Affinity DataKi: 21nMAssay Description:Binding affinity to recombinant FOXM1 DBD (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as disruption of FOXM1-DNA complex prein...More data for this Ligand-Target Pair
Affinity DataKi: 52nMAssay Description:Binding affinity to recombinant FOXM1 DBD (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as disruption of FOXM1-DNA complex prein...More data for this Ligand-Target Pair
TargetCytochrome P450 3A4(Homo sapiens (Human))
Maharishi Markandeshwar (Deemed To Be University)
Curated by ChEMBL
Maharishi Markandeshwar (Deemed To Be University)
Curated by ChEMBL
Affinity DataKi: 6.79E+4nMAssay Description:Inhibition of CYP3A4 in human liver microsomes using midazolam as substrateMore data for this Ligand-Target Pair
TargetPancreatic triacylglycerol lipase(Homo sapiens (Human))
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)
Curated by ChEMBL
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)
Curated by ChEMBL
Affinity DataIC50: 190nMAssay Description:Inhibition of human pancreatic lipase using emulsified olive oil as substrate pretreated with substrate for 5 mins followed by enzyme addition and me...More data for this Ligand-Target Pair
TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)
Curated by ChEMBL
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)
Curated by ChEMBL
Affinity DataIC50: 750nMAssay Description:Inhibition of porcine pancreatic lipase using p-nitrophenyl butyrate as substrate pretreated for 15 mins followed by substrate addition and measured ...More data for this Ligand-Target Pair
TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)
Curated by ChEMBL
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)
Curated by ChEMBL
Affinity DataIC50: 770nMAssay Description:Inhibition of porcine pancreatic lipase using p-nitrophenyl butyrate as substrate pretreated for 15 mins followed by substrate addition and measured ...More data for this Ligand-Target Pair
TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)
Curated by ChEMBL
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)
Curated by ChEMBL
Affinity DataIC50: 800nMAssay Description:Inhibition of porcine pancreatic lipase using p-nitrophenyl butyrate as substrate pretreated for 15 mins followed by substrate addition and measured ...More data for this Ligand-Target Pair
TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)
Curated by ChEMBL
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)
Curated by ChEMBL
Affinity DataIC50: 800nMAssay Description:Inhibition of porcine pancreatic lipase using p-nitrophenyl butyrate as substrate pretreated for 15 mins followed by substrate addition and measured ...More data for this Ligand-Target Pair
TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)
Curated by ChEMBL
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)
Curated by ChEMBL
Affinity DataIC50: 840nMAssay Description:Inhibition of porcine pancreatic lipase using p-nitrophenyl butyrate as substrate pretreated for 15 mins followed by substrate addition and measured ...More data for this Ligand-Target Pair
TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)
Curated by ChEMBL
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)
Curated by ChEMBL
Affinity DataIC50: 850nMAssay Description:Inhibition of porcine pancreatic lipase using p-nitrophenyl butyrate as substrate pretreated for 15 mins followed by substrate addition and measured ...More data for this Ligand-Target Pair
TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)
Curated by ChEMBL
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)
Curated by ChEMBL
Affinity DataIC50: 910nMAssay Description:Inhibition of porcine pancreatic lipase using p-nitrophenyl butyrate as substrate pretreated for 15 mins followed by substrate addition and measured ...More data for this Ligand-Target Pair
TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)
Curated by ChEMBL
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)
Curated by ChEMBL
Affinity DataIC50: 950nMAssay Description:Inhibition of porcine pancreatic lipase using p-nitrophenyl butyrate as substrate pretreated for 15 mins followed by substrate addition and measured ...More data for this Ligand-Target Pair
TargetPancreatic triacylglycerol lipase(Homo sapiens (Human))
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)
Curated by ChEMBL
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of human pancreatic lipase using emulsified olive oil as substrate pretreated with substrate for 5 mins followed by enzyme addition and me...More data for this Ligand-Target Pair
TargetPancreatic triacylglycerol lipase(Homo sapiens (Human))
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)
Curated by ChEMBL
