Affinity DataKi: 0.130nMAssay Description:Displacement of [3H]des-Arg10 Leu9 kallidin from human bradykinin B1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Binding affinity to human bradykinin B1 receptor expressed in rat CNSMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Binding affinity to human bradykinin B1 receptor expressed in rat CNSMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataKi: 0.240nMAssay Description:Compound was evaluated in vitro for the inhibition of HIV-Protease, using a peptide hydrolysis assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Binding affinity to human bradykinin B1 receptor expressed in rat CNSMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Binding affinity to human bradykinin B1 receptor expressed in rat CNSMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Displacement of [3H]des-Arg10 Leu9 kallidin from human bradykinin B1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Displacement of [3H]des-arg10, leu9-kallidin from human bradykinin B1 receptor expresed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Binding affinity to human bradykinin B1 receptor expressed in rat CNSMore data for this Ligand-Target Pair
Affinity DataKi: 0.440nMAssay Description:Displacement of [3H]des-Arg10 Leu9 kallidin from human bradykinin B1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Binding affinity to human bradykinin B1 receptor expressed in rat CNSMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Displacement of [3H]des-arg10, leu9-kallidin from human bradykinin B1 receptor expresed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Displacement of [3H]des-arg10, leu9-kallidin from human bradykinin B1 receptor expresed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.510nMAssay Description:Displacement of [3H]des-Arg10 Leu9 kallidin from human bradykinin B1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.540nMAssay Description:Displacement of [3H]des-Arg10 Leu9 kallidin from human bradykinin B1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.570nMAssay Description:Displacement of [3H]des-Arg10 Leu9 kallidin from human bradykinin B1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Displacement of [3H]des-Arg10 Leu9 kallidin from human bradykinin B1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Binding affinity to human bradykinin B1 receptor expressed in rat CNSMore data for this Ligand-Target Pair
Affinity DataKi: 0.660nMAssay Description:Displacement of [3H]des-Arg10 Leu9 kallidin from human bradykinin B1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.690nMAssay Description:Binding affinity to rabbit bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Displacement of [3H]des-arg10, leu9-kallidin from human bradykinin B1 receptor expresed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Displacement of [3H]des-arg10, leu9-kallidin from human bradykinin B1 receptor expresed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Displacement of [3H]des-arg10, leu9-kallidin from human bradykinin B1 receptor expresed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.810nMAssay Description:Displacement of [3H]des-Arg10 Leu9 kallidin from human bradykinin B1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.810nMAssay Description:Displacement of [3H]des-Arg10 Leu9 kallidin from human bradykinin B1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Binding affinity to human bradykinin B1 receptor expressed in rat CNSMore data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Binding affinity to human bradykinin B1 receptor expressed in rat CNSMore data for this Ligand-Target Pair
Affinity DataKi: 0.930nMAssay Description:Displacement of [3H]des-Arg10 Leu9 kallidin from human bradykinin B1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Displacement of [3H]des-arg10, leu9-kallidin from human bradykinin B1 receptor expresed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Binding affinity to human bradykinin B1 receptor expressed in rat CNSMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Binding affinity to rabbit bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]des-arg10, leu9-kallidin from human bradykinin B1 receptor expresed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Binding affinity to human bradykinin B1 receptor expressed in rat CNSMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Binding affinity to human bradykinin B1 receptor expressed in rat CNSMore data for this Ligand-Target Pair
Affinity DataKi: 1.35nMAssay Description:Displacement of [3H]des-Arg10 Leu9 kallidin from human bradykinin B1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Binding affinity to human bradykinin B1 receptor expressed in rat CNSMore data for this Ligand-Target Pair
Affinity DataKi: 1.44nMAssay Description:Displacement of [3H]des-Arg10 Leu9 kallidin from human bradykinin B1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.47nMAssay Description:Displacement of [3H]des-Arg10 Leu9 kallidin from human bradykinin B1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Binding affinity to human bradykinin B1 receptor expressed in rat CNSMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Binding affinity to human bradykinin B1 receptor expressed in rat CNSMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Displacement of [3H]des-Arg10 Leu9 kallidin from human bradykinin B1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Displacement of [3H]des-Arg10 Leu9 kallidin from human bradykinin B1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Binding affinity to human bradykinin B1 receptor expressed in rat CNSMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Inhibitory constant against human Bradykinin receptor B1 expressed in chinese hamster ovary cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Binding affinity to human bradykinin B1 receptor expressed in rat CNSMore data for this Ligand-Target Pair
Affinity DataKi: 1.95nMAssay Description:Displacement of [3H]des-Arg10 Leu9 kallidin from human bradykinin B1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Binding affinity to rhesus monkey bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Displacement of [3H]des-arg10, leu9-kallidin from human bradykinin B1 receptor expresed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.30nMAssay Description:Binding affinity to human bradykinin B1 receptor expressed in rat CNSMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Displacement of [3H]des-Arg10 Leu9 kallidin from human bradykinin B1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair