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Found 390 with Last Name = 'scheiner' and Initial = 'm'
TargetAcetylcholinesterase(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50514053(CHEMBL4441666)
Affinity DataKi:  3.70nMAssay Description:Inhibition of recombinant human AChE assessed as inhibition constant for enzyme-inhibitor complex using acetylthiocholine iodide as substrate preincu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50514053(CHEMBL4441666)
Affinity DataKi:  7.20nMAssay Description:Inhibition of recombinant human AChE assessed as inhibition constant for enzyme-substrate-inhbitor complex using acetylthiocholine iodide as substrat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50281388(CHEMBL4173258)
Affinity DataKi:  11nMAssay Description:Inhibition of human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50514048(CHEMBL4447210)
Affinity DataKi:  17nMAssay Description:Inhibition of recombinant human AChE assessed as inhibition constant for enzyme-inhibitor complex using acetylthiocholine iodide as substrate preincu...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50508994(CHEMBL4589118)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]-LSD from recombinant human 5HT6 receptor expressed in CHOK1 cells measured after 60 mins by microbeta scintillation counting met...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50200170(5-(4-chloro-3-methyl-phenyl)-1-(4-methyl-benzyl)-1...)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]-CP55940 from human recombinant cannabinoid CB2 receptor expressed in human HEK cells by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50514048(CHEMBL4447210)
Affinity DataKi:  28nMAssay Description:Inhibition of recombinant human AChE assessed as inhibition constant for enzyme-substrate-inhbitor complex using acetylthiocholine iodide as substrat...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50244276(2-(4-ethoxybenzyl)-N,N-diethyl-1-isopentyl-1H-benz...)
Affinity DataKi:  37nMAssay Description:Displacement of [3H]-CP55940 from human recombinant cannabinoid CB2 receptor expressed in human HEK cells by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50244276(2-(4-ethoxybenzyl)-N,N-diethyl-1-isopentyl-1H-benz...)
Affinity DataKi:  37nMAssay Description:Binding affinity in human CB2R expressed in human HEK cells incubated for 3 hrs by microbeta scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50514055(CHEMBL4458217)
Affinity DataKi:  39nMAssay Description:Displacement of [3H]-CP55940 from human recombinant cannabinoid CB2 receptor expressed in human HEK cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50458225(Ciproxifan)
Affinity DataKi:  46nMAssay Description:Inhibition of human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50053435(CHEMBL3323035)
Affinity DataKi:  76nMAssay Description:Inhibition of human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50359391(CHEMBL1929421)
Affinity DataKi:  84nMAssay Description:Inhibition of human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50514057(CHEMBL4456083)
Affinity DataKi:  89nMAssay Description:Inhibition of recombinant human AChE assessed as inhibition constant for enzyme-inhibitor complex using acetylthiocholine iodide as substrate preincu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50508998(CHEMBL3747907)
Affinity DataKi:  128nMAssay Description:Inhibition of human histamine H3 receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM21278(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...)
Affinity DataKi:  143nMAssay Description:Displacement of [3H]-CP55940 from human recombinant cannabinoid CB1 receptor expressed in CHO cells by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetAcetylcholinesterase(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50514057(CHEMBL4456083)
Affinity DataKi:  206nMAssay Description:Inhibition of recombinant human AChE assessed as inhibition constant for enzyme-substrate-inhbitor complex using acetylthiocholine iodide as substrat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50509001(CHEMBL4552323)
Affinity DataKi:  240nMAssay Description:Displacement of [3H]-LSD from recombinant human 5HT6 receptor expressed in CHOK1 cells measured after 60 mins by microbeta scintillation counting met...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50200170(5-(4-chloro-3-methyl-phenyl)-1-(4-methyl-benzyl)-1...)
Affinity DataKi:  687nMAssay Description:Displacement of [3H]-CP55940 from human recombinant cannabinoid CB1 receptor expressed in CHO cells by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50514049(CHEMBL4464883)
Affinity DataKi:  2.40E+3nMAssay Description:Displacement of [3H]-CP55940 from human recombinant cannabinoid CB2 receptor expressed in human HEK cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50053441(CHEMBL3323053)
Affinity DataKi:  2.50E+3nMAssay Description:Inhibition of human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50514056(CHEMBL4588547)
Affinity DataKi:  2.50E+3nMAssay Description:Displacement of [3H]-CP55940 from human recombinant cannabinoid CB2 receptor expressed in human HEK cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50514059(CHEMBL4545532)
Affinity DataKi:  3.00E+3nMAssay Description:Displacement of [3H]-CP55940 from human recombinant cannabinoid CB2 receptor expressed in human HEK cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50514051(CHEMBL4453905)
Affinity DataKi:  4.00E+3nMAssay Description:Displacement of [3H]-CP55940 from human recombinant cannabinoid CB2 receptor expressed in human HEK cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50514057(CHEMBL4456083)
Affinity DataKi:  4.30E+3nMAssay Description:Displacement of [3H]-CP55940 from human recombinant cannabinoid CB2 receptor expressed in human HEK cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50514053(CHEMBL4441666)
Affinity DataKi:  5.00E+3nMAssay Description:Displacement of [3H]-CP55940 from human recombinant cannabinoid CB2 receptor expressed in human HEK cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50514048(CHEMBL4447210)
Affinity DataKi:  6.80E+3nMAssay Description:Displacement of [3H]-CP55940 from human recombinant cannabinoid CB2 receptor expressed in human HEK cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50514050(CHEMBL4583716)
Affinity DataKi:  7.30E+3nMAssay Description:Displacement of [3H]-CP55940 from human recombinant cannabinoid CB2 receptor expressed in human HEK cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50514060(CHEMBL4558335)
Affinity DataKi:  9.60E+3nMAssay Description:Displacement of [3H]-CP55940 from human recombinant cannabinoid CB2 receptor expressed in human HEK cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50514052(CHEMBL4555887)
Affinity DataKi:  1.74E+4nMAssay Description:Displacement of [3H]-CP55940 from human recombinant cannabinoid CB2 receptor expressed in human HEK cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50514061(CHEMBL4473438)
Affinity DataKi:  2.69E+4nMAssay Description:Displacement of [3H]-CP55940 from human recombinant cannabinoid CB2 receptor expressed in human HEK cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50514054(CHEMBL4456433)
Affinity DataKi:  2.87E+4nMAssay Description:Displacement of [3H]-CP55940 from human recombinant cannabinoid CB2 receptor expressed in human HEK cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50514058(CHEMBL4458929)
Affinity DataKi:  3.07E+4nMAssay Description:Displacement of [3H]-CP55940 from human recombinant cannabinoid CB2 receptor expressed in human HEK cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50508995(CHEMBL4591636)
Affinity DataKi:  3.53E+4nMAssay Description:Inhibition of alpha4beta2 nAChR (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50508995(CHEMBL4591636)
Affinity DataKi:  6.68E+4nMAssay Description:Inhibition of alpha7 nAChR (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50359391(CHEMBL1929421)
Affinity DataIC50:  0.300nMAssay Description:Inhibition of human MAOAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50579160(CHEMBL4854913)
Affinity DataIC50:  0.410nMAssay Description:Inhibition of human recombinant AChE using acetylthiocholine iodide as a substrate preincubated for 20 mins followed by substrate addition by spectro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50579161(CHEMBL4848527)
Affinity DataIC50:  0.630nMAssay Description:Inhibition of human recombinant AChE using acetylthiocholine iodide as a substrate preincubated for 20 mins followed by substrate addition by spectro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Julius Maximilian University W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50077257((4-Isopropyl-phenyl)-carbamic acid (S)-3a-methyl-1...)
Affinity DataIC50:  1nMAssay Description:Inhibition of human plasma BChE using s-butyrylthiocholine as substrate preincubated for 30 mins followed by substrate addition and measured after 25...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM10592(7-chloro-15-methyl-10-azatetracyclo[11.3.1.0^{2,11...)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of human recombinant AChE using acetylthiocholine iodide as a substrate preincubated for 20 mins followed by substrate addition by spectro...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50579162(CHEMBL4872514)
Affinity DataIC50:  1.30nMAssay Description:Inhibition of human recombinant AChE using acetylthiocholine iodide as a substrate preincubated for 20 mins followed by substrate addition by spectro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50514055(CHEMBL4458217)
Affinity DataIC50:  1.30nMAssay Description:Inhibition of recombinant human AChE using acetylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and measured...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50579158(CHEMBL4866930)
Affinity DataIC50:  1.80nMAssay Description:Inhibition of human recombinant AChE using acetylthiocholine iodide as a substrate preincubated for 20 mins followed by substrate addition by spectro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50514057(CHEMBL4456083)
Affinity DataIC50:  2nMAssay Description:Inhibition of recombinant human AChE using acetylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and measured...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50579159(CHEMBL4863615)
Affinity DataIC50:  2.40nMAssay Description:Inhibition of human recombinant AChE using acetylthiocholine iodide as a substrate preincubated for 20 mins followed by substrate addition by spectro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50579156(CHEMBL4862716)
Affinity DataIC50:  2.40nMAssay Description:Inhibition of human recombinant AChE using acetylthiocholine iodide as a substrate preincubated for 20 mins followed by substrate addition by spectro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Julius Maximilian University W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50514055(CHEMBL4458217)
Affinity DataIC50:  2.5nMAssay Description:Inhibition of human BChE using butyrylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and measured for 3 mins...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50579157(CHEMBL4859103)
Affinity DataIC50:  2.60nMAssay Description:Inhibition of human recombinant AChE using acetylthiocholine iodide as a substrate preincubated for 20 mins followed by substrate addition by spectro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50514053(CHEMBL4441666)
Affinity DataIC50:  3.20nMAssay Description:Inhibition of recombinant human AChE using acetylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and measured...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50514058(CHEMBL4458929)
Affinity DataIC50:  3.20nMAssay Description:Inhibition of recombinant human AChE using acetylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and measured...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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