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Found 54 with Last Name = 'genovese' and Initial = 'm'
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50604536(CHEMBL5173673)
Affinity DataEC50:  16nMAssay Description:Agonist activity at yeast Gal4-fused human PPARalpha LBD transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM50516908(CHEMBL4444352)
Affinity DataEC50:  1.10E+4nMAssay Description:Potentiation of CFTR F508del mutant (unknown origin) expressed in rat FRT cells assessed as increase in iodide influx in presence of forskolin incuba...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50604538(CHEMBL5191536)
Affinity DataEC50:  250nMAssay Description:Agonist activity at yeast Gal4-fused human PPARalpha LBD transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50604539(CHEMBL5204992)
Affinity DataEC50:  370nMAssay Description:Agonist activity at yeast Gal4-fused human PPARalpha LBD transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50604540(CHEMBL5173134)
Affinity DataEC50:  380nMAssay Description:Agonist activity at yeast Gal4-fused human PPARalpha LBD transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50604541(CHEMBL5207071)
Affinity DataEC50:  580nMAssay Description:Agonist activity at yeast Gal4-fused human PPARalpha LBD transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50604542(CHEMBL5203327)
Affinity DataEC50:  710nMAssay Description:Agonist activity at yeast Gal4-fused human PPARalpha LBD transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50604543(CHEMBL5172173)
Affinity DataEC50:  800nMAssay Description:Agonist activity at yeast Gal4-fused human PPARalpha LBD transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50604544(CHEMBL5191690)
Affinity DataEC50:  940nMAssay Description:Agonist activity at yeast Gal4-fused human PPARalpha LBD transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50604545(CHEMBL5196830)
Affinity DataEC50:  1.45E+3nMAssay Description:Agonist activity at yeast Gal4-fused human PPARalpha LBD transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM24566(2-({4-chloro-6-[(2,3-dimethylphenyl)amino]pyrimidi...)
Affinity DataEC50:  1.56E+3nMAssay Description:Agonist activity at yeast Gal4-fused human PPARalpha LBD transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50604546(CHEMBL5195064)
Affinity DataEC50:  1.60E+3nMAssay Description:Agonist activity at yeast Gal4-fused human PPARalpha LBD transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50604547(CHEMBL1967191)
Affinity DataEC50:  1.60E+3nMAssay Description:Agonist activity at yeast Gal4-fused human PPARalpha LBD transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50604548(CHEMBL5196394)
Affinity DataEC50:  1.90E+3nMAssay Description:Agonist activity at yeast Gal4-fused human PPARalpha LBD transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50604549(CHEMBL5184438)
Affinity DataEC50:  2.55E+3nMAssay Description:Agonist activity at yeast Gal4-fused human PPARalpha LBD transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50604550(CHEMBL5194126)
Affinity DataEC50:  4.80E+3nMAssay Description:Agonist activity at yeast Gal4-fused human PPARalpha LBD transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50604551(CHEMBL5194570)
Affinity DataEC50:  7.20E+3nMAssay Description:Agonist activity at yeast Gal4-fused human PPARalpha LBD transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50604552(CHEMBL5207420)
Affinity DataEC50:  9.10E+3nMAssay Description:Agonist activity at yeast Gal4-fused human PPARalpha LBD transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50604553(CHEMBL5186824)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at yeast Gal4-fused human PPARalpha LBD transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50604554(CHEMBL5199782)
Affinity DataEC50:  1.21E+4nMAssay Description:Agonist activity at yeast Gal4-fused human PPARalpha LBD transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50030474(Avandamet | Avandaryl | Avandia | BRL-49653 | CHEB...)
