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Found 104 with Last Name = 'harris' and Initial = 'ld'
TargetOrotate phosphoribosyltransferase(Plasmodium falciparum)
Albert Einstein College of Medicine

LigandPNGBDBM214779(OPRT inhibitor, 2)
Affinity DataKi:  40nM ΔG°:  -42.2kJ/molepH: 8.0 T: 2°CAssay Description:Inhibition constants (Ki, equivalent to Kd for competitive inhibitors) were measured at 25 °C by adding purified OPRT enzymes (25 nM for PfOPRT a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUridine 5'-monophosphate synthase(Homo sapiens (Human))
Albert Einstein College of Medicine

LigandPNGBDBM214779(OPRT inhibitor, 2)
Affinity DataKi:  41nM ΔG°:  -42.2kJ/molepH: 8.0 T: 2°CAssay Description:Inhibition constants (Ki, equivalent to Kd for competitive inhibitors) were measured at 25 °C by adding purified OPRT enzymes (25 nM for PfOPRT a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUridine 5'-monophosphate synthase(Homo sapiens (Human))
Albert Einstein College of Medicine

LigandPNGBDBM214786(OPRT inhibitor, 9)
Affinity DataKi:  80nM ΔG°:  -40.5kJ/molepH: 8.0 T: 2°CAssay Description:Inhibition constants (Ki, equivalent to Kd for competitive inhibitors) were measured at 25 °C by adding purified OPRT enzymes (25 nM for PfOPRT a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUridine 5'-monophosphate synthase(Homo sapiens (Human))
Albert Einstein College of Medicine

LigandPNGBDBM214791(OPRT inhibitor, 14)
Affinity DataKi:  83nM ΔG°:  -40.4kJ/molepH: 8.0 T: 2°CAssay Description:Inhibition constants (Ki, equivalent to Kd for competitive inhibitors) were measured at 25 °C by adding purified OPRT enzymes (25 nM for PfOPRT a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUridine 5'-monophosphate synthase(Homo sapiens (Human))
Albert Einstein College of Medicine

LigandPNGBDBM214785(OPRT inhibitor, 8)
Affinity DataKi:  90nM ΔG°:  -40.2kJ/molepH: 8.0 T: 2°CAssay Description:Inhibition constants (Ki, equivalent to Kd for competitive inhibitors) were measured at 25 °C by adding purified OPRT enzymes (25 nM for PfOPRT a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUridine 5'-monophosphate synthase(Homo sapiens (Human))
Albert Einstein College of Medicine

LigandPNGBDBM214784(OPRT inhibitor, 7)
Affinity DataKi:  110nM ΔG°:  -39.7kJ/molepH: 8.0 T: 2°CAssay Description:Inhibition constants (Ki, equivalent to Kd for competitive inhibitors) were measured at 25 °C by adding purified OPRT enzymes (25 nM for PfOPRT a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUridine 5'-monophosphate synthase(Homo sapiens (Human))
Albert Einstein College of Medicine

LigandPNGBDBM214778(OPRT inhibitor, 1 )
Affinity DataKi:  120nM ΔG°:  -39.5kJ/molepH: 8.0 T: 2°CAssay Description:Inhibition constants (Ki, equivalent to Kd for competitive inhibitors) were measured at 25 °C by adding purified OPRT enzymes (25 nM for PfOPRT a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUridine 5'-monophosphate synthase(Homo sapiens (Human))
Albert Einstein College of Medicine

LigandPNGBDBM214797(OPRT inhibitor, 20)
Affinity DataKi:  120nM ΔG°:  -39.5kJ/molepH: 8.0 T: 2°CAssay Description:Inhibition constants (Ki, equivalent to Kd for competitive inhibitors) were measured at 25 °C by adding purified OPRT enzymes (25 nM for PfOPRT a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUridine 5'-monophosphate synthase(Homo sapiens (Human))
Albert Einstein College of Medicine

LigandPNGBDBM214783(OPRT inhibitor, 6)
Affinity DataKi:  140nM ΔG°:  -39.1kJ/molepH: 8.0 T: 2°CAssay Description:Inhibition constants (Ki, equivalent to Kd for competitive inhibitors) were measured at 25 °C by adding purified OPRT enzymes (25 nM for PfOPRT a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUridine 5'-monophosphate synthase(Homo sapiens (Human))
Albert Einstein College of Medicine

LigandPNGBDBM214796(OPRT inhibitor, 19)
Affinity DataKi:  150nM ΔG°:  -38.9kJ/molepH: 8.0 T: 2°CAssay Description:Inhibition constants (Ki, equivalent to Kd for competitive inhibitors) were measured at 25 °C by adding purified OPRT enzymes (25 nM for PfOPRT a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOrotate phosphoribosyltransferase(Plasmodium falciparum)
Albert Einstein College of Medicine

LigandPNGBDBM214785(OPRT inhibitor, 8)
Affinity DataKi:  170nM ΔG°:  -38.6kJ/molepH: 8.0 T: 2°CAssay Description:Inhibition constants (Ki, equivalent to Kd for competitive inhibitors) were measured at 25 °C by adding purified OPRT enzymes (25 nM for PfOPRT a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOrotate phosphoribosyltransferase(Plasmodium falciparum)
Albert Einstein College of Medicine

LigandPNGBDBM214778(OPRT inhibitor, 1 )
Affinity DataKi:  190nM ΔG°:  -38.4kJ/molepH: 8.0 T: 2°CAssay Description:Inhibition constants (Ki, equivalent to Kd for competitive inhibitors) were measured at 25 °C by adding purified OPRT enzymes (25 nM for PfOPRT a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUridine 5'-monophosphate synthase(Homo sapiens (Human))
Albert Einstein College of Medicine

LigandPNGBDBM214781(OPRT inhibitor, 4)
Affinity DataKi:  200nM ΔG°:  -38.2kJ/molepH: 8.0 T: 2°CAssay Description:Inhibition constants (Ki, equivalent to Kd for competitive inhibitors) were measured at 25 °C by adding purified OPRT enzymes (25 nM for PfOPRT a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUridine 5'-monophosphate synthase(Homo sapiens (Human))
Albert Einstein College of Medicine

LigandPNGBDBM214794(OPRT inhibitor, 17)
Affinity DataKi:  200nM ΔG°:  -38.2kJ/molepH: 8.0 T: 2°CAssay Description:Inhibition constants (Ki, equivalent to Kd for competitive inhibitors) were measured at 25 °C by adding purified OPRT enzymes (25 nM for PfOPRT a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOrotate phosphoribosyltransferase(Plasmodium falciparum)
Albert Einstein College of Medicine

LigandPNGBDBM214791(OPRT inhibitor, 14)
Affinity DataKi:  220nM ΔG°:  -38.0kJ/molepH: 8.0 T: 2°CAssay Description:Inhibition constants (Ki, equivalent to Kd for competitive inhibitors) were measured at 25 °C by adding purified OPRT enzymes (25 nM for PfOPRT a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUridine 5'-monophosphate synthase(Homo sapiens (Human))
Albert Einstein College of Medicine

LigandPNGBDBM214793(OPRT inhibitor, 16)
Affinity DataKi:  230nM ΔG°:  -37.9kJ/molepH: 8.0 T: 2°CAssay Description:Inhibition constants (Ki, equivalent to Kd for competitive inhibitors) were measured at 25 °C by adding purified OPRT enzymes (25 nM for PfOPRT a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUridine 5'-monophosphate synthase(Homo sapiens (Human))
Albert Einstein College of Medicine

LigandPNGBDBM214795(OPRT inhibitor, 18)
Affinity DataKi:  230nM ΔG°:  -37.9kJ/molepH: 8.0 T: 2°CAssay Description:Inhibition constants (Ki, equivalent to Kd for competitive inhibitors) were measured at 25 °C by adding purified OPRT enzymes (25 nM for PfOPRT a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUridine 5'-monophosphate synthase(Homo sapiens (Human))
Albert Einstein College of Medicine

LigandPNGBDBM214792(OPRT inhibitor, 15)
Affinity DataKi:  240nM ΔG°:  -37.8kJ/molepH: 8.0 T: 2°CAssay Description:Inhibition constants (Ki, equivalent to Kd for competitive inhibitors) were measured at 25 °C by adding purified OPRT enzymes (25 nM for PfOPRT a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUridine 5'-monophosphate synthase(Homo sapiens (Human))
Albert Einstein College of Medicine

LigandPNGBDBM214790(OPRT inhibitor, 13)
Affinity DataKi:  250nM ΔG°:  -37.7kJ/molepH: 8.0 T: 2°CAssay Description:Inhibition constants (Ki, equivalent to Kd for competitive inhibitors) were measured at 25 °C by adding purified OPRT enzymes (25 nM for PfOPRT a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrotate phosphoribosyltransferase(Plasmodium falciparum)
Albert Einstein College of Medicine

