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Found 99 with Last Name = 'kang' and Initial = 'ij'
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50275991(4-chlorophenyl 2-phenylethenesulfonate | CHEMBL469...)
Affinity DataIC50:  302nMAssay Description:Displacement of [3H]BRL49653 from PPARgamma (unknown origin) ligand binding domain by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50276033(3-phenoxyphenyl 2-phenylethenesulfonate | CHEMBL51...)
Affinity DataIC50:  382nMAssay Description:Displacement of [3H]BRL49653 from PPARgamma (unknown origin) ligand binding domain by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50275989(CHEMBL469939 | p-tolyl 2-phenylethenesulfonate)
Affinity DataIC50:  407nMAssay Description:Displacement of [3H]BRL49653 from PPARgamma (unknown origin) ligand binding domain by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50276029(4-(benzyloxy)phenyl 2-phenylethenesulfonate | CHEM...)
Affinity DataIC50:  703nMAssay Description:Displacement of [3H]BRL49653 from PPARgamma (unknown origin) ligand binding domain by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50276030(CHEMBL471829 | ethyl 4-(styrylsulfonyloxy)benzoate)
Affinity DataIC50:  747nMAssay Description:Displacement of [3H]BRL49653 from PPARgamma (unknown origin) ligand binding domain by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50275988(CHEMBL469938 | naphthalen-2-yl 2-phenylethenesulfo...)
Affinity DataIC50:  1.09E+3nMAssay Description:Displacement of [3H]BRL49653 from PPARgamma (unknown origin) ligand binding domain by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50275990(CHEMBL467711 | m-tolyl 2-phenylethenesulfonate)
Affinity DataIC50:  1.19E+3nMAssay Description:Displacement of [3H]BRL49653 from PPARgamma (unknown origin) ligand binding domain by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50275993(4-methoxyphenyl 2-phenylethenesulfonate | CHEMBL46...)
Affinity DataIC50:  1.29E+3nMAssay Description:Displacement of [3H]BRL49653 from PPARgamma (unknown origin) ligand binding domain by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine--tRNA ligase, cytoplasmic(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50111476(1-[5-(4''-Chloro-biphenyl-4-yloxy)-pentyl]-3-pyrid...)
Affinity DataIC50:  1.31E+3nMAssay Description:Inhibitory activity against Echovirus 9 using plaque reduction assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50275950(CHEMBL443343 | phenyl 2-phenylethenesulfonate)
Affinity DataIC50:  1.33E+3nMAssay Description:Displacement of [3H]BRL49653 from PPARgamma (unknown origin) ligand binding domain by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50275992(2,4,6-trichlorophenyl 2-phenylethenesulfonate | CH...)
Affinity DataIC50:  1.44E+3nMAssay Description:Displacement of [3H]BRL49653 from PPARgamma (unknown origin) ligand binding domain by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50276031(4-formylphenyl 2-phenylethenesulfonate | CHEMBL471...)
Affinity DataIC50:  2.10E+3nMAssay Description:Displacement of [3H]BRL49653 from PPARgamma (unknown origin) ligand binding domain by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50276032(4-acetamidophenyl 2-phenylethenesulfonate | CHEMBL...)
Affinity DataIC50:  1.07E+4nMAssay Description:Displacement of [3H]BRL49653 from PPARgamma (unknown origin) ligand binding domain by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50276034(3-(styrylsulfonyloxy)benzoic acid | CHEMBL470575)
Affinity DataIC50:  1.35E+4nMAssay Description:Displacement of [3H]BRL49653 from PPARgamma (unknown origin) ligand binding domain by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine--tRNA ligase, cytoplasmic(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50171204(1-[(R)-5-(4'-Chloro-biphenyl-4-yloxy)-3-methyl-pen...)
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibitory activity against Echovirus 9 using plaque reduction assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine--tRNA ligase, cytoplasmic(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50171203(1-[(S)-5-(4'-Chloro-biphenyl-4-yloxy)-3-methyl-pen...)
