Compile Data Set for Download or QSAR
maximum 50k data
Found 495 with Last Name = 'maddali' and Initial = 'k'
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50482161(CHEMBL1082256)
Affinity DataIC50:  4nMAssay Description:Inhibition of HIV1 integrase strand transfer activity after 1 hr by densitometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50482160(CHEMBL1082257)
Affinity DataIC50:  5nMAssay Description:Inhibition of HIV1 integrase strand transfer activity after 1 hr by densitometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50482160(CHEMBL1082257)
Affinity DataIC50:  6nMAssay Description:Inhibition of HIV1 integrase 3'-end processing activity after 1 hr by densitometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50482161(CHEMBL1082256)
Affinity DataIC50:  8nMAssay Description:Inhibition of HIV1 integrase 3'-end processing activity after 1 hr by densitometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50482699(CHEMBL1241174)
Affinity DataIC50:  10nMAssay Description:Inhibition of HIV1 integrase strand transfer activity expressed in Escherichia coli after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50183273((S)-6-(3-chloro-2-fluorobenzyl)-1-(1-hydroxy-3-met...)
Affinity DataIC50:  28nMAssay Description:Inhibition of HIV1 integrase strand transfer activity by gel-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50482700(CHEMBL1241178)
Affinity DataIC50:  31nMAssay Description:Inhibition of HIV1 integrase strand transfer activity expressed in Escherichia coli after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50482160(CHEMBL1082257)
Affinity DataIC50:  40nMAssay Description:Inhibition of HIV1 integrase strand transfer activity expressed in Escherichia coli after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50050533(6-BENZYL-1-BENZYLOXYMETHYL-5-ISOPROPYL URACIL | 6-...)
Affinity DataIC50:  40nMAssay Description:Inhibition of HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50482700(CHEMBL1241178)
Affinity DataIC50:  40nMAssay Description:Inhibition of HIV1 integrase 3'-processing activity expressed in Escherichia coli after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50486150(CHEMBL2206768)
Affinity DataIC50:  47nMAssay Description:Inhibition of HIV1 recombinant integrase strand transfer activity using [32P]-labeled oligonucleotide a substrate after 30 mins by electrophoretic an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50482714(CHEMBL1241175)
Affinity DataIC50:  47nMAssay Description:Inhibition of HIV1 integrase strand transfer activity expressed in Escherichia coli after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50482698(CHEMBL1241173)
Affinity DataIC50:  50nMAssay Description:Inhibition of HIV1 integrase strand transfer activity expressed in Escherichia coli after 60 minsMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50482710(CHEMBL1241189)
Affinity DataIC50:  50nMAssay Description:Inhibition of HIV1 integrase strand transfer activity expressed in Escherichia coli after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50482699(CHEMBL1241174)
Affinity DataIC50:  50nMAssay Description:Inhibition of HIV1 integrase 3'-processing activity expressed in Escherichia coli after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50004364(CHEMBL3238134)
Affinity DataIC50:  50nMAssay Description:Inhibition of HIV1 integrase strand transfer activity by gel-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50486153(CHEMBL2206761)
Affinity DataIC50:  54nMAssay Description:Inhibition of HIV1 recombinant integrase strand transfer activity using [32P]-labeled oligonucleotide a substrate after 30 mins by electrophoretic an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50486149(CHEMBL2206770)
Affinity DataIC50:  58nMAssay Description:Inhibition of HIV1 recombinant integrase strand transfer activity using [32P]-labeled oligonucleotide a substrate after 30 mins by electrophoretic an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50482709(CHEMBL1241187)
Affinity DataIC50:  60nMAssay Description:Inhibition of HIV1 integrase strand transfer activity expressed in Escherichia coli after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50482720(CHEMBL1241183)
Affinity DataIC50:  60nMAssay Description:Inhibition of HIV1 integrase strand transfer activity expressed in Escherichia coli after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50482161(CHEMBL1082256)
Affinity DataIC50:  60nMAssay Description:Inhibition of HIV1 integrase strand transfer activity expressed in Escherichia coli after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50482704(CHEMBL1241184)
Affinity DataIC50:  60nMAssay Description:Inhibition of HIV1 integrase strand transfer activity expressed in Escherichia coli after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50482703(CHEMBL1241182)
Affinity DataIC50:  60nMAssay Description:Inhibition of HIV1 integrase strand transfer activity expressed in Escherichia coli after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50482701(CHEMBL1241179)
Affinity DataIC50:  60nMAssay Description:Inhibition of HIV1 integrase strand transfer activity expressed in Escherichia coli after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50482719(CHEMBL1241176)
Affinity DataIC50:  65nMAssay Description:Inhibition of HIV1 integrase strand transfer activity expressed in Escherichia coli after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [1148-1435](Human immunodeficiency virus type 1)
National Institutes of Health

LigandPNGBDBM86654(Bicyclic hydroxy-1H-pyrrolopyridine-trione, 1)
Affinity DataIC50:  67nMAssay Description:The compound were evaluated in biochemical IN (integrase) assay that measure inhibitory potency (IC50 values)against both the 3'-processing(3'...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM25351(N-[2-(4-{[(4-fluorophenyl)methyl]carbamoyl}-5-hydr...)