LigandPNGBDBM214786(OPRT inhibitor, 9)
Affinity DataKi:  270nM ΔG°:  -37.5kJ/molepH: 8.0 T: 2°CAssay Description:Inhibition constants (Ki, equivalent to Kd for competitive inhibitors) were measured at 25 °C by adding purified OPRT enzymes (25 nM for PfOPRT a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOrotate phosphoribosyltransferase(Plasmodium falciparum)
Albert Einstein College of Medicine

LigandPNGBDBM214784(OPRT inhibitor, 7)
Affinity DataKi:  270nM ΔG°:  -37.5kJ/molepH: 8.0 T: 2°CAssay Description:Inhibition constants (Ki, equivalent to Kd for competitive inhibitors) were measured at 25 °C by adding purified OPRT enzymes (25 nM for PfOPRT a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUridine 5'-monophosphate synthase(Homo sapiens (Human))
Albert Einstein College of Medicine

LigandPNGBDBM214787(OPRT inhibitor, 10)
Affinity DataKi:  290nM ΔG°:  -37.3kJ/molepH: 8.0 T: 2°CAssay Description:Inhibition constants (Ki, equivalent to Kd for competitive inhibitors) were measured at 25 °C by adding purified OPRT enzymes (25 nM for PfOPRT a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOrotate phosphoribosyltransferase(Plasmodium falciparum)
Albert Einstein College of Medicine

LigandPNGBDBM214782(OPRT inhibitor, 5)
Affinity DataKi:  300nM ΔG°:  -37.2kJ/molepH: 8.0 T: 2°CAssay Description:Inhibition constants (Ki, equivalent to Kd for competitive inhibitors) were measured at 25 °C by adding purified OPRT enzymes (25 nM for PfOPRT a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOrotate phosphoribosyltransferase(Plasmodium falciparum)
Albert Einstein College of Medicine

LigandPNGBDBM214780(OPRT inhibitor, 3)
Affinity DataKi:  350nM ΔG°:  -36.8kJ/molepH: 8.0 T: 2°CAssay Description:Inhibition constants (Ki, equivalent to Kd for competitive inhibitors) were measured at 25 °C by adding purified OPRT enzymes (25 nM for PfOPRT a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOrotate phosphoribosyltransferase(Plasmodium falciparum)
Albert Einstein College of Medicine

LigandPNGBDBM214783(OPRT inhibitor, 6)
Affinity DataKi:  350nM ΔG°:  -36.8kJ/molepH: 8.0 T: 2°CAssay Description:Inhibition constants (Ki, equivalent to Kd for competitive inhibitors) were measured at 25 °C by adding purified OPRT enzymes (25 nM for PfOPRT a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUridine 5'-monophosphate synthase(Homo sapiens (Human))
Albert Einstein College of Medicine

LigandPNGBDBM214782(OPRT inhibitor, 5)
Affinity DataKi:  360nM ΔG°:  -36.8kJ/molepH: 8.0 T: 2°CAssay Description:Inhibition constants (Ki, equivalent to Kd for competitive inhibitors) were measured at 25 °C by adding purified OPRT enzymes (25 nM for PfOPRT a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOrotate phosphoribosyltransferase(Plasmodium falciparum)
Albert Einstein College of Medicine

LigandPNGBDBM214781(OPRT inhibitor, 4)
Affinity DataKi:  370nM ΔG°:  -36.7kJ/molepH: 8.0 T: 2°CAssay Description:Inhibition constants (Ki, equivalent to Kd for competitive inhibitors) were measured at 25 °C by adding purified OPRT enzymes (25 nM for PfOPRT a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOrotate phosphoribosyltransferase(Plasmodium falciparum)
Albert Einstein College of Medicine

LigandPNGBDBM214790(OPRT inhibitor, 13)
Affinity DataKi:  470nM ΔG°:  -36.1kJ/molepH: 8.0 T: 2°CAssay Description:Inhibition constants (Ki, equivalent to Kd for competitive inhibitors) were measured at 25 °C by adding purified OPRT enzymes (25 nM for PfOPRT a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrotate phosphoribosyltransferase(Plasmodium falciparum)
Albert Einstein College of Medicine

