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Found 118 with Last Name = 'saletti' and Initial = 'm'
TargetTranslocator protein(Rattus norvegicus (rat))TBA
LigandPNGBDBM50409614(CHEMBL5288131)
Affinity DataKi:  0.0700nMAssay Description:Inhibitory activity against dihydrofolate reductase (DHFR) from Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetTranslocator protein(Homo sapiens (Human))TBA
LigandPNGBDBM50409613(CHEMBL5275028)
Affinity DataKi:  0.300nMAssay Description:Inhibitory activity against dihydrofolate reductase (DHFR) from Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetTranslocator protein(Homo sapiens (Human))TBA
LigandPNGBDBM22041(2-[6-chloro-2-(4-chlorophenyl)imidazo[1,2-a]pyridi...)
Affinity DataKi:  0.5nMAssay Description:Inhibitory activity against Dihydrofolate reductase of Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetTranslocator protein(Homo sapiens (Human))TBA
LigandPNGBDBM50363523(CHEMBL1944785)
Affinity DataKi:  2.40nMAssay Description:Inhibitory activity against Dihydrofolate reductase of Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetTranslocator protein(Rattus norvegicus (rat))TBA
LigandPNGBDBM50045880(2-[5-Chloro-2-(4-chloro-phenyl)-1H-indol-3-yl]-N,N...)
Affinity DataKi:  3.90nMAssay Description:Inhibitory activity against dihydrofolate reductase (DHFR) of Neisseria gonorrhoeaMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetTranslocator protein(Rattus norvegicus (rat))TBA
LigandPNGBDBM50243007(2-(2-(4-(2-Fluoroethoxy)phenyl)-5,7-dimethylpyrazo...)
Affinity DataKi:  7nMAssay Description:Inhibitory activity against dihydrofolate reductase (DHFR) from rat liverMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetTranslocator protein(Rattus norvegicus (rat))TBA
LigandPNGBDBM22041(2-[6-chloro-2-(4-chlorophenyl)imidazo[1,2-a]pyridi...)
Affinity DataIC50:  0.5nMAssay Description:Inhibitory activity against Dihydrofolate reductase of Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetTranslocator protein(Rattus norvegicus (rat))TBA
LigandPNGBDBM22032(1-(2-chlorophenyl)-N-methyl-N-(1-methylpropyl)isoq...)
Affinity DataIC50:  1.80nMAssay Description:Inhibitory activity against Dihydrofolate reductase of Escherichia coliMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))TBA
LigandPNGBDBM50059754(3-Methyl-4-phenyl-quinoline-2-carboxylic acid sec-...)
Affinity DataIC50:  2.10nMAssay Description:Inhibitory activity against Dihydrofolate reductase of Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetTranslocator protein(Rattus norvegicus (rat))TBA
LigandPNGBDBM50059749(3-Methyl-4-phenyl-quinoline-2-carboxylic acid benz...)
Affinity DataIC50:  2.10nMAssay Description:Inhibition of rat liver Dihydrofolate reductase.More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetTranslocator protein(Rattus norvegicus (rat))TBA
LigandPNGBDBM50131729(4-(2-Fluoro-phenyl)-3-methyl-quinoline-2-carboxyli...)
Affinity DataIC50:  2.20nMAssay Description:Inhibitory activity against dihydrofolate reductase (DHFR) from rat liverMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetTranslocator protein(Rattus norvegicus (rat))TBA
LigandPNGBDBM50059755(4-(2-Fluoro-phenyl)-3-methyl-quinoline-2-carboxyli...)
Affinity DataIC50:  2.90nMAssay Description:Inhibition of rat liver Dihydrofolate reductase.More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProstaglandin G/H synthase 2(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM50589579(CHEMBL5185981)
Affinity DataIC50:  3nMAssay Description:Inhibition of COX2 in LPS-stimulated mouse J774 cells assessed as inhibition of PGE2 production and measured after 24 hrs by enzyme immuno-assay (EIA...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTranslocator protein(Rattus norvegicus (rat))TBA
LigandPNGBDBM50059758(4-Methyl-1-phenyl-isoquinoline-3-carboxylic acid b...)
Affinity DataIC50:  3.10nMAssay Description:Evaluated for the inhibition of chicken liver Dihydrofolate reductase by using standard enzyme assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetTranslocator protein(Rattus norvegicus (rat))TBA
LigandPNGBDBM50059739(4-(2-Fluoro-phenyl)-3-methyl-quinoline-2-carboxyli...)
Affinity DataIC50:  3.40nMAssay Description:Inhibition of rat liver Dihydrofolate reductase.More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetTranslocator protein(Rattus norvegicus (rat))TBA
LigandPNGBDBM50098694(3-[(Benzyl-ethyl-amino)-methyl]-4-phenyl-quinoline...)
Affinity DataIC50:  4.10nMAssay Description:Inhibitory activity against dihydrofolate reductase (DHFR) of Plasmodium bergheiMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProstaglandin G/H synthase 2(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM50589578(CHEMBL5180981)
Affinity DataIC50:  5nMAssay Description:Inhibition of COX2 in LPS-stimulated mouse J774 cells assessed as inhibition of PGE2 production and measured after 24 hrs by enzyme immuno-assay (EIA...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTranslocator protein(Rattus norvegicus (rat))TBA
LigandPNGBDBM50059738(3-Methyl-4-phenyl-quinoline-2-carboxylic acid (4-c...)
Affinity DataIC50:  6.40nMAssay Description:Compound was tested for inhibitory activity against Dihydrofolate Reductase(DHFR) of rat liverMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProstaglandin G/H synthase 2(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM50589575(CHEMBL5176255)
Affinity DataIC50:  8nMAssay Description:Inhibition of COX2 in LPS-stimulated mouse J774 cells assessed as inhibition of PGE2 production and measured after 24 hrs by enzyme immuno-assay (EIA...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTranslocator protein(Rattus norvegicus (rat))TBA
LigandPNGBDBM22032(1-(2-chlorophenyl)-N-methyl-N-(1-methylpropyl)isoq...)
Affinity DataIC50:  8.40nMAssay Description:Inhibitory activity against dihydrofolate reductase (DHFR) from Escherichia coliMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))TBA
LigandPNGBDBM50131721(3-Hydroxymethyl-4-phenyl-quinoline-2-carboxylic ac...)
Affinity DataIC50:  8.70nMAssay Description:Inhibitory activity against dihydrofolate reductase (DHFR) from rat liverMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetTranslocator protein(Rattus norvegicus (rat))TBA
LigandPNGBDBM50059756(3-Methyl-4-phenyl-quinoline-2-carboxylic acid (4-m...)
Affinity DataIC50:  8.80nMAssay Description:Inhibitory activity against Dihydrofolate reductase of Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetTranslocator protein(Rattus norvegicus (rat))TBA
LigandPNGBDBM50059750(7,8-Dihydro-benzo[k]phenanthridine-6-carboxylic ac...)
Affinity DataIC50:  8.90nMAssay Description:Evaluated for the inhibition of chicken liver Dihydrofolate reductase by using standard enzyme assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProstaglandin G/H synthase 2(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM50589572(CHEMBL5189607)
Affinity DataIC50:  9nMAssay Description:Inhibition of COX2 in LPS-stimulated mouse J774 cells assessed as inhibition of PGE2 production and measured after 24 hrs by enzyme immuno-assay (EIA...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTranslocator protein(Rattus norvegicus (rat))TBA
LigandPNGBDBM50131727(3-Methyl-4-phenyl-naphthalene-2-carboxylic acid be...)
Affinity DataIC50:  9.80nMAssay Description:Inhibitory activity against dihydrofolate reductase (DHFR) from Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetTranslocator protein(Rattus norvegicus (rat))TBA
LigandPNGBDBM50059745(3-Methyl-4-phenyl-quinoline-2-carboxylic acid (4-c...)
