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Found 343 with Last Name = 'garnier' and Initial = 'm'
TargetIsoform 1 of Calcitonin receptor (1)(Homo sapiens (Human))
Rutgers University

Curated by ChEMBL
LigandPNGBDBM50110268(CHEMBL2369895 | CSNLSTCVLGKLSQELc[DKLQK]YPRTNTGSGT...)
Affinity DataKi:  0.0230nMAssay Description:Inhibition of [125I]-salmon calcitonin (sCT) binding to human calcitonin receptor I1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoform 1 of Calcitonin receptor (1)(Homo sapiens (Human))
Rutgers University

Curated by ChEMBL
LigandPNGBDBM50024170(CHEMBL2369912)
Affinity DataKi:  0.0500nMAssay Description:Inhibition of [125I]-salmon calcitonin (sCT) binding to human calcitonin receptor I1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoform 1 of Calcitonin receptor (1)(Homo sapiens (Human))
Rutgers University

Curated by ChEMBL
LigandPNGBDBM50110272(CHEMBL2369907 | CSNLSTCVLGKLSQELc[DKLHK]YPRTNTGSGT...)
Affinity DataKi:  0.0510nMAssay Description:Inhibition of [125I]-salmon calcitonin (sCT) binding to human calcitonin receptor I1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoform 1 of Calcitonin receptor (1)(Homo sapiens (Human))
Rutgers University

Curated by ChEMBL
LigandPNGBDBM50110275(CGNLSTCBLGTYTQDF[DKFHO]YPQTAIGVGAP-amide | CHEMBL2...)
Affinity DataKi:  0.0690nMAssay Description:Inhibition of [125I]-salmon calcitonin (sCT) binding to human calcitonin receptor I1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoform 1 of Calcitonin receptor (1)(Homo sapiens (Human))
Rutgers University

Curated by ChEMBL
LigandPNGBDBM50110265(CHEMBL2369886 | CSNLSTCVLGKLSQELc[DKLHO]YPRTNTGSGT...)
Affinity DataKi:  0.0690nMAssay Description:Inhibition of [125I]-salmon calcitonin (sCT) binding to human calcitonin receptor I1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoform 1 of Calcitonin receptor (1)(Homo sapiens (Human))
Rutgers University

Curated by ChEMBL
LigandPNGBDBM50110273(CGNLSTCMLGTYTQDFc[DKFHK]FPQTAIGVGAP-amide | CHEMBL...)
Affinity DataKi:  0.560nMAssay Description:Inhibition of [125I]-salmon calcitonin (sCT) binding to human calcitonin receptor I1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoform 1 of Calcitonin receptor (1)(Homo sapiens (Human))
Rutgers University

Curated by ChEMBL
LigandPNGBDBM50110267(CGNLSTCBLGTYTQDFNKFHZYPQTAIGVGAP-amide | CHEMBL236...)
Affinity DataKi:  5.30nMAssay Description:Inhibition of [125I]-salmon calcitonin (sCT) binding to human calcitonin receptor I1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoform 1 of Calcitonin receptor (1)(Homo sapiens (Human))
Rutgers University

Curated by ChEMBL
LigandPNGBDBM50110271(CGNLSTCMLGTYTQDFNKFHTFPQTAIGVGAP-amide | CHEMBL236...)
Affinity DataKi:  43nMAssay Description:Inhibition of [125I]-salmon calcitonin (sCT) binding to human calcitonin receptor I1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50417543(CHEMBL1632210)
Affinity DataKi:  50.1nMAssay Description:Displacement of [3H]dofetilide from human ERG by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoform 1 of Calcitonin receptor (1)(Homo sapiens (Human))
Rutgers University

Curated by ChEMBL
LigandPNGBDBM50024171(CHEMBL2369899)
Affinity DataKi:  195nMAssay Description:Inhibition of [125I]-salmon calcitonin (sCT) binding to human calcitonin receptor I1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50417549(CHEMBL1632223)
Affinity DataKi:  316nMAssay Description:Displacement of [3H]dofetilide from human ERG by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50417544(CHEMBL1632218)
Affinity DataKi:  316nMAssay Description:Displacement of [3H]dofetilide from human ERG by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoform 1 of Calcitonin receptor (1)(Homo sapiens (Human))
Rutgers University

