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Found 23 with Last Name = 'gyires' and Initial = 'k'
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM13063(4-(5-methyl-3-phenyl-1,2-oxazol-4-yl)benzene-1-sul...)
Affinity DataIC50:  40nMAssay Description:Inhibition of human recombinant COX2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50229774(CHEMBL254418 | N-Hydroxy-4-(5-methyl-3-phenylisoxa...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of human recombinant COX2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMembrane primary amine oxidase(Homo sapiens (Human))
Semmelweis Egyetem

US Patent
LigandPNGBDBM102391(US8536210, 40)
Affinity DataIC50:  3.50E+3nMpH: 7.2 T: 2°CAssay Description:For determining the SSAO/VAP-1 activity, the colorimetric method described by Holt, A (Holt, A., Biochem. 244, 384, 1997) for monoamine oxidase and a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMembrane primary amine oxidase(Homo sapiens (Human))
Semmelweis Egyetem

US Patent
LigandPNGBDBM102357(US8536210, 6)
Affinity DataIC50:  4.30E+3nMpH: 7.2 T: 2°CAssay Description:For determining the SSAO/VAP-1 activity, the colorimetric method described by Holt, A (Holt, A., Biochem. 244, 384, 1997) for monoamine oxidase and a...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMembrane primary amine oxidase(Homo sapiens (Human))
Semmelweis Egyetem

US Patent
LigandPNGBDBM102360(US8536210, 9)
Affinity DataIC50:  1.49E+4nMpH: 7.2 T: 2°CAssay Description:For determining the SSAO/VAP-1 activity, the colorimetric method described by Holt, A (Holt, A., Biochem. 244, 384, 1997) for monoamine oxidase and a...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMembrane primary amine oxidase(Homo sapiens (Human))
Semmelweis Egyetem

US Patent
LigandPNGBDBM102369(US8536210, 18)
Affinity DataIC50:  1.80E+4nMpH: 7.2 T: 2°CAssay Description:For determining the SSAO/VAP-1 activity, the colorimetric method described by Holt, A (Holt, A., Biochem. 244, 384, 1997) for monoamine oxidase and a...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMembrane primary amine oxidase(Homo sapiens (Human))
Semmelweis Egyetem

US Patent
LigandPNGBDBM102370(US8536210, 19)
Affinity DataIC50:  2.90E+4nMpH: 7.2 T: 2°CAssay Description:For determining the SSAO/VAP-1 activity, the colorimetric method described by Holt, A (Holt, A., Biochem. 244, 384, 1997) for monoamine oxidase and a...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMembrane primary amine oxidase(Homo sapiens (Human))
Semmelweis Egyetem

US Patent
LigandPNGBDBM102368(US8536210, 17)
Affinity DataIC50:  3.00E+4nMpH: 7.2 T: 2°CAssay Description:For determining the SSAO/VAP-1 activity, the colorimetric method described by Holt, A (Holt, A., Biochem. 244, 384, 1997) for monoamine oxidase and a...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMembrane primary amine oxidase(Homo sapiens (Human))
Semmelweis Egyetem

US Patent
LigandPNGBDBM102358(US8536210, 7)
Affinity DataIC50:  4.00E+4nMpH: 7.2 T: 2°CAssay Description:For determining the SSAO/VAP-1 activity, the colorimetric method described by Holt, A (Holt, A., Biochem. 244, 384, 1997) for monoamine oxidase and a...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMembrane primary amine oxidase(Homo sapiens (Human))
Semmelweis Egyetem

US Patent
LigandPNGBDBM102378(US8536210, 27)
Affinity DataIC50:  4.10E+4nMpH: 7.2 T: 2°CAssay Description:For determining the SSAO/VAP-1 activity, the colorimetric method described by Holt, A (Holt, A., Biochem. 244, 384, 1997) for monoamine oxidase and a...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails US Patent
TargetMembrane primary amine oxidase(Homo sapiens (Human))
Semmelweis Egyetem

US Patent
LigandPNGBDBM102373(US8536210, 22)
Affinity DataIC50:  4.80E+4nMpH: 7.2 T: 2°CAssay Description:For determining the SSAO/VAP-1 activity, the colorimetric method described by Holt, A (Holt, A., Biochem. 244, 384, 1997) for monoamine oxidase and a...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMembrane primary amine oxidase(Homo sapiens (Human))
Semmelweis Egyetem