Affinity DataIC50:  9.80nMAssay Description:Inhibitory activity against Dihydrofolate reductase of Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetTranslocator protein(Rattus norvegicus (rat))TBA
LigandPNGBDBM50409519(CHEMBL5275613)
Affinity DataIC50:  10nMAssay Description:Evaluated for the inhibition of chicken liver Dihydrofolate reductase by using standard enzyme assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetTranslocator protein(Rattus norvegicus (rat))TBA
LigandPNGBDBM50059743(4-Methyl-1-phenyl-isoquinoline-3-carboxylic acid s...)
Affinity DataIC50:  11nMAssay Description:Inhibitory activity against Dihydrofolate reductase of Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetTranslocator protein(Rattus norvegicus (rat))TBA
LigandPNGBDBM50131730(3-Methyl-4-phenyl-quinoline-2-carboxylic acid dibe...)
Affinity DataIC50:  11nMAssay Description:Inhibitory activity against dihydrofolate reductase (DHFR) of Neisseria gonorrhoeaMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetTranslocator protein(Rattus norvegicus (rat))TBA
LigandPNGBDBM50131726(3-Diethylaminomethyl-4-phenyl-quinoline-2-carboxyl...)
Affinity DataIC50:  12nMAssay Description:Inhibitory activity against dihydrofolate reductase (DHFR) of Neisseria gonorrhoeaMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetTranslocator protein(Rattus norvegicus (rat))TBA
LigandPNGBDBM50059737(4-(2-Fluoro-phenyl)-3-methyl-quinoline-2-carboxyli...)
Affinity DataIC50:  13nMAssay Description:Inhibitory activity against Dihydrofolate reductase of Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProstaglandin G/H synthase 2(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM50430948(CHEMBL2337402)
Affinity DataIC50:  14nMAssay Description:Inhibition of COX2 in LPS-stimulated mouse J774 cells assessed as inhibition of PGE2 production and measured after 24 hrs by enzyme immuno-assay (EIA...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProstaglandin G/H synthase 2(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM50589573(CHEMBL5171792)
Affinity DataIC50:  16nMAssay Description:Inhibition of COX2 in LPS-stimulated mouse J774 cells assessed as inhibition of PGE2 production and measured after 24 hrs by enzyme immuno-assay (EIA...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProstaglandin G/H synthase 2(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM50589576(CHEMBL5180584)
Affinity DataIC50:  17nMAssay Description:Inhibition of COX2 in LPS-stimulated mouse J774 cells assessed as inhibition of PGE2 production and measured after 24 hrs by enzyme immuno-assay (EIA...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProstaglandin G/H synthase 2(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM50430960(CHEMBL2337400)
Affinity DataIC50:  17nMAssay Description:Inhibition of COX2 in LPS-stimulated mouse J774 cells assessed as inhibition of PGE2 production and measured after 24 hrs by enzyme immuno-assay (EIA...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProstaglandin G/H synthase 2(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM50589574(CHEMBL5195567)
Affinity DataIC50:  25nMAssay Description:Inhibition of COX2 in LPS-stimulated mouse J774 cells assessed as inhibition of PGE2 production and measured after 24 hrs by enzyme immuno-assay (EIA...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProstaglandin G/H synthase 2(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM50430954(CHEMBL2337407 | US9162979, 36-II)
Affinity DataIC50:  27nMAssay Description:Inhibition of COX2 in LPS-stimulated mouse J774 cells assessed as inhibition of PGE2 production and measured after 24 hrs by enzyme immuno-assay (EIA...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProstaglandin G/H synthase 2(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM50589571(CHEMBL5179625)
Affinity DataIC50:  29nMAssay Description:Inhibition of COX2 in LPS-stimulated mouse J774 cells assessed as inhibition of PGE2 production and measured after 24 hrs by enzyme immuno-assay (EIA...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTranslocator protein(Rattus norvegicus (rat))TBA
LigandPNGBDBM50131733(4-Phenyl-quinoline-2-carboxylic acid benzyl-methyl...)
