Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
University of Washington
Curated by PDSP Ki Database
University of Washington
Curated by PDSP Ki Database
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Hacettepe University
Curated by ChEMBL
Hacettepe University
Curated by ChEMBL
Affinity DataKi: 0.900nMAssay Description:Competitive inhibition of MAOB in rat liver homogenate by spectrophotometricallyMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Hacettepe University
Curated by ChEMBL
Hacettepe University
Curated by ChEMBL
Affinity DataKi: 0.960nMAssay Description:Competitive inhibition of MAOB in rat liver homogenate by spectrophotometricallyMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Hacettepe University
Curated by ChEMBL
Hacettepe University
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Inhibition of recombinant human MAO-A expressed in baculovirus infected BTI insect cells using p-tyramine as substrate incubated for 30 mins by Ample...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Hacettepe University
Curated by ChEMBL
Hacettepe University
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Inhibition of recombinant human MAO-A expressed in baculovirus infected BTI insect cells using p-tyramine as substrate incubated for 30 mins by Ample...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Hacettepe University
Curated by ChEMBL
Hacettepe University
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Inhibition of recombinant human MAO-A expressed in baculovirus infected BTI insect cells using p-tyramine as substrate incubated for 30 mins by Ample...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Hacettepe University
Curated by ChEMBL
Hacettepe University
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Inhibition of recombinant human MAO-A expressed in baculovirus infected BTI insect cells using p-tyramine as substrate incubated for 30 mins by Ample...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Hacettepe University
Curated by ChEMBL
Hacettepe University
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Inhibition of recombinant human MAO-A expressed in baculovirus infected BTI insect cells using p-tyramine as substrate incubated for 30 mins by Ample...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Hacettepe University
Curated by ChEMBL
Hacettepe University
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Inhibition of recombinant human MAO-A expressed in baculovirus infected BTI insect cells using p-tyramine as substrate incubated for 30 mins by Ample...More data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Displacement of [3H]Lu AE93103 from human NK3 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Displacement of [3H]Lu AE93103 from human NK3 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
University of Washington
Curated by PDSP Ki Database
University of Washington
Curated by PDSP Ki Database
Affinity DataKi: 1.90nMAssay Description:Displacement of [3H]Lu AE93103 from human NK3 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
University of Washington
Curated by PDSP Ki Database
University of Washington
Curated by PDSP Ki Database
Affinity DataKi: 2.80nMAssay Description:Displacement of [3H]Lu AE93103 from human NK3 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.30nMAssay Description:Displacement of [3H]Lu AE93103 from human NK3 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.60nMAssay Description:Displacement of [3H]Lu AE93103 from human NK3 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.70nMAssay Description:Displacement of [3H]Lu AE93103 from human NK3 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Hacettepe University
Curated by ChEMBL
Hacettepe University
Curated by ChEMBL
Affinity DataKi: 4nMAssay Description:Inhibition of recombinant human MAO-A expressed in baculovirus infected BTI insect cells using p-tyramine as substrate incubated for 30 mins by Ample...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Hacettepe University
Curated by ChEMBL
Hacettepe University
Curated by ChEMBL
Affinity DataKi: 4nMAssay Description:Inhibition of recombinant human MAO-A expressed in baculovirus infected BTI insect cells using p-tyramine as substrate incubated for 30 mins by Ample...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Hacettepe University
Curated by ChEMBL
Hacettepe University
Curated by ChEMBL
Affinity DataKi: 4nMAssay Description:Inhibition of recombinant human MAO-A expressed in baculovirus infected BTI insect cells using p-tyramine as substrate incubated for 30 mins by Ample...More data for this Ligand-Target Pair
Affinity DataKi: 4.20nMAssay Description:Displacement of [3H]Lu AE93103 from human NK3 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Hacettepe University
Curated by ChEMBL
Hacettepe University
Curated by ChEMBL
Affinity DataKi: 4.22nMAssay Description:Competitive inhibition of MAOA in rat liver homogenate by spectrophotometricallyMore data for this Ligand-Target Pair
