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Found 33 with Last Name = 'yaqub' and Initial = 'm'
TargetUrease [D459Y,K653P](Canavalia ensiformis (Jack bean))
University of Karachi

LigandPNGBDBM152597(2-(1-(Benzofuran-2-yl)ethylidene)-N-(3-nitrophenyl...)
Affinity DataIC50:  77nMpH: 8.2Assay Description:The mixture of this enzyme inhibition assay was composed of 10 無 of enzyme (5 U/mL) and 10 無 of each test compound in the series (3a-3s) in 40 無 b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease [D459Y,K653P](Canavalia ensiformis (Jack bean))
University of Karachi

LigandPNGBDBM152587(2-(1-(Benzofuran-2-yl)ethylidene)-N-phenylhydrazin...)
Affinity DataIC50:  89nMpH: 8.2Assay Description:The mixture of this enzyme inhibition assay was composed of 10 無 of enzyme (5 U/mL) and 10 無 of each test compound in the series (3a-3s) in 40 無 b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease [D459Y,K653P](Canavalia ensiformis (Jack bean))
University of Karachi

LigandPNGBDBM152600(2-(1-(Benzofuran-2-yl)ethylidene)-N-(3-methoxyphen...)
Affinity DataIC50:  102nMpH: 8.2Assay Description:The mixture of this enzyme inhibition assay was composed of 10 無 of enzyme (5 U/mL) and 10 無 of each test compound in the series (3a-3s) in 40 無 b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5'-nucleotidase(Homo sapiens (Human))
Bahauddin Zakariya University

Curated by ChEMBL
LigandPNGBDBM50561931(CHEMBL4746318)
Affinity DataIC50:  150nMAssay Description:Inhibition of recombinant human ecto-5' nucleotidase expressed in COS7 cell membranes assessed as inorganic phosphate release using AMP as substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrease [D459Y,K653P](Canavalia ensiformis (Jack bean))
University of Karachi

LigandPNGBDBM152591(2-(1-(Benzofuran-2-yl)ethylidene)-N-(4-fluoropheny...)
Affinity DataIC50:  177nMpH: 8.2Assay Description:The mixture of this enzyme inhibition assay was composed of 10 無 of enzyme (5 U/mL) and 10 無 of each test compound in the series (3a-3s) in 40 無 b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5'-nucleotidase(Homo sapiens (Human))
Bahauddin Zakariya University

Curated by ChEMBL
LigandPNGBDBM50561933(CHEMBL4788305)
Affinity DataIC50:  180nMAssay Description:Inhibition of recombinant human ecto-5' nucleotidase expressed in COS7 cell membranes assessed as inorganic phosphate release using AMP as substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrease [D459Y,K653P](Canavalia ensiformis (Jack bean))
University of Karachi

LigandPNGBDBM152598(2-(1-(Benzofuran-2-yl)ethylidene)-N-(4-nitrophenyl...)
Affinity DataIC50:  181nMpH: 8.2Assay Description:The mixture of this enzyme inhibition assay was composed of 10 無 of enzyme (5 U/mL) and 10 無 of each test compound in the series (3a-3s) in 40 無 b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5'-nucleotidase(Rattus norvegicus (Rat))
Bahauddin Zakariya University

Curated by ChEMBL
LigandPNGBDBM50561936(CHEMBL4741833)
Affinity DataIC50:  190nMAssay Description:Inhibition of recombinant rat ecto-5' nucleotidase expressed in COS7 cell membranes assessed as inorganic phosphate release using AMP as substrate uM...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5'-nucleotidase(Homo sapiens (Human))
Bahauddin Zakariya University

Curated by ChEMBL
LigandPNGBDBM50561932(CHEMBL4761451)
Affinity DataIC50:  260nMAssay Description:Inhibition of recombinant human ecto-5' nucleotidase expressed in COS7 cell membranes assessed as inorganic phosphate release using AMP as substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrease [D459Y,K653P](Canavalia ensiformis (Jack bean))
University of Karachi

LigandPNGBDBM57806(1-[1-(1-benzofuran-2-yl)ethylideneamino]-3-(3-meth...)
Affinity DataIC50:  283nMpH: 8.2Assay Description:The mixture of this enzyme inhibition assay was composed of 10 無 of enzyme (5 U/mL) and 10 無 of each test compound in the series (3a-3s) in 40 無 b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease [D459Y,K653P](Canavalia ensiformis (Jack bean))
University of Karachi

LigandPNGBDBM152602(2-(1-(Benzofuran-2-yl)ethylidene)-N-(2-methylpheny...)
Affinity DataIC50:  314nMpH: 8.2Assay Description:The mixture of this enzyme inhibition assay was composed of 10 無 of enzyme (5 U/mL) and 10 無 of each test compound in the series (3a-3s) in 40 無 b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5'-nucleotidase(Homo sapiens (Human))
Bahauddin Zakariya University

Curated by ChEMBL
LigandPNGBDBM50561938(CHEMBL4746633)
Affinity DataIC50:  320nMAssay Description:Inhibition of recombinant human ecto-5' nucleotidase expressed in COS7 cell membranes using AMP as substrate preincubated for 10 mins followed by sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrease [D459Y,K653P](Canavalia ensiformis (Jack bean))
University of Karachi

LigandPNGBDBM152593(2-(1-(Benzofuran-2-yl)ethylidene)-N-(2-fluoropheny...)
Affinity DataIC50:  321nMpH: 8.2Assay Description:The mixture of this enzyme inhibition assay was composed of 10 無 of enzyme (5 U/mL) and 10 無 of each test compound in the series (3a-3s) in 40 無 b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease [D459Y,K653P](Canavalia ensiformis (Jack bean))
University of Karachi

LigandPNGBDBM152594(2-(1-(Benzofuran-2-yl)ethylidene)-N-(2,4-difluorop...)
Affinity DataIC50:  387nMpH: 8.2Assay Description:The mixture of this enzyme inhibition assay was composed of 10 無 of enzyme (5 U/mL) and 10 無 of each test compound in the series (3a-3s) in 40 無 b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5'-nucleotidase(Homo sapiens (Human))
Bahauddin Zakariya University

Curated by ChEMBL
LigandPNGBDBM50561930(CHEMBL4760778)
Affinity DataIC50:  460nMAssay Description:Inhibition of recombinant human ecto-5' nucleotidase expressed in COS7 cell membranes assessed as inorganic phosphate release using AMP as substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5'-nucleotidase(Rattus norvegicus (Rat))
Bahauddin Zakariya University

Curated by ChEMBL
LigandPNGBDBM50561931(CHEMBL4746318)
Affinity DataIC50:  520nMAssay Description:Inhibition of recombinant rat ecto-5' nucleotidase expressed in COS7 cell membranes assessed as inorganic phosphate release using AMP as substrate uM...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrease [D459Y,K653P](Canavalia ensiformis (Jack bean))
University of Karachi

LigandPNGBDBM152596(2-(1-(Benzofuran-2-yl)ethylidene)-N-(2-bromophenyl...)
Affinity DataIC50:  564nMpH: 8.2Assay Description:The mixture of this enzyme inhibition assay was composed of 10 無 of enzyme (5 U/mL) and 10 無 of each test compound in the series (3a-3s) in 40 無 b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease [D459Y,K653P](Canavalia ensiformis (Jack bean))
University of Karachi

LigandPNGBDBM152589(2-(1-(Benzofuran-2-yl)ethylidene)-N-(2,4-dichlorop...)
Affinity DataIC50:  592nMpH: 8.2Assay Description:The mixture of this enzyme inhibition assay was composed of 10 無 of enzyme (5 U/mL) and 10 無 of each test compound in the series (3a-3s) in 40 無 b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5'-nucleotidase(Rattus norvegicus (Rat))
Bahauddin Zakariya University

Curated by ChEMBL
LigandPNGBDBM50561934(CHEMBL4753669)
Affinity DataIC50:  680nMAssay Description:Inhibition of recombinant rat ecto-5' nucleotidase expressed in COS7 cell membranes assessed as inorganic phosphate release using AMP as substrate uM...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5'-nucleotidase(Homo sapiens (Human))
Bahauddin Zakariya University

Curated by ChEMBL
LigandPNGBDBM50561929(CHEMBL4797703)
Affinity DataIC50:  690nMAssay Description:Inhibition of recombinant human ecto-5' nucleotidase expressed in COS7 cell membranes assessed as inorganic phosphate release using AMP as substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrease [D459Y,K653P](Canavalia ensiformis (Jack bean))
University of Karachi

LigandPNGBDBM152603(N-Allyl-2-(1-(benzofuran-2-yl)ethylidene)hydrazine...)
Affinity DataIC50:  694nMpH: 8.2Assay Description:The mixture of this enzyme inhibition assay was composed of 10 無 of enzyme (5 U/mL) and 10 無 of each test compound in the series (3a-3s) in 40 無 b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrease [D459Y,K653P](Canavalia ensiformis (Jack bean))
University of Karachi

LigandPNGBDBM152588(2-(1-(Benzofuran-2-yl)ethylidene)-N-(3-chloropheny...)
Affinity DataIC50:  1.13E+3nMpH: 8.2Assay Description:The mixture of this enzyme inhibition assay was composed of 10 無 of enzyme (5 U/mL) and 10 無 of each test compound in the series (3a-3s) in 40 無 b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease [D459Y,K653P](Canavalia ensiformis (Jack bean))
University of Karachi

