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Found 140 with Last Name = 'abu-serie' and Initial = 'mm'
TargetAcetylcholinesterase(Homo sapiens (Human))
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50509708(CHEMBL4458648)
Affinity DataKi:  121nMAssay Description:Mixed type inhibition of recombinant human AChE assessed as dissociation constant using acetylthiocholine iodide as substrate incubated for 10 mins b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50509708(CHEMBL4458648)
Affinity DataKi:  253nMAssay Description:Mixed type inhibition of recombinant human AChE assessed as dissociation constant for enzyme-substrate-inhibitor complex using acetylthiocholine iodi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50572694(CHEMBL4854379)
Affinity DataIC50:  0.570nMAssay Description:Inhibition of MMP9 (unknown origin) by colorimetric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50327224(4-Benzyl-[1,2,4]triazolo[4,3-a]quinoxaline | CHEMB...)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of MAO-A (unknown origin) by multi-well spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha/RAC-beta/RAC-gamma serine/threonine-protein kinase(Homo sapiens (Human))
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50550738(CHEMBL4792262)
Affinity DataIC50:  1.30nMAssay Description:Inhibition of human AKT assessed as inhibition of substrate phosphorylation using AKTide-2T as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha/RAC-beta/RAC-gamma serine/threonine-protein kinase(Homo sapiens (Human))
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50550740(CHEMBL4780030)
Affinity DataIC50:  2.10nMAssay Description:Inhibition of human AKT assessed as inhibition of substrate phosphorylation using AKTide-2T as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50572691(CHEMBL4862110)
Affinity DataIC50:  4.5nMAssay Description:Inhibition of MMP9 (unknown origin) by colorimetric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50550738(CHEMBL4792262)
Affinity DataIC50:  4.5nMAssay Description:Inhibition of MMP-9 (unknown origin) by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50572689(CHEMBL4871376)
Affinity DataIC50:  5.10nMAssay Description:Inhibition of MMP9 (unknown origin) by colorimetric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073514(CHEMBL3408913)
Affinity DataIC50:  5.30nMAssay Description:Inhibition of MAO-A (unknown origin) by multi-well spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50572690(CHEMBL4852596)
Affinity DataIC50:  5.40nMAssay Description:Inhibition of MAO-A (unknown origin) by multi-well spectrophotometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50550740(CHEMBL4780030)
Affinity DataIC50:  5.60nMAssay Description:Inhibition of MMP-9 (unknown origin) by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50572690(CHEMBL4852596)
Affinity DataIC50:  6.80nMAssay Description:Inhibition of MAO-B (unknown origin) by fluorometric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50572689(CHEMBL4871376)
Affinity DataIC50:  7.10nMAssay Description:Inhibition of MAO-B (unknown origin) by fluorometric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50550739(CHEMBL4788683)
Affinity DataIC50:  7.5nMAssay Description:Inhibition of MMP-9 (unknown origin) by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50572690(CHEMBL4852596)
Affinity DataIC50:  8.40nMAssay Description:Inhibition of MMP9 (unknown origin) by colorimetric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRAC-alpha/RAC-beta/RAC-gamma serine/threonine-protein kinase(Homo sapiens (Human))
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50550739(CHEMBL4788683)
Affinity DataIC50:  8.80nMAssay Description:Inhibition of human AKT assessed as inhibition of substrate phosphorylation using AKTide-2T as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThioredoxin reductase 1, cytoplasmic(Homo sapiens (Human))
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50576853(CHEMBL4859206)
Affinity DataIC50:  9.20nMAssay Description:Inhibition of TrxR1 (unknown origin) assessed as reduction in DTNB to TNB by colorimetric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThioredoxin reductase 1, cytoplasmic(Homo sapiens (Human))
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50576853(CHEMBL4859206)
Affinity DataIC50:  9.20nMAssay Description:Inhibition of TrxR1 (unknown origin) assessed as reduction in DTNB to TNB by colorimetric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50572692(CHEMBL4878125)
Affinity DataIC50:  9.30nMAssay Description:Inhibition of MMP9 (unknown origin) by colorimetric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50572689(CHEMBL4871376)
Affinity DataIC50:  10nMAssay Description:Inhibition of MAO-A (unknown origin) by multi-well spectrophotometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNADPH oxidase 4(Homo sapiens (Human))
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50576853(CHEMBL4859206)
Affinity DataIC50:  11nMAssay Description:Inhibition of human NADPH oxidase 4 by quantitative sandwich enzyme immunoassay techniqueMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNADPH oxidase 4(Homo sapiens (Human))
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50576853(CHEMBL4859206)
Affinity DataIC50:  11nMAssay Description:Inhibition of human NADPH oxidase 4 by quantitative sandwich enzyme immunoassay techniqueMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit alpha(Homo sapiens (Human))
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50576853(CHEMBL4859206)
Affinity DataIC50:  11nMAssay Description:Inhibition of IKKalpha (unknown origin) by ADP-Glo kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit alpha(Homo sapiens (Human))
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50576851(CHEMBL1876217)
Affinity DataIC50:  11nMAssay Description:Inhibition of IKKalpha (unknown origin) by ADP-Glo kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit alpha(Homo sapiens (Human))
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50576853(CHEMBL4859206)