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibitory activity against Echovirus 9 using plaque reduction assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNonstructural protein 5A(Hepatitis C virus)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50522203(CHEMBL4437203)
Affinity DataEC50:  41nMAssay Description:Inhibition of NS5A in HCV genotype 1b infected in human HuH7 replicon cells assessed as reduction in subgenomic viral RNA replication treated for 2 d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNonstructural protein 5A(Hepatitis C virus)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50522204(CHEMBL4546321)
Affinity DataEC50: >5.00E+4nMAssay Description:Inhibition of NS5A in HCV genotype 1b infected in human HuH7 replicon cells assessed as reduction in subgenomic viral RNA replication treated for 2 d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNonstructural protein 5A(Hepatitis C virus)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50522205(CHEMBL4544117)
Affinity DataEC50:  2.60nMAssay Description:Inhibition of NS5A in HCV genotype 1b infected in human HuH7 replicon cells assessed as reduction in subgenomic viral RNA replication treated for 2 d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNonstructural protein 5A(Hepatitis C virus)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50522206(CHEMBL4445388)
Affinity DataEC50:  1.40nMAssay Description:Inhibition of NS5A in HCV genotype 1b infected in human HuH7 replicon cells assessed as reduction in subgenomic viral RNA replication treated for 2 d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNonstructural protein 5A(Hepatitis C virus)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50522207(CHEMBL4468540)
Affinity DataEC50:  0.00700nMAssay Description:Inhibition of NS5A in HCV genotype 1b infected in human HuH7 replicon cells assessed as reduction in subgenomic viral RNA replication treated for 2 d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNonstructural protein 5A(Hepatitis C virus)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50387084(BMS-790052 | DACLATASVIR)
Affinity DataEC50:  0.00900nMAssay Description:Inhibition of NS5A in HCV genotype 1b infected in human HuH7 replicon cells assessed as reduction in subgenomic viral RNA replication treated for 2 d...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNonstructural protein 5A(Hepatitis C virus)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50522208(CHEMBL4440654)
Affinity DataEC50:  1.10nMAssay Description:Inhibition of NS5A in HCV genotype 1b infected in human HuH7 replicon cells assessed as reduction in subgenomic viral RNA replication treated for 2 d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNonstructural protein 5A(Hepatitis C virus)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50522209(CHEMBL4441831)
Affinity DataEC50:  40nMAssay Description:Inhibition of NS5A in HCV genotype 1b infected in human HuH7 replicon cells assessed as reduction in subgenomic viral RNA replication treated for 2 d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNonstructural protein 5A(Hepatitis C virus)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50522210(CHEMBL4448110)
Affinity DataEC50:  7.20nMAssay Description:Inhibition of NS5A in HCV genotype 1b infected in human HuH7 replicon cells assessed as reduction in subgenomic viral RNA replication treated for 2 d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNonstructural protein 5A(Hepatitis C virus)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50522211(CHEMBL4550614)
Affinity DataEC50:  108nMAssay Description:Inhibition of NS5A in HCV genotype 1b infected in human HuH7 replicon cells assessed as reduction in subgenomic viral RNA replication treated for 2 d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNonstructural protein 5A(Hepatitis C virus)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50522212(CHEMBL4443748)
Affinity DataEC50:  0.190nMAssay Description:Inhibition of NS5A in HCV genotype 1b infected in human HuH7 replicon cells assessed as reduction in subgenomic viral RNA replication treated for 2 d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNonstructural protein 5A(Hepatitis C virus)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50522213(CHEMBL4456739)
Affinity DataEC50:  327nMAssay Description:Inhibition of NS5A in HCV genotype 1b infected in human HuH7 replicon cells assessed as reduction in subgenomic viral RNA replication treated for 2 d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNonstructural protein 5A(Hepatitis C virus)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50522214(CHEMBL4551169)
Affinity DataEC50:  2.82E+3nMAssay Description:Inhibition of NS5A in HCV genotype 1b infected in human HuH7 replicon cells assessed as reduction in subgenomic viral RNA replication treated for 2 d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNonstructural protein 5A(Hepatitis C virus)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50522215(CHEMBL4579658)
Affinity DataEC50:  159nMAssay Description:Inhibition of NS5A in HCV genotype 1b infected in human HuH7 replicon cells assessed as reduction in subgenomic viral RNA replication treated for 2 d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNonstructural protein 5A(Hepatitis C virus)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50522216(CHEMBL4517969)
Affinity DataEC50:  123nMAssay Description:Inhibition of NS5A in HCV genotype 1b infected in human HuH7 replicon cells assessed as reduction in subgenomic viral RNA replication treated for 2 d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNonstructural protein 5A(Hepatitis C virus)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50522217(CHEMBL4585945)
Affinity DataEC50:  179nMAssay Description:Inhibition of NS5A in HCV genotype 1b infected in human HuH7 replicon cells assessed as reduction in subgenomic viral RNA replication treated for 2 d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNonstructural protein 5A(Hepatitis C virus)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50522218(CHEMBL4442444)