LigandPNGBDBM152592(2-(1-(Benzofuran-2-yl)ethylidene)-N-(3-fluoropheny...)
Affinity DataIC50:  1.15E+3nMpH: 8.2Assay Description:The mixture of this enzyme inhibition assay was composed of 10 無 of enzyme (5 U/mL) and 10 無 of each test compound in the series (3a-3s) in 40 無 b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5'-nucleotidase(Rattus norvegicus (Rat))
Bahauddin Zakariya University

Curated by ChEMBL
LigandPNGBDBM50561937(CHEMBL4780721)
Affinity DataIC50:  1.56E+3nMAssay Description:Inhibition of recombinant rat ecto-5' nucleotidase expressed in COS7 cell membranes assessed as inorganic phosphate release using AMP as substrate uM...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrease [D459Y,K653P](Canavalia ensiformis (Jack bean))
University of Karachi

LigandPNGBDBM152590(2-(1-(Benzofuran-2-yl)ethylidene)-N-(2,5-dichlorop...)
Affinity DataIC50:  2.01E+3nMpH: 8.2Assay Description:The mixture of this enzyme inhibition assay was composed of 10 無 of enzyme (5 U/mL) and 10 無 of each test compound in the series (3a-3s) in 40 無 b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5'-nucleotidase(Rattus norvegicus (Rat))
Bahauddin Zakariya University

Curated by ChEMBL
LigandPNGBDBM50561935(CHEMBL4761355)
Affinity DataIC50:  2.12E+3nMAssay Description:Inhibition of recombinant rat ecto-5' nucleotidase expressed in COS7 cell membranes assessed as inorganic phosphate release using AMP as substrate uM...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrease [D459Y,K653P](Canavalia ensiformis (Jack bean))
University of Karachi

LigandPNGBDBM152599(2-(1-(Benzofuran-2-yl)ethylidene)-N-(4-methoxyphen...)
Affinity DataIC50:  2.61E+3nMpH: 8.2Assay Description:The mixture of this enzyme inhibition assay was composed of 10 無 of enzyme (5 U/mL) and 10 無 of each test compound in the series (3a-3s) in 40 無 b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease [D459Y,K653P](Canavalia ensiformis (Jack bean))
University of Karachi

LigandPNGBDBM114552(1-[(E)-1-(1-benzofuran-2-yl)ethylideneamino]-3-(4-...)
Affinity DataIC50:  3.47E+3nMpH: 8.2Assay Description:The mixture of this enzyme inhibition assay was composed of 10 無 of enzyme (5 U/mL) and 10 無 of each test compound in the series (3a-3s) in 40 無 b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5'-nucleotidase(Rattus norvegicus (Rat))
Bahauddin Zakariya University

Curated by ChEMBL
LigandPNGBDBM50561933(CHEMBL4788305)
Affinity DataIC50:  3.56E+3nMAssay Description:Inhibition of recombinant rat ecto-5' nucleotidase expressed in COS7 cell membranes assessed as inorganic phosphate release using AMP as substrate uM...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5'-nucleotidase(Rattus norvegicus (Rat))
Bahauddin Zakariya University

Curated by ChEMBL
LigandPNGBDBM50561932(CHEMBL4761451)
Affinity DataIC50:  5.01E+3nMAssay Description:Inhibition of recombinant rat ecto-5' nucleotidase expressed in COS7 cell membranes assessed as inorganic phosphate release using AMP as substrate uM...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5'-nucleotidase(Rattus norvegicus (Rat))
Bahauddin Zakariya University

Curated by ChEMBL
LigandPNGBDBM50561930(CHEMBL4760778)
Affinity DataIC50:  7.99E+3nMAssay Description:Inhibition of recombinant rat ecto-5' nucleotidase expressed in COS7 cell membranes assessed as inorganic phosphate release using AMP as substrate uM...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrease [D459Y,K653P](Canavalia ensiformis (Jack bean))
University of Karachi

LigandPNGBDBM152595(2-(1-(Benzofuran-2-yl)ethylidene)-N-(3-bromophenyl...)
Affinity DataIC50:  1.09E+4nMpH: 8.2Assay Description:The mixture of this enzyme inhibition assay was composed of 10 無 of enzyme (5 U/mL) and 10 無 of each test compound in the series (3a-3s) in 40 無 b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease [D459Y,K653P](Canavalia ensiformis (Jack bean))
University of Karachi

LigandPNGBDBM152601(2-(1-(Benzofuran-2-yl)ethylidene)-N-(2-methoxyphen...)
Affinity DataIC50:  2.40E+4nMpH: 8.2Assay Description:The mixture of this enzyme inhibition assay was composed of 10 無 of enzyme (5 U/mL) and 10 無 of each test compound in the series (3a-3s) in 40 無 b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed