TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Technical University Dortmund
Curated by ChEMBL
Technical University Dortmund
Curated by ChEMBL
Affinity DataIC50: 110nMAssay Description:Inhibition of PI3Kgamma (unknown origin)More data for this Ligand-Target Pair
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Technical University Dortmund
Curated by ChEMBL
Technical University Dortmund
Curated by ChEMBL
Affinity DataIC50: 120nMAssay Description:Inhibition of CK1delta (unknown origin)More data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Technical University Dortmund
Curated by ChEMBL
Technical University Dortmund
Curated by ChEMBL
Affinity DataIC50: 140nMAssay Description:Inhibition of DNA-PK (unknown origin)More data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Technical University Dortmund
Curated by ChEMBL
Technical University Dortmund
Curated by ChEMBL
Affinity DataIC50: 220nMAssay Description:Inhibition of CK1alpha (unknown origin)More data for this Ligand-Target Pair
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Technical University Dortmund
Curated by ChEMBL
Technical University Dortmund
Curated by ChEMBL
Affinity DataIC50: 240nMAssay Description:Inhibition of CK1delta (unknown origin)More data for this Ligand-Target Pair
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Technical University Dortmund
Curated by ChEMBL
Technical University Dortmund
Curated by ChEMBL
Affinity DataIC50: 380nMAssay Description:Inhibition of CK1epsilon (unknown origin)More data for this Ligand-Target Pair
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Technical University Dortmund
Curated by ChEMBL
Technical University Dortmund
Curated by ChEMBL
Affinity DataIC50: 430nMAssay Description:Inhibition of CK1delta (unknown origin)More data for this Ligand-Target Pair
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Technical University Dortmund
Curated by ChEMBL
Technical University Dortmund
Curated by ChEMBL
Affinity DataIC50: 490nMAssay Description:Inhibition of CK1epsilon (unknown origin)More data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Technical University Dortmund
Curated by ChEMBL
Technical University Dortmund
Curated by ChEMBL
Affinity DataIC50: 820nMAssay Description:Inhibition of CK1alpha (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Technical University Dortmund
Curated by ChEMBL
Technical University Dortmund
Curated by ChEMBL
Affinity DataIC50: 970nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Technical University Dortmund
Curated by ChEMBL
Technical University Dortmund
Curated by ChEMBL
Affinity DataIC50: 1.28E+3nMAssay Description:Inhibition of PI3Kalpha (unknown origin)More data for this Ligand-Target Pair
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Technical University Dortmund
Curated by ChEMBL
Technical University Dortmund
Curated by ChEMBL
Affinity DataIC50: 2.07E+3nMAssay Description:Inhibition of CK1epsilon (unknown origin)More data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Technical University Dortmund
Curated by ChEMBL
Technical University Dortmund
Curated by ChEMBL
Affinity DataIC50: 2.92E+3nMAssay Description:Inhibition of CK1alpha (unknown origin)More data for this Ligand-Target Pair
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Technical University Dortmund
Curated by ChEMBL
Technical University Dortmund
Curated by ChEMBL
Affinity DataIC50: 3.64E+3nMAssay Description:Inhibition of CK1delta (unknown origin)More data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Technical University Dortmund
Curated by ChEMBL
Technical University Dortmund
Curated by ChEMBL
Affinity DataIC50: 6.18E+3nMAssay Description:Inhibition of CK1alpha (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Technical University Dortmund
Curated by ChEMBL
Technical University Dortmund
Curated by ChEMBL
Affinity DataIC50: 8.48E+3nMAssay Description:Inhibition of PI3Kbeta (unknown origin)More data for this Ligand-Target Pair
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Technical University Dortmund
Curated by ChEMBL
Technical University Dortmund
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CK1epsilon (unknown origin)More data for this Ligand-Target Pair
TargetAryl hydrocarbon receptor(Mus musculus (Mouse))
Max Planck Institute Of Molecular Physiology
Curated by ChEMBL
Max Planck Institute Of Molecular Physiology
Curated by ChEMBL
Affinity DataEC50: 71nMAssay Description:Activation of AhR in mouse Hepa1c1c7 cells assessed as induction of XRE-dependent reporter activity incubated for 4 hrs by Renilla/Firefly based dual...More data for this Ligand-Target Pair
TargetAryl hydrocarbon receptor(Homo sapiens (Human))
Max Planck Institute Of Molecular Physiology
Curated by ChEMBL
Max Planck Institute Of Molecular Physiology
Curated by ChEMBL
Affinity DataEC50: 3.20nMAssay Description:Activation of AhR in human HepG2 cells assessed as induction of XRE-dependent reporter activity incubated for 4 hrs by Renilla/Firefly based dual-luc...More data for this Ligand-Target Pair
TargetAryl hydrocarbon receptor(Mus musculus (Mouse))
Max Planck Institute Of Molecular Physiology
Curated by ChEMBL
Max Planck Institute Of Molecular Physiology
Curated by ChEMBL
Affinity DataEC50: 0.0580nMAssay Description:Activation of AhR in mouse NIH3T3 cells assessed as induction of XRE-dependent reporter activity incubated for 4 hrs by Renilla/Firefly based dual-lu...More data for this Ligand-Target Pair
TargetAryl hydrocarbon receptor(Homo sapiens (Human))
Max Planck Institute Of Molecular Physiology
Curated by ChEMBL
Max Planck Institute Of Molecular Physiology
Curated by ChEMBL
Affinity DataEC50: 0.700nMAssay Description:Activation of AhR in human HaCaT cells assessed as induction of XRE-dependent reporter activity incubated for 4 hrs by Renilla/Firefly based dual-luc...More data for this Ligand-Target Pair