Affinity DataKi: 0.900nMAssay Description:Tested for inhibition of adenosine A1 receptor binding to rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Binding affinity for adenosine A3 receptor as inhibition of [125I]-AB-MECA binding to human receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Tested for inhibition of adenosine A1 receptor binding to rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]-R-PIA from adenosine A1 receptor of Wistar rat forebrainMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Displacement of [3H]NAMH from human histamine H3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Tested for inhibition of adenosine A1 receptor binding to rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Tested for inhibition of adenosine A1 receptor binding to rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Inhibition of human H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Displacement of [3H]NAMH from human histamine H3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Displacement of [3H]NAMH from human histamine H3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.70nMAssay Description:Antagonist activity at histamine H3 receptor in rat cortical membraneMore data for this Ligand-Target Pair
Affinity DataKi: 2.80nMAssay Description:Displacement of [3H]NAMH from human histamine H3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.10nMAssay Description:Displacement of [3H]-R-PIA from adenosine A1 receptor of Wistar rat forebrainMore data for this Ligand-Target Pair
Affinity DataKi: 3.60nMAssay Description:Displacement of [3H]-R-PIA from adenosine A1 receptor of Wistar rat forebrainMore data for this Ligand-Target Pair
Affinity DataKi: 3.60nMAssay Description:Tested for inhibition of adenosine A1 receptor binding to rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 3.90nMAssay Description:Displacement of [3H]NAMH from human histamine H3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Tested for inhibition of adenosine A1 receptor binding to rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 4.20nMAssay Description:Tested for inhibition of adenosine A1 receptor binding to rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 4.30nMAssay Description:Binding affinity to human adenosine A2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 4.70nMAssay Description:Displacement of [3H]-R-PIA from adenosine A1 receptor of Wistar rat forebrainMore data for this Ligand-Target Pair
Affinity DataKi: 4.80nMAssay Description:Displacement of [3H]NAMH from human histamine H3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 6.10nMAssay Description:Tested for inhibition of adenosine A1 receptor binding to rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:Displacement of [3H]NAMH from rat histamine H3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 6.90nMAssay Description:Displacement of [3H]NAMH from human histamine H3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 7.20nMAssay Description:Displacement of [3H]NAMH from rat histamine H3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 7.60nMAssay Description:Displacement of [3H]NAMH from rat histamine H3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 7.80nMAssay Description:Binding affinity for adenosine A3 receptor as inhibition of [125I]-AB-MECA binding to human receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 7.90nMAssay Description:Displacement of [3H]NAMH from rat histamine H3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 8.10nMAssay Description:Binding affinity to human adenosine A2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 8.5nMAssay Description:Displacement of [3H]NAMH from rat histamine H3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 8.70nMAssay Description:Displacement of [3H]NAMH from human histamine H3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 9.10nMAssay Description:Displacement of [3H]NAMH from human histamine H3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 9.20nMAssay Description:Displacement of [3H]NAMH from human histamine H3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 9.30nMAssay Description:Tested for inhibition of adenosine A1 receptor binding to rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 9.30nMAssay Description:Tested for inhibition of adenosine A1 receptor binding to rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 9.90nMAssay Description:Tested for inhibition of adenosine A1 receptor binding to rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Tested for inhibition of adenosine A1 receptor binding to rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Tested for inhibition of adenosine A1 receptor binding to rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Displacement of [3H]NAMH from rat histamine H3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Binding affinity to human adenosine A2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Displacement of [3H]-CGS- 21680 from adenosine A2A receptor of rat striatal tissueMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Tested for inhibition of adenosine A1 receptor binding to rat brainMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Novo Nordisk
Curated by ChEMBL
Novo Nordisk
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:In vitro inhibition of [3H]GABA uptake at the Sodium- and chloride-dependent GABA transporter 1 (GAT-1) uptake site in rat brain synaptosomesMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Novo Nordisk
Curated by ChEMBL
Novo Nordisk
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:In vitro inhibition of [3H]GABA uptake at the Sodium- and chloride-dependent GABA transporter 1 (GAT-1) uptake site in rat brain synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Displacement of [3H]NAMH from rat histamine H3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Novo Nordisk
Curated by ChEMBL
Novo Nordisk
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:In vitro inhibition of [3H]GABA uptake at the Sodium- and chloride-dependent GABA transporter 1 (GAT-1) uptake site in rat brain synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Tested for inhibition of adenosine A1 receptor binding to rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Tested for inhibition of adenosine A1 receptor binding to rat brainMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Novo Nordisk
Curated by ChEMBL
Novo Nordisk
Curated by ChEMBL
Affinity DataKi: 14nMAssay Description:In vitro inhibition of [3H]GABA uptake at the Sodium- and chloride-dependent GABA transporter 1 (GAT-1) uptake site in rat brain synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Binding affinity to human adenosine A1 receptorMore data for this Ligand-Target Pair