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Found 27 with Last Name = 'molette' and Initial = 'j'
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50151865(CHEMBL172 | MEFLOQUINE)
Affinity DataKi:  1.90E+3nMAssay Description:Inhibition of human ERG expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM79214(1-[1,3-bis(chloranyl)-6-(trifluoromethyl)phenanthr...)
Affinity DataKi:  7.50E+3nMAssay Description:Inhibition of human ERG expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM22985(Aralen | CHEMBL76 | CHLOROQUINE PHOSPHATE | Chloro...)
Affinity DataKi:  7.50E+3nMAssay Description:Inhibition of human ERG expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Ac Immune

Curated by ChEMBL
LigandPNGBDBM50586984(CHEMBL5084771)
Affinity DataIC50:  3.10nMAssay Description:Displacement of [3H]PI-2620 from Tau in human brain homogenate incubated for 60 mins by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Ac Immune

Curated by ChEMBL
LigandPNGBDBM50586985(CHEMBL5082735)
Affinity DataIC50:  3.5nMAssay Description:Displacement of [3H]PI-2620 from Tau in human brain homogenate incubated for 60 mins by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Ac Immune

Curated by ChEMBL
LigandPNGBDBM50586972(CHEMBL5088921)
Affinity DataIC50:  4.90nMAssay Description:Displacement of [3H]PI-2620 from Tau in human brain homogenate incubated for 60 mins by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Mus musculus)
Ac Immune

Curated by ChEMBL
LigandPNGBDBM50586985(CHEMBL5082735)
Affinity DataIC50:  7.80nMAssay Description:Displacement of [18F]-FEH from MAO-A in mouse brain homogenate incubated for 60 mins by imaging analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Ac Immune

Curated by ChEMBL
LigandPNGBDBM50586975(CHEMBL5081662)
Affinity DataIC50:  16nMAssay Description:Displacement of [3H]PI-2620 from Tau in human brain homogenate incubated for 60 mins by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Ac Immune

Curated by ChEMBL
LigandPNGBDBM50586986(CHEMBL5091624)
Affinity DataIC50:  18nMAssay Description:Displacement of [3H]PI-2620 from Tau in human brain homogenate incubated for 60 mins by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Ac Immune

Curated by ChEMBL
LigandPNGBDBM50586979(CHEMBL5084917)
Affinity DataIC50:  36nMAssay Description:Displacement of [3H]PI-2620 from Tau in human brain homogenate incubated for 60 mins by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Mus musculus)
Ac Immune

Curated by ChEMBL
LigandPNGBDBM50586984(CHEMBL5084771)
Affinity DataIC50:  51nMAssay Description:Displacement of [18F]-FEH from MAO-A in mouse brain homogenate incubated for 60 mins by imaging analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Ac Immune

Curated by ChEMBL
LigandPNGBDBM50586982(CHEMBL5083649)
Affinity DataIC50:  70nMAssay Description:Displacement of [3H]PI-2620 from Tau in human brain homogenate incubated for 60 mins by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Ac Immune

Curated by ChEMBL
LigandPNGBDBM50586973(CHEMBL5077904)
Affinity DataIC50:  82nMAssay Description:Displacement of [3H]PI-2620 from Tau in human brain homogenate incubated for 60 mins by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Ac Immune

Curated by ChEMBL
LigandPNGBDBM50586974(CHEMBL5090407)
Affinity DataIC50:  116nMAssay Description:Displacement of [3H]PI-2620 from Tau in human brain homogenate incubated for 60 mins by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Ac Immune

Curated by ChEMBL
LigandPNGBDBM50586978(CHEMBL5080178)
Affinity DataIC50:  260nMAssay Description:Displacement of [3H]PI-2620 from Tau in human brain homogenate incubated for 60 mins by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Ac Immune

Curated by ChEMBL
LigandPNGBDBM50586980(CHEMBL5081126)
Affinity DataIC50:  310nMAssay Description:Displacement of [3H]PI-2620 from Tau in human brain homogenate incubated for 60 mins by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Ac Immune

Curated by ChEMBL
LigandPNGBDBM50586977(CHEMBL5081957)
Affinity DataIC50:  344nMAssay Description:Displacement of [3H]PI-2620 from Tau in human brain homogenate incubated for 60 mins by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Ac Immune

Curated by ChEMBL
LigandPNGBDBM50586981(CHEMBL5094590)
Affinity DataIC50:  559nMAssay Description:Displacement of [3H]PI-2620 from Tau in human brain homogenate incubated for 60 mins by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Ac Immune

Curated by ChEMBL
LigandPNGBDBM50586976(CHEMBL5092563)
Affinity DataIC50:  732nMAssay Description:Displacement of [3H]PI-2620 from Tau in human brain homogenate incubated for 60 mins by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Mus musculus)
Ac Immune

Curated by ChEMBL
LigandPNGBDBM50586974(CHEMBL5090407)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [18F]-FEH from MAO-A in mouse brain homogenate incubated for 60 mins by imaging analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Mus musculus)
Ac Immune

Curated by ChEMBL
LigandPNGBDBM50586975(CHEMBL5081662)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [18F]-FEH from MAO-A in mouse brain homogenate incubated for 60 mins by imaging analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Mus musculus)
Ac Immune

Curated by ChEMBL
LigandPNGBDBM50586976(CHEMBL5092563)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [18F]-FEH from MAO-A in mouse brain homogenate incubated for 60 mins by imaging analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Mus musculus)
Ac Immune

Curated by ChEMBL
LigandPNGBDBM50586977(CHEMBL5081957)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [18F]-FEH from MAO-A in mouse brain homogenate incubated for 60 mins by imaging analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Mus musculus)
Ac Immune

Curated by ChEMBL
LigandPNGBDBM50586972(CHEMBL5088921)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [18F]-FEH from MAO-A in mouse brain homogenate incubated for 60 mins by imaging analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Mus musculus)
Ac Immune

Curated by ChEMBL
LigandPNGBDBM50586986(CHEMBL5091624)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [18F]-FEH from MAO-A in mouse brain homogenate incubated for 60 mins by imaging analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Ac Immune

Curated by ChEMBL
LigandPNGBDBM50586983(CHEMBL5091757)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [3H]PI-2620 from Tau in human brain homogenate incubated for 60 mins by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Mus musculus)
Ac Immune

Curated by ChEMBL
LigandPNGBDBM50586973(CHEMBL5077904)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [18F]-FEH from MAO-A in mouse brain homogenate incubated for 60 mins by imaging analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed