Compile Data Set for Download or QSAR
maximum 50k data
Found 30 with Last Name = 'navratil' and Initial = 'j'
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
Institute of Experimental Botany Ascr and Palacky University

LigandPNGBDBM123786(AAP1742)
Affinity DataIC50:  280nMAssay Description:Cyclin-dependent kinase selectivity was evaluated using CDK1-cyclin B, CDK2-cyclin E, CDK4-cyclin D1, CDK7-cyclin H, and CDK9-cyclin T1.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
Institute of Experimental Botany Ascr and Palacky University

LigandPNGBDBM12028(4-Arylazo-3,5-diamino-1H-pyrazole 31b | 4-[(E)-2-(...)
Affinity DataIC50:  350nMAssay Description:Cyclin-dependent kinase selectivity was evaluated using CDK1-cyclin B, CDK2-cyclin E, CDK4-cyclin D1, CDK7-cyclin H, and CDK9-cyclin T1.More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
Institute of Experimental Botany Ascr and Palacky University

LigandPNGBDBM123786(AAP1742)
Affinity DataIC50:  454nMAssay Description:Cyclin-dependent kinase selectivity was evaluated using CDK1-cyclin B, CDK2-cyclin E, CDK4-cyclin D1, CDK7-cyclin H, and CDK9-cyclin T1.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Institute of Experimental Botany Ascr and Palacky University

LigandPNGBDBM123786(AAP1742)
Affinity DataIC50:  549nMAssay Description:Cyclin-dependent kinase selectivity was evaluated using CDK1-cyclin B, CDK2-cyclin E, CDK4-cyclin D1, CDK7-cyclin H, and CDK9-cyclin T1.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Institute of Experimental Botany Ascr and Palacky University

LigandPNGBDBM123786(AAP1742)
Affinity DataIC50:  1.33E+3nMAssay Description:Cyclin-dependent kinase selectivity was evaluated using CDK1-cyclin B, CDK2-cyclin E, CDK4-cyclin D1, CDK7-cyclin H, and CDK9-cyclin T1.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50353649(CHEMBL1829835)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of PKCzeta in human U937 cells assessed as inhibition of TNFalpha-induced NF-kB activation by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50353651(CHEMBL1829841)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of PKCzeta in human U937 cells assessed as inhibition of TNFalpha-induced NF-kB activation by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
Institute of Experimental Botany Ascr and Palacky University

LigandPNGBDBM12028(4-Arylazo-3,5-diamino-1H-pyrazole 31b | 4-[(E)-2-(...)
Affinity DataIC50:  1.35E+4nMAssay Description:Cyclin-dependent kinase selectivity was evaluated using CDK1-cyclin B, CDK2-cyclin E, CDK4-cyclin D1, CDK7-cyclin H, and CDK9-cyclin T1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50353652(CHEMBL1829842)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibition of PKCzeta in human U937 cells assessed as inhibition of TNFalpha-induced NF-kB activation by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50353647(CHEMBL1829832)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibition of PKCzeta in human U937 cells assessed as inhibition of TNFalpha-induced NF-kB activation by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Institute of Experimental Botany Ascr and Palacky University

LigandPNGBDBM123786(AAP1742)
Affinity DataIC50:  1.49E+4nMAssay Description:Cyclin-dependent kinase selectivity was evaluated using CDK1-cyclin B, CDK2-cyclin E, CDK4-cyclin D1, CDK7-cyclin H, and CDK9-cyclin T1.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50353653(CHEMBL1829843)
Affinity DataIC50:  1.70E+4nMAssay Description:Inhibition of PKCzeta in human U937 cells assessed as inhibition of TNFalpha-induced NF-kB activation by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50353649(CHEMBL1829835)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibition of human PKCzeta assessed as [gamma32P]ATP utilization using myelin basic protein as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Institute of Experimental Botany Ascr and Palacky University

LigandPNGBDBM12028(4-Arylazo-3,5-diamino-1H-pyrazole 31b | 4-[(E)-2-(...)
Affinity DataIC50:  2.00E+4nMAssay Description:Cyclin-dependent kinase selectivity was evaluated using CDK1-cyclin B, CDK2-cyclin E, CDK4-cyclin D1, CDK7-cyclin H, and CDK9-cyclin T1.More data for this Ligand-Target Pair
TargetProtein kinase C zeta type(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50353653(CHEMBL1829843)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of human PKCzeta assessed as [gamma32P]ATP utilization using myelin basic protein as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50353651(CHEMBL1829841)
Affinity DataIC50:  2.30E+4nMAssay Description:Inhibition of human PKCzeta assessed as [gamma32P]ATP utilization using myelin basic protein as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50353653(CHEMBL1829843)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of human PKCzeta assessed as [gamma32P]ATP utilization using myelin basic protein as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50353653(CHEMBL1829843)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of human PKCzeta assessed as [gamma32P]ATP utilization using myelin basic protein as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Institute of Experimental Botany Ascr and Palacky University

LigandPNGBDBM12028(4-Arylazo-3,5-diamino-1H-pyrazole 31b | 4-[(E)-2-(...)
Affinity DataIC50:  2.60E+4nMAssay Description:Cyclin-dependent kinase selectivity was evaluated using CDK1-cyclin B, CDK2-cyclin E, CDK4-cyclin D1, CDK7-cyclin H, and CDK9-cyclin T1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50353650(CHEMBL1829837)
Affinity DataIC50:  2.80E+4nMAssay Description:Inhibition of PKCzeta in human U937 cells assessed as inhibition of TNFalpha-induced NF-kB activation by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50353648(CHEMBL1829833)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibition of PKCzeta in human U937 cells assessed as inhibition of TNFalpha-induced NF-kB activation by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50353655(CHEMBL1829834)
Affinity DataIC50:  3.20E+4nMAssay Description:Inhibition of PKCzeta in human U937 cells assessed as inhibition of TNFalpha-induced NF-kB activation by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50353654(CHEMBL1829822)
Affinity DataIC50:  3.30E+4nMAssay Description:Inhibition of human PKCzeta assessed as [gamma32P]ATP utilization using myelin basic protein as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50353652(CHEMBL1829842)
Affinity DataIC50:  3.30E+4nMAssay Description:Inhibition of human PKCzeta assessed as [gamma32P]ATP utilization using myelin basic protein as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50353647(CHEMBL1829832)
Affinity DataIC50:  3.80E+4nMAssay Description:Inhibition of human PKCzeta assessed as [gamma32P]ATP utilization using myelin basic protein as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50353654(CHEMBL1829822)
Affinity DataIC50:  3.80E+4nMAssay Description:Inhibition of PKCzeta in human U937 cells assessed as inhibition of TNFalpha-induced NF-kB activation by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50353655(CHEMBL1829834)
Affinity DataIC50:  3.90E+4nMAssay Description:Inhibition of human PKCzeta assessed as [gamma32P]ATP utilization using myelin basic protein as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50353650(CHEMBL1829837)
Affinity DataIC50:  4.30E+4nMAssay Description:Inhibition of human PKCzeta assessed as [gamma32P]ATP utilization using myelin basic protein as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Institute of Experimental Botany Ascr and Palacky University

LigandPNGBDBM12028(4-Arylazo-3,5-diamino-1H-pyrazole 31b | 4-[(E)-2-(...)
Affinity DataIC50:  4.40E+4nMAssay Description:Cyclin-dependent kinase selectivity was evaluated using CDK1-cyclin B, CDK2-cyclin E, CDK4-cyclin D1, CDK7-cyclin H, and CDK9-cyclin T1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50353648(CHEMBL1829833)
Affinity DataIC50:  5.50E+4nMAssay Description:Inhibition of human PKCzeta assessed as [gamma32P]ATP utilization using myelin basic protein as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed