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Found 1190 with Last Name = 'khan' and Initial = 'n'
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
University of Washington

Curated by PDSP Ki Database
LigandPNGBDBM78940(METHIOTHEPIN | MLS000859918 | Methiothepin mesylat...)
Affinity DataKi:  0.420nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Hacettepe University

Curated by ChEMBL
LigandPNGBDBM50304157(3-(2-Thienyl)-2-thiocarbamoyl-2,3,4,5,6,7-hexahydr...)
Affinity DataKi:  0.900nMAssay Description:Competitive inhibition of MAOB in rat liver homogenate by spectrophotometricallyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Hacettepe University

Curated by ChEMBL
LigandPNGBDBM50304152(3-(2-Furyl)-2-thiocarbamoyl-2,3,4,5,6,7-hexahydro-...)
Affinity DataKi:  0.960nMAssay Description:Competitive inhibition of MAOB in rat liver homogenate by spectrophotometricallyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Hacettepe University

Curated by ChEMBL
LigandPNGBDBM50557363(CHEMBL4757953)
Affinity DataKi:  1nMAssay Description:Inhibition of recombinant human MAO-A expressed in baculovirus infected BTI insect cells using p-tyramine as substrate incubated for 30 mins by Ample...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Hacettepe University

Curated by ChEMBL
LigandPNGBDBM50557368(CHEMBL4762228)
Affinity DataKi:  1nMAssay Description:Inhibition of recombinant human MAO-A expressed in baculovirus infected BTI insect cells using p-tyramine as substrate incubated for 30 mins by Ample...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Hacettepe University

Curated by ChEMBL
LigandPNGBDBM50557366(CHEMBL4787184)
Affinity DataKi:  1nMAssay Description:Inhibition of recombinant human MAO-A expressed in baculovirus infected BTI insect cells using p-tyramine as substrate incubated for 30 mins by Ample...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Hacettepe University

Curated by ChEMBL
LigandPNGBDBM50557361(CHEMBL4761363)
Affinity DataKi:  1nMAssay Description:Inhibition of recombinant human MAO-A expressed in baculovirus infected BTI insect cells using p-tyramine as substrate incubated for 30 mins by Ample...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Hacettepe University

Curated by ChEMBL
LigandPNGBDBM50557339(CHEMBL4748517)
Affinity DataKi:  1nMAssay Description:Inhibition of recombinant human MAO-A expressed in baculovirus infected BTI insect cells using p-tyramine as substrate incubated for 30 mins by Ample...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Hacettepe University

Curated by ChEMBL
LigandPNGBDBM50557360(CHEMBL4787516)
Affinity DataKi:  1nMAssay Description:Inhibition of recombinant human MAO-A expressed in baculovirus infected BTI insect cells using p-tyramine as substrate incubated for 30 mins by Ample...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50337403(CHEMBL1682668 | methyl 1-(((1R,2S)-2-(benzyl(methy...)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]Lu AE93103 from human NK3 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50337411((1S,2R)-1-(3,4-dichlorophenyl)-N-(4-fluorobenzyl)-...)
Affinity DataKi:  1.80nMAssay Description:Displacement of [3H]Lu AE93103 from human NK3 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
University of Washington

Curated by PDSP Ki Database
LigandPNGBDBM22872(1-(3-chloro-5,6-dihydrobenzo[b][1]benzothiepin-5-y...)
Affinity DataKi:  1.80nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50337418((1S,2R)-1-(3,4-dichlorophenyl)-2-((3-(4-(N,N-dimet...)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]Lu AE93103 from human NK3 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
University of Washington

Curated by PDSP Ki Database
LigandPNGBDBM22872(1-(3-chloro-5,6-dihydrobenzo[b][1]benzothiepin-5-y...)
Affinity DataKi:  2.60nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50337404((1S,2R)-N-benzyl-1-(3,4-dichlorophenyl)-2-((4-(3,3...)
Affinity DataKi:  2.80nMAssay Description:Displacement of [3H]Lu AE93103 from human NK3 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50337409((1S,2R)-1-(3,4-dichlorophenyl)-N-(4-fluorobenzyl)-...)
Affinity DataKi:  3.30nMAssay Description:Displacement of [3H]Lu AE93103 from human NK3 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50337407(CHEMBL1682672 | N1-(1-(((1R,2S)-2-(benzyl(methyl)c...)
Affinity DataKi:  3.60nMAssay Description:Displacement of [3H]Lu AE93103 from human NK3 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50337410((1S,2R)-1-(3,4-dichlorophenyl)-N-(4-fluorobenzyl)-...)
Affinity DataKi:  3.70nMAssay Description:Displacement of [3H]Lu AE93103 from human NK3 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Hacettepe University

Curated by ChEMBL
LigandPNGBDBM50557330(CHEMBL4794193)
Affinity DataKi:  4nMAssay Description:Inhibition of recombinant human MAO-A expressed in baculovirus infected BTI insect cells using p-tyramine as substrate incubated for 30 mins by Ample...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Hacettepe University

Curated by ChEMBL
LigandPNGBDBM50557362(CHEMBL4764828)
Affinity DataKi:  4nMAssay Description:Inhibition of recombinant human MAO-A expressed in baculovirus infected BTI insect cells using p-tyramine as substrate incubated for 30 mins by Ample...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Hacettepe University

Curated by ChEMBL
LigandPNGBDBM50557355(CHEMBL4788778)
Affinity DataKi:  4nMAssay Description:Inhibition of recombinant human MAO-A expressed in baculovirus infected BTI insect cells using p-tyramine as substrate incubated for 30 mins by Ample...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50337401((1S,2R)-N-benzyl-1-(3,4-dichlorophenyl)-N-methyl-2...)
Affinity DataKi:  4.20nMAssay Description:Displacement of [3H]Lu AE93103 from human NK3 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Hacettepe University

Curated by ChEMBL
LigandPNGBDBM50304156(3-(2-Furyl)-2-(N-phenyllthiocarbamoyl)-3,3a,4,5,6,...)
Affinity DataKi:  4.22nMAssay Description:Competitive inhibition of MAOA in rat liver homogenate by spectrophotometricallyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50337435(CHEMBL1682637 | rac-2-((4-acetamido-4-phenylpiperi...)
Affinity DataKi:  4.60nMAssay Description:Displacement of [3H]Lu AE93103 from human NK3 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Hacettepe University

Curated by ChEMBL
LigandPNGBDBM50029816(5-Chloro-pyridine-2-carboxylic acid (2-amino-ethyl...)
Affinity DataKi:  5nMAssay Description:Inhibition of recombinant human MAO-B expressed in baculovirus infected BTI insect cells using p-tyramine as substrate incubated for 30 mins by Ample...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Hacettepe University

Curated by ChEMBL
LigandPNGBDBM50557341(CHEMBL4744188)
Affinity DataKi:  5nMAssay Description:Inhibition of recombinant human MAO-A expressed in baculovirus infected BTI insect cells using p-tyramine as substrate incubated for 30 mins by Ample...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50337425(CHEMBL1682628 | rac-2-((4-acetamido-4-phenylpiperi...)
Affinity DataKi:  5.30nMAssay Description:Displacement of [3H]Lu AE93103 from human NK3 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Hacettepe University