Affinity DataIC50:  11nMAssay Description:Inhibition of IKKalpha (unknown origin) by ADP-Glo kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit alpha(Homo sapiens (Human))
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50576851(CHEMBL1876217)
Affinity DataIC50:  11nMAssay Description:Inhibition of IKKalpha (unknown origin) by ADP-Glo kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50572692(CHEMBL4878125)
Affinity DataIC50:  11nMAssay Description:Inhibition of MAO-B (unknown origin) by fluorometric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50572691(CHEMBL4862110)
Affinity DataIC50:  11nMAssay Description:Inhibition of MAO-B (unknown origin) by fluorometric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50572691(CHEMBL4862110)
Affinity DataIC50:  12nMAssay Description:Inhibition of MAO-A (unknown origin) by multi-well spectrophotometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThioredoxin reductase 1, cytoplasmic(Homo sapiens (Human))
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50576851(CHEMBL1876217)
Affinity DataIC50:  13nMAssay Description:Inhibition of TrxR1 (unknown origin) assessed as reduction in DTNB to TNB by colorimetric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThioredoxin reductase 1, cytoplasmic(Homo sapiens (Human))
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50576851(CHEMBL1876217)
Affinity DataIC50:  13nMAssay Description:Inhibition of TrxR1 (unknown origin) assessed as reduction in DTNB to TNB by colorimetric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073542(CHEMBL3408929)
Affinity DataIC50:  15nMAssay Description:Inhibition of MAO-A (unknown origin) by multi-well spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNADPH oxidase 4(Homo sapiens (Human))
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50576851(CHEMBL1876217)
Affinity DataIC50:  16nMAssay Description:Inhibition of human NADPH oxidase 4 by quantitative sandwich enzyme immunoassay techniqueMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit alpha(Homo sapiens (Human))
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50576852(CHEMBL4849098)
Affinity DataIC50:  16nMAssay Description:Inhibition of IKKalpha (unknown origin) by ADP-Glo kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit alpha(Homo sapiens (Human))
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50576852(CHEMBL4849098)
Affinity DataIC50:  16nMAssay Description:Inhibition of IKKalpha (unknown origin) by ADP-Glo kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNADPH oxidase 4(Homo sapiens (Human))
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50576851(CHEMBL1876217)
Affinity DataIC50:  16nMAssay Description:Inhibition of human NADPH oxidase 4 by quantitative sandwich enzyme immunoassay techniqueMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThioredoxin reductase 1, cytoplasmic(Homo sapiens (Human))
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50576852(CHEMBL4849098)
Affinity DataIC50:  18nMAssay Description:Inhibition of TrxR1 (unknown origin) assessed as reduction in DTNB to TNB by colorimetric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThioredoxin reductase 1, cytoplasmic(Homo sapiens (Human))
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50576852(CHEMBL4849098)
Affinity DataIC50:  18nMAssay Description:Inhibition of TrxR1 (unknown origin) assessed as reduction in DTNB to TNB by colorimetric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNADPH oxidase 4(Homo sapiens (Human))
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50576852(CHEMBL4849098)
Affinity DataIC50:  22nMAssay Description:Inhibition of human NADPH oxidase 4 by quantitative sandwich enzyme immunoassay techniqueMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNADPH oxidase 4(Homo sapiens (Human))
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50576852(CHEMBL4849098)
Affinity DataIC50:  22nMAssay Description:Inhibition of human NADPH oxidase 4 by quantitative sandwich enzyme immunoassay techniqueMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073514(CHEMBL3408913)
Affinity DataIC50:  23nMAssay Description:Inhibition of MMP9 (unknown origin) by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50572692(CHEMBL4878125)
Affinity DataIC50:  24nMAssay Description:Inhibition of MAO-A (unknown origin) by multi-well spectrophotometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50509709(CHEMBL4441059)
Affinity DataIC50:  26nMAssay Description:Inhibition of human serum BChE using butyrylthiocholine iodide as substrate pre-incubated for 20 mins before substrate addition and measured for 180 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073514(CHEMBL3408913)
Affinity DataIC50:  29nMAssay Description:Inhibition of MAO-B (unknown origin) by fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Alexandria University

Curated by ChEMBL
LigandPNGBDBM13080(CGS 27023A Analog 3 | N-hydroxy-2-[(4-methoxybenze...)
Affinity DataIC50:  31nMAssay Description:Inhibition of MMP-1 (unknown origin) by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50509708(CHEMBL4458648)
Affinity DataIC50:  33nMAssay Description:Inhibition of human serum BChE using butyrylthiocholine iodide as substrate pre-incubated for 20 mins before substrate addition and measured for 180 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50509718(CHEMBL4466829)
Affinity DataIC50:  36nMAssay Description:Inhibition of human serum BChE using butyrylthiocholine iodide as substrate pre-incubated for 20 mins before substrate addition and measured for 180 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50509705(CHEMBL4444030)
Affinity DataIC50:  39nMAssay Description:Inhibition of human serum BChE using butyrylthiocholine iodide as substrate pre-incubated for 20 mins before substrate addition and measured for 180 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Alexandria University

Curated by ChEMBL
LigandPNGBDBM17638(2-{1-[(4-chlorophenyl)carbonyl]-5-methoxy-2-methyl...)
Affinity DataIC50:  39nMAssay Description:Inhibition of ovine COX -1 by colorimetric inhibitor screening assay kit methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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