LigandPNGBDBM214793(OPRT inhibitor, 16)
Affinity DataKi:  480nM ΔG°:  -36.1kJ/molepH: 8.0 T: 2°CAssay Description:Inhibition constants (Ki, equivalent to Kd for competitive inhibitors) were measured at 25 °C by adding purified OPRT enzymes (25 nM for PfOPRT a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOrotate phosphoribosyltransferase(Plasmodium falciparum)
Albert Einstein College of Medicine

LigandPNGBDBM214792(OPRT inhibitor, 15)
Affinity DataKi:  500nM ΔG°:  -36.0kJ/molepH: 8.0 T: 2°CAssay Description:Inhibition constants (Ki, equivalent to Kd for competitive inhibitors) were measured at 25 °C by adding purified OPRT enzymes (25 nM for PfOPRT a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOrotate phosphoribosyltransferase(Plasmodium falciparum)
Albert Einstein College of Medicine

LigandPNGBDBM214796(OPRT inhibitor, 19)
Affinity DataKi:  500nM ΔG°:  -36.0kJ/molepH: 8.0 T: 2°CAssay Description:Inhibition constants (Ki, equivalent to Kd for competitive inhibitors) were measured at 25 °C by adding purified OPRT enzymes (25 nM for PfOPRT a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOrotate phosphoribosyltransferase(Plasmodium falciparum)
Albert Einstein College of Medicine

LigandPNGBDBM214797(OPRT inhibitor, 20)
Affinity DataKi:  510nM ΔG°:  -35.9kJ/molepH: 8.0 T: 2°CAssay Description:Inhibition constants (Ki, equivalent to Kd for competitive inhibitors) were measured at 25 °C by adding purified OPRT enzymes (25 nM for PfOPRT a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUridine 5'-monophosphate synthase(Homo sapiens (Human))
Albert Einstein College of Medicine

LigandPNGBDBM214788(OPRT inhibitor, 11)
Affinity DataKi:  520nM ΔG°:  -35.9kJ/molepH: 8.0 T: 2°CAssay Description:Inhibition constants (Ki, equivalent to Kd for competitive inhibitors) were measured at 25 °C by adding purified OPRT enzymes (25 nM for PfOPRT a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUridine 5'-monophosphate synthase(Homo sapiens (Human))
Albert Einstein College of Medicine

LigandPNGBDBM214780(OPRT inhibitor, 3)
Affinity DataKi:  530nM ΔG°:  -35.8kJ/molepH: 8.0 T: 2°CAssay Description:Inhibition constants (Ki, equivalent to Kd for competitive inhibitors) were measured at 25 °C by adding purified OPRT enzymes (25 nM for PfOPRT a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOrotate phosphoribosyltransferase(Plasmodium falciparum)
Albert Einstein College of Medicine

LigandPNGBDBM214795(OPRT inhibitor, 18)
Affinity DataKi:  570nM ΔG°:  -35.6kJ/molepH: 8.0 T: 2°CAssay Description:Inhibition constants (Ki, equivalent to Kd for competitive inhibitors) were measured at 25 °C by adding purified OPRT enzymes (25 nM for PfOPRT a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOrotate phosphoribosyltransferase(Plasmodium falciparum)
Albert Einstein College of Medicine

LigandPNGBDBM214787(OPRT inhibitor, 10)
Affinity DataKi:  690nM ΔG°:  -35.2kJ/molepH: 8.0 T: 2°CAssay Description:Inhibition constants (Ki, equivalent to Kd for competitive inhibitors) were measured at 25 °C by adding purified OPRT enzymes (25 nM for PfOPRT a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOrotate phosphoribosyltransferase(Plasmodium falciparum)
Albert Einstein College of Medicine

LigandPNGBDBM214794(OPRT inhibitor, 17)
Affinity DataKi:  750nM ΔG°:  -35.0kJ/molepH: 8.0 T: 2°CAssay Description:Inhibition constants (Ki, equivalent to Kd for competitive inhibitors) were measured at 25 °C by adding purified OPRT enzymes (25 nM for PfOPRT a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOrotate phosphoribosyltransferase(Plasmodium falciparum)
Albert Einstein College of Medicine

LigandPNGBDBM214788(OPRT inhibitor, 11)
Affinity DataKi:  1.30E+3nM ΔG°:  -33.6kJ/molepH: 8.0 T: 2°CAssay Description:Inhibition constants (Ki, equivalent to Kd for competitive inhibitors) were measured at 25 °C by adding purified OPRT enzymes (25 nM for PfOPRT a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUridine 5'-monophosphate synthase(Homo sapiens (Human))
Albert Einstein College of Medicine