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)
Curated by ChEMBL
Affinity DataIC50: 1.25E+3nMAssay Description:Inhibition of human pancreatic lipase using emulsified olive oil as substrate pretreated with substrate for 5 mins followed by enzyme addition and me...More data for this Ligand-Target Pair
TargetPancreatic triacylglycerol lipase(Homo sapiens (Human))
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)
Curated by ChEMBL
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)
Curated by ChEMBL
Affinity DataIC50: 1.65E+3nMAssay Description:Inhibition of human pancreatic lipase using emulsified olive oil as substrate pretreated with substrate for 5 mins followed by enzyme addition and me...More data for this Ligand-Target Pair
TargetPancreatic triacylglycerol lipase(Homo sapiens (Human))
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)
Curated by ChEMBL
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)
Curated by ChEMBL
Affinity DataIC50: 1.87E+3nMAssay Description:Inhibition of human pancreatic lipase using emulsified olive oil as substrate pretreated with substrate for 5 mins followed by enzyme addition and me...More data for this Ligand-Target Pair
TargetPancreatic triacylglycerol lipase(Homo sapiens (Human))
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)
Curated by ChEMBL
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)
Curated by ChEMBL
Affinity DataIC50: 2.01E+3nMAssay Description:Inhibition of human pancreatic lipase using emulsified olive oil as substrate pretreated with substrate for 5 mins followed by enzyme addition and me...More data for this Ligand-Target Pair
TargetPancreatic triacylglycerol lipase(Homo sapiens (Human))
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)
Curated by ChEMBL
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)
Curated by ChEMBL
Affinity DataIC50: 2.28E+3nMAssay Description:Inhibition of human pancreatic lipase using emulsified olive oil as substrate pretreated with substrate for 5 mins followed by enzyme addition and me...More data for this Ligand-Target Pair
TargetPancreatic triacylglycerol lipase(Homo sapiens (Human))
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)
Curated by ChEMBL
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)
Curated by ChEMBL
Affinity DataIC50: 2.31E+3nMAssay Description:Inhibition of human pancreatic lipase using emulsified olive oil as substrate pretreated with substrate for 5 mins followed by enzyme addition and me...More data for this Ligand-Target Pair
TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)
Curated by ChEMBL
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)
Curated by ChEMBL
Affinity DataIC50: 4.43E+3nMAssay Description:Inhibition of porcine pancreatic lipase using p-nitrophenyl butyrate as substrate pretreated for 15 mins followed by substrate addition and measured ...More data for this Ligand-Target Pair
TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)
Curated by ChEMBL
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)
Curated by ChEMBL
Affinity DataIC50: 5.35E+3nMAssay Description:Inhibition of porcine pancreatic lipase using p-nitrophenyl butyrate as substrate pretreated for 15 mins followed by substrate addition and measured ...More data for this Ligand-Target Pair
TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)
Curated by ChEMBL
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)
Curated by ChEMBL
Affinity DataIC50: 6.22E+3nMAssay Description:Inhibition of porcine pancreatic lipase using p-nitrophenyl butyrate as substrate pretreated for 15 mins followed by substrate addition and measured ...More data for this Ligand-Target Pair
TargetPancreatic triacylglycerol lipase(Homo sapiens (Human))
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)
Curated by ChEMBL
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)
Curated by ChEMBL
Affinity DataIC50: 6.90E+3nMAssay Description:Inhibition of human pancreatic lipase using emulsified olive oil as substrate pretreated with substrate for 5 mins followed by enzyme addition and me...More data for this Ligand-Target Pair
TargetPancreatic triacylglycerol lipase(Homo sapiens (Human))
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)
Curated by ChEMBL
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)
Curated by ChEMBL
Affinity DataIC50: 7.38E+3nMAssay Description:Inhibition of human pancreatic lipase using emulsified olive oil as substrate pretreated with substrate for 5 mins followed by enzyme addition and me...More data for this Ligand-Target Pair
TargetPancreatic triacylglycerol lipase(Homo sapiens (Human))
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)
Curated by ChEMBL
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)
Curated by ChEMBL
Affinity DataIC50: 7.82E+3nMAssay Description:Inhibition of human pancreatic lipase using emulsified olive oil as substrate pretreated with substrate for 5 mins followed by enzyme addition and me...More data for this Ligand-Target Pair
TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)
Curated by ChEMBL
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)
Curated by ChEMBL
Affinity DataIC50: 8.64E+3nMAssay Description:Inhibition of porcine pancreatic lipase using p-nitrophenyl butyrate as substrate pretreated for 15 mins followed by substrate addition and measured ...More data for this Ligand-Target Pair
TargetPancreatic triacylglycerol lipase(Homo sapiens (Human))
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)
Curated by ChEMBL
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)
Curated by ChEMBL
Affinity DataIC50: 9.15E+3nMAssay Description:Inhibition of human pancreatic lipase using emulsified olive oil as substrate pretreated with substrate for 5 mins followed by enzyme addition and me...More data for this Ligand-Target Pair
TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)
Curated by ChEMBL
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)
Curated by ChEMBL
Affinity DataIC50: 1.03E+4nMAssay Description:Inhibition of porcine pancreatic lipase using p-nitrophenyl butyrate as substrate pretreated for 15 mins followed by substrate addition and measured ...More data for this Ligand-Target Pair
TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)
Curated by ChEMBL
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)
Curated by ChEMBL
Affinity DataIC50: 1.04E+4nMAssay Description:Inhibition of porcine pancreatic lipase using p-nitrophenyl butyrate as substrate pretreated for 15 mins followed by substrate addition and measured ...More data for this Ligand-Target Pair
TargetPancreatic triacylglycerol lipase(Homo sapiens (Human))
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)
Curated by ChEMBL
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)
Curated by ChEMBL
Affinity DataIC50: 1.18E+4nMAssay Description:Inhibition of human pancreatic lipase using emulsified olive oil as substrate pretreated with substrate for 5 mins followed by enzyme addition and me...More data for this Ligand-Target Pair
TargetPancreatic triacylglycerol lipase(Homo sapiens (Human))
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)
Curated by ChEMBL
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)
Curated by ChEMBL
Affinity DataIC50: 1.35E+4nMAssay Description:Inhibition of human pancreatic lipase using emulsified olive oil as substrate pretreated with substrate for 5 mins followed by enzyme addition and me...More data for this Ligand-Target Pair
TargetPancreatic triacylglycerol lipase(Homo sapiens (Human))
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)
Curated by ChEMBL
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)
Curated by ChEMBL
Affinity DataIC50: 1.45E+4nMAssay Description:Inhibition of human pancreatic lipase using emulsified olive oil as substrate pretreated with substrate for 5 mins followed by enzyme addition and me...More data for this Ligand-Target Pair
TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)
Curated by ChEMBL
Csir - National Institute For Interdisciplinary Science and Technology (Csir-Niist)
Curated by ChEMBL
Affinity DataIC50: 1.46E+4nMAssay Description:Inhibition of porcine pancreatic lipase using p-nitrophenyl butyrate as substrate pretreated for 15 mins followed by substrate addition and measured ...More data for this Ligand-Target Pair
Affinity DataIC50: 5.05E+4nMAssay Description:Binding affinity to recombinant FOXM1 DBD (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as disruption of FOXM1-DNA complex prein...More data for this Ligand-Target Pair
Affinity DataIC50: 1.22E+5nMAssay Description:Binding affinity to recombinant FOXM1 DBD (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as disruption of FOXM1-DNA complex prein...More data for this Ligand-Target Pair
TargetIntegrase(Human immunodeficiency virus 1)
Maharishi Markandeshwar (Deemed To Be University)
Curated by ChEMBL
Maharishi Markandeshwar (Deemed To Be University)
Curated by ChEMBL
Affinity DataEC50: 1nMAssay Description:Inhibition of HIV-1 integrase mutant strand transfer activity incubated for 10 mins by enzymatic assayMore data for this Ligand-Target Pair
TargetIntegrase(Human immunodeficiency virus 1)
Maharishi Markandeshwar (Deemed To Be University)
Curated by ChEMBL
Maharishi Markandeshwar (Deemed To Be University)
Curated by ChEMBL
Affinity DataEC50: 0.210nMAssay Description:Inhibition of HIV-1 integrase strand transfer activity incubated for 10 mins by enzymatic assayMore data for this Ligand-Target Pair