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Found 37 with Last Name = 'gopal' and Initial = 'k'
TargetForkhead box protein M1(Homo sapiens)
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50562257(CHEMBL4740210)
Affinity DataKi:  21nMAssay Description:Binding affinity to recombinant FOXM1 DBD (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as disruption of FOXM1-DNA complex prein...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetForkhead box protein M1(Homo sapiens)
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50085045(5-((4-((6-hydroxy-2,5,7,8-tetramethyl-3,4-dihydro-...)
Affinity DataKi:  52nMAssay Description:Binding affinity to recombinant FOXM1 DBD (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as disruption of FOXM1-DNA complex prein...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Maharishi Markandeshwar (Deemed To Be University)

Curated by ChEMBL
LigandPNGBDBM50481218(CHEMBL390983 | DX-619)
Affinity DataKi:  6.79E+4nMAssay Description:Inhibition of CYP3A4 in human liver microsomes using midazolam as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPancreatic triacylglycerol lipase(Homo sapiens (Human))
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)

Curated by ChEMBL
LigandPNGBDBM24567((2S)-1-[(2S,3S)-3-hexyl-4-oxooxetan-2-yl]tridecan-...)
Affinity DataIC50:  190nMAssay Description:Inhibition of human pancreatic lipase using emulsified olive oil as substrate pretreated with substrate for 5 mins followed by enzyme addition and me...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)

Curated by ChEMBL
LigandPNGBDBM50367145(CHEMBL4173252)
Affinity DataIC50:  750nMAssay Description:Inhibition of porcine pancreatic lipase using p-nitrophenyl butyrate as substrate pretreated for 15 mins followed by substrate addition and measured ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)

Curated by ChEMBL
LigandPNGBDBM50367138(CHEMBL4160519)
Affinity DataIC50:  770nMAssay Description:Inhibition of porcine pancreatic lipase using p-nitrophenyl butyrate as substrate pretreated for 15 mins followed by substrate addition and measured ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)

Curated by ChEMBL
LigandPNGBDBM24567((2S)-1-[(2S,3S)-3-hexyl-4-oxooxetan-2-yl]tridecan-...)
Affinity DataIC50:  800nMAssay Description:Inhibition of porcine pancreatic lipase using p-nitrophenyl butyrate as substrate pretreated for 15 mins followed by substrate addition and measured ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)

Curated by ChEMBL
LigandPNGBDBM50367133(CHEMBL4164998)
Affinity DataIC50:  800nMAssay Description:Inhibition of porcine pancreatic lipase using p-nitrophenyl butyrate as substrate pretreated for 15 mins followed by substrate addition and measured ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)

Curated by ChEMBL
LigandPNGBDBM50367134(CHEMBL4167341)
Affinity DataIC50:  840nMAssay Description:Inhibition of porcine pancreatic lipase using p-nitrophenyl butyrate as substrate pretreated for 15 mins followed by substrate addition and measured ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)

Curated by ChEMBL
LigandPNGBDBM50367211(CHEMBL4165339)
Affinity DataIC50:  850nMAssay Description:Inhibition of porcine pancreatic lipase using p-nitrophenyl butyrate as substrate pretreated for 15 mins followed by substrate addition and measured ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)

Curated by ChEMBL
LigandPNGBDBM50367212(CHEMBL4168413)
Affinity DataIC50:  910nMAssay Description:Inhibition of porcine pancreatic lipase using p-nitrophenyl butyrate as substrate pretreated for 15 mins followed by substrate addition and measured ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)

Curated by ChEMBL
LigandPNGBDBM50367214(CHEMBL4163899)
Affinity DataIC50:  950nMAssay Description:Inhibition of porcine pancreatic lipase using p-nitrophenyl butyrate as substrate pretreated for 15 mins followed by substrate addition and measured ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Homo sapiens (Human))
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)

Curated by ChEMBL
LigandPNGBDBM50367145(CHEMBL4173252)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of human pancreatic lipase using emulsified olive oil as substrate pretreated with substrate for 5 mins followed by enzyme addition and me...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Homo sapiens (Human))
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)

Curated by ChEMBL
LigandPNGBDBM50367138(CHEMBL4160519)
Affinity DataIC50:  1.25E+3nMAssay Description:Inhibition of human pancreatic lipase using emulsified olive oil as substrate pretreated with substrate for 5 mins followed by enzyme addition and me...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Homo sapiens (Human))
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)

Curated by ChEMBL
LigandPNGBDBM50367133(CHEMBL4164998)
Affinity DataIC50:  1.65E+3nMAssay Description:Inhibition of human pancreatic lipase using emulsified olive oil as substrate pretreated with substrate for 5 mins followed by enzyme addition and me...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Homo sapiens (Human))
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)

Curated by ChEMBL
LigandPNGBDBM50367134(CHEMBL4167341)
Affinity DataIC50:  1.87E+3nMAssay Description:Inhibition of human pancreatic lipase using emulsified olive oil as substrate pretreated with substrate for 5 mins followed by enzyme addition and me...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Homo sapiens (Human))
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)

Curated by ChEMBL
LigandPNGBDBM50367211(CHEMBL4165339)
Affinity DataIC50:  2.01E+3nMAssay Description:Inhibition of human pancreatic lipase using emulsified olive oil as substrate pretreated with substrate for 5 mins followed by enzyme addition and me...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Homo sapiens (Human))
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)

Curated by ChEMBL
LigandPNGBDBM50367212(CHEMBL4168413)
Affinity DataIC50:  2.28E+3nMAssay Description:Inhibition of human pancreatic lipase using emulsified olive oil as substrate pretreated with substrate for 5 mins followed by enzyme addition and me...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Homo sapiens (Human))
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)

Curated by ChEMBL
LigandPNGBDBM50367214(CHEMBL4163899)
Affinity DataIC50:  2.31E+3nMAssay Description:Inhibition of human pancreatic lipase using emulsified olive oil as substrate pretreated with substrate for 5 mins followed by enzyme addition and me...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)

Curated by ChEMBL
LigandPNGBDBM50367213(CHEMBL4175223)
Affinity DataIC50:  4.43E+3nMAssay Description:Inhibition of porcine pancreatic lipase using p-nitrophenyl butyrate as substrate pretreated for 15 mins followed by substrate addition and measured ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)

Curated by ChEMBL
LigandPNGBDBM50367143(CHEMBL4168757)
Affinity DataIC50:  5.35E+3nMAssay Description:Inhibition of porcine pancreatic lipase using p-nitrophenyl butyrate as substrate pretreated for 15 mins followed by substrate addition and measured ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)

Curated by ChEMBL
LigandPNGBDBM50367135(CHEMBL4160094)
Affinity DataIC50:  6.22E+3nMAssay Description:Inhibition of porcine pancreatic lipase using p-nitrophenyl butyrate as substrate pretreated for 15 mins followed by substrate addition and measured ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Homo sapiens (Human))
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)

Curated by ChEMBL
LigandPNGBDBM50367213(CHEMBL4175223)
Affinity DataIC50:  6.90E+3nMAssay Description:Inhibition of human pancreatic lipase using emulsified olive oil as substrate pretreated with substrate for 5 mins followed by enzyme addition and me...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Homo sapiens (Human))
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)

Curated by ChEMBL
LigandPNGBDBM50367216(CHEMBL4176621)
Affinity DataIC50:  7.38E+3nMAssay Description:Inhibition of human pancreatic lipase using emulsified olive oil as substrate pretreated with substrate for 5 mins followed by enzyme addition and me...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Homo sapiens (Human))
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)

Curated by ChEMBL
LigandPNGBDBM50367135(CHEMBL4160094)
Affinity DataIC50:  7.82E+3nMAssay Description:Inhibition of human pancreatic lipase using emulsified olive oil as substrate pretreated with substrate for 5 mins followed by enzyme addition and me...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)

