Affinity DataKi: 27nMAssay Description:Binding affinity against human opioid receptor like 1 (hORL) was determined using [leucyl-3H]nociceptin in vitro in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 45nMAssay Description:Binding affinity against human opioid receptor like 1 (hORL) was determined using [leucyl-3H]nociceptin in vitro in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 72nMAssay Description:Binding affinity against human opioid receptor like 1 (hORL) was determined using [leucyl-3H]nociceptin in vitro in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 78nMAssay Description:Binding affinity against human Opioid receptor kappa 1 (hKOR) was determined using [3H]diprenorphine in vitro in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 78nMAssay Description:Binding affinity against human opioid receptor like 1 (hORL) was determined using [leucyl-3H]nociceptin in vitro in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 78nMAssay Description:Binding affinity against human Opioid receptor mu 1 (hMOR) was determined using [3H]diprenorphine in vitro transfected to COS-1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 85nMAssay Description:Binding affinity against human Opioid receptor mu 1 (hMOR) was determined using [3H]diprenorphine in vitro transfected to COS-1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 90nMAssay Description:Binding affinity against human Opioid receptor mu 1 (hMOR) was determined using [3H]diprenorphine in vitro transfected to COS-1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 105nMAssay Description:Binding affinity against human Opioid receptor kappa 1 (hKOR) was determined using [3H]diprenorphine in vitro in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 153nMAssay Description:Binding affinity against human Opioid receptor kappa 1 (hKOR) was determined using [3H]diprenorphine in vitro in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 222nMAssay Description:Binding affinity against human opioid receptor delta 1 was determined using [3H]diprenorphine in vitro transfected to COS-1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 779nMAssay Description:Binding affinity against human Opioid receptor kappa 1 (hKOR) was determined using [3H]diprenorphine in vitro in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 833nMAssay Description:Binding affinity against human Opioid receptor mu 1 (hMOR) was determined using [3H]diprenorphine in vitro transfected to COS-1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.56E+3nMAssay Description:Binding affinity against human Opioid receptor mu 1 (hMOR) was determined using [3H]diprenorphine in vitro transfected to COS-1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.27E+3nMAssay Description:Binding affinity against human Opioid receptor kappa 1 (hKOR) was determined using [3H]diprenorphine in vitro in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: >5.00E+3nMAssay Description:Binding affinity against human opioid receptor like 1 (hORL) was determined using [leucyl-3H]nociceptin in vitro in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: >5.00E+3nMAssay Description:Binding affinity against human Opioid receptor kappa 1 (hKOR) was determined using [3H]diprenorphine in vitro in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: >5.00E+3nMAssay Description:Binding affinity against human Opioid receptor mu 1 (hMOR) was determined using [3H]diprenorphine in vitro transfected to COS-1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: >5.00E+3nMAssay Description:Binding affinity against human opioid receptor like 1 (hORL) was determined using [leucyl-3H]nociceptin in vitro in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: >5.00E+3nMAssay Description:Binding affinity against human Opioid receptor mu 1 (hMOR) was determined using [3H]diprenorphine in vitro transfected to COS-1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: >5.00E+3nMAssay Description:Binding affinity against human Opioid receptor mu 1 (hMOR) was determined using [3H]diprenorphine in vitro transfected to COS-1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: >5.00E+3nMAssay Description:Binding affinity against human Opioid receptor kappa 1 (hKOR) was determined using [3H]diprenorphine in vitro in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: >5.00E+3nMAssay Description:Binding affinity against human opioid receptor like 1 (hORL) was determined using [leucyl-3H]nociceptin in vitro in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: >5.00E+3nMAssay Description:Binding affinity against human opioid receptor like 1 (hORL) was determined using [leucyl-3H]nociceptin in vitro in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: >5.00E+3nMAssay Description:Binding affinity against human opioid receptor delta 1 was determined using [3H]diprenorphine in vitro transfected to COS-1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: >5.00E+3nMAssay Description:Binding affinity against human opioid receptor delta 1 was determined using [3H]diprenorphine in vitro transfected to COS-1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: >5.00E+3nMAssay Description:Binding affinity against human opioid receptor delta 1 was determined using [3H]diprenorphine in vitro transfected to COS-1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: >5.00E+3nMAssay Description:Binding affinity against human opioid receptor delta 1 was determined using [3H]diprenorphine in vitro transfected to COS-1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: >5.00E+3nMAssay Description:Binding affinity against human opioid receptor delta 1 was determined using [3H]diprenorphine in vitro transfected to COS-1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: >5.00E+3nMAssay Description:Binding affinity against human Opioid receptor kappa 1 (hKOR) was determined using [3H]diprenorphine in vitro in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: >5.00E+3nMAssay Description:Binding affinity against human opioid receptor delta 1 was determined using [3H]diprenorphine in vitro transfected to COS-1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: >5.00E+3nMAssay Description:Binding affinity against human opioid receptor delta 1 was determined using [3H]diprenorphine in vitro transfected to COS-1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of [125I]SDF1 binding to CXCR4 transfected in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibition of [125I]SDF1 binding to CXCR4 transfected in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Inhibition of [125I]SDF1 binding to CXCR4 transfected in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Inhibition of [125I]SDF1 binding to CXCR4 transfected in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Inhibition of [125I]SDF1 binding to CXCR4 transfected in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 21nMAssay Description:Inhibition of [125I]SDF1 binding to CXCR4 transfected in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:Inhibition of [125I]SDF1 binding to CXCR4 transfected in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 47nMAssay Description:Inhibition of [125I]SDF1 binding to CXCR4 transfected in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 63nMAssay Description:Inhibition of [125I]SDF1 binding to CXCR4 transfected in CHO cellsMore data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
Université
Curated by ChEMBL
Université
Curated by ChEMBL
Affinity DataIC50: 68nMAssay Description:Antagonist activity against human CGRP1 expressed in HEK293 cells assessed as inhibition of human alpha-CGRP-promoted cAMP productionMore data for this Ligand-Target Pair
Affinity DataIC50: 92nMAssay Description:Inhibition of [125I]SDF1 binding to CXCR4 transfected in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 99nMAssay Description:Inhibition of [125I]SDF1 binding to CXCR4 transfected in CHO cellsMore data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
Université
Curated by ChEMBL
Université
Curated by ChEMBL
Affinity DataIC50: 107nMAssay Description:Antagonist activity against human CGRP1 expressed in HEK293 cells assessed as inhibition of human alpha-CGRP-promoted cAMP productionMore data for this Ligand-Target Pair
Affinity DataIC50: 128nMAssay Description:Inhibition of [125I]SDF1 binding to CXCR4 transfected in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:Inhibition of [125I]SDF1 binding to CXCR4 transfected in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 157nMAssay Description:Inhibition of [125I]SDF1 binding to CXCR4 transfected in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 167nMAssay Description:Inhibition of [125I]SDF1 binding to CXCR4 transfected in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 170nMAssay Description:Inhibition of [125I]SDF1 binding to CXCR4 transfected in CHO cellsMore data for this Ligand-Target Pair