Affinity DataEC50:  40nMAssay Description:Agonist activity at yeast Gal4-fused human PPARgamma transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase act...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50604538(CHEMBL5191536)
Affinity DataEC50:  2.20E+3nMAssay Description:Agonist activity at yeast Gal4-fused human PPARgamma transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase act...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50604539(CHEMBL5204992)
Affinity DataEC50:  3.20E+3nMAssay Description:Agonist activity at yeast Gal4-fused human PPARgamma transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase act...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50604541(CHEMBL5207071)
Affinity DataEC50:  3.40E+3nMAssay Description:Agonist activity at yeast Gal4-fused human PPARgamma transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase act...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50604542(CHEMBL5203327)
Affinity DataEC50:  3.90E+3nMAssay Description:Agonist activity at yeast Gal4-fused human PPARgamma transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase act...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50604544(CHEMBL5191690)
Affinity DataEC50:  4.60E+3nMAssay Description:Agonist activity at yeast Gal4-fused human PPARgamma transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase act...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50604552(CHEMBL5207420)
Affinity DataEC50:  6.70E+3nMAssay Description:Agonist activity at yeast Gal4-fused human PPARgamma transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase act...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50604540(CHEMBL5173134)
Affinity DataEC50:  7.50E+3nMAssay Description:Agonist activity at yeast Gal4-fused human PPARgamma transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase act...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50604548(CHEMBL5196394)
Affinity DataEC50:  7.90E+3nMAssay Description:Agonist activity at yeast Gal4-fused human PPARgamma transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase act...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50604546(CHEMBL5195064)
Affinity DataEC50:  8.40E+3nMAssay Description:Agonist activity at yeast Gal4-fused human PPARgamma transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase act...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50604543(CHEMBL5172173)
Affinity DataEC50:  1.02E+4nMAssay Description:Agonist activity at yeast Gal4-fused human PPARgamma transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase act...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50604547(CHEMBL1967191)
Affinity DataEC50:  1.03E+4nMAssay Description:Agonist activity at yeast Gal4-fused human PPARgamma transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase act...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50604549(CHEMBL5184438)
Affinity DataEC50:  1.09E+4nMAssay Description:Agonist activity at yeast Gal4-fused human PPARgamma transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase act...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50604550(CHEMBL5194126)
Affinity DataEC50:  1.28E+4nMAssay Description:Agonist activity at yeast Gal4-fused human PPARgamma transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase act...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50604551(CHEMBL5194570)
Affinity DataEC50:  1.30E+4nMAssay Description:Agonist activity at yeast Gal4-fused human PPARgamma transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase act...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50604554(CHEMBL5199782)
Affinity DataEC50:  2.00E+4nMAssay Description:Agonist activity at yeast Gal4-fused human PPARgamma transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase act...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50604545(CHEMBL5196830)
Affinity DataEC50:  2.57E+4nMAssay Description:Agonist activity at yeast Gal4-fused human PPARgamma transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase act...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50085041(2-(4-(3-(4-acetyl-3-hydroxy-2-propylphenoxy)propox...)
Affinity DataEC50:  21nMAssay Description:Agonist activity at yeast Gal4-fused human PPARdelta transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase act...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50604546(CHEMBL5195064)
Affinity DataEC50:  2.80E+4nMAssay Description:Agonist activity at yeast Gal4-fused human PPARdelta transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase act...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Universit£?Degli Studi Di Bari "Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50604547(CHEMBL1967191)
Affinity DataEC50:  3.71E+4nMAssay Description:Agonist activity at yeast Gal4-fused human PPARdelta transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase act...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM50581833(CHEMBL1949980)
Affinity DataEC50:  70nMAssay Description:Potentiation of CFTR F508del mutant in rat FRT cells assessed as increase in iodide influx in presence of forskolinMore data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM19459(5,7-dihydroxy-3-(4-hydroxyphenyl)-4H-chromen-4-one...)
Affinity DataEC50:  7.00E+3nMAssay Description:Potentiation of CFTR F508del mutant activity (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50486732(CHEMBL2068831)
Affinity DataEC50:  90nMAssay Description:Potentiation of CFTR F508del mutant activity (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM50486733(CHEMBL2068832)
Affinity DataEC50:  1.10E+3nMAssay Description:Potentiation of CFTR F508del mutant activity (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM50289534(CHEMBL2018574)
Affinity DataEC50:  2.20E+3nMAssay Description:Corrector activity at CFTR F508del mutant (unknown origin) expressed in rat FRT cells assessed as increase in iodide influx in presence of forskolin ...More data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50516902(CHEMBL1583913)
Affinity DataEC50:  3.80E+3nMAssay Description:Corrector activity at CFTR F508del mutant (unknown origin) expressed in rat FRT cells assessed as increase in iodide influx in presence of forskolin ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM50516901(CHEMBL1403454)
Affinity DataEC50:  3.90E+3nMAssay Description:Corrector activity at CFTR F508del mutant (unknown origin) expressed in rat FRT cells assessed as increase in iodide influx in presence of forskolin ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM50516906(CHEMBL4444246)
Affinity DataEC50:  5.00E+3nMAssay Description:Corrector activity at CFTR F508del mutant (unknown origin) expressed in rat FRT cells assessed as increase in iodide influx in presence of forskolin ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM50516908(CHEMBL4444352)
Affinity DataEC50:  4.20E+3nMAssay Description:Corrector activity at CFTR F508del mutant (unknown origin) expressed in rat FRT cells assessed as increase in iodide influx in presence of forskolin ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM50289534(CHEMBL2018574)
Affinity DataEC50:  1.40E+4nMAssay Description:Potentiation of CFTR F508del mutant (unknown origin) expressed in rat FRT cells assessed as increase in iodide influx in presence of forskolin incuba...More data for this Ligand-Target Pair
In DepthDetails PubMed
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