Curated by ChEMBL
LigandPNGBDBM50110266(CGNLSTCMLGTYTQDFNKPHTFPQTAIGVGAP-amide | CHEMBL236...)
Affinity DataKi:  400nMAssay Description:Inhibition of [125I]-salmon calcitonin (sCT) binding to human calcitonin receptor I1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50417545(CHEMBL1631535)
Affinity DataKi:  501nMAssay Description:Displacement of [3H]dofetilide from human ERG by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50417546(CHEMBL1632220)
Affinity DataKi:  631nMAssay Description:Displacement of [3H]dofetilide from human ERG by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoform 1 of Calcitonin receptor (1)(Homo sapiens (Human))
Rutgers University

Curated by ChEMBL
LigandPNGBDBM50422415(CHEMBL2304022)
Affinity DataKi:  1.23E+3nMAssay Description:Inhibition of [125I]-salmon calcitonin (sCT) binding to human calcitonin receptor I1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50417548(CHEMBL1631542)
Affinity DataKi:  2.00E+3nMAssay Description:Displacement of [3H]dofetilide from human ERG by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoform 1 of Calcitonin receptor (1)(Homo sapiens (Human))
Rutgers University

Curated by ChEMBL
LigandPNGBDBM50110276(CGNLSTCMLGTYTQDFNPKHTFPQTAIGVGAP-amide | CHEMBL236...)
Affinity DataKi: >2.50E+3nMAssay Description:Inhibition of [125I]-salmon calcitonin (sCT) binding to human calcitonin receptor I1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoform 1 of Calcitonin receptor (1)(Homo sapiens (Human))
Rutgers University

Curated by ChEMBL
LigandPNGBDBM50110274(CGNLSTCMLGTYTQDFNPGHTFPQTAIGVGAP-amide | CHEMBL236...)
Affinity DataKi:  2.57E+3nMAssay Description:Inhibition of [125I]-salmon calcitonin (sCT) binding to human calcitonin receptor I1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50417547(CHEMBL1632206)
Affinity DataKi:  3.98E+3nMAssay Description:Displacement of [3H]dofetilide from human ERG by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50333015(1-(3-{2-[4-(2-Methyl-5-quinolinyl)-1-piperazinyl]e...)
Affinity DataKi:  1.26E+4nMAssay Description:Displacement of [3H]dofetilide from human ERG by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalcitonin receptor(Rattus norvegicus)
Rutgers University

Curated by ChEMBL
LigandPNGBDBM50024170(CHEMBL2369912)
Affinity DataIC50:  0.180nMAssay Description:Displacement of [125I]-salmon calcitonin (sCT) from calcitonin receptor of rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalcitonin receptor(Rattus norvegicus)
Rutgers University

Curated by ChEMBL
LigandPNGBDBM50110265(CHEMBL2369886 | CSNLSTCVLGKLSQELc[DKLHO]YPRTNTGSGT...)
Affinity DataIC50:  0.249nMAssay Description:Displacement of [125I]-salmon calcitonin (sCT) from calcitonin receptor of rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalcitonin receptor(Rattus norvegicus)
Rutgers University

Curated by ChEMBL
LigandPNGBDBM50110268(CHEMBL2369895 | CSNLSTCVLGKLSQELc[DKLQK]YPRTNTGSGT...)
Affinity DataIC50:  0.326nMAssay Description:Displacement of [125I]-salmon calcitonin (sCT) from calcitonin receptor of rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalcitonin receptor(Rattus norvegicus)
Rutgers University

Curated by ChEMBL
LigandPNGBDBM50110272(CHEMBL2369907 | CSNLSTCVLGKLSQELc[DKLHK]YPRTNTGSGT...)
Affinity DataIC50:  0.377nMAssay Description:Displacement of [125I]-salmon calcitonin (sCT) from calcitonin receptor of rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalcitonin receptor(Rattus norvegicus)
Rutgers University

Curated by ChEMBL
LigandPNGBDBM50110275(CGNLSTCBLGTYTQDF[DKFHO]YPQTAIGVGAP-amide | CHEMBL2...)
Affinity DataIC50:  0.408nMAssay Description:Displacement of [125I]-salmon calcitonin (sCT) from calcitonin receptor of rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter and Eliza Hall Institute of Medical Research

Curated by ChEMBL
LigandPNGBDBM313798(US10167292, Example 42)
Affinity DataIC50:  2nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter and Eliza Hall Institute of Medical Research

Curated by ChEMBL
LigandPNGBDBM313807(US10167292, Example 51B)
Affinity DataIC50:  2nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Walter and Eliza Hall Institute of Medical Research

Curated by ChEMBL
LigandPNGBDBM313791(US10167292, Example 35)
Affinity DataIC50:  3nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter and Eliza Hall Institute of Medical Research

Curated by ChEMBL
LigandPNGBDBM313807(US10167292, Example 51B)
Affinity DataIC50:  3nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Walter and Eliza Hall Institute of Medical Research

Curated by ChEMBL
LigandPNGBDBM313789(US10167292, Example 33)
Affinity DataIC50:  4nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCalcitonin receptor(Rattus norvegicus)
Rutgers University

Curated by ChEMBL
LigandPNGBDBM50110273(CGNLSTCMLGTYTQDFc[DKFHK]FPQTAIGVGAP-amide | CHEMBL...)
Affinity DataIC50:  5.40nMAssay Description:Displacement of [125I]-salmon calcitonin (sCT) from calcitonin receptor of rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter and Eliza Hall Institute of Medical Research

Curated by ChEMBL
LigandPNGBDBM313791(US10167292, Example 35)
Affinity DataIC50:  6nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter and Eliza Hall Institute of Medical Research

Curated by ChEMBL
LigandPNGBDBM313798(US10167292, Example 42)
Affinity DataIC50:  6nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Walter and Eliza Hall Institute of Medical Research

Curated by ChEMBL
LigandPNGBDBM313807(US10167292, Example 51B)
Affinity DataIC50:  6nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter and Eliza Hall Institute of Medical Research

Curated by ChEMBL
LigandPNGBDBM313774(US10167292, Example 8)
Affinity DataIC50:  6nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter and Eliza Hall Institute of Medical Research

Curated by ChEMBL
LigandPNGBDBM313797(US10167292, Example 41)
Affinity DataIC50:  7nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter and Eliza Hall Institute of Medical Research

Curated by ChEMBL
LigandPNGBDBM313775(US10167292, Example 10)
Affinity DataIC50:  7nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Walter and Eliza Hall Institute of Medical Research

Curated by ChEMBL
LigandPNGBDBM313807(US10167292, Example 51B)
Affinity DataIC50:  7nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter and Eliza Hall Institute of Medical Research

Curated by ChEMBL
LigandPNGBDBM313779(US10167292, Example 16)
Affinity DataIC50:  7nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter and Eliza Hall Institute of Medical Research

Curated by ChEMBL
LigandPNGBDBM313773(US10167292, Example 7)
Affinity DataIC50:  7nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Walter and Eliza Hall Institute of Medical Research

Curated by ChEMBL
LigandPNGBDBM313774(US10167292, Example 8)
Affinity DataIC50:  9nMAssay Description:Inhibition of human His-tagged Brd3 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter and Eliza Hall Institute of Medical Research

Curated by ChEMBL
LigandPNGBDBM313778(US10167292, Example 13)
Affinity DataIC50:  10nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter and Eliza Hall Institute of Medical Research

Curated by ChEMBL
LigandPNGBDBM313796(US10167292, Example 40)
Affinity DataIC50:  10nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Walter and Eliza Hall Institute of Medical Research

Curated by ChEMBL
LigandPNGBDBM313775(US10167292, Example 10)
Affinity DataIC50:  10nMAssay Description:Inhibition of human His-tagged Brd3 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter and Eliza Hall Institute of Medical Research

Curated by ChEMBL
LigandPNGBDBM313791(US10167292, Example 35)
Affinity DataIC50:  10nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Walter and Eliza Hall Institute of Medical Research

Curated by ChEMBL
LigandPNGBDBM313773(US10167292, Example 7)
Affinity DataIC50:  10nMAssay Description:Inhibition of human His-tagged Brd3 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Walter and Eliza Hall Institute of Medical Research

Curated by ChEMBL
LigandPNGBDBM313779(US10167292, Example 16)
Affinity DataIC50:  11nMAssay Description:Inhibition of human His-tagged Brd3 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter and Eliza Hall Institute of Medical Research

Curated by ChEMBL
LigandPNGBDBM313803(US10167292, Example 47)
Affinity DataIC50:  11nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Walter and Eliza Hall Institute of Medical Research

Curated by ChEMBL
LigandPNGBDBM313791(US10167292, Example 35)
Affinity DataIC50:  12nMAssay Description:Inhibition of human His-tagged Brd3 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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