Compile Data Set for Download or QSAR
maximum 50k data
Found 394 with Last Name = 'fernández' and Initial = 'm'
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Pavia

Curated by ChEMBL
LigandPNGBDBM50357453(CHEMBL1917719)
Affinity DataKi:  0.700nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Pavia

Curated by ChEMBL
LigandPNGBDBM50357441(CHEMBL1917705)
Affinity DataKi:  0.860nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Pavia

Curated by ChEMBL
LigandPNGBDBM50357440(CHEMBL1917704)
Affinity DataKi:  0.970nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Pavia

Curated by ChEMBL
LigandPNGBDBM50357430(CHEMBL1917711)
Affinity DataKi:  1.07nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Pavia

Curated by ChEMBL
LigandPNGBDBM50198061((E)-N,N-dimethyl-3-(biphen-4-yl)but-2-en-1-ylamine...)
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Pavia

Curated by ChEMBL
LigandPNGBDBM50357431(CHEMBL1917712)
Affinity DataKi:  4.14nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Pavia

Curated by ChEMBL
LigandPNGBDBM50357429(CHEMBL1917702)
Affinity DataKi:  5.25nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Pavia

Curated by ChEMBL
LigandPNGBDBM50198065(4(E)-N-Benzyl-3-(biphenyl-4-yl)-N-methylbut-2-en-1...)
Affinity DataKi:  6.32nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Pavia

Curated by ChEMBL
LigandPNGBDBM50357446(CHEMBL1917710)
Affinity DataKi:  7.02nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Pavia

Curated by ChEMBL
LigandPNGBDBM50357447(CHEMBL1917713)
Affinity DataKi:  7.70nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Pavia

Curated by ChEMBL
LigandPNGBDBM50198058((E)-N-benzyl-N-methyl-3-(naphthalen-2-yl)but-2-en-...)
Affinity DataKi:  7.88nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Pavia

Curated by ChEMBL
LigandPNGBDBM50357448(CHEMBL1917714)
Affinity DataKi:  9.60nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Instituto De Qu£Mica M£Dica

Curated by ChEMBL
LigandPNGBDBM50380548(CHEMBL2019055)
Affinity DataKi:  9.70nMAssay Description:Competitive inhibition of human recombinant BChE using panvera peptide as substrate preincubated for 60 mins before substrate addition by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Pavia

Curated by ChEMBL
LigandPNGBDBM50357432(CHEMBL1917703)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Pavia

Curated by ChEMBL
LigandPNGBDBM50357449(CHEMBL1917715)
Affinity DataKi:  11.6nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Pavia

Curated by ChEMBL
LigandPNGBDBM50357443(CHEMBL1917707)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Pavia

Curated by ChEMBL
LigandPNGBDBM50198068((E)-N,N-dimethyl-3-(naphthalen-2-yl)but-2-en-1-ami...)
Affinity DataKi:  19.8nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Sus scrofa (pig))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50326300(3-(Benzyloxycarbonyl-L-leucylamino)-N-(3-(6-amino-...)
Affinity DataKi:  23nMAssay Description:Inhibition of porcine erythrocyte calpain 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Pavia

Curated by ChEMBL
LigandPNGBDBM50357445(CHEMBL1917709)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Sus scrofa (pig))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50326298(3-(Benzyloxycarbonyl-L-leucylamino)-N-(3-(6-amino-...)
Affinity DataKi:  41nMAssay Description:Inhibition of porcine erythrocyte calpain 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-2 catalytic subunit(Sus scrofa)
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50084684(CHEMBL333627 | {3-Methyl-1-[1-(3-morpholin-4-yl-pr...)
Affinity DataKi:  41nMAssay Description:Inhibition of porcine kidney calpain 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Sus scrofa (pig))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50326303(3-(Benzyloxycarbonyl-L-leucylamino)-N-(3-(6-amino-...)
Affinity DataKi:  53nMAssay Description:Inhibition of porcine erythrocyte calpain 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Sus scrofa (pig))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50326304(3-(Benzyloxycarbonyl-L-leucylamino)-N-(3-(6-amino-...)
Affinity DataKi:  55nMAssay Description:Inhibition of porcine erythrocyte calpain 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-2 catalytic subunit(Sus scrofa)
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50326304(3-(Benzyloxycarbonyl-L-leucylamino)-N-(3-(6-amino-...)
Affinity DataKi:  68nMAssay Description:Inhibition of porcine kidney calpain 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-2 catalytic subunit(Sus scrofa)
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50326303(3-(Benzyloxycarbonyl-L-leucylamino)-N-(3-(6-amino-...)
Affinity DataKi:  70nMAssay Description:Inhibition of porcine kidney calpain 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-2 catalytic subunit(Sus scrofa)
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50326300(3-(Benzyloxycarbonyl-L-leucylamino)-N-(3-(6-amino-...)
Affinity DataKi:  77nMAssay Description:Inhibition of porcine kidney calpain 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Pavia

Curated by ChEMBL
LigandPNGBDBM50357444(CHEMBL1917708)
Affinity DataKi:  91nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Pavia

Curated by ChEMBL
LigandPNGBDBM50357428(CHEMBL1917701)
Affinity DataKi:  92nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Pavia