Affinity DataEC50:  27nMAssay Description:Inhibition of NS5A in HCV genotype 1b infected in human HuH7 replicon cells assessed as reduction in subgenomic viral RNA replication treated for 2 d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNonstructural protein 5A(Hepatitis C virus)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50522219(CHEMBL4462939)
Affinity DataEC50:  732nMAssay Description:Inhibition of NS5A in HCV genotype 1b infected in human HuH7 replicon cells assessed as reduction in subgenomic viral RNA replication treated for 2 d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNonstructural protein 5A(Hepatitis C virus)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50522220(CHEMBL4592667)
Affinity DataEC50:  92nMAssay Description:Inhibition of NS5A in HCV genotype 1b infected in human HuH7 replicon cells assessed as reduction in subgenomic viral RNA replication treated for 2 d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNonstructural protein 5A(Hepatitis C virus)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50522221(CHEMBL4570173)
Affinity DataEC50:  433nMAssay Description:Inhibition of NS5A in HCV genotype 1b infected in human HuH7 replicon cells assessed as reduction in subgenomic viral RNA replication treated for 2 d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNonstructural protein 5A(Hepatitis C virus)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50522222(CHEMBL4443293)
Affinity DataEC50:  16nMAssay Description:Inhibition of NS5A in HCV genotype 1b infected in human HuH7 replicon cells assessed as reduction in subgenomic viral RNA replication treated for 2 d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNonstructural protein 5A(Hepatitis C virus)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50522223(CHEMBL4457196)
Affinity DataEC50:  23nMAssay Description:Inhibition of NS5A in HCV genotype 1b infected in human HuH7 replicon cells assessed as reduction in subgenomic viral RNA replication treated for 2 d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNonstructural protein 5A(Hepatitis C virus)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50522224(CHEMBL4449784)
Affinity DataEC50:  0.230nMAssay Description:Inhibition of NS5A in HCV genotype 1b infected in human HuH7 replicon cells assessed as reduction in subgenomic viral RNA replication treated for 2 d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNonstructural protein 5A(Hepatitis C virus)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50522225(CHEMBL4553591)
Affinity DataEC50:  1.90nMAssay Description:Inhibition of NS5A in HCV genotype 1b infected in human HuH7 replicon cells assessed as reduction in subgenomic viral RNA replication treated for 2 d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNonstructural protein 5A(Hepatitis C virus)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50522226(CHEMBL4435415)
Affinity DataEC50:  1.30nMAssay Description:Inhibition of NS5A in HCV genotype 1b infected in human HuH7 replicon cells assessed as reduction in subgenomic viral RNA replication treated for 2 d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNonstructural protein 5A(Hepatitis C virus)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50522227(CHEMBL4586142)
Affinity DataEC50:  110nMAssay Description:Inhibition of NS5A in HCV genotype 1b infected in human HuH7 replicon cells assessed as reduction in subgenomic viral RNA replication treated for 2 d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNonstructural protein 5A(Hepatitis C virus)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50522228(CHEMBL4568524)
Affinity DataEC50:  0.630nMAssay Description:Inhibition of NS5A in HCV genotype 1b infected in human HuH7 replicon cells assessed as reduction in subgenomic viral RNA replication treated for 2 d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNonstructural protein 5A(Hepatitis C virus)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50522229(CHEMBL4436675)
Affinity DataEC50:  1.70nMAssay Description:Inhibition of NS5A in HCV genotype 1b infected in human HuH7 replicon cells assessed as reduction in subgenomic viral RNA replication treated for 2 d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNonstructural protein 5A(Hepatitis C virus)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50522230(CHEMBL4474586)
Affinity DataEC50:  2.10nMAssay Description:Inhibition of NS5A in HCV genotype 1b infected in human HuH7 replicon cells assessed as reduction in subgenomic viral RNA replication treated for 2 d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNonstructural protein 5A(Hepatitis C virus)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50522231(CHEMBL4469566)
Affinity DataEC50:  272nMAssay Description:Inhibition of NS5A in HCV genotype 1b infected in human HuH7 replicon cells assessed as reduction in subgenomic viral RNA replication treated for 2 d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNonstructural protein 5A(Hepatitis C virus)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50522232(CHEMBL4592569)
Affinity DataEC50:  0.450nMAssay Description:Inhibition of NS5A in HCV genotype 1b infected in human HuH7 replicon cells assessed as reduction in subgenomic viral RNA replication treated for 2 d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNonstructural protein 5A(Hepatitis C virus)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50522233(CHEMBL4473401)
Affinity DataEC50:  1.5nMAssay Description:Inhibition of NS5A in HCV genotype 1b infected in human HuH7 replicon cells assessed as reduction in subgenomic viral RNA replication treated for 2 d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNonstructural protein 5A(Hepatitis C virus)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50522234(CHEMBL4517067)
Affinity DataEC50:  52nMAssay Description:Inhibition of NS5A in HCV genotype 1b infected in human HuH7 replicon cells assessed as reduction in subgenomic viral RNA replication treated for 2 d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNonstructural protein 5A(Hepatitis C virus)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50522235(CHEMBL4445786)
Affinity DataEC50:  7.60nMAssay Description:Inhibition of NS5A in HCV genotype 1b infected in human HuH7 replicon cells assessed as reduction in subgenomic viral RNA replication treated for 2 d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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