Curated by ChEMBL
LigandPNGBDBM50367216(CHEMBL4176621)
Affinity DataIC50:  8.64E+3nMAssay Description:Inhibition of porcine pancreatic lipase using p-nitrophenyl butyrate as substrate pretreated for 15 mins followed by substrate addition and measured ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Homo sapiens (Human))
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)

Curated by ChEMBL
LigandPNGBDBM50367143(CHEMBL4168757)
Affinity DataIC50:  9.15E+3nMAssay Description:Inhibition of human pancreatic lipase using emulsified olive oil as substrate pretreated with substrate for 5 mins followed by enzyme addition and me...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)

Curated by ChEMBL
LigandPNGBDBM50367136(CHEMBL4172103)
Affinity DataIC50:  1.03E+4nMAssay Description:Inhibition of porcine pancreatic lipase using p-nitrophenyl butyrate as substrate pretreated for 15 mins followed by substrate addition and measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)

Curated by ChEMBL
LigandPNGBDBM50367215(CHEMBL4170734)
Affinity DataIC50:  1.04E+4nMAssay Description:Inhibition of porcine pancreatic lipase using p-nitrophenyl butyrate as substrate pretreated for 15 mins followed by substrate addition and measured ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Homo sapiens (Human))
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)

Curated by ChEMBL
LigandPNGBDBM50367136(CHEMBL4172103)
Affinity DataIC50:  1.18E+4nMAssay Description:Inhibition of human pancreatic lipase using emulsified olive oil as substrate pretreated with substrate for 5 mins followed by enzyme addition and me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Homo sapiens (Human))
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)

Curated by ChEMBL
LigandPNGBDBM50367215(CHEMBL4170734)
Affinity DataIC50:  1.35E+4nMAssay Description:Inhibition of human pancreatic lipase using emulsified olive oil as substrate pretreated with substrate for 5 mins followed by enzyme addition and me...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Homo sapiens (Human))
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)

Curated by ChEMBL
LigandPNGBDBM50367142(CHEMBL4161505)
Affinity DataIC50:  1.45E+4nMAssay Description:Inhibition of human pancreatic lipase using emulsified olive oil as substrate pretreated with substrate for 5 mins followed by enzyme addition and me...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)

Curated by ChEMBL
LigandPNGBDBM50367142(CHEMBL4161505)
Affinity DataIC50:  1.46E+4nMAssay Description:Inhibition of porcine pancreatic lipase using p-nitrophenyl butyrate as substrate pretreated for 15 mins followed by substrate addition and measured ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetForkhead box protein M1(Homo sapiens)
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50562257(CHEMBL4740210)
Affinity DataIC50:  5.05E+4nMAssay Description:Binding affinity to recombinant FOXM1 DBD (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as disruption of FOXM1-DNA complex prein...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetForkhead box protein M1(Homo sapiens)
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50085045(5-((4-((6-hydroxy-2,5,7,8-tetramethyl-3,4-dihydro-...)
Affinity DataIC50:  1.22E+5nMAssay Description:Binding affinity to recombinant FOXM1 DBD (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as disruption of FOXM1-DNA complex prein...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Maharishi Markandeshwar (Deemed To Be University)

Curated by ChEMBL
LigandPNGBDBM50183273((S)-6-(3-chloro-2-fluorobenzyl)-1-(1-hydroxy-3-met...)
Affinity DataEC50:  1nMAssay Description:Inhibition of HIV-1 integrase mutant strand transfer activity incubated for 10 mins by enzymatic assayMore data for this Ligand-Target Pair
In DepthDetails PubMedDrugBank

TargetIntegrase(Human immunodeficiency virus 1)
Maharishi Markandeshwar (Deemed To Be University)

Curated by ChEMBL
LigandPNGBDBM50183273((S)-6-(3-chloro-2-fluorobenzyl)-1-(1-hydroxy-3-met...)
Affinity DataEC50:  0.210nMAssay Description:Inhibition of HIV-1 integrase strand transfer activity incubated for 10 mins by enzymatic assayMore data for this Ligand-Target Pair
In DepthDetails PubMedDrugBank