TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 0.180nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 0.270nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 0.280nMAssay Description:Displacement of [3H]-PK11195 from TSPO in rat C6 cell lysate after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 2.20nMAssay Description:Displacement of [3H]-PK11195 from TSPO in rat C6 cell lysate after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 5.60nMAssay Description:Displacement of [3H]-PK11195 from TSPO in rat C6 cell lysate after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 6.40nMAssay Description:Displacement of [3H]-PK11195 from TSPO in rat C6 cell lysate after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 7.30nMAssay Description:Displacement of [3H]-PK11195 from TSPO in rat C6 cell lysate after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 9.70nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:Displacement of [3H]-PK11195 from TSPO in rat C6 cell lysate after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 14nMAssay Description:Displacement of [3H]-PK11195 from TSPO in rat C6 cell lysate after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 19nMAssay Description:Displacement of [3H]-PK11195 from TSPO in rat C6 cell lysate after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Displacement of [3H]-PK11195 from TSPO in rat C6 cell lysate after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 38nMAssay Description:Displacement of [3H]-PK11195 from TSPO in rat C6 cell lysate after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 49nMAssay Description:Displacement of [3H]-PK11195 from TSPO in rat C6 cell lysate after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 55nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 59nMAssay Description:Displacement of [3H]-PK11195 from TSPO in rat C6 cell lysate after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 68nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 83nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 88nMAssay Description:Displacement of [3H]-PK11195 from TSPO in rat C6 cell lysate after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 94nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 95nMAssay Description:Displacement of [3H]-PK11195 from TSPO in rat C6 cell lysate after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 127nMAssay Description:Displacement of [3H]-PK11195 from TSPO in rat C6 cell lysate after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 157nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 201nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 252nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 277nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 397nMAssay Description:Displacement of [3H]-PK11195 from TSPO in rat C6 cell lysate after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: >500nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: >500nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-flunitrazepam from TSPO in rat C6 cell lysate by liquid scintillation countingMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-flunitrazepam from TSPO in rat C6 cell lysate by liquid scintillation countingMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-flunitrazepam from TSPO in rat C6 cell lysate by liquid scintillation countingMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-flunitrazepam from TSPO in rat C6 cell lysate by liquid scintillation countingMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-flunitrazepam from TSPO in rat C6 cell lysate by liquid scintillation countingMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-flunitrazepam from TSPO in rat C6 cell lysate by liquid scintillation countingMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-flunitrazepam from TSPO in rat C6 cell lysate by liquid scintillation countingMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-flunitrazepam from TSPO in rat C6 cell lysate by liquid scintillation countingMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-flunitrazepam from TSPO in rat C6 cell lysate by liquid scintillation countingMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-flunitrazepam from TSPO in rat C6 cell lysate by liquid scintillation countingMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-flunitrazepam from TSPO in rat C6 cell lysate by liquid scintillation countingMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-flunitrazepam from TSPO in rat C6 cell lysate by liquid scintillation countingMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-flunitrazepam from TSPO in rat C6 cell lysate by liquid scintillation countingMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-flunitrazepam from TSPO in rat C6 cell lysate by liquid scintillation countingMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-flunitrazepam from TSPO in rat C6 cell lysate by liquid scintillation countingMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-flunitrazepam from TSPO in rat C6 cell lysate by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+3nMAssay Description:Live-cell amino acid uptake assays using HEK293 cells were carried out in 96-well plates (CulturPlate-96, Perkin Elmer). 96-well plates were coated w...More data for this Ligand-Target Pair
TargetAmino acid transporter(Rattus norvegicus)
Vanderbilt University Medical Center
Curated by ChEMBL
Vanderbilt University Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of ASCT2-mediated glutamine transport in rat C6 cells using [3H]-glutamine after 15 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 1.80E+3nMAssay Description:Live-cell amino acid uptake assays using HEK293 cells were carried out in 96-well plates (CulturPlate-96, Perkin Elmer). 96-well plates were coated w...More data for this Ligand-Target Pair
TargetAmino acid transporter(Rattus norvegicus)
Vanderbilt University Medical Center
Curated by ChEMBL
Vanderbilt University Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of ASCT2-mediated glutamine transport in rat C6 cells using [3H]-glutamine after 15 mins by scintillation countingMore data for this Ligand-Target Pair