US Patent
LigandPNGBDBM102367(US8536210, 16)
Affinity DataIC50:  5.30E+4nMpH: 7.2 T: 2°CAssay Description:For determining the SSAO/VAP-1 activity, the colorimetric method described by Holt, A (Holt, A., Biochem. 244, 384, 1997) for monoamine oxidase and a...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMembrane primary amine oxidase(Homo sapiens (Human))
Semmelweis Egyetem

US Patent
LigandPNGBDBM102372(US8536210, 21)
Affinity DataIC50:  5.80E+4nMpH: 7.2 T: 2°CAssay Description:For determining the SSAO/VAP-1 activity, the colorimetric method described by Holt, A (Holt, A., Biochem. 244, 384, 1997) for monoamine oxidase and a...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMembrane primary amine oxidase(Homo sapiens (Human))
Semmelweis Egyetem

US Patent
LigandPNGBDBM102359(US8536210, 8)
Affinity DataIC50:  9.50E+4nMpH: 7.2 T: 2°CAssay Description:For determining the SSAO/VAP-1 activity, the colorimetric method described by Holt, A (Holt, A., Biochem. 244, 384, 1997) for monoamine oxidase and a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50229774(CHEMBL254418 | N-Hydroxy-4-(5-methyl-3-phenylisoxa...)
Affinity DataIC50:  9.62E+4nMAssay Description:Inhibition of ovine COX1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMembrane primary amine oxidase(Homo sapiens (Human))
Semmelweis Egyetem

US Patent
LigandPNGBDBM102352(US8536210, 1)
Affinity DataIC50:  1.02E+5nMpH: 7.2 T: 2°CAssay Description:For determining the SSAO/VAP-1 activity, the colorimetric method described by Holt, A (Holt, A., Biochem. 244, 384, 1997) for monoamine oxidase and a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMembrane primary amine oxidase(Homo sapiens (Human))
Semmelweis Egyetem

US Patent
LigandPNGBDBM102375(US8536210, 24)
Affinity DataIC50:  1.06E+5nMpH: 7.2 T: 2°CAssay Description:For determining the SSAO/VAP-1 activity, the colorimetric method described by Holt, A (Holt, A., Biochem. 244, 384, 1997) for monoamine oxidase and a...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails US Patent
TargetMembrane primary amine oxidase(Homo sapiens (Human))
Semmelweis Egyetem

US Patent
LigandPNGBDBM102374(US8536210, 23)
Affinity DataIC50:  1.11E+5nMpH: 7.2 T: 2°CAssay Description:For determining the SSAO/VAP-1 activity, the colorimetric method described by Holt, A (Holt, A., Biochem. 244, 384, 1997) for monoamine oxidase and a...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMembrane primary amine oxidase(Homo sapiens (Human))
Semmelweis Egyetem

US Patent
LigandPNGBDBM102376(US8536210, 25)
Affinity DataIC50:  1.13E+5nMpH: 7.2 T: 2°CAssay Description:For determining the SSAO/VAP-1 activity, the colorimetric method described by Holt, A (Holt, A., Biochem. 244, 384, 1997) for monoamine oxidase and a...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM13063(4-(5-methyl-3-phenyl-1,2-oxazol-4-yl)benzene-1-sul...)
Affinity DataIC50:  1.57E+5nMAssay Description:Inhibition of ovine COX1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMembrane primary amine oxidase(Homo sapiens (Human))
Semmelweis Egyetem

US Patent
LigandPNGBDBM102363(US8536210, 12)
Affinity DataIC50:  1.80E+5nMpH: 7.2 T: 2°CAssay Description:For determining the SSAO/VAP-1 activity, the colorimetric method described by Holt, A (Holt, A., Biochem. 244, 384, 1997) for monoamine oxidase and a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMembrane primary amine oxidase(Homo sapiens (Human))
Semmelweis Egyetem

US Patent
LigandPNGBDBM102380(US8536210, 29)
Affinity DataIC50:  2.40E+5nMpH: 7.2 T: 2°CAssay Description:For determining the SSAO/VAP-1 activity, the colorimetric method described by Holt, A (Holt, A., Biochem. 244, 384, 1997) for monoamine oxidase and a...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMembrane primary amine oxidase(Homo sapiens (Human))
Semmelweis Egyetem

US Patent
LigandPNGBDBM102383(US8536210, 32)
Affinity DataIC50:  2.63E+5nMpH: 7.2 T: 2°CAssay Description:For determining the SSAO/VAP-1 activity, the colorimetric method described by Holt, A (Holt, A., Biochem. 244, 384, 1997) for monoamine oxidase and a...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails US Patent