Affinity DataIC50:  67nMAssay Description:Inhibition of HIV1 recombinant integrase strand transfer activity expressed in Escherichia coli after 30 mins using [32P]-labeled oligonucleotide as ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM25351(N-[2-(4-{[(4-fluorophenyl)methyl]carbamoyl}-5-hydr...)
Affinity DataIC50:  67nMAssay Description:Inhibition of HIV1 recombinant integrase strand transfer activity expressed in Escherichia coli after 60 mins using [32P]-labeled oligonucleotide as ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50482712(CHEMBL1241169)
Affinity DataIC50:  70nMAssay Description:Inhibition of HIV1 integrase strand transfer activity expressed in Escherichia coli after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50482716(CHEMBL1240540)
Affinity DataIC50:  70nMAssay Description:Inhibition of HIV1 integrase strand transfer activity expressed in Escherichia coli after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50482713(CHEMBL1241172)
Affinity DataIC50:  70nMAssay Description:Inhibition of HIV1 integrase strand transfer activity expressed in Escherichia coli after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM25351(N-[2-(4-{[(4-fluorophenyl)methyl]carbamoyl}-5-hydr...)
Affinity DataIC50:  74nMAssay Description:Inhibition of HIV1 recombinant integrase strand transfer activity expressed in Escherichia coli after 60 mins using [32P]-labeled oligonucleotide as ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50482698(CHEMBL1241173)
Affinity DataIC50:  80nMAssay Description:Inhibition of HIV1 integrase 3'-processing activity expressed in Escherichia coli after 60 minsMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50486160(CHEMBL2206769)
Affinity DataIC50:  80nMAssay Description:Inhibition of HIV1 recombinant integrase strand transfer activity using [32P]-labeled oligonucleotide a substrate after 30 mins by electrophoretic an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50482717(CHEMBL1241180)
Affinity DataIC50:  80nMAssay Description:Inhibition of HIV1 integrase strand transfer activity expressed in Escherichia coli after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50482702(CHEMBL1241181)
Affinity DataIC50:  80nMAssay Description:Inhibition of HIV1 integrase strand transfer activity expressed in Escherichia coli after 60 minsMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50004360(CHEMBL3238130)
Affinity DataIC50:  80nMAssay Description:Inhibition of HIV1 integrase strand transfer activity by gel-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50004362(CHEMBL3238132)
Affinity DataIC50:  80nMAssay Description:Inhibition of HIV1 integrase strand transfer activity by gel-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM25351(N-[2-(4-{[(4-fluorophenyl)methyl]carbamoyl}-5-hydr...)
Affinity DataIC50:  87nMAssay Description:Inhibition of HIV1 integrase strand transfer activity by gel-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50482708(CHEMBL1241191)
Affinity DataIC50:  90nMAssay Description:Inhibition of HIV1 integrase 3'-processing activity expressed in Escherichia coli after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50482160(CHEMBL1082257)
Affinity DataIC50:  90nMAssay Description:Inhibition of HIV1 integrase 3'-processing activity expressed in Escherichia coli after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50482708(CHEMBL1241191)
Affinity DataIC50:  90nMAssay Description:Inhibition of HIV1 integrase strand transfer activity expressed in Escherichia coli after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50480538(CHEMBL557899)
Affinity DataIC50:  100nMAssay Description:Inhibition of HIV1 integrase strand transfer activity in presence of magnesiumMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50482712(CHEMBL1241169)
Affinity DataIC50:  100nMAssay Description:Inhibition of HIV1 integrase 3'-processing activity expressed in Escherichia coli after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50480524(CHEMBL562366)
Affinity DataIC50:  100nMAssay Description:Inhibition of HIV1 integrase strand transfer activity in presence of magnesiumMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50482720(CHEMBL1241183)
Affinity DataIC50:  100nMAssay Description:Inhibition of HIV1 integrase 3'-processing activity expressed in Escherichia coli after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50004358(CHEMBL3238128)
Affinity DataIC50:  100nMAssay Description:Inhibition of HIV1 integrase strand transfer activity by gel-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50482710(CHEMBL1241189)
Affinity DataIC50:  110nMAssay Description:Inhibition of HIV1 integrase 3'-processing activity expressed in Escherichia coli after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50482713(CHEMBL1241172)
Affinity DataIC50:  110nMAssay Description:Inhibition of HIV1 integrase 3'-processing activity expressed in Escherichia coli after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50482711(CHEMBL1241170)
Affinity DataIC50:  110nMAssay Description:Inhibition of HIV1 integrase strand transfer activity expressed in Escherichia coli after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 495 total ) | Next | Last >>
Jump to: