TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Affinity DataEC50: 16nMAssay Description:Agonist activity at yeast Gal4-fused human PPARalpha LBD transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase...More data for this Ligand-Target Pair
Affinity DataEC50: 1.10E+4nMAssay Description:Potentiation of CFTR F508del mutant (unknown origin) expressed in rat FRT cells assessed as increase in iodide influx in presence of forskolin incuba...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Affinity DataEC50: 250nMAssay Description:Agonist activity at yeast Gal4-fused human PPARalpha LBD transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Affinity DataEC50: 370nMAssay Description:Agonist activity at yeast Gal4-fused human PPARalpha LBD transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Affinity DataEC50: 380nMAssay Description:Agonist activity at yeast Gal4-fused human PPARalpha LBD transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Affinity DataEC50: 580nMAssay Description:Agonist activity at yeast Gal4-fused human PPARalpha LBD transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Affinity DataEC50: 710nMAssay Description:Agonist activity at yeast Gal4-fused human PPARalpha LBD transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Affinity DataEC50: 800nMAssay Description:Agonist activity at yeast Gal4-fused human PPARalpha LBD transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Affinity DataEC50: 940nMAssay Description:Agonist activity at yeast Gal4-fused human PPARalpha LBD transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Affinity DataEC50: 1.45E+3nMAssay Description:Agonist activity at yeast Gal4-fused human PPARalpha LBD transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Affinity DataEC50: 1.56E+3nMAssay Description:Agonist activity at yeast Gal4-fused human PPARalpha LBD transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Affinity DataEC50: 1.60E+3nMAssay Description:Agonist activity at yeast Gal4-fused human PPARalpha LBD transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Affinity DataEC50: 1.60E+3nMAssay Description:Agonist activity at yeast Gal4-fused human PPARalpha LBD transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Affinity DataEC50: 1.90E+3nMAssay Description:Agonist activity at yeast Gal4-fused human PPARalpha LBD transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Affinity DataEC50: 2.55E+3nMAssay Description:Agonist activity at yeast Gal4-fused human PPARalpha LBD transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Affinity DataEC50: 4.80E+3nMAssay Description:Agonist activity at yeast Gal4-fused human PPARalpha LBD transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Affinity DataEC50: 7.20E+3nMAssay Description:Agonist activity at yeast Gal4-fused human PPARalpha LBD transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Affinity DataEC50: 9.10E+3nMAssay Description:Agonist activity at yeast Gal4-fused human PPARalpha LBD transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Affinity DataEC50: 1.00E+4nMAssay Description:Agonist activity at yeast Gal4-fused human PPARalpha LBD transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Affinity DataEC50: 1.21E+4nMAssay Description:Agonist activity at yeast Gal4-fused human PPARalpha LBD transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Affinity DataEC50: 40nMAssay Description:Agonist activity at yeast Gal4-fused human PPARgamma transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase act...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Affinity DataEC50: 2.20E+3nMAssay Description:Agonist activity at yeast Gal4-fused human PPARgamma transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase act...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Affinity DataEC50: 3.20E+3nMAssay Description:Agonist activity at yeast Gal4-fused human PPARgamma transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase act...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Affinity DataEC50: 3.40E+3nMAssay Description:Agonist activity at yeast Gal4-fused human PPARgamma transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase act...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Affinity DataEC50: 3.90E+3nMAssay Description:Agonist activity at yeast Gal4-fused human PPARgamma transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase act...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Affinity DataEC50: 4.60E+3nMAssay Description:Agonist activity at yeast Gal4-fused human PPARgamma transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase act...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Affinity DataEC50: 6.70E+3nMAssay Description:Agonist activity at yeast Gal4-fused human PPARgamma transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase act...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Affinity DataEC50: 7.50E+3nMAssay Description:Agonist activity at yeast Gal4-fused human PPARgamma transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase act...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Affinity DataEC50: 7.90E+3nMAssay Description:Agonist activity at yeast Gal4-fused human PPARgamma transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase act...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Affinity DataEC50: 8.40E+3nMAssay Description:Agonist activity at yeast Gal4-fused human PPARgamma transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase act...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Affinity DataEC50: 1.02E+4nMAssay Description:Agonist activity at yeast Gal4-fused human PPARgamma transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase act...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Affinity DataEC50: 1.03E+4nMAssay Description:Agonist activity at yeast Gal4-fused human PPARgamma transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase act...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Affinity DataEC50: 1.09E+4nMAssay Description:Agonist activity at yeast Gal4-fused human PPARgamma transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase act...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Affinity DataEC50: 1.28E+4nMAssay Description:Agonist activity at yeast Gal4-fused human PPARgamma transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase act...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Affinity DataEC50: 1.30E+4nMAssay Description:Agonist activity at yeast Gal4-fused human PPARgamma transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase act...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Affinity DataEC50: 2.00E+4nMAssay Description:Agonist activity at yeast Gal4-fused human PPARgamma transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase act...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Affinity DataEC50: 2.57E+4nMAssay Description:Agonist activity at yeast Gal4-fused human PPARgamma transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase act...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Affinity DataEC50: 21nMAssay Description:Agonist activity at yeast Gal4-fused human PPARdelta transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase act...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Affinity DataEC50: 2.80E+4nMAssay Description:Agonist activity at yeast Gal4-fused human PPARdelta transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase act...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Universit£?Degli Studi Di Bari "Aldo Moro
Curated by ChEMBL
Affinity DataEC50: 3.71E+4nMAssay Description:Agonist activity at yeast Gal4-fused human PPARdelta transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase act...More data for this Ligand-Target Pair
Affinity DataEC50: 70nMAssay Description:Potentiation of CFTR F508del mutant in rat FRT cells assessed as increase in iodide influx in presence of forskolinMore data for this Ligand-Target Pair
Affinity DataEC50: 7.00E+3nMAssay Description:Potentiation of CFTR F508del mutant activity (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 90nMAssay Description:Potentiation of CFTR F508del mutant activity (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 1.10E+3nMAssay Description:Potentiation of CFTR F508del mutant activity (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 2.20E+3nMAssay Description:Corrector activity at CFTR F508del mutant (unknown origin) expressed in rat FRT cells assessed as increase in iodide influx in presence of forskolin ...More data for this Ligand-Target Pair
Affinity DataEC50: 3.80E+3nMAssay Description:Corrector activity at CFTR F508del mutant (unknown origin) expressed in rat FRT cells assessed as increase in iodide influx in presence of forskolin ...More data for this Ligand-Target Pair
Affinity DataEC50: 3.90E+3nMAssay Description:Corrector activity at CFTR F508del mutant (unknown origin) expressed in rat FRT cells assessed as increase in iodide influx in presence of forskolin ...More data for this Ligand-Target Pair
Affinity DataEC50: 5.00E+3nMAssay Description:Corrector activity at CFTR F508del mutant (unknown origin) expressed in rat FRT cells assessed as increase in iodide influx in presence of forskolin ...More data for this Ligand-Target Pair
Affinity DataEC50: 4.20E+3nMAssay Description:Corrector activity at CFTR F508del mutant (unknown origin) expressed in rat FRT cells assessed as increase in iodide influx in presence of forskolin ...More data for this Ligand-Target Pair
Affinity DataEC50: 1.40E+4nMAssay Description:Potentiation of CFTR F508del mutant (unknown origin) expressed in rat FRT cells assessed as increase in iodide influx in presence of forskolin incuba...More data for this Ligand-Target Pair
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