Curated by ChEMBL
LigandPNGBDBM15613(4-chloro-N-(2-morpholin-4-ylethyl)benzamide | 4-ch...)
Affinity DataKi:  5.53nMAssay Description:Competitive inhibition of MAOA in rat liver homogenate by spectrophotometricallyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50337405((1S,2R)-N-benzyl-1-(3,4-dichlorophenyl)-N-methyl-2...)
Affinity DataKi:  5.60nMAssay Description:Displacement of [3H]Lu AE93103 from human NK3 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50337431((1S,2R)-2-((4-acetamido-4-phenylpiperidin-1-yl)met...)
Affinity DataKi:  5.80nMAssay Description:Displacement of [3H]Lu AE93103 from human NK3 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50337416((1S,2R)-1-(3,4-dichlorophenyl)-N-(4-fluorobenzyl)-...)
Affinity DataKi:  5.80nMAssay Description:Displacement of [3H]Lu AE93103 from human NK3 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50337441(CHEMBL1682643 | rac-2-((4-acetamido-4-phenylpiperi...)
Affinity DataKi:  5.90nMAssay Description:Displacement of [3H]Lu AE93103 from human NK3 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50337421((1S,2R)-2-((4-acetamido-4-phenylpiperidin-1-yl)met...)
Affinity DataKi:  5.90nMAssay Description:Displacement of [3H]Lu AE93103 from human NK3 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50337402((1S,2R)-N-benzyl-1-(3,4-dichlorophenyl)-N-methyl-2...)
Affinity DataKi:  6.10nMAssay Description:Displacement of [3H]Lu AE93103 from human NK3 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50337397((1S,2R)-2-((4-acetamido-4-phenylpiperidin-1-yl)met...)
Affinity DataKi:  7.30nMAssay Description:Displacement of [3H]Lu AE93103 from human NK3 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50337413((1S,2R)-1-(3,4-dichlorophenyl)-N-(4-fluorobenzyl)-...)
Affinity DataKi:  7.30nMAssay Description:Displacement of [3H]Lu AE93103 from human NK3 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50337433(CHEMBL1681797 | rac-2-((4-acetamido-4-phenylpiperi...)
Affinity DataKi:  7.5nMAssay Description:Displacement of [3H]Lu AE93103 from human NK3 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50337415((1S,2R)-1-(3,4-dichlorophenyl)-2-((4-(N,N-dimethyl...)
Affinity DataKi:  7.60nMAssay Description:Displacement of [3H]Lu AE93103 from human NK3 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50337408((1S,2R)-N-benzyl-1-(3,4-dichlorophenyl)-N-methyl-2...)
Affinity DataKi:  7.80nMAssay Description:Displacement of [3H]Lu AE93103 from human NK3 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Hacettepe University

Curated by ChEMBL
LigandPNGBDBM50557331(CHEMBL4740141)
Affinity DataKi:  8nMAssay Description:Inhibition of recombinant human MAO-A expressed in baculovirus infected BTI insect cells using p-tyramine as substrate incubated for 30 mins by Ample...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Hacettepe University

Curated by ChEMBL
LigandPNGBDBM50557340(CHEMBL4778941)
Affinity DataKi:  8nMAssay Description:Inhibition of recombinant human MAO-A expressed in baculovirus infected BTI insect cells using p-tyramine as substrate incubated for 30 mins by Ample...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50337417((1S,2R)-2-((4-(2-(azepan-1-yl)acetyl)piperazin-1-y...)
Affinity DataKi:  8.70nMAssay Description:Displacement of [3H]Lu AE93103 from human NK3 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Hacettepe University

Curated by ChEMBL
LigandPNGBDBM50557332(CHEMBL4783604)
Affinity DataKi:  9nMAssay Description:Inhibition of recombinant human MAO-A expressed in baculovirus infected BTI insect cells using p-tyramine as substrate incubated for 30 mins by Ample...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Hacettepe University

Curated by ChEMBL
LigandPNGBDBM50557346(CHEMBL4763998)
Affinity DataKi:  9nMAssay Description:Inhibition of recombinant human MAO-A expressed in baculovirus infected BTI insect cells using p-tyramine as substrate incubated for 30 mins by Ample...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
University of Washington

Curated by PDSP Ki Database
LigandPNGBDBM22869(6-chloro-10-(4-methylpiperazin-1-yl)-2,9-diazatric...)
Affinity DataKi:  9.5nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Hacettepe University

Curated by ChEMBL
LigandPNGBDBM50557367(CHEMBL4753849)
Affinity DataKi:  10nMAssay Description:Inhibition of recombinant human MAO-A expressed in baculovirus infected BTI insect cells using p-tyramine as substrate incubated for 30 mins by Ample...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
University of Washington

Curated by PDSP Ki Database
LigandPNGBDBM82479(CAS_132539-06-1 | NSC_4585 | OLANZAPINE | USRE4934...)
Affinity DataKi:  10nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50337432(CHEMBL1682635 | rac-2-((4-acetamido-4-phenylpiperi...)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]Lu AE93103 from human NK3 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
University of Washington

Curated by PDSP Ki Database
LigandPNGBDBM84945(CAS_122265 | ICI 169,369 | NSC_122265)
Affinity DataKi:  11nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Hacettepe University

Curated by ChEMBL
LigandPNGBDBM50557365(CHEMBL4751649)
Affinity DataKi:  11nMAssay Description:Inhibition of recombinant human MAO-A expressed in baculovirus infected BTI insect cells using p-tyramine as substrate incubated for 30 mins by Ample...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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