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Found 497 with Last Name = 'jean' and Initial = 'm'
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50340329(4-azamelatonin | CHEMBL1760944)
Affinity DataKi:  0.200nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human MT1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM9019(CHEMBL45 | Melatonin | N-[2-(5-methoxy-1H-indol-3-...)
Affinity DataKi:  0.25nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human MT1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetMelatonin receptor type 1B(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50340324(CHEMBL1760946 | N-(2-(6-Methoxy-1H-pyrrolo[2,3-b]p...)
Affinity DataKi:  0.280nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human MT2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50340329(4-azamelatonin | CHEMBL1760944)
Affinity DataKi:  0.300nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human MT2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50340338(CHEMBL1760947 | N-(2-(6-Methoxy-1H-pyrrolo[2,3-b]p...)
Affinity DataKi:  0.300nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human MT2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM9019(CHEMBL45 | Melatonin | N-[2-(5-methoxy-1H-indol-3-...)
Affinity DataKi:  0.340nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human MT2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetD(2) dopamine receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50325758(CHEMBL1223616 | N-(4-(4-(2,3-dichlorophenyl)pipera...)
Affinity DataKi:  0.400nMAssay Description:Displacement of [3H]spiperone from human dopamine D2S receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50325753(CHEMBL1223856 | N-(4-(4-(2,3-dichlorophenyl)pipera...)
Affinity DataKi:  0.550nMAssay Description:Displacement of [3H]spiperone from human dopamine D2S receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50325750(CHEMBL1223800 | N-(4-(4-(2,3-dichlorophenyl)pipera...)
Affinity DataKi:  0.590nMAssay Description:Displacement of [3H]spiperone from human dopamine D2S receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50325744(CHEMBL1223683 | N-(4-(4-(2,3-dichlorophenyl)pipera...)
Affinity DataKi:  0.600nMAssay Description:Displacement of [3H]spiperone from human dopamine D2S receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50340325(CHEMBL1760945 | N-(2-(6-Methoxy-1H-pyrrolo[2,3-b]p...)
Affinity DataKi:  0.600nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human MT2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50340327(CHEMBL1760957 | N-(2-(5,6,7,8-Tetrahydro-2-methoxy...)
Affinity DataKi:  0.680nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human MT2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50325754(4-phenyl-N-(4-(4-(3-(trifluoromethyl)phenyl)pipera...)
Affinity DataKi:  0.760nMAssay Description:Displacement of [3H]spiperone from human dopamine D2S receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50325757(CHEMBL1223615 | N-(4-(4-(2-methoxyphenyl)piperazin...)
Affinity DataKi:  0.800nMAssay Description:Displacement of [3H]spiperone from human dopamine D2S receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50325746(CHEMBL1223748 | N-(4-(4-(2-methoxyphenyl)piperazin...)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]spiperone from human dopamine D2S receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50325748(CHEMBL1223750 | N-(4-(4-(3-(trifluoromethyl)phenyl...)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]spiperone from human dopamine D2S receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50325751(5-phenyl-N-(4-(4-(3-(trifluoromethyl)phenyl)pipera...)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]spiperone from human dopamine D2S receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50340338(CHEMBL1760947 | N-(2-(6-Methoxy-1H-pyrrolo[2,3-b]p...)
Affinity DataKi:  1.30nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human MT1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50340325(CHEMBL1760945 | N-(2-(6-Methoxy-1H-pyrrolo[2,3-b]p...)
Affinity DataKi:  1.40nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human MT1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50325752(CHEMBL1223802 | N-(4-(4-(2-fluorophenyl)piperazin-...)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]spiperone from human dopamine D2S receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50325745(CHEMBL1223747 | N-(4-(4-(3-(trifluoromethyl)phenyl...)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]spiperone from human dopamine D2S receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50325749(CHEMBL1223799 | N-(4-(4-(2-fluorophenyl)piperazin-...)
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]spiperone from human dopamine D2S receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50325747(CHEMBL1223749 | N-(4-(4-(2,3-dichlorophenyl)pipera...)
Affinity DataKi:  3.10nMAssay Description:Displacement of [3H]spiperone from human dopamine D2S receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50340324(CHEMBL1760946 | N-(2-(6-Methoxy-1H-pyrrolo[2,3-b]p...)