Affinity DataKi: 4.60nMAssay Description:Displacement of [3H]Lu AE93103 from human NK3 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Hacettepe University
Curated by ChEMBL
Hacettepe University
Curated by ChEMBL
Affinity DataKi: 5nMAssay Description:Inhibition of recombinant human MAO-B expressed in baculovirus infected BTI insect cells using p-tyramine as substrate incubated for 30 mins by Ample...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Hacettepe University
Curated by ChEMBL
Hacettepe University
Curated by ChEMBL
Affinity DataKi: 5nMAssay Description:Inhibition of recombinant human MAO-A expressed in baculovirus infected BTI insect cells using p-tyramine as substrate incubated for 30 mins by Ample...More data for this Ligand-Target Pair
Affinity DataKi: 5.30nMAssay Description:Displacement of [3H]Lu AE93103 from human NK3 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Hacettepe University
Curated by ChEMBL
Hacettepe University
Curated by ChEMBL
Affinity DataKi: 5.53nMAssay Description:Competitive inhibition of MAOA in rat liver homogenate by spectrophotometricallyMore data for this Ligand-Target Pair
Affinity DataKi: 5.60nMAssay Description:Displacement of [3H]Lu AE93103 from human NK3 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5.80nMAssay Description:Displacement of [3H]Lu AE93103 from human NK3 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5.80nMAssay Description:Displacement of [3H]Lu AE93103 from human NK3 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5.90nMAssay Description:Displacement of [3H]Lu AE93103 from human NK3 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5.90nMAssay Description:Displacement of [3H]Lu AE93103 from human NK3 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 6.10nMAssay Description:Displacement of [3H]Lu AE93103 from human NK3 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 7.30nMAssay Description:Displacement of [3H]Lu AE93103 from human NK3 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 7.30nMAssay Description:Displacement of [3H]Lu AE93103 from human NK3 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 7.5nMAssay Description:Displacement of [3H]Lu AE93103 from human NK3 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 7.60nMAssay Description:Displacement of [3H]Lu AE93103 from human NK3 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 7.80nMAssay Description:Displacement of [3H]Lu AE93103 from human NK3 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Hacettepe University
Curated by ChEMBL
Hacettepe University
Curated by ChEMBL
Affinity DataKi: 8nMAssay Description:Inhibition of recombinant human MAO-A expressed in baculovirus infected BTI insect cells using p-tyramine as substrate incubated for 30 mins by Ample...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Hacettepe University
Curated by ChEMBL
Hacettepe University
Curated by ChEMBL
Affinity DataKi: 8nMAssay Description:Inhibition of recombinant human MAO-A expressed in baculovirus infected BTI insect cells using p-tyramine as substrate incubated for 30 mins by Ample...More data for this Ligand-Target Pair
Affinity DataKi: 8.70nMAssay Description:Displacement of [3H]Lu AE93103 from human NK3 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Hacettepe University
Curated by ChEMBL
Hacettepe University
Curated by ChEMBL
Affinity DataKi: 9nMAssay Description:Inhibition of recombinant human MAO-A expressed in baculovirus infected BTI insect cells using p-tyramine as substrate incubated for 30 mins by Ample...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Hacettepe University
Curated by ChEMBL
Hacettepe University
Curated by ChEMBL
Affinity DataKi: 9nMAssay Description:Inhibition of recombinant human MAO-A expressed in baculovirus infected BTI insect cells using p-tyramine as substrate incubated for 30 mins by Ample...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
University of Washington
Curated by PDSP Ki Database
University of Washington
Curated by PDSP Ki Database
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Hacettepe University
Curated by ChEMBL
Hacettepe University
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Inhibition of recombinant human MAO-A expressed in baculovirus infected BTI insect cells using p-tyramine as substrate incubated for 30 mins by Ample...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
University of Washington
Curated by PDSP Ki Database
University of Washington
Curated by PDSP Ki Database
Affinity DataKi: 11nMAssay Description:Displacement of [3H]Lu AE93103 from human NK3 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
University of Washington
Curated by PDSP Ki Database
University of Washington
Curated by PDSP Ki Database
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Hacettepe University
Curated by ChEMBL
Hacettepe University
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:Inhibition of recombinant human MAO-A expressed in baculovirus infected BTI insect cells using p-tyramine as substrate incubated for 30 mins by Ample...More data for this Ligand-Target Pair