LigandPNGBDBM214789(OPRT inhibitor, 12)
Affinity DataKi:  4.30E+3nM ΔG°:  -30.6kJ/molepH: 8.0 T: 2°CAssay Description:Inhibition constants (Ki, equivalent to Kd for competitive inhibitors) were measured at 25 °C by adding purified OPRT enzymes (25 nM for PfOPRT a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOrotate phosphoribosyltransferase(Plasmodium falciparum)
Albert Einstein College of Medicine

LigandPNGBDBM214789(OPRT inhibitor, 12)
Affinity DataKi:  1.55E+4nM ΔG°:  -27.5kJ/molepH: 8.0 T: 2°CAssay Description:Inhibition constants (Ki, equivalent to Kd for competitive inhibitors) were measured at 25 °C by adding purified OPRT enzymes (25 nM for PfOPRT a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Victoria University Of Wellington

Curated by ChEMBL
LigandPNGBDBM50281297(CHEMBL4170114)
Affinity DataIC50:  8nMAssay Description:Inhibition of G9a (unknown origin) using biotinylated histone monomethyl-H3K9 peptide by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA (cytosine-5)-methyltransferase 1(Homo sapiens (Human))
Victoria University Of Wellington

Curated by ChEMBL
LigandPNGBDBM50281297(CHEMBL4170114)
Affinity DataIC50:  382nMAssay Description:Inhibition of DNMT1 (unknown origin) using biotinylated histone monomethyl-H3K9 peptide by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2C(RAT)
Emory University

Curated by ChEMBL
LigandPNGBDBM50436060(CHEMBL2397100 | US10273214, Example 1390)
Affinity DataEC50:  5.01E+3nMAssay Description:Positive allosteric modulation of recombinant rat GluN1a/GluN2C receptor expressed in Xenopus laevis oocytes assessed as increase in glycine/L-glutam...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2D(RAT)
Emory University

Curated by ChEMBL
LigandPNGBDBM50545719(CHEMBL4635888)
Affinity DataEC50:  3.16E+3nMAssay Description:Positive allosteric modulation of recombinant rat GluN1a/GluN2D receptor expressed in Xenopus laevis oocytes assessed as increase in glycine/L-glutam...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2C(RAT)
Emory University

Curated by ChEMBL
LigandPNGBDBM50436102(CHEMBL2397256 | US10273214, Example 1180-26)
Affinity DataEC50:  1.26E+3nMAssay Description:Positive allosteric modulation of recombinant rat GluN1a/GluN2C receptor expressed in Xenopus laevis oocytes assessed as increase in glycine/L-glutam...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2C(RAT)
Emory University

Curated by ChEMBL
LigandPNGBDBM50545697(CHEMBL4649350)
Affinity DataEC50:  2.00E+3nMAssay Description:Positive allosteric modulation of recombinant rat GluN1a/GluN2C receptor expressed in Xenopus laevis oocytes assessed as increase in glycine/L-glutam...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2C(RAT)
Emory University

Curated by ChEMBL
LigandPNGBDBM50238337(CHEMBL4095932)
Affinity DataEC50:  2.00E+3nMAssay Description:Positive allosteric modulation of recombinant rat GluN1a/GluN2C receptor expressed in Xenopus laevis oocytes assessed as increase in glycine/L-glutam...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2C(RAT)
Emory University

Curated by ChEMBL
LigandPNGBDBM50545698(CHEMBL4637429)
Affinity DataEC50:  398nMAssay Description:Positive allosteric modulation of recombinant rat GluN1a/GluN2C receptor expressed in Xenopus laevis oocytes assessed as increase in glycine/L-glutam...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2C(RAT)
Emory University

Curated by ChEMBL
LigandPNGBDBM50238338(CHEMBL4068612)
Affinity DataEC50:  1.00E+3nMAssay Description:Positive allosteric modulation of recombinant rat GluN1a/GluN2C receptor expressed in Xenopus laevis oocytes assessed as increase in glycine/L-glutam...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2C(RAT)
Emory University

Curated by ChEMBL
LigandPNGBDBM50545699(CHEMBL4636021)
Affinity DataEC50:  398nMAssay Description:Positive allosteric modulation of recombinant rat GluN1a/GluN2C receptor expressed in Xenopus laevis oocytes assessed as increase in glycine/L-glutam...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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