TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Pfizer
Curated by ChEMBL
Pfizer
Curated by ChEMBL
Affinity DataKi: 0.190nMAssay Description:Binding affinity to Alpha-1 adrenergic receptor by displacement of [3H]prazosinMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Pfizer
Curated by ChEMBL
Pfizer
Curated by ChEMBL
Affinity DataKi: 4.10nMAssay Description:Binding affinity to Alpha-1 adrenergic receptor by displacement of [3H]prazosinMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Pfizer
Curated by ChEMBL
Pfizer
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:Binding affinity to Alpha-1 adrenergic receptor by displacement of [3H]prazosinMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Pfizer
Curated by ChEMBL
Pfizer
Curated by ChEMBL
Affinity DataKi: 160nMAssay Description:Binding affinity to Alpha-1 adrenergic receptor by displacement of [3H]prazosinMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
Pfizer
Curated by ChEMBL
Pfizer
Curated by ChEMBL
Affinity DataKi: 4.83E+3nMAssay Description:Binding affinity to alpha-2 adrenergic receptor by displacement of [3H]clonidineMore data for this Ligand-Target Pair
Affinity DataIC50: 10.2nMAssay Description:Inhibition of rabbit NEPMore data for this Ligand-Target Pair
Affinity DataIC50: 14.3nMAssay Description:Inhibition of rat NEPMore data for this Ligand-Target Pair
Affinity DataIC50: 18.9nMAssay Description:Inhibition of human NEPMore data for this Ligand-Target Pair
Affinity DataIC50: 19nMAssay Description:Inhibitory activity against human platelet microsomal TXA2 synthaseMore data for this Ligand-Target Pair
Affinity DataIC50: 19.7nMAssay Description:Inhibition of human recombinant NEPMore data for this Ligand-Target Pair
Affinity DataIC50: 28nMAssay Description:Inhibitory activity against human platelet microsomal TXA2 synthaseMore data for this Ligand-Target Pair
Affinity DataIC50: 34nMAssay Description:Inhibitory activity against human platelet microsomal TXA2 synthaseMore data for this Ligand-Target Pair
Affinity DataIC50: 48nMAssay Description:Inhibitory activity against human platelet microsomal TXA2 synthaseMore data for this Ligand-Target Pair
Affinity DataIC50: 114nMAssay Description:Inhibition of dog NEPMore data for this Ligand-Target Pair
Affinity DataIC50: 120nMAssay Description:Inhibition of dog NEPMore data for this Ligand-Target Pair
Affinity DataIC50: 124nMAssay Description:Inhibition of dog NEPMore data for this Ligand-Target Pair
Affinity DataIC50: 150nMAssay Description:Inhibition of dog NEPMore data for this Ligand-Target Pair
Affinity DataIC50: 176nMAssay Description:Inhibition of dog NEPMore data for this Ligand-Target Pair
Affinity DataIC50: 184nMAssay Description:Inhibition of dog NEPMore data for this Ligand-Target Pair
Affinity DataIC50: 195nMAssay Description:Inhibition of dog NEPMore data for this Ligand-Target Pair
Affinity DataIC50: 205nMAssay Description:Inhibition of dog NEPMore data for this Ligand-Target Pair
Affinity DataIC50: 213nMAssay Description:Inhibition of dog NEPMore data for this Ligand-Target Pair
Affinity DataIC50: 237nMAssay Description:Inhibition of dog NEPMore data for this Ligand-Target Pair
Affinity DataIC50: 283nMAssay Description:Inhibition of dog NEPMore data for this Ligand-Target Pair
Affinity DataIC50: 286nMAssay Description:Inhibition of dog NEPMore data for this Ligand-Target Pair
Affinity DataIC50: 292nMAssay Description:Inhibition of dog NEPMore data for this Ligand-Target Pair
Affinity DataIC50: 297nMAssay Description:Inhibition of dog NEPMore data for this Ligand-Target Pair
Affinity DataIC50: 313nMAssay Description:Inhibition of dog NEPMore data for this Ligand-Target Pair
Affinity DataIC50: 313nMAssay Description:Inhibition of dog NEPMore data for this Ligand-Target Pair
Affinity DataIC50: 370nMAssay Description:Inhibition of dog NEPMore data for this Ligand-Target Pair
Affinity DataIC50: 374nMAssay Description:Inhibition of dog NEPMore data for this Ligand-Target Pair
Affinity DataIC50: 377nMAssay Description:Inhibition of dog NEPMore data for this Ligand-Target Pair
Affinity DataIC50: 384nMAssay Description:Inhibition of dog NEPMore data for this Ligand-Target Pair
Affinity DataIC50: 530nMAssay Description:Inhibition of dog NEPMore data for this Ligand-Target Pair
Affinity DataIC50: 700nMAssay Description:Inhibition of dog NEPMore data for this Ligand-Target Pair
Affinity DataIC50: 890nMAssay Description:Inhibition of dog NEPMore data for this Ligand-Target Pair
Affinity DataIC50: 1.06E+3nMAssay Description:Inhibition of dog NEPMore data for this Ligand-Target Pair
Affinity DataIC50: 1.14E+3nMAssay Description:Inhibition of dog NEPMore data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of dog NEPMore data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of dog NEPMore data for this Ligand-Target Pair