Curated by ChEMBL
LigandPNGBDBM50357429(CHEMBL1917702)
Affinity DataKi:  92nMAssay Description:Displacement of [3H]-DAMGO from mu opioid receptor in guinea pig brain membrane after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Pavia

Curated by ChEMBL
LigandPNGBDBM50357428(CHEMBL1917701)
Affinity DataKi:  119nMAssay Description:Displacement of [3H]-DAMGO from mu opioid receptor in guinea pig brain membrane after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Pavia

Curated by ChEMBL
LigandPNGBDBM50357431(CHEMBL1917712)
Affinity DataKi:  149nMAssay Description:Displacement of [3H]-DAMGO from mu opioid receptor in guinea pig brain membrane after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Sus scrofa (pig))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50084684(CHEMBL333627 | {3-Methyl-1-[1-(3-morpholin-4-yl-pr...)
Affinity DataKi:  150nMAssay Description:Inhibition of porcine erythrocyte calpain 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Pavia

Curated by ChEMBL
LigandPNGBDBM50357430(CHEMBL1917711)
Affinity DataKi:  152nMAssay Description:Displacement of [3H]-DAMGO from mu opioid receptor in guinea pig brain membrane after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Pavia

Curated by ChEMBL
LigandPNGBDBM50357431(CHEMBL1917712)
Affinity DataKi:  157nMAssay Description:Displacement of [3H]-U69593 from kappa opioid receptor in guinea pig brain membrane after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Sus scrofa (pig))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50326299(3-(Benzyloxycarbonyl-L-leucylamino)-N-(3-(4-amino-...)
Affinity DataKi:  165nMAssay Description:Inhibition of porcine erythrocyte calpain 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Pavia

Curated by ChEMBL
LigandPNGBDBM50357430(CHEMBL1917711)
Affinity DataKi:  189nMAssay Description:Displacement of [3H]-U69593 from kappa opioid receptor in guinea pig brain membrane after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Pavia

Curated by ChEMBL
LigandPNGBDBM50357429(CHEMBL1917702)
Affinity DataKi:  197nMAssay Description:Displacement of [3H]-U69593 from kappa opioid receptor in guinea pig brain membrane after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-2 catalytic subunit(Sus scrofa)
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50326298(3-(Benzyloxycarbonyl-L-leucylamino)-N-(3-(6-amino-...)
Affinity DataKi:  209nMAssay Description:Inhibition of porcine kidney calpain 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Pavia

Curated by ChEMBL
LigandPNGBDBM50357447(CHEMBL1917713)
Affinity DataKi:  214nMAssay Description:Displacement of [3H]-U69593 from kappa opioid receptor in guinea pig brain membrane after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Sus scrofa (pig))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50326306(3-(Benzyloxycarbonyl-L-leucylamino)-N-(3-(dimethyl...)
Affinity DataKi:  226nMAssay Description:Inhibition of porcine erythrocyte calpain 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-2 catalytic subunit(Sus scrofa)
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50326302(3-(Benzyloxycarbonyl-L-leucylamino)-N-(3-(4-methyl...)
Affinity DataKi:  286nMAssay Description:Inhibition of porcine kidney calpain 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Pavia

Curated by ChEMBL
LigandPNGBDBM50357432(CHEMBL1917703)
Affinity DataKi:  301nMAssay Description:Displacement of [3H]-U69593 from kappa opioid receptor in guinea pig brain membrane after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Pavia

Curated by ChEMBL
LigandPNGBDBM50357428(CHEMBL1917701)
Affinity DataKi:  438nMAssay Description:Displacement of [3H]-U69593 from kappa opioid receptor in guinea pig brain membrane after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-2 catalytic subunit(Sus scrofa)
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50326301(3-(Benzyloxycarbonyl-L-leucylamino)-N-(3-(4-amino-...)
Affinity DataKi:  438nMAssay Description:Inhibition of porcine kidney calpain 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50326301(3-(Benzyloxycarbonyl-L-leucylamino)-N-(3-(4-amino-...)
Affinity DataKi:  440nMAssay Description:Inhibition of human liver cathepsin BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Pavia

Curated by ChEMBL
LigandPNGBDBM50357442(CHEMBL1917706)
Affinity DataKi:  459nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Sus scrofa (pig))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50326301(3-(Benzyloxycarbonyl-L-leucylamino)-N-(3-(4-amino-...)
Affinity DataKi:  480nMAssay Description:Inhibition of porcine erythrocyte calpain 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Instituto De Qu£Mica M£Dica

Curated by ChEMBL
LigandPNGBDBM50380542(CHEMBL2019037)
Affinity DataKi:  620nMAssay Description:Competitive inhibition of human recombinant BChE using panvera peptide as substrate preincubated for 60 mins before substrate addition by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Sus scrofa (pig))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50326302(3-(Benzyloxycarbonyl-L-leucylamino)-N-(3-(4-methyl...)
Affinity DataKi:  640nMAssay Description:Inhibition of porcine erythrocyte calpain 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Sus scrofa (pig))
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50326305(3-(Benzyloxycarbonyl-L-leucylamino)-N-(2-(dimethyl...)
Affinity DataKi:  711nMAssay Description:Inhibition of porcine erythrocyte calpain 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 394 total ) | Next | Last >>
Jump to: