Affinity DataKi: 0.170nMAssay Description:Tested for binding affinity against recombinant human Alpha-1A adrenergic receptor using [125I]HEAT in competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Compound was evaluated for its ability to displace [125I]-HEAT binding from rat Alpha-1B adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Compound was tested for binding affinity utilizing cloned receptor binding assays by using [125 I]HEAT as radioligand to the human Alpha-1D adrenergi...More data for this Ligand-Target Pair
Affinity DataKi: 0.210nMAssay Description:Compound was tested for binding affinity utilizing cloned receptor binding assays by using [125 I]HEAT as radioligand to the human Alpha-1B adrenergi...More data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Compound was evaluated for its ability to displace [125I]-HEAT binding from rat Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Compound was evaluated for its ability to displace [125I]-HEAT binding from rat Alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.390nMAssay Description:Compound was tested for binding affinity utilizing cloned receptor binding assays by using [125 I]HEAT as radioligand to the human Alpha-1A adrenergi...More data for this Ligand-Target Pair
Affinity DataKi: 0.480nMAssay Description:In vitro binding affinity towards cloned human Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.510nMAssay Description:Binding affinity against human Alpha-1a adrenergic receptor was evaluated by cloned receptor binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.580nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.830nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Tested for binding affinity against recombinant human Alpha-1A adrenergic receptor using [125I]HEAT in competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.990nMAssay Description:Inhibition of binding of [125I]-HEAT to cloned human alpha-1A adrenergic receptor.More data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Inhibition of binding of [125I]-HEAT to cloned human alpha-1A adrenergic receptor.More data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Compound was tested for its binding affinity utilizing cloned receptor binding assays by using [125 I]HEAT as radioligand to the human Alpha-1B adren...More data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Inhibition of binding of [125I]-HEAT to cloned human alpha-1A adrenergic receptor.More data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Compound was tested for its binding affinity utilizing cloned receptor binding assays by using [125 I]HEAT as radioligand to the human Alpha-1D adren...More data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:In vitro binding affinity towards cloned human Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Compound was evaluated for its ability to displace [125I]-HEAT binding from rat Alpha-1B adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Inhibition of binding of [125I]-HEAT to cloned human alpha-1A adrenergic receptor.More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Inhibition of binding of [125I]-HEAT to cloned human alpha-1B adrenergic receptor.More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:In vitro binding affinity towards cloned human Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Compound was tested for its binding affinity utilizing cloned receptor binding assays by using [125 I]HEAT as radioligand to the human Alpha-1B adren...More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Compound was tested for its binding affinity utilizing cloned receptor binding assays by using [125 I]HEAT as radioligand to the human Alpha-1D adren...More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Inhibition of binding of [125I]-HEAT to cloned human alpha-1A adrenergic receptor.More data for this Ligand-Target Pair
Affinity DataKi: 2.40nMAssay Description:Compound was evaluated for its ability to displace [125I]-HEAT binding from rat Alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.80nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Binding affinity against human Alpha-1a adrenergic receptor was evaluated by cloned receptor binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 3.20nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 3.40nMAssay Description:Compound was evaluated for its ability to displace [125I]-HEAT binding from rat Alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.40nMAssay Description:Inhibition of binding of [125I]-HEAT to cloned human alpha-1A adrenergic receptor.More data for this Ligand-Target Pair
Affinity DataKi: 3.5nMAssay Description:Compound was tested for binding affinity utilizing cloned receptor binding assays by using [125 I]HEAT as radioligand to the human Alpha-1B adrenergi...More data for this Ligand-Target Pair
Affinity DataKi: 3.60nMAssay Description:Inhibition of binding of [125I]-HEAT to cloned human alpha-1A adrenergic receptor.More data for this Ligand-Target Pair
Affinity DataKi: 3.90nMAssay Description:Compound was evaluated for its ability to displace [125I]-HEAT binding from rat Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 4.20nMAssay Description:Compound was tested for its binding affinity utilizing cloned receptor binding assays by using [125 I]HEAT as radioligand to the human Alpha-1A adren...More data for this Ligand-Target Pair
Affinity DataKi: 4.30nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 5.10nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 5.10nMAssay Description:Inhibition of binding of [125I]-HEAT to cloned human alpha-1A adrenergic receptor.More data for this Ligand-Target Pair
Affinity DataKi: 5.40nMAssay Description:Compound was evaluated for its ability to displace [125I]-HEAT binding from rat Alpha-1B adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5.70nMAssay Description:In vitro binding affinity towards cloned human Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 8(Homo sapiens (Human))
Millennium Pharmaceuticals
Curated by ChEMBL
Millennium Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 6nMAssay Description:Displacement of [125I]I309 from human CCR8 expressed in L1.2 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 6.40nMAssay Description:Inhibition of binding of [125I]-HEAT to cloned human alpha-1A adrenergic receptor.More data for this Ligand-Target Pair
Affinity DataKi: 6.60nMAssay Description:Inhibition of binding of [125I]-HEAT to cloned human alpha-1B adrenergic receptor.More data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Compound was evaluated for its ability to displace [125I]-HEAT binding from rat Alpha-1B adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 7.30nMAssay Description:Inhibition of binding of [125I]-HEAT to cloned human alpha-1A adrenergic receptor.More data for this Ligand-Target Pair
Affinity DataKi: 7.30nMAssay Description:In vitro binding affinity towards cloned human Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 7.40nMAssay Description:Inhibition of binding of [125I]-HEAT to cloned human alpha-1A adrenergic receptor.More data for this Ligand-Target Pair
Affinity DataKi: 7.5nMAssay Description:Inhibition of binding of [125I]-HEAT to cloned human alpha-1A adrenergic receptor.More data for this Ligand-Target Pair
Affinity DataKi: 8.80nMAssay Description:Inhibition of binding of [125I]-HEAT to cloned human alpha-1A adrenergic receptor.More data for this Ligand-Target Pair
TargetC-C chemokine receptor type 8(Homo sapiens (Human))
Millennium Pharmaceuticals
Curated by ChEMBL
Millennium Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 9nMAssay Description:Displacement of [125I]I309 from human CCR8 expressed in L1.2 cellsMore data for this Ligand-Target Pair