Affinity DataIC50:  38nMAssay Description:Inhibitory activity against dihydrofolate reductase (DHFR) from Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetTranslocator protein(Rattus norvegicus (rat))TBA
LigandPNGBDBM50054128(2-[2-(4-Chloro-phenyl)-1-oxo-1,2-dihydro-pyrrolo[3...)
Affinity DataIC50:  40nMAssay Description:Inhibition of rat liver Dihydrofolate reductase.More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetTranslocator protein(Rattus norvegicus (rat))TBA
LigandPNGBDBM50059751(8-Benzyl-5-phenyl-8,11-dihydro-6,8-diaza-cyclohept...)
Affinity DataIC50:  45nMAssay Description:Inhibitory activity against Dihydrofolate reductase of Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProstaglandin G/H synthase 2(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM11639(4-[5-(4-methylphenyl)-3-(trifluoromethyl)-1H-pyraz...)
Affinity DataIC50:  61nMAssay Description:Inhibition of COX2 in LPS-stimulated mouse J774 cells assessed as inhibition of PGE2 production and measured after 24 hrs by enzyme immuno-assay (EIA...More data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))TBA
LigandPNGBDBM50131731(4-Phenyl-naphthalene-2-carboxylic acid benzyl-meth...)
Affinity DataIC50:  64nMAssay Description:Inhibitory activity against dihydrofolate reductase (DHFR) from Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProstaglandin G/H synthase 2(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM50589577(CHEMBL5202601)
Affinity DataIC50:  74nMAssay Description:Inhibition of COX2 in LPS-stimulated mouse J774 cells assessed as inhibition of PGE2 production and measured after 24 hrs by enzyme immuno-assay (EIA...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProstaglandin G/H synthase 2(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM50430947(CHEMBL2337409 | US9162979, 37-II)
Affinity DataIC50:  89nMAssay Description:Inhibition of COX2 in LPS-stimulated mouse J774 cells assessed as inhibition of PGE2 production and measured after 24 hrs by enzyme immuno-assay (EIA...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProstaglandin G/H synthase 2(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM50589582(CHEMBL5176195)
Affinity DataIC50:  140nMAssay Description:Inhibition of COX2 in LPS-stimulated mouse J774 cells assessed as inhibition of PGE2 production and measured after 24 hrs by enzyme immuno-assay (EIA...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTranslocator protein(Rattus norvegicus (rat))TBA
LigandPNGBDBM50054130((E)-2-(2-(4-chlorophenyl)-1-oxo-1,2-dihydropyrrolo...)
Affinity DataIC50:  150nMAssay Description:Inhibition of rat liver Dihydrofolate reductase.More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetTranslocator protein(Rattus norvegicus (rat))TBA
LigandPNGBDBM50059740(7-Benzyl-11-phenyl-7,8,9,10-tetrahydro-5,7-diaza-c...)
Affinity DataIC50:  170nMAssay Description:Inhibitory activity against Dihydrofolate reductase of Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetTranslocator protein(Rattus norvegicus (rat))TBA
LigandPNGBDBM50098699(2-[(Benzyl-ethyl-amino)-methyl]-4-phenyl-quinoline...)
Affinity DataIC50:  229nMAssay Description:Evaluated for the inhibition of chicken liver Dihydrofolate reductase by using standard enzyme assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetTranslocator protein(Rattus norvegicus (rat))TBA
LigandPNGBDBM50059744(3-Methyl-4-phenyl-quinoline-2-carboxylic acid sec-...)
Affinity DataIC50:  230nMAssay Description:Inhibition of rat liver Dihydrofolate reductase.More data for this Ligand-Target Pair
In DepthDetails PubMed
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