Affinity DataKi:  3.30nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human MT1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50340326(CHEMBL1760956 | N-(2-(3-iodo-6-methoxy-1H-pyrrolo[...)
Affinity DataKi:  5nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human MT2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50325743(CHEMBL271989 | N-(4-(4-(2-methoxyphenyl)piperazin-...)
Affinity DataKi:  5.60nMAssay Description:Displacement of [3H]spiperone from human dopamine D2S receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50325746(CHEMBL1223748 | N-(4-(4-(2-methoxyphenyl)piperazin...)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]prazosin from human adrenergic alpha1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50325743(CHEMBL271989 | N-(4-(4-(2-methoxyphenyl)piperazin-...)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]prazosin from human adrenergic alpha1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50340327(CHEMBL1760957 | N-(2-(5,6,7,8-Tetrahydro-2-methoxy...)
Affinity DataKi:  9nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human MT1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50325752(CHEMBL1223802 | N-(4-(4-(2-fluorophenyl)piperazin-...)
Affinity DataKi:  9nMAssay Description:Displacement of [3H]prazosin from human adrenergic alpha1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50325755(5-phenyl-N-(4-(4-(3-(trifluoromethyl)phenyl)pipera...)
Affinity DataKi:  9.60nMAssay Description:Displacement of [3H]spiperone from human dopamine D2S receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50325749(CHEMBL1223799 | N-(4-(4-(2-fluorophenyl)piperazin-...)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]prazosin from human adrenergic alpha1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50325760(CHEMBL1223680 | N-(4-(4-(2-fluorophenyl)piperazin-...)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]spiperone from human dopamine D2S receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50325745(CHEMBL1223747 | N-(4-(4-(3-(trifluoromethyl)phenyl...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]prazosin from human adrenergic alpha1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50325742(CHEMBL1223682 | N-(4-(4-(2,3-dimethylphenyl)pipera...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]spiperone from human dopamine D2S receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50325756(4-phenyl-N-(4-(4-(3-(trifluoromethyl)phenyl)pipera...)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]spiperone from human dopamine D2S receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50325761(CHEMBL1223681 | N-(4-(4-o-tolylpiperazin-1-yl)buty...)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]prazosin from human adrenergic alpha1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50325743(CHEMBL271989 | N-(4-(4-(2-methoxyphenyl)piperazin-...)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]spiperone from human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50340326(CHEMBL1760956 | N-(2-(3-iodo-6-methoxy-1H-pyrrolo[...)
Affinity DataKi:  16nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human MT1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50325759(CHEMBL1223617 | N-(4-(4-(3-(trifluoromethyl)phenyl...)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]spiperone from human dopamine D2S receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50325760(CHEMBL1223680 | N-(4-(4-(2-fluorophenyl)piperazin-...)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]prazosin from human adrenergic alpha1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50325747(CHEMBL1223749 | N-(4-(4-(2,3-dichlorophenyl)pipera...)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]spiperone from human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50325750(CHEMBL1223800 | N-(4-(4-(2,3-dichlorophenyl)pipera...)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]prazosin from human adrenergic alpha1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50325744(CHEMBL1223683 | N-(4-(4-(2,3-dichlorophenyl)pipera...)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]spiperone from human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50325757(CHEMBL1223615 | N-(4-(4-(2-methoxyphenyl)piperazin...)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]prazosin from human adrenergic alpha1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50325758(CHEMBL1223616 | N-(4-(4-(2,3-dichlorophenyl)pipera...)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]spiperone from human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50340328(CHEMBL1760955 | N-(2-(6-methoxy-3-(2,2,2-trifluoro...)
Affinity DataKi:  30nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human MT2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50325761(CHEMBL1223681 | N-(4-(4-o-tolylpiperazin-1-yl)buty...)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]spiperone from human dopamine D2S receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50325758(CHEMBL1223616 | N-(4-(4-(2,3-dichlorophenyl)pipera...)
Affinity DataKi:  33nMAssay Description:Displacement of [3H]prazosin from human adrenergic alpha1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50340330(7-azamelatonin | CHEMBL137969 | N-[2-(5-Methoxy-1H...)
Affinity DataKi:  40nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human MT1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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