Compile Data Set for Download or QSAR
maximum 50k data
Found 37 with Last Name = 'lodewyk' and Initial = 'mw'
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50497944(CHEMBL3323418)
Affinity DataIC50:  900nMAssay Description:Correction of defective trafficking of human deltaF508 mutant CFTR protein expressed in FRT epithelial cells coexpressing YFP-H148Q/I152L protein ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50497947(CHEMBL3323415)
Affinity DataIC50:  2.10E+3nMAssay Description:Correction of defective trafficking of human deltaF508 mutant CFTR protein expressed in FRT epithelial cells coexpressing YFP-H148Q/I152L protein ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50497960(CHEMBL3323413)
Affinity DataIC50:  2.20E+3nMAssay Description:Correction of defective trafficking of human deltaF508 mutant CFTR protein expressed in FRT epithelial cells coexpressing YFP-H148Q/I152L protein ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50482138(CHEMBL495336)
Affinity DataIC50:  2.30E+3nMAssay Description:Correction of defective trafficking of human deltaF508 mutant CFTR protein expressed in FRT epithelial cells coexpressing YFP-H148Q/I152L protein ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50497962(CHEMBL3323408)
Affinity DataIC50:  2.90E+3nMAssay Description:Correction of defective trafficking of human deltaF508 mutant CFTR protein expressed in FRT epithelial cells coexpressing YFP-H148Q/I152L protein ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50497946(CHEMBL3323414)
Affinity DataIC50:  3.60E+3nMAssay Description:Correction of defective trafficking of human deltaF508 mutant CFTR protein expressed in FRT epithelial cells coexpressing YFP-H148Q/I152L protein ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50497952(CHEMBL3323405)
Affinity DataIC50:  4.10E+3nMAssay Description:Correction of defective trafficking of human deltaF508 mutant CFTR protein expressed in FRT epithelial cells coexpressing YFP-H148Q/I152L protein ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50497953(CHEMBL3323406)
Affinity DataIC50:  4.50E+3nMAssay Description:Correction of defective trafficking of human deltaF508 mutant CFTR protein expressed in FRT epithelial cells coexpressing YFP-H148Q/I152L protein ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50497951(CHEMBL3323403)
Affinity DataIC50:  4.80E+3nMAssay Description:Correction of defective trafficking of human deltaF508 mutant CFTR protein expressed in FRT epithelial cells coexpressing YFP-H148Q/I152L protein ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50497948(CHEMBL3323417)
Affinity DataIC50:  5.20E+3nMAssay Description:Correction of defective trafficking of human deltaF508 mutant CFTR protein expressed in FRT epithelial cells coexpressing YFP-H148Q/I152L protein ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50497961(CHEMBL3323416)
Affinity DataIC50:  5.20E+3nMAssay Description:Correction of defective trafficking of human deltaF508 mutant CFTR protein expressed in FRT epithelial cells coexpressing YFP-H148Q/I152L protein ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50497950(CHEMBL3323400)
Affinity DataIC50:  5.80E+3nMAssay Description:Correction of defective trafficking of human deltaF508 mutant CFTR protein expressed in FRT epithelial cells coexpressing YFP-H148Q/I152L protein ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50289704(CHEMBL260775)
Affinity DataIC50:  6.00E+3nMAssay Description:Correction of defective trafficking of human deltaF508 mutant CFTR protein expressed in FRT epithelial cells coexpressing YFP-H148Q/I152L protein ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50497943(CHEMBL3323410)
Affinity DataIC50:  6.60E+3nMAssay Description:Correction of defective trafficking of human deltaF508 mutant CFTR protein expressed in FRT epithelial cells coexpressing YFP-H148Q/I152L protein ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50497942(CHEMBL3323401)
Affinity DataIC50:  6.60E+3nMAssay Description:Correction of defective trafficking of human deltaF508 mutant CFTR protein expressed in FRT epithelial cells coexpressing YFP-H148Q/I152L protein ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50497954(CHEMBL3323411)
Affinity DataIC50:  6.90E+3nMAssay Description:Correction of defective trafficking of human deltaF508 mutant CFTR protein expressed in FRT epithelial cells coexpressing YFP-H148Q/I152L protein ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50497958(CHEMBL3323412)
Affinity DataIC50:  7.20E+3nMAssay Description:Correction of defective trafficking of human deltaF508 mutant CFTR protein expressed in FRT epithelial cells coexpressing YFP-H148Q/I152L protein ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50497959(CHEMBL3323409)
Affinity DataIC50:  8.30E+3nMAssay Description:Correction of defective trafficking of human deltaF508 mutant CFTR protein expressed in FRT epithelial cells coexpressing YFP-H148Q/I152L protein ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50497957(CHEMBL3323407)
Affinity DataIC50:  8.70E+3nMAssay Description:Correction of defective trafficking of human deltaF508 mutant CFTR protein expressed in FRT epithelial cells coexpressing YFP-H148Q/I152L protein ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50497956(CHEMBL3323402)
Affinity DataIC50:  8.80E+3nMAssay Description:Correction of defective trafficking of human deltaF508 mutant CFTR protein expressed in FRT epithelial cells coexpressing YFP-H148Q/I152L protein ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50497949(CHEMBL3323399)
Affinity DataIC50:  8.90E+3nMAssay Description:Correction of defective trafficking of human deltaF508 mutant CFTR protein expressed in FRT epithelial cells coexpressing YFP-H148Q/I152L protein ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50497945(CHEMBL3323404)
Affinity DataIC50:  9.20E+3nMAssay Description:Correction of defective trafficking of human deltaF508 mutant CFTR protein expressed in FRT epithelial cells coexpressing YFP-H148Q/I152L protein ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50497955(CHEMBL3323398)
Affinity DataIC50:  1.10E+4nMAssay Description:Correction of defective trafficking of human deltaF508 mutant CFTR protein expressed in FRT epithelial cells coexpressing YFP-H148Q/I152L protein ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50289534(CHEMBL2018574)
Affinity DataEC50:  2.20E+3nMAssay Description:Activity at human CFTR delta F508 mutant expressed in forskolin-stimulated FRT cells assessed as increase in iodine influx measured as decrease in YF...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50290134(CHEMBL2018580)
Affinity DataEC50:  4.20E+3nMAssay Description:Activity at human CFTR delta F508 mutant expressed in forskolin-stimulated FRT cells assessed as increase in iodine influx measured as decrease in YF...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50289860(CHEMBL2018582)
Affinity DataEC50:  6.70E+3nMAssay Description:Activity at human CFTR delta F508 mutant expressed in forskolin-stimulated FRT cells assessed as increase in iodine influx measured as decrease in YF...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50290145(CHEMBL2018584)
Affinity DataEC50:  3.70E+3nMAssay Description:Activity at human CFTR delta F508 mutant expressed in forskolin-stimulated FRT cells assessed as increase in iodine influx measured as decrease in YF...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50289868(CHEMBL2018590)
Affinity DataEC50:  4.30E+3nMAssay Description:Activity at human CFTR delta F508 mutant expressed in forskolin-stimulated FRT cells assessed as increase in iodine influx measured as decrease in YF...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50289861(CHEMBL2018583)
Affinity DataEC50:  2.70E+3nMAssay Description:Activity at human CFTR delta F508 mutant expressed in forskolin-stimulated FRT cells assessed as increase in iodine influx measured as decrease in YF...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50290132(CHEMBL2018577)
Affinity DataEC50:  2.70E+3nMAssay Description:Activity at human CFTR delta F508 mutant expressed in forskolin-stimulated FRT cells assessed as increase in iodine influx measured as decrease in YF...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50290144(CHEMBL2018578)
Affinity DataEC50:  7.30E+3nMAssay Description:Activity at human CFTR delta F508 mutant expressed in forskolin-stimulated FRT cells assessed as increase in iodine influx measured as decrease in YF...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50290147(CHEMBL2018589)
Affinity DataEC50:  4.60E+3nMAssay Description:Activity at human CFTR delta F508 mutant expressed in forskolin-stimulated FRT cells assessed as increase in iodine influx measured as decrease in YF...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50289859(CHEMBL2018581)
Affinity DataEC50:  1.50E+3nMAssay Description:Activity at human CFTR delta F508 mutant expressed in forskolin-stimulated FRT cells assessed as increase in iodine influx measured as decrease in YF...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50290130(CHEMBL2018575)
Affinity DataEC50:  3.00E+3nMAssay Description:Activity at human CFTR delta F508 mutant expressed in forskolin-stimulated FRT cells assessed as increase in iodine influx measured as decrease in YF...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50289959(CHEMBL2018593)
Affinity DataEC50:  8.20E+3nMAssay Description:Activity at human CFTR delta F508 mutant expressed in forskolin-stimulated FRT cells assessed as increase in iodine influx measured as decrease in YF...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50289958(CHEMBL2018592)
Affinity DataEC50:  3.00E+3nMAssay Description:Activity at human CFTR delta F508 mutant expressed in forskolin-stimulated FRT cells assessed as increase in iodine influx measured as decrease in YF...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM75164(MLS001204421 | N-[2-(3-Cyano-5,7-dimethyl-quinolin...)
Affinity DataEC50:  1.10E+4nMAssay Description:Activity at human CFTR delta F508 mutant expressed in forskolin-stimulated FRT cells assessed as increase in iodine influx measured as decrease in YF...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed