Compile Data Set for Download or QSAR
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Found 19 with Last Name = 'hiratake' and Initial = 'j'
TargetAsparagine synthetase [glutamine-hydrolyzing](Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50378579(CHEMBL1627258)
Affinity DataKi:  2.5nMAssay Description:Inhibition of human recombinant ASNS expressed in Sf9 cells assessed as assessed as overall inhibition constant for ammonia dependent production of i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAsparagine synthetase [glutamine-hydrolyzing](Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50392270(CHEMBL2153507)
Affinity DataKi:  8nMAssay Description:Inhibition of human recombinant ASNS expressed in Sf9 cells assessed as overall inhibition constant for glutamine dependent production of inorganic p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAsparagine synthetase [glutamine-hydrolyzing](Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50378579(CHEMBL1627258)
Affinity DataKi:  24nMAssay Description:Inhibition of human recombinant ASNS expressed in Sf9 cells assessed as overall inhibition constant for glutamine dependent production of inorganic p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAsparagine synthetase [glutamine-hydrolyzing](Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50392270(CHEMBL2153507)
Affinity DataKi:  33nMAssay Description:Inhibition of human recombinant ASNS expressed in Sf9 cells assessed as assessed as overall inhibition constant for ammonia dependent production of i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAsparagine synthetase [glutamine-hydrolyzing](Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50378579(CHEMBL1627258)
Affinity DataKi:  280nMAssay Description:Inhibition of human recombinant ASNS expressed in Sf9 cells assessed as assessed as initial inhibition constant for ammonia dependent production of i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAsparagine synthetase [glutamine-hydrolyzing](Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50392271(CHEMBL2153508)
Affinity DataKi:  310nMAssay Description:Inhibition of human recombinant ASNS expressed in Sf9 cells assessed as assessed as overall inhibition constant for ammonia dependent production of i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate--cysteine ligase catalytic subunit(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50366432(CHEMBL1627263)
Affinity DataKi:  390nMAssay Description:Tested for inhibition of Escherichia coli gamma-glutamylcysteine synthetase at a concentration of 5.1 uMMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAsparagine synthetase [glutamine-hydrolyzing](Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50392270(CHEMBL2153507)
Affinity DataKi:  450nMAssay Description:Inhibition of human recombinant ASNS expressed in Sf9 cells assessed as assessed as initial inhibition constant for ammonia dependent production of i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAsparagine synthetase [glutamine-hydrolyzing](Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50392270(CHEMBL2153507)
Affinity DataKi:  490nMAssay Description:Inhibition of human recombinant ASNS expressed in Sf9 cells assessed as initial inhibition constant for glutamine dependent production of inorganic p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAsparagine synthetase [glutamine-hydrolyzing](Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50392271(CHEMBL2153508)
Affinity DataKi:  840nMAssay Description:Inhibition of human recombinant ASNS expressed in Sf9 cells assessed as overall inhibition constant for glutamine dependent production of inorganic p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAsparagine synthetase [glutamine-hydrolyzing](Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50378579(CHEMBL1627258)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of human recombinant ASNS expressed in Sf9 cells assessed as initial inhibition constant for glutamine dependent production of inorganic p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAsparagine synthetase [glutamine-hydrolyzing](Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50392271(CHEMBL2153508)
Affinity DataKi:  3.04E+3nMAssay Description:Inhibition of human recombinant ASNS expressed in Sf9 cells assessed as assessed as initial inhibition constant for ammonia dependent production of i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAsparagine synthetase [glutamine-hydrolyzing](Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50392271(CHEMBL2153508)
Affinity DataKi:  4.50E+3nMAssay Description:Inhibition of human recombinant ASNS expressed in Sf9 cells assessed as initial inhibition constant for glutamine dependent production of inorganic p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate--cysteine ligase catalytic subunit(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287274((2S)-2-ammonio-4-[(2-carboxylatobutyl)phosphinato]...)
Affinity DataKi:  4.95E+3nMAssay Description:Tested for inhibition of Escherichia coli gamma-glutamylcysteine synthetase at a concentration of 5.7 uMMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGlutamate--cysteine ligase catalytic subunit(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287275(2-ammonio-4-[(2-carboxylatobutyl)sulfonyl]butanoat...)
Affinity DataKi:  9.23E+3nMAssay Description:Tested for inhibition of Escherichia coli gamma-glutamylcysteine synthetase at a concentration of 16.3 uMMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAsparagine synthetase [glutamine-hydrolyzing](Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50378579(CHEMBL1627258)
Affinity DataKi:  1.00E+4nMAssay Description:Inhibition of human recombinant ASNS expressed in Sf9 insect cells assessed as overall inhibition constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAsparagine synthetase [glutamine-hydrolyzing](Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50378579(CHEMBL1627258)
Affinity DataKi:  2.00E+4nMAssay Description:Inhibition of human recombinant ASNS expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate--cysteine ligase catalytic subunit(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50366433(CHEMBL1609891)
Affinity DataKi:  4.93E+4nMAssay Description:Tested for inhibition of Escherichia coli gamma-glutamylcysteine synthetase at a concentration of 25.0 uMMore data for this Ligand-Target Pair
In DepthDetails Article
TargetExo-1,4-beta-xylosidase xlnD(Aspergillus niger)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50096896(2-phenyl-1-{[3,4,5-trihydroxy-6-(hydroxymethyl)tet...)
Affinity DataKi:  1.00E+6nMAssay Description:Compound was evaluated for the selective and competitive inhibition of Beta-xylosidase from A. pulverulentusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed