for 15 mins followed by ATP addition by ADP Glo luminescent assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50615026(CHEMBL5286202)
Affinity DataIC50:  5.40nMAssay Description:Inhibition of human full length GST-tagged WEE1 expressed in insect cells incubated for 15 mins followed by ATP addition by ADP Glo luminescent assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50615067(CHEMBL5275152)
Affinity DataIC50:  5.90nMAssay Description:Inhibition of human full length GST-tagged WEE1 expressed in insect cells incubated for 15 mins followed by ATP addition by ADP Glo luminescent assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50615028(CHEMBL5285865)
Affinity DataIC50:  6nMAssay Description:Inhibition of human full length GST-tagged WEE1 expressed in insect cells incubated for 15 mins followed by ATP addition by ADP Glo luminescent assayMore data for this Ligand-Target Pair
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TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM21998(6-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-5-{[(4S)-...)
Affinity DataIC50:  6.20nMAssay Description:Inhibition of human MCT4 in human SNU-398 cells assessed as inhibition of lactate efflux preincubated for 30 mins followed by D(+)glucose and measure...More data for this Ligand-Target Pair
In DepthDetails PubMed
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